4,5-Dihydroxypyrimidine Carboxamides and N-Alkyl-5-hydroxypyrimidinone Carboxamides Are Potent, Selective HIV Integrase Inhibitors with Good Pharmacokinetic Profiles in Preclinical Species / Summa, V., Petrocchi, ., Alessia, ., Matassa, ., Victor, G., Gardelli, ., Cristina, ., Muraglia, ., Ester, ., Rowley, ., Michael, ., Paz, ., Odalys, G., Laufer, ., Ralph, ., Monteagudo, ., Edith, ., Pace, ., Paola,. - In: JOURNAL OF MEDICINAL CHEMISTRY. - ISSN 0022-2623. - 49:23(2006), pp. 6646-6649. [10.1021/jm060854f]
4,5-Dihydroxypyrimidine Carboxamides and N-Alkyl-5-hydroxypyrimidinone Carboxamides Are Potent, Selective HIV Integrase Inhibitors with Good Pharmacokinetic Profiles in Preclinical Species
Summa V
;
2006
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