Sfoglia per Autore
Chiral phenoxyacetic acid analogues inhibit colon cancer cell proliferation acting as PPARγ partial agonists
2019 Sabatino, L.; Ziccardi, P.; Cerchia, C.; Muccillo, L.; Piemontese, L.; Loiodice, F.; Colantuoni, V.; Lupo, A.; Lavecchia, A.
Recent advances in developing PCSK9 inhibitors for lipid-lowering therapy
2019 Lavecchia, A.; Cerchia, C.
Development of novel amides as noncovalent inhibitors of immunoproteasomes
2019 Ettari, R.; Cerchia, C.; Maiorana, S.; Guccione, M.; Novellino, E.; Bitto, A.; Grasso, S.; Lavecchia, A.; Zappala, M.
Novel Phenyldiazenyl Fibrate Analogues as PPAR α/γ/δ Pan-Agonists for the Amelioration of Metabolic Syndrome
2019 Giampietro, L.; Laghezza, A.; Cerchia, C.; Florio, R.; Recinella, L.; Capone, F.; Ammazzalorso, A.; Bruno, I.; De Filippis, B.; Fantacuzzi, M.; Ferrante, C.; Maccallini, C.; Tortorella, P.; Verginelli, F.; Brunetti, L.; Cama, A.; Amoroso, R.; Loiodice, F.; Lavecchia, A.
Discovery of Novel Naphthylphenylketone and Naphthylphenylamine Derivatives as Cell Division Cycle 25B (CDC25B) Phosphatase Inhibitors: Design, Synthesis, Inhibition Mechanism, and in Vitro Efficacy against Melanoma Cell Lines
2019 Cerchia, Carmen; Nasso, Rosarita; Mori, Matteo; Villa, Stefania; Gelain, Arianna; Capasso, Alessandra; Aliotta, Federica; Simonetti, Martina; Rullo, Rosario; Masullo, Mariorosario; DE VENDITTIS, Emmanuele; Ruocco, MARIA ROSARIA; Lavecchia, Antonio
Identification of the First PPARα/γ Dual Agonist Able to Bind to Canonical and Alternate Sites of PPARγ and to Inhibit its Cdk5-Mediated Phosphorylation
2018 Laghezza, Antonio; Piemontese, Luca; Cerchia, Carmen; Montanari, Roberta; Capelli, Davide; Giudici, Marco; Crestani, Maurizio; Tortorella, Paolo; Peiretti, Franck; Pochetti, Giorgio; Lavecchia, Antonio; Loiodice, Fulvio
Selective PPARγ modulators for Type 2 diabetes treatment: How far have we come and what does the future hold?
2018 Lavecchia, Antonio; Cerchia, Carmen
Characterization of novel inhibitors of CDC25 phosphatases: biochemical and biological analysis
2017 Nasso, Rosarita; Masullo, Mariorosario; Rullo, Rosario; Simonetti, Martina; Arcucci, Alessandro; Granato, Giuseppina; Cerchia, Carmen; Lavecchia, Antonio; Ruocco, MARIA ROSARIA; DE VENDITTIS, Emmanuele
New diphenylmethane derivatives as peroxisome proliferator-activated receptor alpha/gamma dual agonists endowed with anti-proliferative effects and mitochondrial activity
2017 Piemontese, Luca; Cerchia, Carmen; Laghezza, Antonio; Ziccardi, Pamela; Sblano, Sabina; Tortorella, Paolo; Iacobazzi, Vito; Infantino, Vittoria; Convertini, Paolo; Dal Piaz, Fabrizio; Lupo, Angelo; Colantuoni, Vittorio; Lavecchia, Antonio; Loiodice, Fulvio
Exploring the Role of N(6)-Substituents in Potent Dual Acting 5'-C-Ethyltetrazolyladenosine Derivatives: Synthesis, Binding, Functional Assays, and Antinociceptive Effects in Mice
2017 Petrelli, Riccardo; Scortichini, Mirko; Kachler, Sonja; Boccella, Serena; Cerchia, Carmen; Torquati, Ilaria; Del Bello, Fabio; Salvemini, Daniela; Novellino, Ettore; Luongo, Livio; Maione, Sabatino; Jacobson, Kenneth A; Lavecchia, Antonio; Klotz, Karl-Norbert; Cappellacci, Loredana
Small Molecule Drugs And Targeted Therapy For Melanoma: Current Strategies And Future Directions
2017 Cerchia, Carmen; Lavecchia, Antonio
Exploring structural relationships between bioactive and commercial chemical space and developing target hypotheses for compound acquisition
2017 Cerchia, Carmen; Dimova, Dilyana; Lavecchia, Antonio; Bajorath, Jürgen
A compound-based proteomic approach discloses 15-ketoatractyligenin methyl ester as a new PPARγ partial agonist with anti-proliferative ability
2017 Vasaturo, Michele; Fiengo, Lorenzo; De Tommasi, Nunziatina; Sabatino, Lina; Ziccardi, Pamela; Colantuoni, Vittorio; Bruno, Maurizio; Cerchia, Carmen; Novellino, Ettore; Lupo, Angelo; Lavecchia, Antonio; Piaz, Fabrizio Dal
Structural basis for PPAR partial or full activation revealed by a novel ligand binding mode
2016 Capelli, Davide; Cerchia, Carmen; Montanari, Roberta; Loiodice, Fulvio; Tortorella, Paolo; Laghezza, Antonio; Cervoni, Laura; Pochetti, Giorgio; Lavecchia, Antonio
In silico methods to address polypharmacology: Current status, applications and future perspectives
2016 Lavecchia, Antonio; Cerchia, Carmen
Novel Non-Peptide Small Molecules Preventing IKKβ/NEMO Association Inhibit NF-κB Activation in LPS-Stimulated J774 Macrophages
2016 DE FALCO, Francesca; DI GIOVANNI, Carmen; Cerchia, Carmen; DE STEFANO, Daniela; Capuozzo, Antonella; Irace, Carlo; Iuvone, Teresa; Santamaria, Rita; Carnuccio, Rosa; Lavecchia, Antonio
The antiproliferative and proapoptotic effects of cladosporols A and B are related to their different binding mode as PPARγ ligands
2016 Zurlo, Diana; Ziccardi, Pamela; Votino, Carolina; Colangelo, Tommaso; Cerchia, Carmen; Dal Piaz, Fabrizio; Dallavalle, Sabrina; Moricca, Salvatore; Novellino, Ettore; Lavecchia, Antonio; Colantuoni, Vittorio; Lupo, Angelo
Ligand-based chemoinformatic discovery of a novel small molecule inhibitor targeting CDC25 dual specificity phosphatases and displaying in vitro efficacy against melanoma cells
2015 Capasso, Alessandra; Cerchia, Carmen; Di Giovanni, Carmen; Granato, Giuseppina; Albano, Francesco; Romano, Simona; De Vendittis, Emmanuele; Ruocco, Maria Rosaria; Lavecchia, Antonio
Cdc25 inhibitors in melanoma cells
2014 Capasso, Alessandra; Cerchia, Carmen; DI GIOVANNI, Carmen; Granato, Giuseppina; Bertoni, Alessandra; Albano, Francesco; DE VENDITTIS, Emmanuele; Ruocco, MARIA ROSARIA; Lavecchia, Antonio
Novel inhibitors of signal transducer and activator of transcription 3 signaling pathway: an update on the recent patent literature
2014 Lavecchia, Antonio; DI GIOVANNI, Carmen; Cerchia, Carmen
Titolo | Tipologia | Data di pubblicazione | Autore(i) | File |
---|---|---|---|---|
Chiral phenoxyacetic acid analogues inhibit colon cancer cell proliferation acting as PPARγ partial agonists | 1.1 Articolo in rivista | 2019 | Sabatino, L.; Ziccardi, P.; Cerchia, C.; Muccillo, L.; Piemontese, L.; Loiodice, F.; Colantuoni, V.; Lupo, A.; Lavecchia, A. | |
Recent advances in developing PCSK9 inhibitors for lipid-lowering therapy | 1.1 Articolo in rivista | 2019 | Lavecchia, A.; Cerchia, C. | |
Development of novel amides as noncovalent inhibitors of immunoproteasomes | 1.1 Articolo in rivista | 2019 | Ettari, R.; Cerchia, C.; Maiorana, S.; Guccione, M.; Novellino, E.; Bitto, A.; Grasso, S.; Lavecchia, A.; Zappala, M. | |
Novel Phenyldiazenyl Fibrate Analogues as PPAR α/γ/δ Pan-Agonists for the Amelioration of Metabolic Syndrome | 1.1 Articolo in rivista | 2019 | Giampietro, L.; Laghezza, A.; Cerchia, C.; Florio, R.; Recinella, L.; Capone, F.; Ammazzalorso, A.; Bruno, I.; De Filippis, B.; Fantacuzzi, M.; Ferrante, C.; Maccallini, C.; Tortorella, P.; Verginelli, F.; Brunetti, L.; Cama, A.; Amoroso, R.; Loiodice, F.; Lavecchia, A. | |
Discovery of Novel Naphthylphenylketone and Naphthylphenylamine Derivatives as Cell Division Cycle 25B (CDC25B) Phosphatase Inhibitors: Design, Synthesis, Inhibition Mechanism, and in Vitro Efficacy against Melanoma Cell Lines | 1.1 Articolo in rivista | 2019 | Cerchia, Carmen; Nasso, Rosarita; Mori, Matteo; Villa, Stefania; Gelain, Arianna; Capasso, Alessandra; Aliotta, Federica; Simonetti, Martina; Rullo, Rosario; Masullo, Mariorosario; DE VENDITTIS, Emmanuele; Ruocco, MARIA ROSARIA; Lavecchia, Antonio | |
Identification of the First PPARα/γ Dual Agonist Able to Bind to Canonical and Alternate Sites of PPARγ and to Inhibit its Cdk5-Mediated Phosphorylation | 1.1 Articolo in rivista | 2018 | Laghezza, Antonio; Piemontese, Luca; Cerchia, Carmen; Montanari, Roberta; Capelli, Davide; Giudici, Marco; Crestani, Maurizio; Tortorella, Paolo; Peiretti, Franck; Pochetti, Giorgio; Lavecchia, Antonio; Loiodice, Fulvio | |
Selective PPARγ modulators for Type 2 diabetes treatment: How far have we come and what does the future hold? | 1.1 Articolo in rivista | 2018 | Lavecchia, Antonio; Cerchia, Carmen | |
Characterization of novel inhibitors of CDC25 phosphatases: biochemical and biological analysis | 4.2 Abstract in Atti di convegno | 2017 | Nasso, Rosarita; Masullo, Mariorosario; Rullo, Rosario; Simonetti, Martina; Arcucci, Alessandro; Granato, Giuseppina; Cerchia, Carmen; Lavecchia, Antonio; Ruocco, MARIA ROSARIA; DE VENDITTIS, Emmanuele | |
New diphenylmethane derivatives as peroxisome proliferator-activated receptor alpha/gamma dual agonists endowed with anti-proliferative effects and mitochondrial activity | 1.1 Articolo in rivista | 2017 | Piemontese, Luca; Cerchia, Carmen; Laghezza, Antonio; Ziccardi, Pamela; Sblano, Sabina; Tortorella, Paolo; Iacobazzi, Vito; Infantino, Vittoria; Convertini, Paolo; Dal Piaz, Fabrizio; Lupo, Angelo; Colantuoni, Vittorio; Lavecchia, Antonio; Loiodice, Fulvio | |
Exploring the Role of N(6)-Substituents in Potent Dual Acting 5'-C-Ethyltetrazolyladenosine Derivatives: Synthesis, Binding, Functional Assays, and Antinociceptive Effects in Mice | 1.1 Articolo in rivista | 2017 | Petrelli, Riccardo; Scortichini, Mirko; Kachler, Sonja; Boccella, Serena; Cerchia, Carmen; Torquati, Ilaria; Del Bello, Fabio; Salvemini, Daniela; Novellino, Ettore; Luongo, Livio; Maione, Sabatino; Jacobson, Kenneth A; Lavecchia, Antonio; Klotz, Karl-Norbert; Cappellacci, Loredana | |
Small Molecule Drugs And Targeted Therapy For Melanoma: Current Strategies And Future Directions | 1.1 Articolo in rivista | 2017 | Cerchia, Carmen; Lavecchia, Antonio | |
Exploring structural relationships between bioactive and commercial chemical space and developing target hypotheses for compound acquisition | 1.1 Articolo in rivista | 2017 | Cerchia, Carmen; Dimova, Dilyana; Lavecchia, Antonio; Bajorath, Jürgen | |
A compound-based proteomic approach discloses 15-ketoatractyligenin methyl ester as a new PPARγ partial agonist with anti-proliferative ability | 1.1 Articolo in rivista | 2017 | Vasaturo, Michele; Fiengo, Lorenzo; De Tommasi, Nunziatina; Sabatino, Lina; Ziccardi, Pamela; Colantuoni, Vittorio; Bruno, Maurizio; Cerchia, Carmen; Novellino, Ettore; Lupo, Angelo; Lavecchia, Antonio; Piaz, Fabrizio Dal | |
Structural basis for PPAR partial or full activation revealed by a novel ligand binding mode | 1.1 Articolo in rivista | 2016 | Capelli, Davide; Cerchia, Carmen; Montanari, Roberta; Loiodice, Fulvio; Tortorella, Paolo; Laghezza, Antonio; Cervoni, Laura; Pochetti, Giorgio; Lavecchia, Antonio | |
In silico methods to address polypharmacology: Current status, applications and future perspectives | 1.1 Articolo in rivista | 2016 | Lavecchia, Antonio; Cerchia, Carmen | |
Novel Non-Peptide Small Molecules Preventing IKKβ/NEMO Association Inhibit NF-κB Activation in LPS-Stimulated J774 Macrophages | 1.1 Articolo in rivista | 2016 | DE FALCO, Francesca; DI GIOVANNI, Carmen; Cerchia, Carmen; DE STEFANO, Daniela; Capuozzo, Antonella; Irace, Carlo; Iuvone, Teresa; Santamaria, Rita; Carnuccio, Rosa; Lavecchia, Antonio | |
The antiproliferative and proapoptotic effects of cladosporols A and B are related to their different binding mode as PPARγ ligands | 1.1 Articolo in rivista | 2016 | Zurlo, Diana; Ziccardi, Pamela; Votino, Carolina; Colangelo, Tommaso; Cerchia, Carmen; Dal Piaz, Fabrizio; Dallavalle, Sabrina; Moricca, Salvatore; Novellino, Ettore; Lavecchia, Antonio; Colantuoni, Vittorio; Lupo, Angelo | |
Ligand-based chemoinformatic discovery of a novel small molecule inhibitor targeting CDC25 dual specificity phosphatases and displaying in vitro efficacy against melanoma cells | 1.1 Articolo in rivista | 2015 | Capasso, Alessandra; Cerchia, Carmen; Di Giovanni, Carmen; Granato, Giuseppina; Albano, Francesco; Romano, Simona; De Vendittis, Emmanuele; Ruocco, Maria Rosaria; Lavecchia, Antonio | |
Cdc25 inhibitors in melanoma cells | 1.5 Abstract in rivista | 2014 | Capasso, Alessandra; Cerchia, Carmen; DI GIOVANNI, Carmen; Granato, Giuseppina; Bertoni, Alessandra; Albano, Francesco; DE VENDITTIS, Emmanuele; Ruocco, MARIA ROSARIA; Lavecchia, Antonio | |
Novel inhibitors of signal transducer and activator of transcription 3 signaling pathway: an update on the recent patent literature | 1.1 Articolo in rivista | 2014 | Lavecchia, Antonio; DI GIOVANNI, Carmen; Cerchia, Carmen |
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