SEVERINO, BEATRICE

SEVERINO, BEATRICE  

DIPARTIMENTO DI FARMACIA  

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Risultati 1 - 20 di 124 (tempo di esecuzione: 0.049 secondi).
Titolo Tipologia Data di pubblicazione Autore(i) File
Synthesis and biological activity of pseudopeptides inhibitors of Ras farnesyl transferase containing unconventional amino acids. 1.1 Articolo in rivista 1999 Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; De Luca, S; Giuliano, A; Santelli, G; Califano, D; Severino, Beatrice; Santagada, Vincenzo
Synthesis of substituted benzamides as anti-inflammatory agents that inhibit preferentially cyclooxygenase 1 but do not cause gastric damage. 1.1 Articolo in rivista 2001 Caliendo, Giuseppe; Santagada, Vincenzo; Perissutti, Elisa; Severino, Beatrice; Fiorino, Ferdinando; Warner, T. D.; Wallace, J. L.; Ifa, D. R.; Antunes, E; Cirino, Giuseppe; de Nucci, G.
Conformation-activity relationship of peptide T and new pseudocyclic hexapeptide analogs. 1.1 Articolo in rivista 2007 D'Ursi, A; Caliendo, Giuseppe; Perissutti, Elisa; Santagada, Vincenzo; Severino, Beatrice; Albrizio, Stefania; Bifulco, G; Spisani, S; Temussi, PIERO ANDREA
A convenient synthesis of N-Fmoc-N,N'-bis-Boc-7-guanyl-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid (Fmoc-N,N'-bis-Boc-7-guanyl-Tic-OH, GTIC). 1.1 Articolo in rivista 2001 Santagada, Vincenzo; Fiorino, Ferdinando; Severino, Beatrice; Salvadori, S; Lazarus, L. H.; Bryant, S. D.; Caliendo, Giuseppe
A nitro-arginine derivative of trimebutine (NO2-Arg-Trim) attenuates pain induced by colorectal distension in conscious rats. 1.1 Articolo in rivista 2009 Distrutti, E.; Mencarelli, A.; Renga, B.; Caliendo, Giuseppe; Santagada, Vincenzo; Severino, Beatrice; Fiorucci, S.
Synthetic peptides as probes for conformational preferences of domains of membrane receptors 1.1 Articolo in rivista 2005 F., Naider; S., Khare; B., Arshava; Severino, Beatrice; J., Russo; J. M., Becker
PAR1 Antagonism Protects Against Experimental Liver Fibrosis. Role of Proteinase Receptors in Stellate Cell Activation 1.1 Articolo in rivista 2004 Fiorucci, S.; Antonelli, E.; Distrutti, E.; Severino, Beatrice; Fiorentina, R.; Baldoni, M.; Caliendo, Giuseppe; Santagada, Vincenzo; Morelli, A.; Cirino, Giuseppe
A convenient strategy of dimerization by microwave heating and using 2,5-diketopiperazine as scaffold. 1.1 Articolo in rivista 2003 Santagada, Vincenzo; Fiorino, Ferdinando; Perissutti, Elisa; Severino, Beatrice; Terracciano, Sara; Cirino, Giuseppe; Caliendo, Giuseppe
Probing the shape of a hydrophobic pocket in the active site of delta-opioid antagonists 1.1 Articolo in rivista 2001 V., Santagada; G., Caliendo; Severino, Beatrice; E., Perissutti; F., Ceccarelli; L., Giusti; M. R., Mazzoni; S., Salvadori; P. A., Temussi
Synthesis, Pharmacological Evaluation, and Molecular Modeling Studies of Novel Peptidic CAAX Analogues as Farnesyl-Protein-Transferase Inhibitors 1.1 Articolo in rivista 2006 Santagada, Vincenzo; Caliendo, Giuseppe; Severino, Beatrice; Lavecchia, Antonio; Perissutti, Elisa; Fiorino, Ferdinando; Zampella, Angela; Sepe, Valentina; Califano, D.; Santelli, G.; Novellino, Ettore
5‑HT1A Receptor: An Old Target as a New Attractive Tool in Drug Discovery from Central Nervous System to Cancer 1.1 Articolo in rivista 2014 Fiorino, Ferdinando; Severino, Beatrice; Magli, Elisa; Ciano, Antonio; Caliendo, Giuseppe; Santagada, Vincenzo; Frecentese, Francesco; Perissutti, Elisa
Design of inhibitors for human tissue kallikrein using non-natural aromatic and basic amino acids. 1.1 Articolo in rivista 2002 Daniel C., Pimenta; Robson L., Melo; Caliendo, Giuseppe; Santagada, Vincenzo; Fiorino, Ferdinando; Severino, Beatrice; Gilberto De, Nucci; Luiz, Juliano; Maria, A. J. u. l. i. a. n. o.
Synthesis, Biological Evaluation and Docking Studies of PAR2-AP Derived Pseudopeptides as Inhibitors of Kallikrein 5 and 6 1.1 Articolo in rivista 2015 Severino, Beatrice; Fiorino, Ferdinando; Corvino, Angela; Caliendo, Giuseppe; Santagada, Vincenzo; Diego Magno, Assis; Juliana R., Oliveira; Luiz, Juliano; Serena, Manganelli; Emilio, Benfenati; Frecentese, Francesco; Perissutti, Elisa; Maria Aparecida, Juliano
Microwave-enhanced solution coupling of the a,a-dialkyl amino acid, Aib 1.1 Articolo in rivista 2001 Santagada, Vincenzo; Fiorino, Ferdinando; Perissutti, Elisa; Severino, Beatrice; De Filippis, V; Vivenzio, B; Caliendo, Giuseppe
Synthesis of new 1,2,3-benzotriazin-4-one-arylpiperazine derivatives as 5-HT1A serotonin receptor ligands. 1.1 Articolo in rivista 2000 Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; Santagada, Vincenzo; Severino, Beatrice; Bruni, G; Romeo, M. R.
A convenient synthesis by microwave heating and pharmacological evaluation of novel benzoyltriazole and saccharine derivatives as 5-HT1A receptor ligands. 1.1 Articolo in rivista 2002 Caliendo, Giuseppe; Fiorino, Ferdinando; Perissutti, Elisa; Severino, Beatrice; Daniela, Scolaro; Stefania, Gessi; Elena, Cattabriga; Pier Andrea, Borea; Santagada, Vincenzo
A convenient synthesis by microwave irradiation of an active metabolite (EXP-3174) of losartan. 1.1 Articolo in rivista 2003 Santagada, Vincenzo; Fiorino, Ferdinando; Perissutti, Elisa; Severino, Beatrice; Terracciano, Sara; Cleber Evandro, Teixeira; Caliendo, Giuseppe
Thrombin receptors and their antagonists: an update on the patent literature 1.1 Articolo in rivista 2010 Cirino, Giuseppe; Severino, Beatrice
Effect of positive charge in VIP 16g-glutamyl diamino derivatives on hVPAC1 and hVPAC2 receptor function 1.1 Articolo in rivista 2008 S., De Maria; V., Metafora; S., Metafora; G., Ravagnan; M., Carteni; G., Pontoni; A., Facchiano; M., Lepretti; Severino, Beatrice; Caliendo, Giuseppe; Santagada, Vincenzo; I., Langer; P. R. o. b. b. e. r. e. c. h., T.
Synthesis by microwave irradiation and binding properties of novel 5-HT1A receptor ligands. 1.1 Articolo in rivista 2001 Caliendo, Giuseppe; Fiorino, Ferdinando; Perissutti, Elisa; Severino, Beatrice; Gessi, S; Cattabriga, E; Borea, P. A.; Santagada, Vincenzo