FIORINO, FERDINANDO
FIORINO, FERDINANDO
DIPARTIMENTO DI FARMACIA
A convenient synthesis of N-Fmoc-N,N'-bis-Boc-7-guanyl-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid (Fmoc-N,N'-bis-Boc-7-guanyl-Tic-OH, GTIC).
2001 Santagada, Vincenzo; Fiorino, Ferdinando; Severino, Beatrice; Salvadori, S; Lazarus L., H; Bryant S., D; Caliendo, Giuseppe
Preparation and local anesthetic activity of benzotriazinone and benzoyltriazole derivatives.
1999 Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; Santagada, Vincenzo; Meli, Rosaria; MATTACE RASO, Giuseppina; Zanesco, A; De Nucci, G.
X-ray Structural Analysis of Ethyl [2,2-dimethyl-6-(D2-thiazolin-2-yl)-4H-1,4-benzoxazin-3-one-4-yl]butyrate.
1998 Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; Albrizio, Stefania; Giordano, M.; Santagada, Vincenzo; Santini, Antonello
A convenient synthesis by microwave irradiation of an active metabolite (EXP-3174) of losartan.
2003 Santagada, Vincenzo; Fiorino, Ferdinando; Perissutti, Elisa; Severino, Beatrice; Terracciano, Sara; Cleber Evandro, Teixeira; Caliendo, Giuseppe
Design of inhibitors for human tissue kallikrein using non-natural aromatic and basic amino acids.
2002 Daniel C., Pimenta; Robson L., Melo; Caliendo, Giuseppe; Santagada, Vincenzo; Fiorino, Ferdinando; Severino, Beatrice; Gilberto De, Nucci; Luiz, Juliano; Maria, A. J. u. l. i. a. n. o.
Identification of a pepducin acting as S1P3 receptor antagonist
2013 Severino, Beatrice; Giuseppina Maria Incisivo, ; Fiorino, Ferdinando; Bertolino, Antonio; Frecentese, Francesco; Barbato, Francesco; Serena, Manganelli; Giada, Maggioni; Capasso, Domenica; Caliendo, Giuseppe; Santagada, Vincenzo; Sorrentino, Raffaella; Roviezzo, Fiorentina; Perissutti, Elisa
Microwave-enhanced solution coupling of the a,a-dialkyl amino acid, Aib
2001 Santagada, Vincenzo; Fiorino, Ferdinando; Perissutti, Elisa; Severino, Beatrice; De Filippis, V; Vivenzio, B; Caliendo, Giuseppe
Synthesis, Pharmacological Evaluation, and Molecular Modeling Studies of Novel Peptidic CAAX Analogues as Farnesyl-Protein-Transferase Inhibitors
2006 Santagada, Vincenzo; Caliendo, Giuseppe; Severino, Beatrice; Lavecchia, Antonio; Perissutti, Elisa; Fiorino, Ferdinando; Zampella, Angela; Sepe, Valentina; Califano, D.; Santelli, G.; Novellino, Ettore
Synthesis and Binding Affinities for 5-HT1A, 5-HT2A and 5-HT2C receptors of a series of 1- and 2-(4-arylpiperazinylalkyl)-4-(benzoyl)-1,2,3-triazole derivatives.
1999 Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; Santagada, Vincenzo; Albrizio, Stefania; Spadola, L.; Bruni, G.; Romeo, M. R.
Synthesis by microwave irradiation and binding properties of novel 5-HT1A receptor ligands.
2001 Caliendo, Giuseppe; Fiorino, Ferdinando; Perissutti, Elisa; Severino, Beatrice; Gessi, S; Cattabriga, E; Borea, P. A.; Santagada, Vincenzo
Phenol derived CVFM analogs inhibitors of ras farnesyl transferase possessing cellular in vitro activity.
1998 Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; Ramunno, Anna; Santagada, Vincenzo; Albrizio, Stefania; Califano, D.; Giuliano, A.; Santelli, G.
A convenient synthesis by microwave heating and pharmacological evaluation of novel benzoyltriazole and saccharine derivatives as 5-HT1A receptor ligands.
2002 Caliendo, Giuseppe; Fiorino, Ferdinando; Perissutti, Elisa; Severino, Beatrice; Daniela, Scolaro; Stefania, Gessi; Elena, Cattabriga; Pier Andrea, Borea; Santagada, Vincenzo
Synthesis and in vitro activities of NK-1 antagonists derived from L-Triptophan.
1997 Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; Santagada, Vincenzo; Calignano, Antonio; Mancuso, F.; Albrizio, Stefania
Microwave enhanced solution synthesis of 1,4-benzodiazepin-5-ones.
2001 Santagada, Vincenzo; Perissutti, Elisa; Fiorino, Ferdinando; Vivenzio, B; Caliendo, Giuseppe
Inhibition of rat vas deferens contractions by flavonoids in-vitro
2006 Capasso, Raffaele; Fiorino, Ferdinando; V., Ascione; Frecentese, Francesco; Borrelli, Francesca
Synthesis and vasorelaxant activity of new 1,4-benzoxazine derivatives potassium channel openers.
2002 Caliendo, Giuseppe; Perissutti, Elisa; Santagada, Vincenzo; Fiorino, Ferdinando; Severino, Beatrice; D'EMMANUELE DI VILLA BIANCA, Roberta; Laura, Lippolis; Aldo, Pinto; Sorrentino, Raffaella
Synthesis and biological activity of pseudopeptides inhibitors of Ras farnesyl transferase containing unconventional amino acids.
1999 Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; De Luca, S; Giuliano, A; Santelli, G; Califano, D; Severino, Beatrice; Santagada, Vincenzo
Synthesis, Biological Evaluation and Docking Studies of PAR2-AP Derived Pseudopeptides as Inhibitors of Kallikrein 5 and 6
2015 Severino, Beatrice; Fiorino, Ferdinando; Corvino, Angela; Caliendo, Giuseppe; Santagada, Vincenzo; Diego Magno, Assis; Juliana R., Oliveira; Luiz, Juliano; Serena, Manganelli; Emilio, Benfenati; Frecentese, Francesco; Perissutti, Elisa; Maria Aparecida, Juliano
Thrombin and PAR-1 activating peptide increase iNOS expression in cytokine-stimulated C6 glioma cells.
2001 Meli, Rosaria; MATTACE RASO, Giuseppina; Cicala, Carla; Esposito, Emanuela; Fiorino, Ferdinando; Cirino, Giuseppe
A convenient strategy of dimerization by microwave heating and using 2,5-diketopiperazine as scaffold.
2003 Santagada, Vincenzo; Fiorino, Ferdinando; Perissutti, Elisa; Severino, Beatrice; Terracciano, Sara; Cirino, Giuseppe; Caliendo, Giuseppe
Titolo | Tipologia | Data di pubblicazione | Autore(i) | File |
---|---|---|---|---|
A convenient synthesis of N-Fmoc-N,N'-bis-Boc-7-guanyl-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid (Fmoc-N,N'-bis-Boc-7-guanyl-Tic-OH, GTIC). | 1.1 Articolo in rivista | 2001 | Santagada, Vincenzo; Fiorino, Ferdinando; Severino, Beatrice; Salvadori, S; Lazarus L., H; Bryant S., D; Caliendo, Giuseppe | |
Preparation and local anesthetic activity of benzotriazinone and benzoyltriazole derivatives. | 1.1 Articolo in rivista | 1999 | Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; Santagada, Vincenzo; Meli, Rosaria; MATTACE RASO, Giuseppina; Zanesco, A; De Nucci, G. | |
X-ray Structural Analysis of Ethyl [2,2-dimethyl-6-(D2-thiazolin-2-yl)-4H-1,4-benzoxazin-3-one-4-yl]butyrate. | 1.1 Articolo in rivista | 1998 | Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; Albrizio, Stefania; Giordano, M.; Santagada, Vincenzo; Santini, Antonello | |
A convenient synthesis by microwave irradiation of an active metabolite (EXP-3174) of losartan. | 1.1 Articolo in rivista | 2003 | Santagada, Vincenzo; Fiorino, Ferdinando; Perissutti, Elisa; Severino, Beatrice; Terracciano, Sara; Cleber Evandro, Teixeira; Caliendo, Giuseppe | |
Design of inhibitors for human tissue kallikrein using non-natural aromatic and basic amino acids. | 1.1 Articolo in rivista | 2002 | Daniel C., Pimenta; Robson L., Melo; Caliendo, Giuseppe; Santagada, Vincenzo; Fiorino, Ferdinando; Severino, Beatrice; Gilberto De, Nucci; Luiz, Juliano; Maria, A. J. u. l. i. a. n. o. | |
Identification of a pepducin acting as S1P3 receptor antagonist | 1.1 Articolo in rivista | 2013 | Severino, Beatrice; Giuseppina Maria Incisivo, ; Fiorino, Ferdinando; Bertolino, Antonio; Frecentese, Francesco; Barbato, Francesco; Serena, Manganelli; Giada, Maggioni; Capasso, Domenica; Caliendo, Giuseppe; Santagada, Vincenzo; Sorrentino, Raffaella; Roviezzo, Fiorentina; Perissutti, Elisa | |
Microwave-enhanced solution coupling of the a,a-dialkyl amino acid, Aib | 1.1 Articolo in rivista | 2001 | Santagada, Vincenzo; Fiorino, Ferdinando; Perissutti, Elisa; Severino, Beatrice; De Filippis, V; Vivenzio, B; Caliendo, Giuseppe | |
Synthesis, Pharmacological Evaluation, and Molecular Modeling Studies of Novel Peptidic CAAX Analogues as Farnesyl-Protein-Transferase Inhibitors | 1.1 Articolo in rivista | 2006 | Santagada, Vincenzo; Caliendo, Giuseppe; Severino, Beatrice; Lavecchia, Antonio; Perissutti, Elisa; Fiorino, Ferdinando; Zampella, Angela; Sepe, Valentina; Califano, D.; Santelli, G.; Novellino, Ettore | |
Synthesis and Binding Affinities for 5-HT1A, 5-HT2A and 5-HT2C receptors of a series of 1- and 2-(4-arylpiperazinylalkyl)-4-(benzoyl)-1,2,3-triazole derivatives. | 1.1 Articolo in rivista | 1999 | Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; Santagada, Vincenzo; Albrizio, Stefania; Spadola, L.; Bruni, G.; Romeo, M. R. | |
Synthesis by microwave irradiation and binding properties of novel 5-HT1A receptor ligands. | 1.1 Articolo in rivista | 2001 | Caliendo, Giuseppe; Fiorino, Ferdinando; Perissutti, Elisa; Severino, Beatrice; Gessi, S; Cattabriga, E; Borea, P. A.; Santagada, Vincenzo | |
Phenol derived CVFM analogs inhibitors of ras farnesyl transferase possessing cellular in vitro activity. | 1.1 Articolo in rivista | 1998 | Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; Ramunno, Anna; Santagada, Vincenzo; Albrizio, Stefania; Califano, D.; Giuliano, A.; Santelli, G. | |
A convenient synthesis by microwave heating and pharmacological evaluation of novel benzoyltriazole and saccharine derivatives as 5-HT1A receptor ligands. | 1.1 Articolo in rivista | 2002 | Caliendo, Giuseppe; Fiorino, Ferdinando; Perissutti, Elisa; Severino, Beatrice; Daniela, Scolaro; Stefania, Gessi; Elena, Cattabriga; Pier Andrea, Borea; Santagada, Vincenzo | |
Synthesis and in vitro activities of NK-1 antagonists derived from L-Triptophan. | 1.1 Articolo in rivista | 1997 | Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; Santagada, Vincenzo; Calignano, Antonio; Mancuso, F.; Albrizio, Stefania | |
Microwave enhanced solution synthesis of 1,4-benzodiazepin-5-ones. | 1.1 Articolo in rivista | 2001 | Santagada, Vincenzo; Perissutti, Elisa; Fiorino, Ferdinando; Vivenzio, B; Caliendo, Giuseppe | |
Inhibition of rat vas deferens contractions by flavonoids in-vitro | 1.1 Articolo in rivista | 2006 | Capasso, Raffaele; Fiorino, Ferdinando; V., Ascione; Frecentese, Francesco; Borrelli, Francesca | |
Synthesis and vasorelaxant activity of new 1,4-benzoxazine derivatives potassium channel openers. | 1.1 Articolo in rivista | 2002 | Caliendo, Giuseppe; Perissutti, Elisa; Santagada, Vincenzo; Fiorino, Ferdinando; Severino, Beatrice; D'EMMANUELE DI VILLA BIANCA, Roberta; Laura, Lippolis; Aldo, Pinto; Sorrentino, Raffaella | |
Synthesis and biological activity of pseudopeptides inhibitors of Ras farnesyl transferase containing unconventional amino acids. | 1.1 Articolo in rivista | 1999 | Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; De Luca, S; Giuliano, A; Santelli, G; Califano, D; Severino, Beatrice; Santagada, Vincenzo | |
Synthesis, Biological Evaluation and Docking Studies of PAR2-AP Derived Pseudopeptides as Inhibitors of Kallikrein 5 and 6 | 1.1 Articolo in rivista | 2015 | Severino, Beatrice; Fiorino, Ferdinando; Corvino, Angela; Caliendo, Giuseppe; Santagada, Vincenzo; Diego Magno, Assis; Juliana R., Oliveira; Luiz, Juliano; Serena, Manganelli; Emilio, Benfenati; Frecentese, Francesco; Perissutti, Elisa; Maria Aparecida, Juliano | |
Thrombin and PAR-1 activating peptide increase iNOS expression in cytokine-stimulated C6 glioma cells. | 1.1 Articolo in rivista | 2001 | Meli, Rosaria; MATTACE RASO, Giuseppina; Cicala, Carla; Esposito, Emanuela; Fiorino, Ferdinando; Cirino, Giuseppe | |
A convenient strategy of dimerization by microwave heating and using 2,5-diketopiperazine as scaffold. | 1.1 Articolo in rivista | 2003 | Santagada, Vincenzo; Fiorino, Ferdinando; Perissutti, Elisa; Severino, Beatrice; Terracciano, Sara; Cirino, Giuseppe; Caliendo, Giuseppe |