CASERTANO, MARCELLO
CASERTANO, MARCELLO
Dipartimento di Farmacia
Antiproliferative effects of synthetic prenylated quinones and thiazinoquinones inspired by marine natural products
2020 Casertano, M.; Imperatore, C.; Della Sala, G.; Aiello, A.; Menna, M.
Cis-trans photodynamics of benzodiazopyrrole derivatives in view of biomedical applications
2020 Altucci, C.; Imperatore, C.; Valadan, M.; Tartaglione, L.; Persico, M.; Ramunno, A.; Menna, M.; Casertano, M.; Dell’Aversano, Carmela.; Singh, M.; d’Ausilio Garigliota, M. L.; Bajardi, F.; Morelli, E.; Fattorusso, C.; Varra, M
Synthesis of functionalized polyols to explore the potential of a bioactive marine-derived polyketide as multitarget drug candidate
2021 Casertano, Marcello; Imperatore, Concetta; Vito, Alessio; Genovese, Massimo; Del Corso, Antonella; Menna, Marialuisa
Microwave-Assisted Synthesis of 2-Methyl-1H-indole-3-carboxylate Derivatives via Pd-Catalyzed Heterocyclization
2022 Bellavita, Rosa; Casertano, Marcello; Grasso, Nicola; Gillick-Healy, Malachi; Kelly, Brian G.; Adamo, Mauro F. A.; Menna, Marialuisa; Merlino, Francesco; Grieco, Paolo
Identifying Human PTP1B Enzyme Inhibitors from Marine Natural Products: Perspectives for Developing of Novel Insulin-Mimetic Drugs
2022 Casertano, Marcello; Genovese, Massimo; Piazza, Lucia; Balestri, Francesco; Del Corso, Antonella; Vito, Alessio; Paoli, Paolo; Santi, Alice; Imperatore, Concetta; Menna, Marialuisa
Toward marine inspired multitarget drugs for diabetes mellitus and its complications: design and synthesis of novel dual Protein Tyrosine Phosphatase 1B and Aldose Reductase ligands
2021 Imperatore, Concetta; Casertano, Marcello; Paoli, Paolo; Del Corso, Antonella; Menna, Marialuisa
Insights into Cytotoxic Behavior of Lepadins and Structure Elucidation of the New Alkaloid Lepadin L from the Mediterranean Ascidian Clavelina lepadiformis
2022 Casertano, Marcello; Genovese, Massimo; Paoli, Paolo; Santi, Alice; Aiello, Anna; Menna, Marialuisa; Imperatore, Concetta
Exploitation of natural products in the search of drug-like molecules and leads: a fascinating resource
2020 Casertano, Marcello
Dual Targeting of PTP1B and Aldose Reductase with Marine Drug Phosphoeleganin: A Promising Strategy for Treatment of Type 2 Diabetes
2021 Genovese, Massimo; Imperatore, Concetta; Casertano, Marcello; Aiello, Anna; Balestri, Francesco; Piazza, Lucia; Menna, Marialuisa; Del Corso, Antonella; Paoli, Paolo
Exploring the antimalarial potential of the methoxy-thiazinoquinone scaffold: Identification of a new lead candidate
2019 Imperatore, Concetta; Persico, Marco; Senese, Maria; Aiello, Anna; Casertano, Marcello; Luciano, Paolo; Basilico, Nicoletta; Parapini, Silvia; Paladino, Antonella; Fattorusso, Caterina; Menna, Marialuisa
Exploring the photodynamic properties of two antiproliferative benzodiazopyrrole derivatives
2020 Imperatore, Concetta; Valadan, Mohammadhassan; Tartaglione, Luciana; Persico, Marco; Ramunno, Anna; Menna, Marialuisa; Casertano, Marcello; Dell'Aversano, Carmela; Singh, Manjot; Luisa d’Aulisio Garigliota, Maria; Bajardi, Francesco; Morelli, Elena; Fattorusso, Caterina; Altucci, Carlo; Varra, Michela
Chemical Investigation of the Indonesian Tunicate Polycarpa aurata and Evaluation of the Effects Against Schistosoma mansoni of the Novel Alkaloids Polyaurines A and B
2019 Casertano, Marcello; Imperatore, Concetta; Luciano, Paolo; Aiello, Anna; Yunovilsa Putra, Masteria; Gimmelli, Roberto; Ruberti, Giovina; Menna, Marialuisa
In Vitro Antiproliferative Evaluation of Synthetic Meroterpenes Inspired by Marine Natural Products
2019 Imperatore, Concetta; DELLA SALA, Gerardo; Casertano, Marcello; Luciano, Paolo; Aiello, Anna; Laurenzana, Ilaria; Piccoli, Claudia; Menna, Marialuisa
Antiplasmodial activity of p-substituted benzyl thiazinoquinone derivatives and their potential against parasitic infections
2020 Casertano, Marcello; Menna, Marialuisa; Fattorusso, Caterina; Basilico, Nicoletta; Parapini, Silvia; Persico, Marco; Imperatore, Concetta
Assignment of the Absolute Configuration of Phosphoeleganin via Synthesis of Model Compounds
2017 Luciano, Paolo; Imperatore, Concetta; Senese, Maria; Aiello, Anna; Casertano, Marcello; Guo, Yue W; Menna, Marialuisa
Investigating the antiparasitic potential of the marine sesquiterpene avarone, its reduced form avarol, and the novel semisynthetic thiazinoquinone analogue thiazoavarone
2020 Imperatore, Concetta; Gimmelli, Roberto; Persico, Marco; Casertano, Marcello; Guidi, Alessandra; Saccoccia, Fulvio; Ruberti, Giovina; Luciano, Paolo; Aiello, Anna; Parapini, Silvia; Avunduk, Sibel; Basilico, Nicoletta; Fattorusso, Caterina; Menna, Marialuisa
The ascidian-derived metabolites with antimicrobial properties
2020 Casertano, Marcello; Menna, Marialuisa; Imperatore, Concetta
Spectroscopic properties of two 5′-(4-dimethylamino)azobenzene conjugated G-quadruplex forming oligonucleotides
2020 Imperatore, Concetta; Varriale, Antonio; Rivieccio, Elisa; Pennacchio, Angela; Staiano, MARIA TERESA; D'Auria, Sabato; Casertano, Marcello; Altucci, Carlo; Valadan, Mohammadhassan; Singh, Manjot; Menna, Marialuisa; Varra, Michela
Fighting Multiparasitism, a Neglected Reality in Marginalised Community: New Tools from the Sea
2020 Imperatore, Concetta; Casertano, Marcello; Luciano, Paolo; Aiello, Anna; Gimmelli, Roberto; Ruberti, Giovina; Parapini, Silvia; Basilico, Nicoletta; Avunduk, Sibel; Persico, Marco; Fattorusso, Caterina; Menna, Marialuisa
Thiazinoquinones as New Promising Multistage Schistosomicidal Compounds Impacting Schistosoma mansoni and Egg Viability
2020 Roberto, Gimmelli; Persico, Marco; Imperatore, Concetta; Fulvio, Saccoccia; Guidi, Alessandra; Casertano, Marcello; Luciano, Paolo; Agostina, Pietrantoni; Lucia, Bertuccini; Antonella, Paladino; Giuliana, Papoff; Menna, Marialuisa; Fattorusso, Caterina; Giovina, Ruberti
Titolo | Tipologia | Data di pubblicazione | Autore(i) | File |
---|---|---|---|---|
Antiproliferative effects of synthetic prenylated quinones and thiazinoquinones inspired by marine natural products | 8.02 Comunicazioni a Convegni o Seminari | 2020 | Casertano, M.; Imperatore, C.; Della Sala, G.; Aiello, A.; Menna, M. | |
Cis-trans photodynamics of benzodiazopyrrole derivatives in view of biomedical applications | 8.02 Comunicazioni a Convegni o Seminari | 2020 | Altucci, C.; Imperatore, C.; Valadan, M.; Tartaglione, L.; Persico, M.; Ramunno, A.; Menna, M.; Casertano, M.; Dell’Aversano, Carmela.; Singh, M.; d’Ausilio Garigliota, M. L.; Bajardi, F.; Morelli, E.; Fattorusso, C.; Varra, M | |
Synthesis of functionalized polyols to explore the potential of a bioactive marine-derived polyketide as multitarget drug candidate | 8.02 Comunicazioni a Convegni o Seminari | 2021 | Casertano, Marcello; Imperatore, Concetta; Vito, Alessio; Genovese, Massimo; Del Corso, Antonella; Menna, Marialuisa | |
Microwave-Assisted Synthesis of 2-Methyl-1H-indole-3-carboxylate Derivatives via Pd-Catalyzed Heterocyclization | 1.1 Articolo in rivista | 2022 | Bellavita, Rosa; Casertano, Marcello; Grasso, Nicola; Gillick-Healy, Malachi; Kelly, Brian G.; Adamo, Mauro F. A.; Menna, Marialuisa; Merlino, Francesco; Grieco, Paolo | |
Identifying Human PTP1B Enzyme Inhibitors from Marine Natural Products: Perspectives for Developing of Novel Insulin-Mimetic Drugs | 1.1 Articolo in rivista | 2022 | Casertano, Marcello; Genovese, Massimo; Piazza, Lucia; Balestri, Francesco; Del Corso, Antonella; Vito, Alessio; Paoli, Paolo; Santi, Alice; Imperatore, Concetta; Menna, Marialuisa | |
Toward marine inspired multitarget drugs for diabetes mellitus and its complications: design and synthesis of novel dual Protein Tyrosine Phosphatase 1B and Aldose Reductase ligands | 8.02 Comunicazioni a Convegni o Seminari | 2021 | Imperatore, Concetta; Casertano, Marcello; Paoli, Paolo; Del Corso, Antonella; Menna, Marialuisa | |
Insights into Cytotoxic Behavior of Lepadins and Structure Elucidation of the New Alkaloid Lepadin L from the Mediterranean Ascidian Clavelina lepadiformis | 1.1 Articolo in rivista | 2022 | Casertano, Marcello; Genovese, Massimo; Paoli, Paolo; Santi, Alice; Aiello, Anna; Menna, Marialuisa; Imperatore, Concetta | |
Exploitation of natural products in the search of drug-like molecules and leads: a fascinating resource | 8.10 Tesi di Dottorato | 2020 | Casertano, Marcello | |
Dual Targeting of PTP1B and Aldose Reductase with Marine Drug Phosphoeleganin: A Promising Strategy for Treatment of Type 2 Diabetes | 1.1 Articolo in rivista | 2021 | Genovese, Massimo; Imperatore, Concetta; Casertano, Marcello; Aiello, Anna; Balestri, Francesco; Piazza, Lucia; Menna, Marialuisa; Del Corso, Antonella; Paoli, Paolo | |
Exploring the antimalarial potential of the methoxy-thiazinoquinone scaffold: Identification of a new lead candidate | 1.1 Articolo in rivista | 2019 | Imperatore, Concetta; Persico, Marco; Senese, Maria; Aiello, Anna; Casertano, Marcello; Luciano, Paolo; Basilico, Nicoletta; Parapini, Silvia; Paladino, Antonella; Fattorusso, Caterina; Menna, Marialuisa | |
Exploring the photodynamic properties of two antiproliferative benzodiazopyrrole derivatives | 1.1 Articolo in rivista | 2020 | Imperatore, Concetta; Valadan, Mohammadhassan; Tartaglione, Luciana; Persico, Marco; Ramunno, Anna; Menna, Marialuisa; Casertano, Marcello; Dell'Aversano, Carmela; Singh, Manjot; Luisa d’Aulisio Garigliota, Maria; Bajardi, Francesco; Morelli, Elena; Fattorusso, Caterina; Altucci, Carlo; Varra, Michela | |
Chemical Investigation of the Indonesian Tunicate Polycarpa aurata and Evaluation of the Effects Against Schistosoma mansoni of the Novel Alkaloids Polyaurines A and B | 1.1 Articolo in rivista | 2019 | Casertano, Marcello; Imperatore, Concetta; Luciano, Paolo; Aiello, Anna; Yunovilsa Putra, Masteria; Gimmelli, Roberto; Ruberti, Giovina; Menna, Marialuisa | |
In Vitro Antiproliferative Evaluation of Synthetic Meroterpenes Inspired by Marine Natural Products | 1.1 Articolo in rivista | 2019 | Imperatore, Concetta; DELLA SALA, Gerardo; Casertano, Marcello; Luciano, Paolo; Aiello, Anna; Laurenzana, Ilaria; Piccoli, Claudia; Menna, Marialuisa | |
Antiplasmodial activity of p-substituted benzyl thiazinoquinone derivatives and their potential against parasitic infections | 1.1 Articolo in rivista | 2020 | Casertano, Marcello; Menna, Marialuisa; Fattorusso, Caterina; Basilico, Nicoletta; Parapini, Silvia; Persico, Marco; Imperatore, Concetta | |
Assignment of the Absolute Configuration of Phosphoeleganin via Synthesis of Model Compounds | 1.1 Articolo in rivista | 2017 | Luciano, Paolo; Imperatore, Concetta; Senese, Maria; Aiello, Anna; Casertano, Marcello; Guo, Yue W; Menna, Marialuisa | |
Investigating the antiparasitic potential of the marine sesquiterpene avarone, its reduced form avarol, and the novel semisynthetic thiazinoquinone analogue thiazoavarone | 1.1 Articolo in rivista | 2020 | Imperatore, Concetta; Gimmelli, Roberto; Persico, Marco; Casertano, Marcello; Guidi, Alessandra; Saccoccia, Fulvio; Ruberti, Giovina; Luciano, Paolo; Aiello, Anna; Parapini, Silvia; Avunduk, Sibel; Basilico, Nicoletta; Fattorusso, Caterina; Menna, Marialuisa | |
The ascidian-derived metabolites with antimicrobial properties | 1.1 Articolo in rivista | 2020 | Casertano, Marcello; Menna, Marialuisa; Imperatore, Concetta | |
Spectroscopic properties of two 5′-(4-dimethylamino)azobenzene conjugated G-quadruplex forming oligonucleotides | 1.1 Articolo in rivista | 2020 | Imperatore, Concetta; Varriale, Antonio; Rivieccio, Elisa; Pennacchio, Angela; Staiano, MARIA TERESA; D'Auria, Sabato; Casertano, Marcello; Altucci, Carlo; Valadan, Mohammadhassan; Singh, Manjot; Menna, Marialuisa; Varra, Michela | |
Fighting Multiparasitism, a Neglected Reality in Marginalised Community: New Tools from the Sea | 1.5 Abstract in rivista | 2020 | Imperatore, Concetta; Casertano, Marcello; Luciano, Paolo; Aiello, Anna; Gimmelli, Roberto; Ruberti, Giovina; Parapini, Silvia; Basilico, Nicoletta; Avunduk, Sibel; Persico, Marco; Fattorusso, Caterina; Menna, Marialuisa | |
Thiazinoquinones as New Promising Multistage Schistosomicidal Compounds Impacting Schistosoma mansoni and Egg Viability | 1.1 Articolo in rivista | 2020 | Roberto, Gimmelli; Persico, Marco; Imperatore, Concetta; Fulvio, Saccoccia; Guidi, Alessandra; Casertano, Marcello; Luciano, Paolo; Agostina, Pietrantoni; Lucia, Bertuccini; Antonella, Paladino; Giuliana, Papoff; Menna, Marialuisa; Fattorusso, Caterina; Giovina, Ruberti |