SUMMA, Vincenzo
SUMMA, Vincenzo
Dipartimento di Farmacia
Validation of an LC-MS/MS Method for the Determination of Abscisic Acid Concentration in a Real-World Setting
2023 Schiano, Elisabetta; Neri, Ilaria; Maisto, Maria; Novellino, Ettore; Iannuzzo, Fortuna; Piccolo, Vincenzo; Summa, Vincenzo; Grumetto, Lucia; Tenore, GIAN CARLO
A Food-Grade Method for Enhancing the Levels of Low Molecular Weight Proanthocyanidins with Potentially High Intestinal Bioavailability
2022 Iannuzzo, Fortuna; Piccolo, Vincenzo; Novellino, Ettore; Schiano, Elisabetta; Salviati, Emanuela; Summa, Vincenzo; Campiglia, Pietro; Carlo Tenore, Gian; Maisto, Maria
Continuous-Flow Technology for Chemical Rearrangements: A Powerful Tool to Generate Pharmaceutically Relevant Compounds
2023 Alfano, Antonella Ilenia; Pelliccia, Sveva; Rossino, Giacomo; Chianese, Orazio; Summa, Vincenzo; Collina, Simona; Brindisi, Margherita
Efficacy of selective histone deacetylase 6 inhibition in mouse models of Pseudomonas aeruginosa infection: A new glimpse for reducing inflammation and infection in cystic fibrosis
2022 Brindisi, Margherita; Barone, Simona; Rossi, Alice; Cassese, Emilia; Del Gaudio, Nunzio; Feliz Morel, Álvaro Javier; Filocamo, Gessica; Alberico, Alessia; De Fino, Ida; Gugliandolo, Davide; Babaei, Mehrad; Bove, Guglielmo; Croce, Martina; Montesano, Camilla; Altucci, Lucia; Bragonzi, Alessandra; Summa, Vincenzo
Beneficial Contribution to Glucose Homeostasis by an Agro-Food Waste Product Rich in Abscisic Acid: Results from a Randomized Controlled Trial
2022 Schiano, E.; Maisto, M.; Piccolo, V.; Novellino, E.; Annunziata, G.; Ciampaglia, R.; Montesano, C.; Croce, M.; Caruso, G.; Iannuzzo, F.; Summa, V.; Tenore, G. C.
Publisher Correction: 6-Bromoindirubin-3?-oxime intercepts GSK3 signaling to promote and enhance skeletal muscle differentiation affecting miR-206 expression in mice (Scientific Reports, (2019), 9, 1, (18091), 10.1038/s41598-019-54574-4)
2020 Ragozzino, E.; Brancaccio, M.; Di Costanzo, A.; Scalabr(`i), F.; Andolfi, G.; Wanderlingh, L. G.; Patriarca, E. J.; Minchiotti, G.; Altamura, S.; Summa, V.; Varrone, F.
Easy access to α-ketoamides as SARS-CoV-2 and MERS Mpro inhibitors via the PADAM oxidation route
2022 Pelliccia, Sveva; Cerchia, Carmen; Esposito, Francesca; Cannalire, Rolando; Corona, Angela; Costanzi, Elisa; Kuzikov, Maria; Gribbon, Philip; Zaliani, Andrea; Brindisi, Margherita; Storici, Paola; Tramontano, Enzo; Summa, Vincenzo
Discovery and Antiviral Profile of New Sulfamoylbenzamide Derivatives as HBV Capsid Assembly Modulators
2022 Ivanova Bencheva, Leda; Donnici, Lorena; Ferrante, Luca; Prandi, Adolfo; Sinisi, Roberta; De Matteo, Marilenia; Randazzo, Pietro; Conti, Matteo; Di Lucia, Pietro; Bono, Elisa; Giustini, Leonardo; Vittoria Orsale, Maria; Patsilinakos, Alexandros; Monteagudo, Edith; Iannacone, Matteo; Summa, Vincenzo; Guidotti, Luca G; De Francesco, Raffaele; Di Fabio, Romano
Cytopathic SARS-CoV-2 screening on VERO-E6 cells in a large-scale repurposing effort
2022 Zaliani, Andrea; Vangeel, Laura; Reinshagen, Jeanette; Iaconis, Daniela; Kuzikov, Maria; Keminer, Oliver; Wolf, Markus; Ellinger, Bernhard; Esposito, Francesca; Corona, Angela; Tramontano, Enzo; Manelfi, Candida; Herzog, Katja; Jochmans, Dirk; De Jonghe, Steven; Chiu, Winston; Francken, Thibault; Schepers, Joost; Collard, Caroline; Abbasi, Kayvan; Clausses, Carsten; Summa, Vincenzo; Beccari, Andrea R.; Neyts, Johan; Gribbon, Philip; Leyssen, Pieter
Application of a Rapid and Simple Technological Process to Increase Levels and Bioccessibility of Free Phenolic Compounds in Annurca Apple Nutraceutical Product
2022 Maisto, Maria; Schiano, Elisabetta; Novellino, Ettore; Piccolo, Vincenzo; Iannuzzo, Fortuna; Salviati, Emanuela; Summa, Vincenzo; Annunziata, Giuseppe; Tenore, GIAN CARLO
Anti-inflammatory and immunomodulatory activity of Mangifera indica L. reveals the modulation of COX-2/mPGES-1 axis and Th17/Treg ratio
2022 Saviano, Anella; Raucci, Federica; Casillo, Gian Marco; Mansour, Adel Abo; Piccolo, Vincenzo; Montesano, Camilla; Smimmo, Martina; Vellecco, Valentina; Capasso, Gennaro; Boscaino, Amedeo; Summa, Vincenzo; Mascolo, Nicola; Iqbal, Asif Jilani; Sorrentino, Raffaella; d'Emmanuele di Villa Bianca, Roberta; Bucci, Mariarosaria; Brancaleone, Vincenzo; Maione, Francesco
Identification and in vitro characterization of a new series of potent and highly selective G9a inhibitors as novel anti-fibroadipogenic agents
2022 Randazzo, Pietro; Sinisi, Roberta; Gornati, Davide; Bertuolo, Stefania; Bencheva, Leda; De Matteo, Marilenia; Nibbio, Martina; Monteagudo, Edith; Turcano, Lorenzo; Bianconi, Valeria; Peruzzi, Giovanna; Summa, Vincenzo; Bresciani, Alberto; Mozzetta, Chiara; Di Fabio, Romano
Natural Compounds Inhibit SARS-CoV-2 nsp13 Unwinding and ATPase Enzyme Activities
2022 Corona, Angela; Wycisk, Krzysztof; Talarico, Carmine; Manelfi, Candida; Milia, Jessica; Cannalire, Rolando; Esposito, Francesca; Gribbon, Philip; Zaliani, Andrea; Iaconis, Daniela; Beccari, Andrea R.; Summa, Vincenzo; Nowotny, Marcin; Tramontano, Enzo
Antiretroviral activity, pharmacokinetics, and tolerability of MK-0518, a novel inhibitor of HIV-1 integrase, dosed as monotherapy for 10 days in treatment-naive HIV-1-infected individuals
2006 Markowitz, M.; Morales-Ramirez, J. O.; Nguyen, B. -Y.; Kovacs, C. M.; Steigbigel, R. T.; Cooper, D. A.; Liporace, R.; Schwartz, R.; Isaacs, R.; Gilde, L. R.; Wenning, L.; Zhao, J.; Teppler, H.; Tsoukas, C.; Galpin, J.; Hicks, C.; Brown, S.; Chen, J.; Miller, M.; Hazuda, D.; Vacca, J.; Iwamoto, M.; Rowley, M.; Summa, V.
Studies of metabolism and disposition of potent human immunodeficiency virus (HIV) integrase inhibitors using 19F-NMR spectroscopy
2007 Monteagudo, ; Pesci, ; Taliani, ; Fiore, ; Petrocchi, ; Nizi, ; Rowley, ; Laufer, ; Summa, V
Thinned Nectarines, an Agro-Food Waste with Antidiabetic Potential: HPLC-HESI-MS/MS Phenolic Characterization and In Vitro Evaluation of Their Beneficial Activities
2022 Schiano, Elisabetta; Piccolo, Vincenzo; Novellino, Ettore; Maisto, Maria; Iannuzzo, Fortuna; Summa, Vincenzo; Tenore, Gian Carlo
A Focus on Severe Acute Respiratory Syndrome ( SARS ) Coronavirus ( SARS‐CoVs ) 1 and 2
2022 Cannalire, Rolando; Tramontano, Enzo; Summa, Vincenzo
Identification of Inhibitors of SARS-CoV-2 3CL-Pro Enzymatic Activity Using a Small Molecule in Vitro Repurposing Screen
2021 Kuzikov, M.; Costanzi, E.; Reinshagen, J.; Esposito, F.; Vangeel, L.; Wolf, M.; Ellinger, B.; Claussen, C.; Geisslinger, G.; Corona, A.; Iaconis, D.; Talarico, C.; Manelfi, C.; Cannalire, R.; Rossetti, G.; Gossen, J.; Albani, S.; Musiani, F.; Herzog, K.; Ye, Y.; Giabbai, B.; Demitri, N.; Jochmans, D.; Jonghe, S. D.; Rymenants, J.; Summa, V.; Tramontano, E.; Beccari, A. R.; Leyssen, P.; Storici, P.; Neyts, J.; Gribbon, P.; Zaliani, A.
Prdm16-mediated H3K9 methylation controls fibro-adipogenic progenitors identity during skeletal muscle repair
2021 Biferali, B.; Bianconi, V.; Perez, D. F.; Kronawitter, S. P.; Marullo, F.; Maggio, R.; Santini, T.; Polverino, F.; Biagioni, S.; Summa, V.; Toniatti, C.; Pasini, D.; Stricker, S.; Fabio, R. D.; Chiacchiera, F.; Peruzzi, G.; Mozzetta, C.
Personalized metabolic profile by synergic use of nmr and hrms
2021 Petrella, G.; Montesano, C.; Lentini, S.; Ciufolini, G.; Vanni, D.; Speziale, R.; Salonia, A.; Montorsi, F.; Summa, V.; Vago, R.; Orsatti, L.; Monteagudo, E.; Cicero, D. O.
Titolo | Tipologia | Data di pubblicazione | Autore(i) | File |
---|---|---|---|---|
Validation of an LC-MS/MS Method for the Determination of Abscisic Acid Concentration in a Real-World Setting | 1.1 Articolo in rivista | 2023 | Schiano, Elisabetta; Neri, Ilaria; Maisto, Maria; Novellino, Ettore; Iannuzzo, Fortuna; Piccolo, Vincenzo; Summa, Vincenzo; Grumetto, Lucia; Tenore, GIAN CARLO | |
A Food-Grade Method for Enhancing the Levels of Low Molecular Weight Proanthocyanidins with Potentially High Intestinal Bioavailability | 1.1 Articolo in rivista | 2022 | Iannuzzo, Fortuna; Piccolo, Vincenzo; Novellino, Ettore; Schiano, Elisabetta; Salviati, Emanuela; Summa, Vincenzo; Campiglia, Pietro; Carlo Tenore, Gian; Maisto, Maria | |
Continuous-Flow Technology for Chemical Rearrangements: A Powerful Tool to Generate Pharmaceutically Relevant Compounds | 1.1 Articolo in rivista | 2023 | Alfano, Antonella Ilenia; Pelliccia, Sveva; Rossino, Giacomo; Chianese, Orazio; Summa, Vincenzo; Collina, Simona; Brindisi, Margherita | |
Efficacy of selective histone deacetylase 6 inhibition in mouse models of Pseudomonas aeruginosa infection: A new glimpse for reducing inflammation and infection in cystic fibrosis | 1.1 Articolo in rivista | 2022 | Brindisi, Margherita; Barone, Simona; Rossi, Alice; Cassese, Emilia; Del Gaudio, Nunzio; Feliz Morel, Álvaro Javier; Filocamo, Gessica; Alberico, Alessia; De Fino, Ida; Gugliandolo, Davide; Babaei, Mehrad; Bove, Guglielmo; Croce, Martina; Montesano, Camilla; Altucci, Lucia; Bragonzi, Alessandra; Summa, Vincenzo | |
Beneficial Contribution to Glucose Homeostasis by an Agro-Food Waste Product Rich in Abscisic Acid: Results from a Randomized Controlled Trial | 1.1 Articolo in rivista | 2022 | Schiano, E.; Maisto, M.; Piccolo, V.; Novellino, E.; Annunziata, G.; Ciampaglia, R.; Montesano, C.; Croce, M.; Caruso, G.; Iannuzzo, F.; Summa, V.; Tenore, G. C. | |
Publisher Correction: 6-Bromoindirubin-3?-oxime intercepts GSK3 signaling to promote and enhance skeletal muscle differentiation affecting miR-206 expression in mice (Scientific Reports, (2019), 9, 1, (18091), 10.1038/s41598-019-54574-4) | 1.7 Commento, erratum, replica e simili | 2020 | Ragozzino, E.; Brancaccio, M.; Di Costanzo, A.; Scalabr(`i), F.; Andolfi, G.; Wanderlingh, L. G.; Patriarca, E. J.; Minchiotti, G.; Altamura, S.; Summa, V.; Varrone, F. | |
Easy access to α-ketoamides as SARS-CoV-2 and MERS Mpro inhibitors via the PADAM oxidation route | 1.1 Articolo in rivista | 2022 | Pelliccia, Sveva; Cerchia, Carmen; Esposito, Francesca; Cannalire, Rolando; Corona, Angela; Costanzi, Elisa; Kuzikov, Maria; Gribbon, Philip; Zaliani, Andrea; Brindisi, Margherita; Storici, Paola; Tramontano, Enzo; Summa, Vincenzo | |
Discovery and Antiviral Profile of New Sulfamoylbenzamide Derivatives as HBV Capsid Assembly Modulators | 1.1 Articolo in rivista | 2022 | Ivanova Bencheva, Leda; Donnici, Lorena; Ferrante, Luca; Prandi, Adolfo; Sinisi, Roberta; De Matteo, Marilenia; Randazzo, Pietro; Conti, Matteo; Di Lucia, Pietro; Bono, Elisa; Giustini, Leonardo; Vittoria Orsale, Maria; Patsilinakos, Alexandros; Monteagudo, Edith; Iannacone, Matteo; Summa, Vincenzo; Guidotti, Luca G; De Francesco, Raffaele; Di Fabio, Romano | |
Cytopathic SARS-CoV-2 screening on VERO-E6 cells in a large-scale repurposing effort | 1.1 Articolo in rivista | 2022 | Zaliani, Andrea; Vangeel, Laura; Reinshagen, Jeanette; Iaconis, Daniela; Kuzikov, Maria; Keminer, Oliver; Wolf, Markus; Ellinger, Bernhard; Esposito, Francesca; Corona, Angela; Tramontano, Enzo; Manelfi, Candida; Herzog, Katja; Jochmans, Dirk; De Jonghe, Steven; Chiu, Winston; Francken, Thibault; Schepers, Joost; Collard, Caroline; Abbasi, Kayvan; Clausses, Carsten; Summa, Vincenzo; Beccari, Andrea R.; Neyts, Johan; Gribbon, Philip; Leyssen, Pieter | |
Application of a Rapid and Simple Technological Process to Increase Levels and Bioccessibility of Free Phenolic Compounds in Annurca Apple Nutraceutical Product | 1.1 Articolo in rivista | 2022 | Maisto, Maria; Schiano, Elisabetta; Novellino, Ettore; Piccolo, Vincenzo; Iannuzzo, Fortuna; Salviati, Emanuela; Summa, Vincenzo; Annunziata, Giuseppe; Tenore, GIAN CARLO | |
Anti-inflammatory and immunomodulatory activity of Mangifera indica L. reveals the modulation of COX-2/mPGES-1 axis and Th17/Treg ratio | 1.1 Articolo in rivista | 2022 | Saviano, Anella; Raucci, Federica; Casillo, Gian Marco; Mansour, Adel Abo; Piccolo, Vincenzo; Montesano, Camilla; Smimmo, Martina; Vellecco, Valentina; Capasso, Gennaro; Boscaino, Amedeo; Summa, Vincenzo; Mascolo, Nicola; Iqbal, Asif Jilani; Sorrentino, Raffaella; d'Emmanuele di Villa Bianca, Roberta; Bucci, Mariarosaria; Brancaleone, Vincenzo; Maione, Francesco | |
Identification and in vitro characterization of a new series of potent and highly selective G9a inhibitors as novel anti-fibroadipogenic agents | 1.1 Articolo in rivista | 2022 | Randazzo, Pietro; Sinisi, Roberta; Gornati, Davide; Bertuolo, Stefania; Bencheva, Leda; De Matteo, Marilenia; Nibbio, Martina; Monteagudo, Edith; Turcano, Lorenzo; Bianconi, Valeria; Peruzzi, Giovanna; Summa, Vincenzo; Bresciani, Alberto; Mozzetta, Chiara; Di Fabio, Romano | |
Natural Compounds Inhibit SARS-CoV-2 nsp13 Unwinding and ATPase Enzyme Activities | 1.1 Articolo in rivista | 2022 | Corona, Angela; Wycisk, Krzysztof; Talarico, Carmine; Manelfi, Candida; Milia, Jessica; Cannalire, Rolando; Esposito, Francesca; Gribbon, Philip; Zaliani, Andrea; Iaconis, Daniela; Beccari, Andrea R.; Summa, Vincenzo; Nowotny, Marcin; Tramontano, Enzo | |
Antiretroviral activity, pharmacokinetics, and tolerability of MK-0518, a novel inhibitor of HIV-1 integrase, dosed as monotherapy for 10 days in treatment-naive HIV-1-infected individuals | 1.2 Recensione in rivista | 2006 | Markowitz, M.; Morales-Ramirez, J. O.; Nguyen, B. -Y.; Kovacs, C. M.; Steigbigel, R. T.; Cooper, D. A.; Liporace, R.; Schwartz, R.; Isaacs, R.; Gilde, L. R.; Wenning, L.; Zhao, J.; Teppler, H.; Tsoukas, C.; Galpin, J.; Hicks, C.; Brown, S.; Chen, J.; Miller, M.; Hazuda, D.; Vacca, J.; Iwamoto, M.; Rowley, M.; Summa, V. | |
Studies of metabolism and disposition of potent human immunodeficiency virus (HIV) integrase inhibitors using 19F-NMR spectroscopy | 1.1 Articolo in rivista | 2007 | Monteagudo, ; Pesci, ; Taliani, ; Fiore, ; Petrocchi, ; Nizi, ; Rowley, ; Laufer, ; Summa, V | |
Thinned Nectarines, an Agro-Food Waste with Antidiabetic Potential: HPLC-HESI-MS/MS Phenolic Characterization and In Vitro Evaluation of Their Beneficial Activities | 1.1 Articolo in rivista | 2022 | Schiano, Elisabetta; Piccolo, Vincenzo; Novellino, Ettore; Maisto, Maria; Iannuzzo, Fortuna; Summa, Vincenzo; Tenore, Gian Carlo | |
A Focus on Severe Acute Respiratory Syndrome ( SARS ) Coronavirus ( SARS‐CoVs ) 1 and 2 | 3.1 Monografia o trattato scientifico | 2022 | Cannalire, Rolando; Tramontano, Enzo; Summa, Vincenzo | |
Identification of Inhibitors of SARS-CoV-2 3CL-Pro Enzymatic Activity Using a Small Molecule in Vitro Repurposing Screen | 1.1 Articolo in rivista | 2021 | Kuzikov, M.; Costanzi, E.; Reinshagen, J.; Esposito, F.; Vangeel, L.; Wolf, M.; Ellinger, B.; Claussen, C.; Geisslinger, G.; Corona, A.; Iaconis, D.; Talarico, C.; Manelfi, C.; Cannalire, R.; Rossetti, G.; Gossen, J.; Albani, S.; Musiani, F.; Herzog, K.; Ye, Y.; Giabbai, B.; Demitri, N.; Jochmans, D.; Jonghe, S. D.; Rymenants, J.; Summa, V.; Tramontano, E.; Beccari, A. R.; Leyssen, P.; Storici, P.; Neyts, J.; Gribbon, P.; Zaliani, A. | |
Prdm16-mediated H3K9 methylation controls fibro-adipogenic progenitors identity during skeletal muscle repair | 1.1 Articolo in rivista | 2021 | Biferali, B.; Bianconi, V.; Perez, D. F.; Kronawitter, S. P.; Marullo, F.; Maggio, R.; Santini, T.; Polverino, F.; Biagioni, S.; Summa, V.; Toniatti, C.; Pasini, D.; Stricker, S.; Fabio, R. D.; Chiacchiera, F.; Peruzzi, G.; Mozzetta, C. | |
Personalized metabolic profile by synergic use of nmr and hrms | 1.1 Articolo in rivista | 2021 | Petrella, G.; Montesano, C.; Lentini, S.; Ciufolini, G.; Vanni, D.; Speziale, R.; Salonia, A.; Montorsi, F.; Summa, V.; Vago, R.; Orsatti, L.; Monteagudo, E.; Cicero, D. O. |