CALIENDO, GIUSEPPE

CALIENDO, GIUSEPPE  

DIPARTIMENTO DI FARMACIA  

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Risultati 1 - 20 di 192 (tempo di esecuzione: 0.037 secondi).
Titolo Tipologia Data di pubblicazione Autore(i) File
Synthesis of novel anti-inflammatory peptides derived from the amino-acid sequence of the bioactive protein SV-IV 1.1 Articolo in rivista 2001 Ialenti, Armando; Santagada, Vincenzo; Caliendo, Giuseppe; Severino, Beatrice; Fiorino, Ferdinando; Maffia, Pasquale; Ianaro, Angela; Morelli, F; DI MICCO, B; Carteni', M; Stiuso, P; Metafora, V; Metafora, S.
Phenol derived CVFM analogs inhibitors of ras farnesyl transferase possessing cellular in vitro activity. 1.1 Articolo in rivista 1998 Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; Ramunno, Anna; Santagada, Vincenzo; Albrizio, Stefania; Califano, D.; Giuliano, A.; Santelli, G.
Synthesis of substituted benzamides as anti-inflammatory agents that inhibit preferentially cyclooxygenase 1 but do not cause gastric damage. 1.1 Articolo in rivista 2001 Caliendo, Giuseppe; Santagada, Vincenzo; Perissutti, Elisa; Severino, Beatrice; Fiorino, Ferdinando; Warner, T. D.; Wallace, J. L.; Ifa, D. R.; Antunes, E; Cirino, Giuseppe; de Nucci, G.
Synthesis and Binding Affinities for 5-HT1A, 5-HT2A and 5-HT2C receptors of a series of 1- and 2-(4-arylpiperazinylalkyl)-4-(benzoyl)-1,2,3-triazole derivatives. 1.1 Articolo in rivista 1999 Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; Santagada, Vincenzo; Albrizio, Stefania; Spadola, L.; Bruni, G.; Romeo, M. R.
Probing the shape of a hydrophobic pocket in the active site of delta-opioid antagonists 1.1 Articolo in rivista 2001 Santagada, V; Caliendo, G; Severino, B; Perissutti, Elisa; E, Ceccarelli; F, Giusti; L, Mazzoni; Mr, Salvadori; S, Temussi; Pa,
The application of microwave irradiation as new convenient synthetic procedure in drug discovery 1.1 Articolo in rivista 2002 Santagada, Vincenzo; Perissutti, Elisa; Caliendo, Giuseppe
Synthesis, Biological Activity and Conformational Study of 1,4-Benzoxazine Derivatives as Potassium Channel Modulators 1.5 Abstract in rivista 1999 Caliendo, G; Grieco, P; Perissutti, E; Santagada, V; Santini, A; Albrizio, S; Fattorusso, C; Pinto, A; Sorrentino, R
The nitric oxide related therapeutic phenomenon: a challenging task. 1.1 Articolo in rivista 2002 Cirino, Giuseppe; Santagada, Vincenzo; Caliendo, Giuseppe
A convenient synthesis by microwave irradiation of an active metabolite (EXP-3174) of losartan. 1.1 Articolo in rivista 2003 Santagada, Vincenzo; Fiorino, Ferdinando; Perissutti, Elisa; Severino, Beatrice; Terracciano, Sara; Cleber Evandro, Teixeira; Caliendo, Giuseppe
A nitro-arginine derivative of trimebutine (NO2-Arg-Trim) attenuates pain induced by colorectal distension in conscious rats. 1.1 Articolo in rivista 2009 Distrutti, E.; Mencarelli, A.; Renga, B.; Caliendo, Giuseppe; Santagada, Vincenzo; Severino, Beatrice; Fiorucci, S.
Synthesis and biological activity of pseudopeptides inhibitors of Ras farnesyl transferase containing unconventional amino acids. 1.1 Articolo in rivista 1999 Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; De Luca, S; Giuliano, A; Santelli, G; Califano, D; Severino, Beatrice; Santagada, Vincenzo
Molecular Structure and Conformation of the (Z) and (E) Geometric Isomers of 2-(2-Phenylbenzylidene)-3-quinuclidinone. 1.1 Articolo in rivista 1995 Santini, Antonello; Benedetti, Ettore; Pedone, Carlo; Giordano, M.; Caliendo, Giuseppe; Santagada, Vincenzo; Grieco, Paolo; Greco, Giovanni
Pharmacological evaluation of benzotriazole derivatives structurally related to trazodone 1.1 Articolo in rivista 1992 Perissutti, Elisa; Meli, Rosaria; Maggetti, S.; Caliendo, Giuseppe; Cappello, B.; Silipo, C.; Vittoria, A.; Di Carlo, R.
A convenient synthesis of N-Fmoc-N,N'-bis-Boc-7-guanyl-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid (Fmoc-N,N'-bis-Boc-7-guanyl-Tic-OH, GTIC). 1.1 Articolo in rivista 2001 Santagada, Vincenzo; Fiorino, Ferdinando; Severino, Beatrice; Salvadori, S; Lazarus, L. H.; Bryant, S. D.; Caliendo, Giuseppe
Microwave enhanced solution synthesis of 1,4-benzodiazepin-5-ones. 1.1 Articolo in rivista 2001 Santagada, Vincenzo; Perissutti, Elisa; Fiorino, Ferdinando; Vivenzio, B; Caliendo, Giuseppe
Synthesis and Structure-Activity Relationships of Antiinflammatory 1-Methyl-2-(4-X-benzoyl)imidazole-5-acetic Acids. 1.1 Articolo in rivista 1994 Caliendo, Giuseppe; Cirino, Giuseppe; Greco, Giovanni; Novellino, Ettore; Perissutti, Elisa; Pinto, A.; Santagada, Vincenzo; Silipo, Carlo; Sorrentino, Ludovico
Synthesis of benzamide derivatives and their evaluation as antiprion agents 1.1 Articolo in rivista 2012 Fiorino, Ferdinando; M., Eiden; A., Giese; Severino, Beatrice; A., Esposito; M. H., Groschup; Perissutti, Elisa; Magli, Elisa; Incisivo, GIUSEPPINA MARIA; Ciano, Antonio; Frecentese, Francesco; H. A., Kretzschmar; J., Wagner; Santagada, Vincenzo; Caliendo, Giuseppe
Comparative bioavailability of two losartan formulations in healthy human volunteers after a single dose administration. 1.1 Articolo in rivista 2006 Oliveira, Ch; MEDEIROS SILVA, R; Santagada, Vincenzo; Caliendo, Giuseppe; Perissutti, Elisa; PRADO GALOPPO, M; MARCONDES REZENDE, V; BARRIENTOS ASTIGARRAGA, Re; Duarte, Mendes; DE NUCCI, G.
Structure-Affinity Relationship Studies on Benzotriazole Derivatives Binding to 5-HT Receptor Subtypes. 1.1 Articolo in rivista 1996 Caliendo, Giuseppe; Greco, Giovanni; Grieco, Paolo; Novellino, Ettore; Perissutti, Elisa; Santagada, Vincenzo; Barbarulo, D.; Esposito, E.; De Blasi, A.
Synthesis, Pharmacological Evaluation, and Molecular Modeling Studies of Novel Peptidic CAAX Analogues as Farnesyl-Protein-Transferase Inhibitors 1.1 Articolo in rivista 2006 Santagada, Vincenzo; Caliendo, Giuseppe; Severino, Beatrice; Lavecchia, Antonio; Perissutti, Elisa; Fiorino, Ferdinando; Zampella, Angela; Sepe, Valentina; Califano, D.; Santelli, G.; Novellino, Ettore