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Combined Use of Factorial Design and Comparative Molecular Field Analysis (CoMFA): a Case Study.
1994 Caliendo, Giuseppe; Greco, Giovanni; Novellino, Ettore; Perissutti, Elisa; Santagada, Vincenzo; Silipo, Carlo
Linking CoMFA and Protein Homology Models of Enzyme-Inhibitor Interactions: an Application to Non-Steroidal Aromatase Inhibitors.
2000 Cavalli, A.; Greco, Giovanni; Novellino, Ettore; Recanatini, M.
Nanocarriers Conjugated with Cell Penetrating Peptides: New Trojan Horses by Modern Ulysses
2016 Zappavigna, Silvia; Misso, Gabriella; Falanga, Annarita; Perillo, Emiliana; Novellino, Ettore; Galdiero, Massimiliano; Grieco, Paolo; Caraglia, Michele; Galdiero, Stefania
Lactofermented annurca apple puree as a functional food indicated for the control of plasma lipid and oxidative amine levels: Results from a randomised clinical trial
2019 Carlo Tenore, Gian; Caruso, Domenico; Buonomo, Giuseppe; D’Avino, Maria; Ciampaglia, Roberto; Maisto, Maria; Schisano, Connie; Bocchino, Bruno; Novellino, Ettore
Structure-Activity Relationship Studies Optimizing the Antiproliferative Activity of Novel Cyclic Somatostatin Analogues Containing a Restrained Cyclic β -Amino Acid
2005 Sukopp, Martin; Schwab, Richard; Marinelli, Luciana; Biron, Eric; Heller, Markus; Varkondi, Edit; Pap, Akos; Novellino, Ettore; Keri, Gyoergy; Kessler, Horst
Annurca Apple Nutraceutical Formulation Enhances Keratin Expression in a Human Model of Skin and Promotes Hair Growth and Tropism in a Randomized Clinical Trial
2018 Tenore, Gian Carlo; Caruso, Domenico; Buonomo, Giuseppe; D'Avino, Maria; Santamaria, Rita; Irace, Carlo; Piccolo, Marialuisa; Maisto, Maria; Novellino, Ettore
Development of piperazine-tethered heterodimers as potent antimalarials against chloroquine-resistant P. falciparum strains. Synthesis and molecular modeling
2007 S., Gemma; G., Kukreja; G., Campiani; S., Butini; M., Bernetti; B. P., Joshi; L., Savini; N., Basilico; D., Taramelli; V., Ardley; Bertamino, Alessia; Novellino, Ettore; Persico, Marco; Catalanotti, Bruno; Fattorusso, Caterina
Plasma lipid lowering effect by a novel chia seed based nutraceutical formulation
2018 Tenore, Gian Carlo; Caruso, Domenico; Buonomo, Giuseppe; D'Avino, Maria; Ciampaglia, Roberto; Novellino, Ettore
Multicomponent Reaction of Z-Chlorooximes, Isocyanides, and Hydroxylamines as Hypernucleophilic Traps. A One-Pot Route to Aminodioximes and Their Transformation into 5-Amino-1,2,4-oxadiazoles by Mitsunobu-Beckmann Rearrangement
2015 Mercalli, Valentina; Massarotti, Alberto; Varese, Monica; Giustiniano, Mariateresa; Meneghetti, Fiorella; Novellino, Ettore; Tron, Gian Cesare
Diarylheterocycle Core Ring Features Effect in Selective COX-1 Inhibition
2012 Perrone, M. G.; Vitale., P; Malerba, P.; Altomare, A.; Rizzi, R.; Lavecchia, Antonio; DI GIOVANNI, Carmen; Novellino, Ettore; Scilimati, A.
Titolo | Tipologia | Data di pubblicazione | Autore(i) | File |
---|---|---|---|---|
Combined Use of Factorial Design and Comparative Molecular Field Analysis (CoMFA): a Case Study. | 1.1 Articolo in rivista | 1994 | Caliendo, Giuseppe; Greco, Giovanni; Novellino, Ettore; Perissutti, Elisa; Santagada, Vincenzo; Silipo, Carlo | |
Linking CoMFA and Protein Homology Models of Enzyme-Inhibitor Interactions: an Application to Non-Steroidal Aromatase Inhibitors. | 1.1 Articolo in rivista | 2000 | Cavalli, A.; Greco, Giovanni; Novellino, Ettore; Recanatini, M. | |
Nanocarriers Conjugated with Cell Penetrating Peptides: New Trojan Horses by Modern Ulysses | 1.1 Articolo in rivista | 2016 | Zappavigna, Silvia; Misso, Gabriella; Falanga, Annarita; Perillo, Emiliana; Novellino, Ettore; Galdiero, Massimiliano; Grieco, Paolo; Caraglia, Michele; Galdiero, Stefania | |
Lactofermented annurca apple puree as a functional food indicated for the control of plasma lipid and oxidative amine levels: Results from a randomised clinical trial | 1.1 Articolo in rivista | 2019 | Carlo Tenore, Gian; Caruso, Domenico; Buonomo, Giuseppe; D’Avino, Maria; Ciampaglia, Roberto; Maisto, Maria; Schisano, Connie; Bocchino, Bruno; Novellino, Ettore | |
Structure-Activity Relationship Studies Optimizing the Antiproliferative Activity of Novel Cyclic Somatostatin Analogues Containing a Restrained Cyclic β -Amino Acid | 1.1 Articolo in rivista | 2005 | Sukopp, Martin; Schwab, Richard; Marinelli, Luciana; Biron, Eric; Heller, Markus; Varkondi, Edit; Pap, Akos; Novellino, Ettore; Keri, Gyoergy; Kessler, Horst | |
Annurca Apple Nutraceutical Formulation Enhances Keratin Expression in a Human Model of Skin and Promotes Hair Growth and Tropism in a Randomized Clinical Trial | 1.1 Articolo in rivista | 2018 | Tenore, Gian Carlo; Caruso, Domenico; Buonomo, Giuseppe; D'Avino, Maria; Santamaria, Rita; Irace, Carlo; Piccolo, Marialuisa; Maisto, Maria; Novellino, Ettore | |
Development of piperazine-tethered heterodimers as potent antimalarials against chloroquine-resistant P. falciparum strains. Synthesis and molecular modeling | 1.1 Articolo in rivista | 2007 | S., Gemma; G., Kukreja; G., Campiani; S., Butini; M., Bernetti; B. P., Joshi; L., Savini; N., Basilico; D., Taramelli; V., Ardley; Bertamino, Alessia; Novellino, Ettore; Persico, Marco; Catalanotti, Bruno; Fattorusso, Caterina | |
Plasma lipid lowering effect by a novel chia seed based nutraceutical formulation | 1.1 Articolo in rivista | 2018 | Tenore, Gian Carlo; Caruso, Domenico; Buonomo, Giuseppe; D'Avino, Maria; Ciampaglia, Roberto; Novellino, Ettore | |
Multicomponent Reaction of Z-Chlorooximes, Isocyanides, and Hydroxylamines as Hypernucleophilic Traps. A One-Pot Route to Aminodioximes and Their Transformation into 5-Amino-1,2,4-oxadiazoles by Mitsunobu-Beckmann Rearrangement | 1.1 Articolo in rivista | 2015 | Mercalli, Valentina; Massarotti, Alberto; Varese, Monica; Giustiniano, Mariateresa; Meneghetti, Fiorella; Novellino, Ettore; Tron, Gian Cesare | |
Diarylheterocycle Core Ring Features Effect in Selective COX-1 Inhibition | 1.1 Articolo in rivista | 2012 | Perrone, M. G.; Vitale., P; Malerba, P.; Altomare, A.; Rizzi, R.; Lavecchia, Antonio; DI GIOVANNI, Carmen; Novellino, Ettore; Scilimati, A. |
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Tipologia
- 1 Contributo su Rivista 788
- 1 Contributo su Rivista::1.1 Arti... 788
Data di pubblicazione
- 2020 - 2024 73
- 2010 - 2019 460
- 2000 - 2009 190
- 1990 - 1999 38
- 1980 - 1989 24
- 1977 - 1979 3
Editore
- American Chemical Society:1155 Si... 29
- Elsevier Science Limited:Oxford F... 7
- Editions Scientifique & Medical E... 4
- WILEY-VCH Verlag GmbH & Co. KGaA,... 3
- Amer Soc Pharmacognosy 2
- Bentham Science Publishers BV:PO ... 2
- John Wiley & Sons Incorporated:Cu... 2
- -SPRINGER, VAN GODEWIJCKSTRAAT 30... 1
- Amer Chemical Soc 1
- ARKAT USA INC, C/O ALAN R KATRITZ... 1
Rivista
- JOURNAL OF MEDICINAL CHEMISTRY 205
- EUROPEAN JOURNAL OF MEDICINAL CHE... 53
- CHEMMEDCHEM 26
- TETRAHEDRON LETTERS 17
- NUTRIENTS 16
- BIOORGANIC & MEDICINAL CHEMISTRY 11
- BIOORGANIC & MEDICINAL CHEMISTRY ... 11
- FOOD CHEMISTRY 11
- SCIENTIFIC REPORTS 11
- ACS MEDICINAL CHEMISTRY LETTERS 10
Keyword
- Humans 45
- Animals 23
- Organic Chemistry 23
- drug design 19
- Drug Discovery3003 Pharmaceutical... 19
- Structure-Activity Relationship 18
- Biochemistry 16
- molecular docking 16
- Molecular Medicine 16
- Pharmacology 15
Lingua
- eng 712
- enm 2
- ita 2
Accesso al fulltext
- no fulltext 588
- reserved 84
- open 58
- restricted 58