BRINDISI, MARGHERITA

BRINDISI, MARGHERITA  

Dipartimento di Farmacia  

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Titolo Tipologia Data di pubblicazione Autore(i) File
Achmatowicz reaction and its application in the syntheses of bioactive molecules 1.1 Articolo in rivista 2016 Ghosh Arun, K.; Brindisi, Margherita
Activation of the Wnt pathway by small peptides: rational design, synthesis and biological evaluation 1.1 Articolo in rivista 2017 Brogi, Simone; Maramai, Samuele; Brindisi, Margherita; Chemi, Giulia; Porcari, Valentina; Corallo, Claudio; Gennari, Luigi; Novellino, Ettore; Ramunno, Anna; Butini, Stefania; Campiani, Giuseppe; Gemma, Sandra
Allosteric Modulation of Ionotropic Glutamate Receptors: An Outlook on New Therapeutic Approaches To Treat Central Nervous System Disorders 1.1 Articolo in rivista 2019 Brogi, Simone; Campiani, Giuseppe; Brindisi, Margherita; Butini, Stefania
Amide Bonds Meet Flow Chemistry: A Journey into Methodologies and Sustainable Evolution 1.1 Articolo in rivista 2022 Alfano, A. L.; Lange, H.; Brindisi, M.
An efficient approach to chiral C8/C9-piperazino-substituted 1,4-benzodiazepin-2-ones as peptidomimetic scaffolds. 1.1 Articolo in rivista 2008 Butini, S.; Gabellieri, E.; Huleatt, P. B.; Campiani, G.; Franceschini, S.; Brindisi, M.; Ros, S.; Sanna Coccone, S.; Fiorini, I.; Novellino, Ettore; Giorgi, G.; Gemma, S.
Antimalarial agents against both sexual and asexual parasites stages: structure-activity relationships and biological studies of the Malaria Box compound 1-[5-(4-bromo-2-chlorophenyl)furan-2-yl]- N -[(piperidin-4-yl)methyl]methanamine (MMV019918) and analogues 1.1 Articolo in rivista 2018 Vallone, Alessandra; D'Alessandro, Sarah; Brogi, Simone; Brindisi, Margherita; Chemi, Giulia; Alfano, Gloria; Lamponi, Stefania; Lee, Soon Goo; Jez, Joseph M.; Koolen, Karin J. M.; Dechering, Koen J.; Saponara, Simona; Fusi, Fabio; Gorelli, Beatrice; Taramelli, Donatella; Parapini, Silvia; Caldelari, Reto; Campiani, Giuseppe; Gemma, Sandra; Butini, Stefania
Asymmetric Diels-Alder reaction of 3-(acyloxy)acryloyl oxazolidinones: Optically active synthesis of a high-affinity ligand for potent HIV-1 protease inhibitors 1.1 Articolo in rivista 2019 Ghosh, A. K.; Grillo, A.; Kovela, S.; Brindisi, M.
Autophagy modulators for the treatment of oral and esophageal squamous cell carcinomas 1.1 Articolo in rivista 2020 Khan, T.; Relitti, N.; Brindisi, M.; Magnano, S.; Zisterer, D.; Gemma, S.; Butini, S.; Campiani, G.
Breakthroughs in medicinal chemistry: New targets and mechanisms, new drugs, new hopes-7 1.2 Recensione in rivista 2020 Gutschow, M.; Eynde, J. J. V.; Jampilek, J.; Kang, C.; Mangoni, A. A.; Fossa, P.; Karaman, R.; Trabocchi, A.; Scott, P. J. H.; Reynisson, J.; Rapposelli, S.; Galdiero, S.; Winum, J. -Y.; Brullo, C.; Prokai-Tatrai, K.; Sharma, A. K.; Schapira, M.; Azuma, Y. -T.; Cerchia, L.; Spete, M.; Torri, G.; Collina, S.; Geronikaki, A.; Garcia-Sosa, A. T.; Helena Vasconcelos, M.; Sousa, M. E.; Kosalec, I.; Tuccinardi, T.; Duarte, I. F.; Salvador, J. A. R.; Bertinaria, M.; Pellecchia, M.; Amato, J.; Rastelli, G.; Gomes, P. A. C.; Guedes, R. C.; Sabatier, J. -M.; Estevez-Braun, A.; Pagano, B.; Mangani, S.; Ragno, R.; Kokotos, G.; Brindisi, M.; Gonzalez, F. V.; Borges, F.; Miloso, M.; Rautio, J.; Munoz-Torrero, D.
Bridged bicyclic 2,3-dioxabicyclo[3.3.1]nonanes as antiplasmodial agents: Synthesis, structure-activity relationships and studies on their biomimetic reaction with Fe(II) 1.1 Articolo in rivista 2019 D'Alessandro, S.; Alfano, G.; Di Cerbo, L.; Brogi, S.; Chemi, G.; Relitti, N.; Brindisi, M.; Lamponi, S.; Novellino, E.; Campiani, G.; Gemma, S.; Basilico, N.; Taramelli, D.; Baratto, M. C.; Pogni, R.; Butini, S.
Chasing a Breath of Fresh Air in Cystic Fibrosis (CF): Therapeutic Potential of Selective HDAC6 Inhibitors to Tackle Multiple Pathways in CF Pathophysiology 1.1 Articolo in rivista 2022 Barone, S.; Cassese, E.; Alfano, A. I.; Brindisi, M.; Summa, V.
Computational tool for fast in silico evaluation of hERG K+ channel affinity 1.1 Articolo in rivista 2017 Chemi, Giulia; Gemma, Sandra; Campiani, Giuseppe; Brogi, Simone; Butini, Stefania; Brindisi, Margherita
Coupling Interrupted Fischer and Multicomponent Joullié-Ugi to Chase Chemical Diversity: from Batch to Sustainable Flow Synthesis of Peptidomimetics 1.1 Articolo in rivista 2021 Alfano, A. I.; Buommino, E.; Ferraro, M. G.; Irace, C.; Zampella, A.; Lange, H.; Brindisi, M.
The Curtius Rearrangement: Applications in Modern Drug Discovery and Medicinal Chemistry 1.1 Articolo in rivista 2018 Ghosh, A. K.; Brindisi, M.; Sarkar, A.
The Curtius rearrangement: mechanistic insight and recent applications in natural product syntheses 1.1 Articolo in rivista 2018 Ghosh, Arun K.; Sarkar, Anindya; Brindisi, Margherita
Dealing with schistosomiasis: Current drug discovery strategies 2.1 Contributo in volume (Capitolo o Saggio) 2019 Gemma, S.; Federico, S.; Brogi, S.; Brindisi, M.; Butini, S.; Campiani, G.
Design and Synthesis of Highly Potent HIV-1 Protease Inhibitors Containing Tricyclic Fused Ring Systems as Novel P2 Ligands: Structure-Activity Studies, Biological and X-ray Structural Analysis 1.1 Articolo in rivista 2018 Ghosh, A. K.; Nyalapatla, R. P.; Kovela, S.; Rao, K. V.; Brindisi, M.; Osswald, H. L.; Amano, M.; Aoki, M.; Agniswamy, J.; Wang, Y. -F.; Weber, I. T.; Mitsuya, H.
Design of Highly Potent, Dual-Acting and Central-Nervous-System-Penetrating HIV-1 Protease Inhibitors with Excellent Potency against Multidrug-Resistant HIV-1 Variants 1.1 Articolo in rivista 2018 Ghosh, Arun K; Rao, Kalapala Venkateswara; Nyalapatla, Prasanth R; Kovela, Satish; Brindisi, Margherita; Osswald, Heather L; Sekhara Reddy, Bhavanam; Agniswamy, Johnson; Wang, Yuan-Fang; Aoki, Manabu; Hattori, Shin-Ichiro; Weber, Irene T; Mitsuya, Hiroaki
Design of novel HIV-1 protease inhibitors incorporating isophthalamide-derived P2-P3 ligands: Synthesis, biological evaluation and X-ray structural studies of inhibitor-HIV-1 protease complex 1.1 Articolo in rivista 2017 Ghosh, Arun K.; Brindisi, Margherita; Nyalapatla, Prasanth R.; Takayama, Jun; Ella-Menye, Jean-Rene; Yashchuk, Sofiya; Agniswamy, Johnson; Wang, Yuan-Fang; Aoki, Manabu; Amano, Masayuki; Weber, Irene T.; Mitsuya, Hiroaki
Design, Synthesis and Structure-Activity Relationship Studies of 4-Quinolinyl- and 9-Acrydinylhydrazones as Potent Antimalarial Agents 1.1 Articolo in rivista 2008 Fattorusso, Caterina; Campiani, G; Kukreja, G; Persico, Marco; Butini, S; Romano, Mp; Altarelli, M; Ros, S; Brindisi, Margherita; Savini, L; Novellino, Ettore; Nacci, V; Fattorusso, Ernesto; Parapini, S; Basilico, N; Taramelli, D; Yardley, V; Croft, S; Borriello, M; AND GEMMA, S.