FIORINO, FERDINANDO
FIORINO, FERDINANDO
DIPARTIMENTO DI FARMACIA
Minimal structural requirements for agonist activity of PAR-2 activating peptides.
2002 Santagada, Vincenzo; Caliendo, Giuseppe; Severino, Beatrice; Perissutti, Elisa; Fiorino, Ferdinando; Cicala, Carla; De Filippis, V; Cirino, Giuseppe
Synthesis and biological activity of pseudopeptides inhibitors of Ras farnesyl transferase containing unconventional amino acids.
1999 Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; De Luca, S; Giuliano, A; Santelli, G; Califano, D; Severino, Beatrice; Santagada, Vincenzo
A convenient synthesis of N-Fmoc-N,N'-bis-Boc-7-guanyl-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid (Fmoc-N,N'-bis-Boc-7-guanyl-Tic-OH, GTIC).
2001 Santagada, Vincenzo; Fiorino, Ferdinando; Severino, Beatrice; Salvadori, S; Lazarus, L. H.; Bryant, S. D.; Caliendo, Giuseppe
Microwave enhanced solution synthesis of 1,4-benzodiazepin-5-ones.
2001 Santagada, Vincenzo; Perissutti, Elisa; Fiorino, Ferdinando; Vivenzio, B; Caliendo, Giuseppe
Synthesis of substituted benzamides as anti-inflammatory agents that inhibit preferentially cyclooxygenase 1 but do not cause gastric damage.
2001 Caliendo, Giuseppe; Santagada, Vincenzo; Perissutti, Elisa; Severino, Beatrice; Fiorino, Ferdinando; Warner, T. D.; Wallace, J. L.; Ifa, D. R.; Antunes, E; Cirino, Giuseppe; de Nucci, G.
Synthesis and Binding Affinities for 5-HT1A, 5-HT2A and 5-HT2C receptors of a series of 1- and 2-(4-arylpiperazinylalkyl)-4-(benzoyl)-1,2,3-triazole derivatives.
1999 Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; Santagada, Vincenzo; Albrizio, Stefania; Spadola, L.; Bruni, G.; Romeo, M. R.
A convenient strategy of dimerization by microwave heating and using 2,5-diketopiperazine as scaffold.
2003 Santagada, Vincenzo; Fiorino, Ferdinando; Perissutti, Elisa; Severino, Beatrice; Terracciano, Sara; Cirino, Giuseppe; Caliendo, Giuseppe
Synthesis, Pharmacological Evaluation, and Molecular Modeling Studies of Novel Peptidic CAAX Analogues as Farnesyl-Protein-Transferase Inhibitors
2006 Santagada, Vincenzo; Caliendo, Giuseppe; Severino, Beatrice; Lavecchia, Antonio; Perissutti, Elisa; Fiorino, Ferdinando; Zampella, Angela; Sepe, Valentina; Califano, D.; Santelli, G.; Novellino, Ettore
Preparation and local anesthetic activity of benzotriazinone and benzoyltriazole derivatives.
1999 Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; Santagada, Vincenzo; Meli, Rosaria; MATTACE RASO, Giuseppina; Zanesco, A; De Nucci, G.
New Potent 5-HT2A Receptor Ligands Containing a N'-Cyanopicolinamidine Nucleus: Synthesis and In Vitro Pharmacological Evaluation
2012 Fiorino, Ferdinando; Severino, Beatrice; Magli, Elisa; Perissutti, Elisa; Frecentese, Francesco; A., Esposito; Incisivo, GIUSEPPINA MARIA; Ciano, Antonio; P., Massarelli; C., Nencini; Santagada, Vincenzo; Caliendo, Giuseppe
Synthesis of 1-naphthylpiperazine derivatives as serotoninergic ligands and their evaluation as antiproliferative agents.
2011 Fiorino, Ferdinando; Magli, Elisa; Perissutti, Elisa; Severino, Beatrice; Frecentese, Francesco; Esposito, A.; De Angelis, F.; Incisivo, GIUSEPPINA MARIA; Massarelli, P.; Nencini, C.; Di Gennaro, E.; Budillon, A.; Di Cintio, A.; Santagada, Vincenzo; Caliendo, Giuseppe
Synthesis of benzamide derivatives and their evaluation as antiprion agents
2012 Fiorino, Ferdinando; M., Eiden; A., Giese; Severino, Beatrice; A., Esposito; M. H., Groschup; Perissutti, Elisa; Magli, Elisa; Incisivo, GIUSEPPINA MARIA; Ciano, Antonio; Frecentese, Francesco; H. A., Kretzschmar; J., Wagner; Santagada, Vincenzo; Caliendo, Giuseppe
A convenient synthesis by microwave irradiation of an active metabolite (EXP-3174) of losartan.
2003 Santagada, Vincenzo; Fiorino, Ferdinando; Perissutti, Elisa; Severino, Beatrice; Terracciano, Sara; Cleber Evandro, Teixeira; Caliendo, Giuseppe
Synthesis by microwave irradiation and binding properties of novel 5-HT1A receptor ligands.
2001 Caliendo, Giuseppe; Fiorino, Ferdinando; Perissutti, Elisa; Severino, Beatrice; Gessi, S; Cattabriga, E; Borea, P. A.; Santagada, Vincenzo
Microwave-enhanced solution coupling of the a,a-dialkyl amino acid, Aib
2001 Santagada, Vincenzo; Fiorino, Ferdinando; Perissutti, Elisa; Severino, Beatrice; De Filippis, V; Vivenzio, B; Caliendo, Giuseppe
Inhibition of rat vas deferens contractions by flavonoids in-vitro
2006 Capasso, Raffaele; Fiorino, Ferdinando; V., Ascione; Frecentese, Francesco; Borrelli, Francesca
Design of inhibitors for human tissue kallikrein using non-natural aromatic and basic amino acids.
2002 Daniel C., Pimenta; Robson L., Melo; Caliendo, Giuseppe; Santagada, Vincenzo; Fiorino, Ferdinando; Severino, Beatrice; Gilberto De, Nucci; Luiz, Juliano; Maria, A. J. u. l. i. a. n. o.
Thrombin and PAR-1 activating peptide increase iNOS expression in cytokine-stimulated C6 glioma cells.
2001 Meli, Rosaria; MATTACE RASO, Giuseppina; Cicala, Carla; Esposito, Emanuela; Fiorino, Ferdinando; Cirino, Giuseppe
Synthesis of new 1,2,3-benzotriazin-4-one-arylpiperazine derivatives as 5-HT1A serotonin receptor ligands.
2000 Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; Santagada, Vincenzo; Severino, Beatrice; Bruni, G; Romeo, M. R.
Synthesis and in vitro activities of NK-1 antagonists derived from L-Triptophan.
1997 Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; Santagada, Vincenzo; Calignano, Antonio; Mancuso, F.; Albrizio, Stefania
Titolo | Tipologia | Data di pubblicazione | Autore(i) | File |
---|---|---|---|---|
Minimal structural requirements for agonist activity of PAR-2 activating peptides. | 1.1 Articolo in rivista | 2002 | Santagada, Vincenzo; Caliendo, Giuseppe; Severino, Beatrice; Perissutti, Elisa; Fiorino, Ferdinando; Cicala, Carla; De Filippis, V; Cirino, Giuseppe | |
Synthesis and biological activity of pseudopeptides inhibitors of Ras farnesyl transferase containing unconventional amino acids. | 1.1 Articolo in rivista | 1999 | Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; De Luca, S; Giuliano, A; Santelli, G; Califano, D; Severino, Beatrice; Santagada, Vincenzo | |
A convenient synthesis of N-Fmoc-N,N'-bis-Boc-7-guanyl-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid (Fmoc-N,N'-bis-Boc-7-guanyl-Tic-OH, GTIC). | 1.1 Articolo in rivista | 2001 | Santagada, Vincenzo; Fiorino, Ferdinando; Severino, Beatrice; Salvadori, S; Lazarus, L. H.; Bryant, S. D.; Caliendo, Giuseppe | |
Microwave enhanced solution synthesis of 1,4-benzodiazepin-5-ones. | 1.1 Articolo in rivista | 2001 | Santagada, Vincenzo; Perissutti, Elisa; Fiorino, Ferdinando; Vivenzio, B; Caliendo, Giuseppe | |
Synthesis of substituted benzamides as anti-inflammatory agents that inhibit preferentially cyclooxygenase 1 but do not cause gastric damage. | 1.1 Articolo in rivista | 2001 | Caliendo, Giuseppe; Santagada, Vincenzo; Perissutti, Elisa; Severino, Beatrice; Fiorino, Ferdinando; Warner, T. D.; Wallace, J. L.; Ifa, D. R.; Antunes, E; Cirino, Giuseppe; de Nucci, G. | |
Synthesis and Binding Affinities for 5-HT1A, 5-HT2A and 5-HT2C receptors of a series of 1- and 2-(4-arylpiperazinylalkyl)-4-(benzoyl)-1,2,3-triazole derivatives. | 1.1 Articolo in rivista | 1999 | Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; Santagada, Vincenzo; Albrizio, Stefania; Spadola, L.; Bruni, G.; Romeo, M. R. | |
A convenient strategy of dimerization by microwave heating and using 2,5-diketopiperazine as scaffold. | 1.1 Articolo in rivista | 2003 | Santagada, Vincenzo; Fiorino, Ferdinando; Perissutti, Elisa; Severino, Beatrice; Terracciano, Sara; Cirino, Giuseppe; Caliendo, Giuseppe | |
Synthesis, Pharmacological Evaluation, and Molecular Modeling Studies of Novel Peptidic CAAX Analogues as Farnesyl-Protein-Transferase Inhibitors | 1.1 Articolo in rivista | 2006 | Santagada, Vincenzo; Caliendo, Giuseppe; Severino, Beatrice; Lavecchia, Antonio; Perissutti, Elisa; Fiorino, Ferdinando; Zampella, Angela; Sepe, Valentina; Califano, D.; Santelli, G.; Novellino, Ettore | |
Preparation and local anesthetic activity of benzotriazinone and benzoyltriazole derivatives. | 1.1 Articolo in rivista | 1999 | Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; Santagada, Vincenzo; Meli, Rosaria; MATTACE RASO, Giuseppina; Zanesco, A; De Nucci, G. | |
New Potent 5-HT2A Receptor Ligands Containing a N'-Cyanopicolinamidine Nucleus: Synthesis and In Vitro Pharmacological Evaluation | 1.1 Articolo in rivista | 2012 | Fiorino, Ferdinando; Severino, Beatrice; Magli, Elisa; Perissutti, Elisa; Frecentese, Francesco; A., Esposito; Incisivo, GIUSEPPINA MARIA; Ciano, Antonio; P., Massarelli; C., Nencini; Santagada, Vincenzo; Caliendo, Giuseppe | |
Synthesis of 1-naphthylpiperazine derivatives as serotoninergic ligands and their evaluation as antiproliferative agents. | 1.1 Articolo in rivista | 2011 | Fiorino, Ferdinando; Magli, Elisa; Perissutti, Elisa; Severino, Beatrice; Frecentese, Francesco; Esposito, A.; De Angelis, F.; Incisivo, GIUSEPPINA MARIA; Massarelli, P.; Nencini, C.; Di Gennaro, E.; Budillon, A.; Di Cintio, A.; Santagada, Vincenzo; Caliendo, Giuseppe | |
Synthesis of benzamide derivatives and their evaluation as antiprion agents | 1.1 Articolo in rivista | 2012 | Fiorino, Ferdinando; M., Eiden; A., Giese; Severino, Beatrice; A., Esposito; M. H., Groschup; Perissutti, Elisa; Magli, Elisa; Incisivo, GIUSEPPINA MARIA; Ciano, Antonio; Frecentese, Francesco; H. A., Kretzschmar; J., Wagner; Santagada, Vincenzo; Caliendo, Giuseppe | |
A convenient synthesis by microwave irradiation of an active metabolite (EXP-3174) of losartan. | 1.1 Articolo in rivista | 2003 | Santagada, Vincenzo; Fiorino, Ferdinando; Perissutti, Elisa; Severino, Beatrice; Terracciano, Sara; Cleber Evandro, Teixeira; Caliendo, Giuseppe | |
Synthesis by microwave irradiation and binding properties of novel 5-HT1A receptor ligands. | 1.1 Articolo in rivista | 2001 | Caliendo, Giuseppe; Fiorino, Ferdinando; Perissutti, Elisa; Severino, Beatrice; Gessi, S; Cattabriga, E; Borea, P. A.; Santagada, Vincenzo | |
Microwave-enhanced solution coupling of the a,a-dialkyl amino acid, Aib | 1.1 Articolo in rivista | 2001 | Santagada, Vincenzo; Fiorino, Ferdinando; Perissutti, Elisa; Severino, Beatrice; De Filippis, V; Vivenzio, B; Caliendo, Giuseppe | |
Inhibition of rat vas deferens contractions by flavonoids in-vitro | 1.1 Articolo in rivista | 2006 | Capasso, Raffaele; Fiorino, Ferdinando; V., Ascione; Frecentese, Francesco; Borrelli, Francesca | |
Design of inhibitors for human tissue kallikrein using non-natural aromatic and basic amino acids. | 1.1 Articolo in rivista | 2002 | Daniel C., Pimenta; Robson L., Melo; Caliendo, Giuseppe; Santagada, Vincenzo; Fiorino, Ferdinando; Severino, Beatrice; Gilberto De, Nucci; Luiz, Juliano; Maria, A. J. u. l. i. a. n. o. | |
Thrombin and PAR-1 activating peptide increase iNOS expression in cytokine-stimulated C6 glioma cells. | 1.1 Articolo in rivista | 2001 | Meli, Rosaria; MATTACE RASO, Giuseppina; Cicala, Carla; Esposito, Emanuela; Fiorino, Ferdinando; Cirino, Giuseppe | |
Synthesis of new 1,2,3-benzotriazin-4-one-arylpiperazine derivatives as 5-HT1A serotonin receptor ligands. | 1.1 Articolo in rivista | 2000 | Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; Santagada, Vincenzo; Severino, Beatrice; Bruni, G; Romeo, M. R. | |
Synthesis and in vitro activities of NK-1 antagonists derived from L-Triptophan. | 1.1 Articolo in rivista | 1997 | Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; Santagada, Vincenzo; Calignano, Antonio; Mancuso, F.; Albrizio, Stefania |