GRIECO, PAOLO
GRIECO, PAOLO
DIPARTIMENTO DI FARMACIA
Cyclic peptides acting as urotensin-II antagonists.
2005 Novellino, Ettore; Grieco, Paolo; Rovero, P.
D-Amino Acid Scan of g-Melanocyte-Stimulating hormone:importance of the Trp8
2000 Grieco, Paolo; Balse, P. M.; Weinberg, D.; Macneil, T.
" Molecular Modelingof the Urotensin-II receptor Complex"
2004 Grieco, Paolo; Lavecchia, A.; Campiglia, P.; Lama, T.; Rovero, P.; Carotenuto, Alfonso; Patacchini, R.; Maggi, C. A.; Novellino, Ettore
A structure – activity relationship study on position –2 of the Gas C-terminal peptide able to inhibit Gs activation by A2A adenosine receptor.
2003 Grieco, Paolo; Albrizio, Stefania; D’Ursi, A. M.; Giusti, L.; Mazzoni, M. R.; Novellino, E.; Rovero, P.
Unraveling the active conformation of urotensin II
2004 Carotenuto, Alfonso; Grieco, Paolo; Campiglia, Pietro; Novellino, Ettore; Ettore, Rovero; Paolo,
Phenol derived CVFM analogs inhibitors of ras farnesyl transferase possessing cellular in vitro activity.
1998 Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; Ramunno, Anna; Santagada, Vincenzo; Albrizio, Stefania; Califano, D.; Giuliano, A.; Santelli, G.
Synthesis and Binding Affinities for 5-HT1A, 5-HT2A and 5-HT2C receptors of a series of 1- and 2-(4-arylpiperazinylalkyl)-4-(benzoyl)-1,2,3-triazole derivatives.
1999 Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; Santagada, Vincenzo; Albrizio, Stefania; Spadola, L.; Bruni, G.; Romeo, M. R.
Structure-Activity Relationships of Novel Cyclic alpha-MSH/gamma-MSH Hybrid Analogues which Lead to Potent and Selective Ligands for the Human MC3R and Human MC5R
2003 Balse, Srinivasan; P., M.; Grieco, Paolo; P, Cai; M, Trivedi; D, Hruby; V., J.
Extensive Structure-Activity Studies of Lactam Derivatives of MT-II and SHU9119: Their activity and Selectivity at Human Melanocortin Receptors 3,4 and, 5.
2003 Grieco, Paolo; P, Balsesrinivasan; P, Han; G, Weinberg; D, Macnail; T, ; VAN DER, Ploeg; L. H. T, Hruby; V., J.
NMR analysis of synthetic peptides agonist to PTPRJ, a receptor-type protein tyrosine phosphatase with tumor suppressor activity
2011 Brancaccio, Diego; Carotenuto, Alfonso; Grieco, Paolo; Campiglia, P; Trapasso, F; Novellino, Ettore
Melanocortin type 3 receptor null mice are refractory to the inhibitory actions of a selective receptor agonist in experimental acute inflammation
2006 Getting, J. S.; Lam, C. W.; Chen, A. S.; Grieco, Paolo; Perretti, M.
New melanocortin peptides useful as medicament against Staphylococcus aureus, Candida albicans, Pseudomonas aeruginosa, Candida glabrata or Candida krusei
2010 Bonino, F.; Catania, A.; Grieco, Paolo; Novellino, Ettore
New dimensions in the design of potent and receptor selective melanotropin analogues
2000 Grieco, Paolo; Han, G.; Hruby, V. J.
Novel peptidomimetic as MMP2 inhibitors
2007 K., Kaia; P., Campiglia; GOMEZ MONTERREY, ISABEL MARIA; M., D'Ursi; Grieco, Paolo; Novellino, Ettore
Further structure-activity studies of lactam derivatives of MT-II and SHU-9119: Their activity and selectivity at human melanocortin receptors 3, 4, and 5.
2007 Grieco, Paolo; Cai, M.; Han, G.; Trivedi, D.; Campiglia, P.; Novellino, Ettore; Hruby, V. J.
Urokinase receptor activation by a novel interaction between connecting peptide region of Urokinase and αvβ5 Integrin Journal of Cell Science, 119, 3424-3434, 2006
2006 Franco, P; Vocca, I; Carriero, M. V; Alfano, D; Cito, L; Longanesi, Cattani; I, ; Grieco, Paolo; P, Ossowski; L, Stoppelli; M., P.
Substitution of Arginine with Proline and Proline Derivatives in MSH Leads to Selectivity for Human Melanocortin 4 Receptor (hMC4R)
2009 H., Qu; M., Cai; A. V., Mayorov; Grieco, Paolo; M., Zingsheim; D., Trivedi; V. J., Hruby
Spiro[(dihydropyrazin-2,5-dione)-6,3’-(2’,3’-dihydrothieno[2,3-b]naphtho-4’,9’-dione)]-Based Cytotoxic Agents: Structure-Activity Relationship Studies on the Substituent at N4-Position of the Diketopiperazine Domain
2008 GOMEZ MONTERREY, ISABEL MARIA; P., Campiglia; Carotenuto, Alfonso; P., Stiuso; A., Bertamino; M., Sala; C., Aaquino; Grieco, Paolo; S., Morello; Pinto, Antonio; P., Ianelli; Novellino, Ettore
Design, synthesis and Cytotoxic Evaluation of a New Series of 3-Substituted-spiro[(dihydropirazin-2,5-dione)-6,3’-(2’,3’-dihydrothieno[2,3-b]naphtho-4’,9’-dione)] Derivatives
2007 GOMEZ MONTERREY, ISABEL MARIA; P., Campiglia; Carotenuto, Alfonso; D., Califano; C., Pisano; L., Vesci; T., Lama; A., Bertamino; M., Sala; A., MAZZELLA di BOSCO; Grieco, Paolo; Novellino, Ettore
Design and Synthesis of Spirotryprostatin-inspired Diketopiperazine Systemsfrom Prolyl Spirooxoindolethiazolidine Derivatives
2010 Bertamino, Alessia; Aquino, Claudio; M., Sala; N., de Simone; C. A., Mattia; L., Erra; S., Musella; P., Iannelli; Carotenuto, Alfonso; Grieco, Paolo; Novellino, Ettore; P., Campiglia; GOMEZ MONTERREY, ISABEL MARIA
| Titolo | Tipologia | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|---|
| Cyclic peptides acting as urotensin-II antagonists. | 6.1 Brevetto | 2005 | Novellino, Ettore; Grieco, Paolo; Rovero, P. | |
| D-Amino Acid Scan of g-Melanocyte-Stimulating hormone:importance of the Trp8 | 1.1 Articolo in rivista | 2000 | Grieco, Paolo; Balse, P. M.; Weinberg, D.; Macneil, T. | |
| " Molecular Modelingof the Urotensin-II receptor Complex" | 4.1 Articoli in Atti di convegno | 2004 | Grieco, Paolo; Lavecchia, A.; Campiglia, P.; Lama, T.; Rovero, P.; Carotenuto, Alfonso; Patacchini, R.; Maggi, C. A.; Novellino, Ettore | |
| A structure – activity relationship study on position –2 of the Gas C-terminal peptide able to inhibit Gs activation by A2A adenosine receptor. | 1.1 Articolo in rivista | 2003 | Grieco, Paolo; Albrizio, Stefania; D’Ursi, A. M.; Giusti, L.; Mazzoni, M. R.; Novellino, E.; Rovero, P. | |
| Unraveling the active conformation of urotensin II | 1.1 Articolo in rivista | 2004 | Carotenuto, Alfonso; Grieco, Paolo; Campiglia, Pietro; Novellino, Ettore; Ettore, Rovero; Paolo, | |
| Phenol derived CVFM analogs inhibitors of ras farnesyl transferase possessing cellular in vitro activity. | 1.1 Articolo in rivista | 1998 | Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; Ramunno, Anna; Santagada, Vincenzo; Albrizio, Stefania; Califano, D.; Giuliano, A.; Santelli, G. | |
| Synthesis and Binding Affinities for 5-HT1A, 5-HT2A and 5-HT2C receptors of a series of 1- and 2-(4-arylpiperazinylalkyl)-4-(benzoyl)-1,2,3-triazole derivatives. | 1.1 Articolo in rivista | 1999 | Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; Santagada, Vincenzo; Albrizio, Stefania; Spadola, L.; Bruni, G.; Romeo, M. R. | |
| Structure-Activity Relationships of Novel Cyclic alpha-MSH/gamma-MSH Hybrid Analogues which Lead to Potent and Selective Ligands for the Human MC3R and Human MC5R | 1.1 Articolo in rivista | 2003 | Balse, Srinivasan; P., M.; Grieco, Paolo; P, Cai; M, Trivedi; D, Hruby; V., J. | |
| Extensive Structure-Activity Studies of Lactam Derivatives of MT-II and SHU9119: Their activity and Selectivity at Human Melanocortin Receptors 3,4 and, 5. | 1.1 Articolo in rivista | 2003 | Grieco, Paolo; P, Balsesrinivasan; P, Han; G, Weinberg; D, Macnail; T, ; VAN DER, Ploeg; L. H. T, Hruby; V., J. | |
| NMR analysis of synthetic peptides agonist to PTPRJ, a receptor-type protein tyrosine phosphatase with tumor suppressor activity | 1.5 Abstract in rivista | 2011 | Brancaccio, Diego; Carotenuto, Alfonso; Grieco, Paolo; Campiglia, P; Trapasso, F; Novellino, Ettore | |
| Melanocortin type 3 receptor null mice are refractory to the inhibitory actions of a selective receptor agonist in experimental acute inflammation | 1.1 Articolo in rivista | 2006 | Getting, J. S.; Lam, C. W.; Chen, A. S.; Grieco, Paolo; Perretti, M. | |
| New melanocortin peptides useful as medicament against Staphylococcus aureus, Candida albicans, Pseudomonas aeruginosa, Candida glabrata or Candida krusei | 6.1 Brevetto | 2010 | Bonino, F.; Catania, A.; Grieco, Paolo; Novellino, Ettore | |
| New dimensions in the design of potent and receptor selective melanotropin analogues | 2.1 Contributo in volume (Capitolo o Saggio) | 2000 | Grieco, Paolo; Han, G.; Hruby, V. J. | |
| Novel peptidomimetic as MMP2 inhibitors | 4.1 Articoli in Atti di convegno | 2007 | K., Kaia; P., Campiglia; GOMEZ MONTERREY, ISABEL MARIA; M., D'Ursi; Grieco, Paolo; Novellino, Ettore | |
| Further structure-activity studies of lactam derivatives of MT-II and SHU-9119: Their activity and selectivity at human melanocortin receptors 3, 4, and 5. | 1.1 Articolo in rivista | 2007 | Grieco, Paolo; Cai, M.; Han, G.; Trivedi, D.; Campiglia, P.; Novellino, Ettore; Hruby, V. J. | |
| Urokinase receptor activation by a novel interaction between connecting peptide region of Urokinase and αvβ5 Integrin Journal of Cell Science, 119, 3424-3434, 2006 | 1.1 Articolo in rivista | 2006 | Franco, P; Vocca, I; Carriero, M. V; Alfano, D; Cito, L; Longanesi, Cattani; I, ; Grieco, Paolo; P, Ossowski; L, Stoppelli; M., P. | |
| Substitution of Arginine with Proline and Proline Derivatives in MSH Leads to Selectivity for Human Melanocortin 4 Receptor (hMC4R) | 1.1 Articolo in rivista | 2009 | H., Qu; M., Cai; A. V., Mayorov; Grieco, Paolo; M., Zingsheim; D., Trivedi; V. J., Hruby | |
| Spiro[(dihydropyrazin-2,5-dione)-6,3’-(2’,3’-dihydrothieno[2,3-b]naphtho-4’,9’-dione)]-Based Cytotoxic Agents: Structure-Activity Relationship Studies on the Substituent at N4-Position of the Diketopiperazine Domain | 1.1 Articolo in rivista | 2008 | GOMEZ MONTERREY, ISABEL MARIA; P., Campiglia; Carotenuto, Alfonso; P., Stiuso; A., Bertamino; M., Sala; C., Aaquino; Grieco, Paolo; S., Morello; Pinto, Antonio; P., Ianelli; Novellino, Ettore | |
| Design, synthesis and Cytotoxic Evaluation of a New Series of 3-Substituted-spiro[(dihydropirazin-2,5-dione)-6,3’-(2’,3’-dihydrothieno[2,3-b]naphtho-4’,9’-dione)] Derivatives | 1.1 Articolo in rivista | 2007 | GOMEZ MONTERREY, ISABEL MARIA; P., Campiglia; Carotenuto, Alfonso; D., Califano; C., Pisano; L., Vesci; T., Lama; A., Bertamino; M., Sala; A., MAZZELLA di BOSCO; Grieco, Paolo; Novellino, Ettore | |
| Design and Synthesis of Spirotryprostatin-inspired Diketopiperazine Systemsfrom Prolyl Spirooxoindolethiazolidine Derivatives | 1.1 Articolo in rivista | 2010 | Bertamino, Alessia; Aquino, Claudio; M., Sala; N., de Simone; C. A., Mattia; L., Erra; S., Musella; P., Iannelli; Carotenuto, Alfonso; Grieco, Paolo; Novellino, Ettore; P., Campiglia; GOMEZ MONTERREY, ISABEL MARIA |