SEVERINO, BEATRICE
SEVERINO, BEATRICE
DIPARTIMENTO DI FARMACIA
Effect of positive charge in VIP 16g-glutamyl diamino derivatives on hVPAC1 and hVPAC2 receptor function
2008 S., De Maria; V., Metafora; S., Metafora; G., Ravagnan; M., Carteni; G., Pontoni; A., Facchiano; M., Lepretti; Severino, Beatrice; Caliendo, Giuseppe; Santagada, Vincenzo; I., Langer; P. R. o. b. b. e. r. e. c. h., T.
Synthesis and biological activity of pseudopeptides inhibitors of Ras farnesyl transferase containing unconventional amino acids.
1999 Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; De Luca, S; Giuliano, A; Santelli, G; Califano, D; Severino, Beatrice; Santagada, Vincenzo
A convenient synthesis of N-Fmoc-N,N'-bis-Boc-7-guanyl-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid (Fmoc-N,N'-bis-Boc-7-guanyl-Tic-OH, GTIC).
2001 Santagada, Vincenzo; Fiorino, Ferdinando; Severino, Beatrice; Salvadori, S; Lazarus, L. H.; Bryant, S. D.; Caliendo, Giuseppe
Thrombin receptors and their antagonists: an update on the patent literature
2010 Cirino, Giuseppe; Severino, Beatrice
A nitro-arginine derivative of trimebutine (NO2-Arg-Trim) attenuates pain induced by colorectal distension in conscious rats.
2009 Distrutti, E.; Mencarelli, A.; Renga, B.; Caliendo, Giuseppe; Santagada, Vincenzo; Severino, Beatrice; Fiorucci, S.
Synthesis and vasorelaxant activity of new 1,4-benzoxazine derivatives potassium channel openers.
2002 Caliendo, Giuseppe; Perissutti, Elisa; Santagada, Vincenzo; Fiorino, Ferdinando; Severino, Beatrice; D'EMMANUELE DI VILLA BIANCA, Roberta; Laura, Lippolis; Aldo, Pinto; Sorrentino, Raffaella
Synthesis of novel anti-inflammatory peptides derived from the amino-acid sequence of the bioactive protein SV-IV
2001 Ialenti, Armando; Santagada, Vincenzo; Caliendo, Giuseppe; Severino, Beatrice; Fiorino, Ferdinando; Maffia, Pasquale; Ianaro, Angela; Morelli, F; DI MICCO, B; Carteni', M; Stiuso, P; Metafora, V; Metafora, S.
Conformation-activity relationship of peptide T and new pseudocyclic hexapeptide analogs.
2007 D'Ursi, A; Caliendo, Giuseppe; Perissutti, Elisa; Santagada, Vincenzo; Severino, Beatrice; Albrizio, Stefania; Bifulco, G; Spisani, S; Temussi, PIERO ANDREA
Synthesis, Biological Evaluation and Docking Studies of PAR2-AP Derived Pseudopeptides as Inhibitors of Kallikrein 5 and 6
2015 Severino, Beatrice; Fiorino, Ferdinando; Corvino, Angela; Caliendo, Giuseppe; Santagada, Vincenzo; Diego Magno, Assis; Juliana R., Oliveira; Luiz, Juliano; Serena, Manganelli; Emilio, Benfenati; Frecentese, Francesco; Perissutti, Elisa; Maria Aparecida, Juliano
Synthesis of 1-naphthylpiperazine derivatives as serotoninergic ligands and their evaluation as antiproliferative agents.
2011 Fiorino, Ferdinando; Magli, Elisa; Perissutti, Elisa; Severino, Beatrice; Frecentese, Francesco; Esposito, A.; De Angelis, F.; Incisivo, GIUSEPPINA MARIA; Massarelli, P.; Nencini, C.; Di Gennaro, E.; Budillon, A.; Di Cintio, A.; Santagada, Vincenzo; Caliendo, Giuseppe
New Potent 5-HT2A Receptor Ligands Containing a N'-Cyanopicolinamidine Nucleus: Synthesis and In Vitro Pharmacological Evaluation
2012 Fiorino, Ferdinando; Severino, Beatrice; Magli, Elisa; Perissutti, Elisa; Frecentese, Francesco; A., Esposito; Incisivo, GIUSEPPINA MARIA; Ciano, Antonio; P., Massarelli; C., Nencini; Santagada, Vincenzo; Caliendo, Giuseppe
Synthesis of substituted benzamides as anti-inflammatory agents that inhibit preferentially cyclooxygenase 1 but do not cause gastric damage.
2001 Caliendo, Giuseppe; Santagada, Vincenzo; Perissutti, Elisa; Severino, Beatrice; Fiorino, Ferdinando; Warner, T. D.; Wallace, J. L.; Ifa, D. R.; Antunes, E; Cirino, Giuseppe; de Nucci, G.
A convenient strategy of dimerization by microwave heating and using 2,5-diketopiperazine as scaffold.
2003 Santagada, Vincenzo; Fiorino, Ferdinando; Perissutti, Elisa; Severino, Beatrice; Terracciano, Sara; Cirino, Giuseppe; Caliendo, Giuseppe
Synthesis, Pharmacological Evaluation, and Molecular Modeling Studies of Novel Peptidic CAAX Analogues as Farnesyl-Protein-Transferase Inhibitors
2006 Santagada, Vincenzo; Caliendo, Giuseppe; Severino, Beatrice; Lavecchia, Antonio; Perissutti, Elisa; Fiorino, Ferdinando; Zampella, Angela; Sepe, Valentina; Califano, D.; Santelli, G.; Novellino, Ettore
Synthesis of benzamide derivatives and their evaluation as antiprion agents
2012 Fiorino, Ferdinando; M., Eiden; A., Giese; Severino, Beatrice; A., Esposito; M. H., Groschup; Perissutti, Elisa; Magli, Elisa; Incisivo, GIUSEPPINA MARIA; Ciano, Antonio; Frecentese, Francesco; H. A., Kretzschmar; J., Wagner; Santagada, Vincenzo; Caliendo, Giuseppe
5‑HT1A Receptor: An Old Target as a New Attractive Tool in Drug Discovery from Central Nervous System to Cancer
2014 Fiorino, Ferdinando; Severino, Beatrice; Magli, Elisa; Ciano, Antonio; Caliendo, Giuseppe; Santagada, Vincenzo; Frecentese, Francesco; Perissutti, Elisa
Minimal structural requirements for agonist activity of PAR-2 activating peptides.
2002 Santagada, Vincenzo; Caliendo, Giuseppe; Severino, Beatrice; Perissutti, Elisa; Fiorino, Ferdinando; Cicala, Carla; De Filippis, V; Cirino, Giuseppe
PAR1 Antagonism Protects Against Experimental Liver Fibrosis. Role of Proteinase Receptors in Stellate Cell Activation
2004 Fiorucci, S.; Antonelli, E.; Distrutti, E.; Severino, Beatrice; Fiorentina, R.; Baldoni, M.; Caliendo, Giuseppe; Santagada, Vincenzo; Morelli, A.; Cirino, Giuseppe
Identification of a pepducin acting as S1P3 receptor antagonist
2013 Severino, Beatrice; Giuseppina Maria Incisivo, ; Fiorino, Ferdinando; Bertolino, Antonio; Frecentese, Francesco; Barbato, Francesco; Manganelli, Serena; Maggioni, Giada; Capasso, Domenica; Caliendo, Giuseppe; Santagada, Vincenzo; Sorrentino, Raffaella; Roviezzo, Fiorentina; Perissutti, Elisa
Effects of N- and C-terminal addition of oligolysines or native loop residues on the biophysical properties of transmembrane domain peptides from a G-protein coupled receptor
2006 P., CANO SANCHEZ; Severino, Beatrice; V. V., Sureshbabu; J., Russo; T., Inui; F. X., Ding; B., Arshava; J., Becker; F., Naider
| Titolo | Tipologia | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|---|
| Effect of positive charge in VIP 16g-glutamyl diamino derivatives on hVPAC1 and hVPAC2 receptor function | 1.1 Articolo in rivista | 2008 | S., De Maria; V., Metafora; S., Metafora; G., Ravagnan; M., Carteni; G., Pontoni; A., Facchiano; M., Lepretti; Severino, Beatrice; Caliendo, Giuseppe; Santagada, Vincenzo; I., Langer; P. R. o. b. b. e. r. e. c. h., T. | |
| Synthesis and biological activity of pseudopeptides inhibitors of Ras farnesyl transferase containing unconventional amino acids. | 1.1 Articolo in rivista | 1999 | Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; De Luca, S; Giuliano, A; Santelli, G; Califano, D; Severino, Beatrice; Santagada, Vincenzo | |
| A convenient synthesis of N-Fmoc-N,N'-bis-Boc-7-guanyl-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid (Fmoc-N,N'-bis-Boc-7-guanyl-Tic-OH, GTIC). | 1.1 Articolo in rivista | 2001 | Santagada, Vincenzo; Fiorino, Ferdinando; Severino, Beatrice; Salvadori, S; Lazarus, L. H.; Bryant, S. D.; Caliendo, Giuseppe | |
| Thrombin receptors and their antagonists: an update on the patent literature | 1.1 Articolo in rivista | 2010 | Cirino, Giuseppe; Severino, Beatrice | |
| A nitro-arginine derivative of trimebutine (NO2-Arg-Trim) attenuates pain induced by colorectal distension in conscious rats. | 1.1 Articolo in rivista | 2009 | Distrutti, E.; Mencarelli, A.; Renga, B.; Caliendo, Giuseppe; Santagada, Vincenzo; Severino, Beatrice; Fiorucci, S. | |
| Synthesis and vasorelaxant activity of new 1,4-benzoxazine derivatives potassium channel openers. | 1.1 Articolo in rivista | 2002 | Caliendo, Giuseppe; Perissutti, Elisa; Santagada, Vincenzo; Fiorino, Ferdinando; Severino, Beatrice; D'EMMANUELE DI VILLA BIANCA, Roberta; Laura, Lippolis; Aldo, Pinto; Sorrentino, Raffaella | |
| Synthesis of novel anti-inflammatory peptides derived from the amino-acid sequence of the bioactive protein SV-IV | 1.1 Articolo in rivista | 2001 | Ialenti, Armando; Santagada, Vincenzo; Caliendo, Giuseppe; Severino, Beatrice; Fiorino, Ferdinando; Maffia, Pasquale; Ianaro, Angela; Morelli, F; DI MICCO, B; Carteni', M; Stiuso, P; Metafora, V; Metafora, S. | |
| Conformation-activity relationship of peptide T and new pseudocyclic hexapeptide analogs. | 1.1 Articolo in rivista | 2007 | D'Ursi, A; Caliendo, Giuseppe; Perissutti, Elisa; Santagada, Vincenzo; Severino, Beatrice; Albrizio, Stefania; Bifulco, G; Spisani, S; Temussi, PIERO ANDREA | |
| Synthesis, Biological Evaluation and Docking Studies of PAR2-AP Derived Pseudopeptides as Inhibitors of Kallikrein 5 and 6 | 1.1 Articolo in rivista | 2015 | Severino, Beatrice; Fiorino, Ferdinando; Corvino, Angela; Caliendo, Giuseppe; Santagada, Vincenzo; Diego Magno, Assis; Juliana R., Oliveira; Luiz, Juliano; Serena, Manganelli; Emilio, Benfenati; Frecentese, Francesco; Perissutti, Elisa; Maria Aparecida, Juliano | |
| Synthesis of 1-naphthylpiperazine derivatives as serotoninergic ligands and their evaluation as antiproliferative agents. | 1.1 Articolo in rivista | 2011 | Fiorino, Ferdinando; Magli, Elisa; Perissutti, Elisa; Severino, Beatrice; Frecentese, Francesco; Esposito, A.; De Angelis, F.; Incisivo, GIUSEPPINA MARIA; Massarelli, P.; Nencini, C.; Di Gennaro, E.; Budillon, A.; Di Cintio, A.; Santagada, Vincenzo; Caliendo, Giuseppe | |
| New Potent 5-HT2A Receptor Ligands Containing a N'-Cyanopicolinamidine Nucleus: Synthesis and In Vitro Pharmacological Evaluation | 1.1 Articolo in rivista | 2012 | Fiorino, Ferdinando; Severino, Beatrice; Magli, Elisa; Perissutti, Elisa; Frecentese, Francesco; A., Esposito; Incisivo, GIUSEPPINA MARIA; Ciano, Antonio; P., Massarelli; C., Nencini; Santagada, Vincenzo; Caliendo, Giuseppe | |
| Synthesis of substituted benzamides as anti-inflammatory agents that inhibit preferentially cyclooxygenase 1 but do not cause gastric damage. | 1.1 Articolo in rivista | 2001 | Caliendo, Giuseppe; Santagada, Vincenzo; Perissutti, Elisa; Severino, Beatrice; Fiorino, Ferdinando; Warner, T. D.; Wallace, J. L.; Ifa, D. R.; Antunes, E; Cirino, Giuseppe; de Nucci, G. | |
| A convenient strategy of dimerization by microwave heating and using 2,5-diketopiperazine as scaffold. | 1.1 Articolo in rivista | 2003 | Santagada, Vincenzo; Fiorino, Ferdinando; Perissutti, Elisa; Severino, Beatrice; Terracciano, Sara; Cirino, Giuseppe; Caliendo, Giuseppe | |
| Synthesis, Pharmacological Evaluation, and Molecular Modeling Studies of Novel Peptidic CAAX Analogues as Farnesyl-Protein-Transferase Inhibitors | 1.1 Articolo in rivista | 2006 | Santagada, Vincenzo; Caliendo, Giuseppe; Severino, Beatrice; Lavecchia, Antonio; Perissutti, Elisa; Fiorino, Ferdinando; Zampella, Angela; Sepe, Valentina; Califano, D.; Santelli, G.; Novellino, Ettore | |
| Synthesis of benzamide derivatives and their evaluation as antiprion agents | 1.1 Articolo in rivista | 2012 | Fiorino, Ferdinando; M., Eiden; A., Giese; Severino, Beatrice; A., Esposito; M. H., Groschup; Perissutti, Elisa; Magli, Elisa; Incisivo, GIUSEPPINA MARIA; Ciano, Antonio; Frecentese, Francesco; H. A., Kretzschmar; J., Wagner; Santagada, Vincenzo; Caliendo, Giuseppe | |
| 5‑HT1A Receptor: An Old Target as a New Attractive Tool in Drug Discovery from Central Nervous System to Cancer | 1.1 Articolo in rivista | 2014 | Fiorino, Ferdinando; Severino, Beatrice; Magli, Elisa; Ciano, Antonio; Caliendo, Giuseppe; Santagada, Vincenzo; Frecentese, Francesco; Perissutti, Elisa | |
| Minimal structural requirements for agonist activity of PAR-2 activating peptides. | 1.1 Articolo in rivista | 2002 | Santagada, Vincenzo; Caliendo, Giuseppe; Severino, Beatrice; Perissutti, Elisa; Fiorino, Ferdinando; Cicala, Carla; De Filippis, V; Cirino, Giuseppe | |
| PAR1 Antagonism Protects Against Experimental Liver Fibrosis. Role of Proteinase Receptors in Stellate Cell Activation | 1.1 Articolo in rivista | 2004 | Fiorucci, S.; Antonelli, E.; Distrutti, E.; Severino, Beatrice; Fiorentina, R.; Baldoni, M.; Caliendo, Giuseppe; Santagada, Vincenzo; Morelli, A.; Cirino, Giuseppe | |
| Identification of a pepducin acting as S1P3 receptor antagonist | 1.1 Articolo in rivista | 2013 | Severino, Beatrice; Giuseppina Maria Incisivo, ; Fiorino, Ferdinando; Bertolino, Antonio; Frecentese, Francesco; Barbato, Francesco; Manganelli, Serena; Maggioni, Giada; Capasso, Domenica; Caliendo, Giuseppe; Santagada, Vincenzo; Sorrentino, Raffaella; Roviezzo, Fiorentina; Perissutti, Elisa | |
| Effects of N- and C-terminal addition of oligolysines or native loop residues on the biophysical properties of transmembrane domain peptides from a G-protein coupled receptor | 1.1 Articolo in rivista | 2006 | P., CANO SANCHEZ; Severino, Beatrice; V. V., Sureshbabu; J., Russo; T., Inui; F. X., Ding; B., Arshava; J., Becker; F., Naider |