GIUSTINIANO, MARIATERESA
GIUSTINIANO, MARIATERESA
Dipartimento di Farmacia
1H NMR-based metabolomics study on follicular fluid from patients with Polycystic Ovary Syndrome
2018 Iaccarino, Nunzia; Amato, Jussara; Pagano, Bruno; Pagano, Alessia; D'Oriano, Laura; Pelliccia, Sveva; Giustiniano, Mariateresa; Brancaccio, Diego; Merlino, Francesco; Novellino, Ettore; Alviggi, Carlo; Randazzo, Antonio
Alanine scanning analysis and structure-function relationships of the frog-skin antimicrobial peptide temporin-1Ta
2011 Giustiniano, Mariateresa; Brancaccio, Diego; Mangoni Maria, Luisa; Auriemma, Luigia; Carotenuto, Alfonso; Campiglia, P; Novellino, Ettore; Grieco, Paolo
Amino acid derivatives as new zinc binding groups for the design of selective matrix metalloproteinase inhibitors
2013 Giustiniano, Mariateresa; P., Tortorella; M., Agamennone; A., Di Pizio; A., Rossello; E., Nuti; GOMEZ MONTERREY, ISABEL MARIA; Novellino, Ettore; P., Campiglia; E., Vernieri; M., Sala; A., Bertamino; Carotenuto, Alfonso
Amphoteric 2-(sulfonylamino)benzaldehydes, secondary amines and isocyanides in the multicomponent synthesis of elusive N-alkyl-2,3-diaminoindoles
2017 Giustiniano, Mariateresa; Pelliccia, Sveva; Sangaletti, Luca; Meneghetti, Fiorella; Amato, Jussara; Novellino, Ettore; Tron, Gian Cesare
Aryl Azides as Forgotten Electrophiles in the Van Leusen Reaction: A Multicomponent Transformation Affording 4-Tosyl-1-arylimidazoles
2019 Necardo, C.; Alfano, A. I.; Del Grosso, E.; Pelliccia, S.; Galli, U.; Novellino, E.; Meneghetti, F.; Giustiniano, M.; Tron, G. C.
Bax Activation Blocks Self-Renewal and Induces Apoptosis of Human Glioblastoma Stem Cells
2017 Daniele, Simona; Pietrobono, Deborah; Costa, Barbara; Giustiniano, Mariateresa; LA PIETRA, Valeria; Giacomelli, Chiara; La Regina, Giuseppe; Silvestri, Romano; Taliani, Sabrina; Trincavelli, Maria Letizia; Da Settimo, Federico; Novellino, Ettore; Martini, Claudia; Marinelli, Luciana
Bio-Inspired Dual-Selective BCL-2/c-MYC G-Quadruplex Binders: Design, Synthesis, and Anticancer Activity of Drug-like Imidazo[2,1-i]purine Derivatives
2020 Pelliccia, Sveva; Amato, Jussara; Capasso, Domenica; Di Gaetano, Sonia; Massarotti, Alberto; Piccolo, Marialuisa; Irace, Carlo; Tron, Gian Cesare; Pagano, Bruno; Randazzo, Antonio; Novellino, Ettore; Giustiniano, Mariateresa
Computer-Aided Identification and Lead Optimization of Dual Murine Double Minute 2 and 4 Binders: Structure-Activity Relationship Studies and Pharmacological Activity
2017 Giustiniano, Mariateresa; Daniele, Simona; Pelliccia, Sveva; La Pietra, Valeria; Pietrobono, Deborah; Brancaccio, Diego; Cosconati, Sandro; Messere, Anna; Giuntini, Stefano; Cerofolini, Linda; Fragai, Marco; Luchinat, Claudio; Taliani, Sabrina; La Regina, Giuseppe; Da Settimo, Federico; Silvestri, Romano; Martini, Claudia; Novellino, Ettore; Marinelli, Luciana
The Dark Side of Isocyanides: Visible-Light Photocatalytic Activity in the Oxidative Functionalization of C(sp3)–H Bonds
2021 Russo, C.; Amato, J.; Tron, G. C.; Giustiniano, M.
An efficient synthesis of 1-arylindazole-3-carboxamides using nitrile imines, isocyanides and 2-hydroxymethylbenzoic acid, followed by a chemoselective Buchwald–Hartwig intramolecular cyclization
2016 Giustiniano, Mariateresa; Mercalli, V.; Novellino, Ettore; Tron, G. C.
Enriching the arsenal of pharmacological tools against mical2
2021 Barravecchia, I.; Barresi, E.; Russo, C.; Scebba, F.; De Cesari, C.; Mignucci, V.; De Luca, D.; Salerno, S.; La Pietra, V.; Giustiniano, M.; Pelliccia, S.; Brancaccio, D.; Donati, G.; Da Settimo, F.; Taliani, S.; Angeloni, D.; Marinelli, L.
Exploiting the Electrophilic and Nucleophilic Dual Role of Nitrile Imines: One-Pot, Three-Component Synthesis of Furo[2,3-d]pyridazin-4(5H)-ones
2015 Giustiniano, Mariateresa; Mercalli, Valentina; Amato, Jussara; Novellino, Ettore; Tron, Gian Cesare
Exploiting the nucleophilicity of the nitrogen atom of imidazoles: One-pot three-component synthesis of imidazo-pyrazines
2019 Galli, U.; Hysenlika, R.; Meneghetti, F.; Grosso, E. D.; Pelliccia, S.; Novellino, E.; Giustiniano, M.; Tron, G. C.
A fast route for the synthesis of tetrazolyl oximes by a novel multicomponent reaction between Z-chlorooximes, isocyanides and trimethylsilyl azide
2017 Giustiniano, Mariateresa; Pelliccia, Sveva; MUNOZ GARCIA, ANA BELEN; Pavone, Michele; Pagano, Bruno; Galli, Ubaldina; Novellino, Ettore; Tron, Gian Cesare
Interrupted Ugi and Passerini Reactions: An Underexplored Treasure Island
2018 Giustiniano, Mariateresa; Moni, Lisa; Sangaletti, Luca; Pelliccia, Sveva; Basso, Andrea; Novellino, Ettore; Tron, Gian Cesare
Multicomponent Reaction of Z-Chlorooximes, Isocyanides, and Hydroxylamines as Hypernucleophilic Traps. A One-Pot Route to Aminodioximes and Their Transformation into 5-Amino-1,2,4-oxadiazoles by Mitsunobu-Beckmann Rearrangement
2015 Mercalli, Valentina; Massarotti, Alberto; Varese, Monica; Giustiniano, Mariateresa; Meneghetti, Fiorella; Novellino, Ettore; Tron, Gian Cesare
Nitrile N-Oxides and Nitrile Imines as New Fuels for the Discovery of Novel Isocyanide-Based Multicomponent Reactions
2016 Tron, Gian; Giustiniano, Mariateresa; Novellino, Ettore
Non-hydrolytic chemoselective cleavage of Ugi tertiary amides: A mild access to N-substituted α-amino acid amides
2018 Giustiniano, Mariateresa; Pelliccia, Sveva; Novellino, Ettore; Cesare Tron, Gian
Novel peptidomimetics as BACE-1 inhibitors: synthesis, molecular modeling, and biological studies
2013 Butini, S.; Gabellieri, E.; Brindisi, M.; Casagni, A.; Guarino, E.; Huleatt, P. B.; Relitti, N.; LA PIETRA, Valeria; Marinelli, Luciana; Giustiniano, Mariateresa; Novellino, Ettore; Campiani, G.; Gemma, S.
On-water pyrrolidine-mediated domino synthesis of 2-iminoisatins
2018 Pelliccia, Sveva; Abbate, Vincenzo; Meneghetti, Fiorella; Frascione, Nunzianda; Hider, Robert Charles; Novellino, Ettore; Tron, Gian Cesare; Giustiniano, Mariateresa
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
1H NMR-based metabolomics study on follicular fluid from patients with Polycystic Ovary Syndrome | 1-gen-2018 | Iaccarino, Nunzia; Amato, Jussara; Pagano, Bruno; Pagano, Alessia; D'Oriano, Laura; Pelliccia, Sveva; Giustiniano, Mariateresa; Brancaccio, Diego; Merlino, Francesco; Novellino, Ettore; Alviggi, Carlo; Randazzo, Antonio | |
Alanine scanning analysis and structure-function relationships of the frog-skin antimicrobial peptide temporin-1Ta | 1-gen-2011 | Giustiniano, Mariateresa; Brancaccio, Diego; Mangoni Maria, Luisa; Auriemma, Luigia; Carotenuto, Alfonso; Campiglia, P; Novellino, Ettore; Grieco, Paolo | |
Amino acid derivatives as new zinc binding groups for the design of selective matrix metalloproteinase inhibitors | 1-gen-2013 | Giustiniano, Mariateresa; P., Tortorella; M., Agamennone; A., Di Pizio; A., Rossello; E., Nuti; GOMEZ MONTERREY, ISABEL MARIA; Novellino, Ettore; P., Campiglia; E., Vernieri; M., Sala; A., Bertamino; Carotenuto, Alfonso | |
Amphoteric 2-(sulfonylamino)benzaldehydes, secondary amines and isocyanides in the multicomponent synthesis of elusive N-alkyl-2,3-diaminoindoles | 1-gen-2017 | Giustiniano, Mariateresa; Pelliccia, Sveva; Sangaletti, Luca; Meneghetti, Fiorella; Amato, Jussara; Novellino, Ettore; Tron, Gian Cesare | |
Aryl Azides as Forgotten Electrophiles in the Van Leusen Reaction: A Multicomponent Transformation Affording 4-Tosyl-1-arylimidazoles | 1-gen-2019 | Necardo, C.; Alfano, A. I.; Del Grosso, E.; Pelliccia, S.; Galli, U.; Novellino, E.; Meneghetti, F.; Giustiniano, M.; Tron, G. C. | |
Bax Activation Blocks Self-Renewal and Induces Apoptosis of Human Glioblastoma Stem Cells | 1-gen-2017 | Daniele, Simona; Pietrobono, Deborah; Costa, Barbara; Giustiniano, Mariateresa; LA PIETRA, Valeria; Giacomelli, Chiara; La Regina, Giuseppe; Silvestri, Romano; Taliani, Sabrina; Trincavelli, Maria Letizia; Da Settimo, Federico; Novellino, Ettore; Martini, Claudia; Marinelli, Luciana | |
Bio-Inspired Dual-Selective BCL-2/c-MYC G-Quadruplex Binders: Design, Synthesis, and Anticancer Activity of Drug-like Imidazo[2,1-i]purine Derivatives | 1-gen-2020 | Pelliccia, Sveva; Amato, Jussara; Capasso, Domenica; Di Gaetano, Sonia; Massarotti, Alberto; Piccolo, Marialuisa; Irace, Carlo; Tron, Gian Cesare; Pagano, Bruno; Randazzo, Antonio; Novellino, Ettore; Giustiniano, Mariateresa | |
Computer-Aided Identification and Lead Optimization of Dual Murine Double Minute 2 and 4 Binders: Structure-Activity Relationship Studies and Pharmacological Activity | 1-gen-2017 | Giustiniano, Mariateresa; Daniele, Simona; Pelliccia, Sveva; La Pietra, Valeria; Pietrobono, Deborah; Brancaccio, Diego; Cosconati, Sandro; Messere, Anna; Giuntini, Stefano; Cerofolini, Linda; Fragai, Marco; Luchinat, Claudio; Taliani, Sabrina; La Regina, Giuseppe; Da Settimo, Federico; Silvestri, Romano; Martini, Claudia; Novellino, Ettore; Marinelli, Luciana | |
The Dark Side of Isocyanides: Visible-Light Photocatalytic Activity in the Oxidative Functionalization of C(sp3)–H Bonds | 1-gen-2021 | Russo, C.; Amato, J.; Tron, G. C.; Giustiniano, M. | |
An efficient synthesis of 1-arylindazole-3-carboxamides using nitrile imines, isocyanides and 2-hydroxymethylbenzoic acid, followed by a chemoselective Buchwald–Hartwig intramolecular cyclization | 1-gen-2016 | Giustiniano, Mariateresa; Mercalli, V.; Novellino, Ettore; Tron, G. C. | |
Enriching the arsenal of pharmacological tools against mical2 | 1-gen-2021 | Barravecchia, I.; Barresi, E.; Russo, C.; Scebba, F.; De Cesari, C.; Mignucci, V.; De Luca, D.; Salerno, S.; La Pietra, V.; Giustiniano, M.; Pelliccia, S.; Brancaccio, D.; Donati, G.; Da Settimo, F.; Taliani, S.; Angeloni, D.; Marinelli, L. | |
Exploiting the Electrophilic and Nucleophilic Dual Role of Nitrile Imines: One-Pot, Three-Component Synthesis of Furo[2,3-d]pyridazin-4(5H)-ones | 1-gen-2015 | Giustiniano, Mariateresa; Mercalli, Valentina; Amato, Jussara; Novellino, Ettore; Tron, Gian Cesare | |
Exploiting the nucleophilicity of the nitrogen atom of imidazoles: One-pot three-component synthesis of imidazo-pyrazines | 1-gen-2019 | Galli, U.; Hysenlika, R.; Meneghetti, F.; Grosso, E. D.; Pelliccia, S.; Novellino, E.; Giustiniano, M.; Tron, G. C. | |
A fast route for the synthesis of tetrazolyl oximes by a novel multicomponent reaction between Z-chlorooximes, isocyanides and trimethylsilyl azide | 1-gen-2017 | Giustiniano, Mariateresa; Pelliccia, Sveva; MUNOZ GARCIA, ANA BELEN; Pavone, Michele; Pagano, Bruno; Galli, Ubaldina; Novellino, Ettore; Tron, Gian Cesare | |
Interrupted Ugi and Passerini Reactions: An Underexplored Treasure Island | 1-gen-2018 | Giustiniano, Mariateresa; Moni, Lisa; Sangaletti, Luca; Pelliccia, Sveva; Basso, Andrea; Novellino, Ettore; Tron, Gian Cesare | |
Multicomponent Reaction of Z-Chlorooximes, Isocyanides, and Hydroxylamines as Hypernucleophilic Traps. A One-Pot Route to Aminodioximes and Their Transformation into 5-Amino-1,2,4-oxadiazoles by Mitsunobu-Beckmann Rearrangement | 1-gen-2015 | Mercalli, Valentina; Massarotti, Alberto; Varese, Monica; Giustiniano, Mariateresa; Meneghetti, Fiorella; Novellino, Ettore; Tron, Gian Cesare | |
Nitrile N-Oxides and Nitrile Imines as New Fuels for the Discovery of Novel Isocyanide-Based Multicomponent Reactions | 1-gen-2016 | Tron, Gian; Giustiniano, Mariateresa; Novellino, Ettore | |
Non-hydrolytic chemoselective cleavage of Ugi tertiary amides: A mild access to N-substituted α-amino acid amides | 1-gen-2018 | Giustiniano, Mariateresa; Pelliccia, Sveva; Novellino, Ettore; Cesare Tron, Gian | |
Novel peptidomimetics as BACE-1 inhibitors: synthesis, molecular modeling, and biological studies | 1-gen-2013 | Butini, S.; Gabellieri, E.; Brindisi, M.; Casagni, A.; Guarino, E.; Huleatt, P. B.; Relitti, N.; LA PIETRA, Valeria; Marinelli, Luciana; Giustiniano, Mariateresa; Novellino, Ettore; Campiani, G.; Gemma, S. | |
On-water pyrrolidine-mediated domino synthesis of 2-iminoisatins | 1-gen-2018 | Pelliccia, Sveva; Abbate, Vincenzo; Meneghetti, Fiorella; Frascione, Nunzianda; Hider, Robert Charles; Novellino, Ettore; Tron, Gian Cesare; Giustiniano, Mariateresa |