GRIECO, PAOLO

GRIECO, PAOLO  

DIPARTIMENTO DI FARMACIA  

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Titolo Tipologia Data di pubblicazione Autore(i) File
Cyclic peptides acting as urotensin-II antagonists. 6.1 Brevetto 2005 Novellino, Ettore; Grieco, Paolo; Rovero, P.
D-Amino Acid Scan of g-Melanocyte-Stimulating hormone:importance of the Trp8 1.1 Articolo in rivista 2000 Grieco, Paolo; Balse, P. M.; Weinberg, D.; Macneil, T.
" Molecular Modelingof the Urotensin-II receptor Complex" 4.1 Articoli in Atti di convegno 2004 Grieco, Paolo; Lavecchia, A.; Campiglia, P.; Lama, T.; Rovero, P.; Carotenuto, Alfonso; Patacchini, R.; Maggi, C. A.; Novellino, Ettore
A structure – activity relationship study on position –2 of the Gas C-terminal peptide able to inhibit Gs activation by A2A adenosine receptor. 1.1 Articolo in rivista 2003 Grieco, Paolo; Albrizio, Stefania; D’Ursi, A. M.; Giusti, L.; Mazzoni, M. R.; Novellino, E.; Rovero, P.
Phenol derived CVFM analogs inhibitors of ras farnesyl transferase possessing cellular in vitro activity. 1.1 Articolo in rivista 1998 Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; Ramunno, Anna; Santagada, Vincenzo; Albrizio, Stefania; Califano, D.; Giuliano, A.; Santelli, G.
Synthesis and Binding Affinities for 5-HT1A, 5-HT2A and 5-HT2C receptors of a series of 1- and 2-(4-arylpiperazinylalkyl)-4-(benzoyl)-1,2,3-triazole derivatives. 1.1 Articolo in rivista 1999 Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; Santagada, Vincenzo; Albrizio, Stefania; Spadola, L.; Bruni, G.; Romeo, M. R.
Structure-Activity Relationships of Novel Cyclic alpha-MSH/gamma-MSH Hybrid Analogues which Lead to Potent and Selective Ligands for the Human MC3R and Human MC5R 1.1 Articolo in rivista 2003 Balse, Srinivasan; P., M.; Grieco, Paolo; P, Cai; M, Trivedi; D, Hruby; V., J.
Extensive Structure-Activity Studies of Lactam Derivatives of MT-II and SHU9119: Their activity and Selectivity at Human Melanocortin Receptors 3,4 and, 5. 1.1 Articolo in rivista 2003 Grieco, Paolo; P, Balsesrinivasan; P, Han; G, Weinberg; D, Macnail; T, ; VAN DER, Ploeg; L. H. T, Hruby; V., J.
Melanocortin type 3 receptor null mice are refractory to the inhibitory actions of a selective receptor agonist in experimental acute inflammation 1.1 Articolo in rivista 2006 Getting, J. S.; Lam, C. W.; Chen, A. S.; Grieco, Paolo; Perretti, M.
New melanocortin peptides useful as medicament against Staphylococcus aureus, Candida albicans, Pseudomonas aeruginosa, Candida glabrata or Candida krusei 6.1 Brevetto 2010 Bonino, F.; Catania, A.; Grieco, Paolo; Novellino, Ettore
New dimensions in the design of potent and receptor selective melanotropin analogues 2.1 Contributo in volume (Capitolo o Saggio) 2000 Grieco, Paolo; Han, G.; Hruby, V. J.
Novel peptidomimetic as MMP2 inhibitors 4.1 Articoli in Atti di convegno 2007 K., Kaia; P., Campiglia; GOMEZ MONTERREY, ISABEL MARIA; M., D'Ursi; Grieco, Paolo; Novellino, Ettore
Further structure-activity studies of lactam derivatives of MT-II and SHU-9119: Their activity and selectivity at human melanocortin receptors 3, 4, and 5. 1.1 Articolo in rivista 2007 Grieco, Paolo; Cai, M.; Han, G.; Trivedi, D.; Campiglia, P.; Novellino, Ettore; Hruby, V. J.
Substitution of Arginine with Proline and Proline Derivatives in MSH Leads to Selectivity for Human Melanocortin 4 Receptor (hMC4R) 1.1 Articolo in rivista 2009 H., Qu; M., Cai; A. V., Mayorov; Grieco, Paolo; M., Zingsheim; D., Trivedi; V. J., Hruby
Design, synthesis and Cytotoxic Evaluation of a New Series of 3-Substituted-spiro[(dihydropirazin-2,5-dione)-6,3’-(2’,3’-dihydrothieno[2,3-b]naphtho-4’,9’-dione)] Derivatives 1.1 Articolo in rivista 2007 GOMEZ MONTERREY, ISABEL MARIA; P., Campiglia; Carotenuto, Alfonso; D., Califano; C., Pisano; L., Vesci; T., Lama; A., Bertamino; M., Sala; A., MAZZELLA di BOSCO; Grieco, Paolo; Novellino, Ettore
Design and Synthesis of Spirotryprostatin-inspired Diketopiperazine Systemsfrom Prolyl Spirooxoindolethiazolidine Derivatives 1.1 Articolo in rivista 2010 Bertamino, Alessia; Aquino, Claudio; M., Sala; N., de Simone; C. A., Mattia; L., Erra; S., Musella; P., Iannelli; Carotenuto, Alfonso; Grieco, Paolo; Novellino, Ettore; P., Campiglia; GOMEZ MONTERREY, ISABEL MARIA
Further Evidence that Melanocortins Prevent Myocardial Reperfusion Injury by Activating MC3 Receptors: Irrelevance of the C-terminal Arg-Phe sequenze 1.1 Articolo in rivista 2003 Mioni, C; Giuliani, D; Cainazzo, M. M; Leone, S; Iannone, C; Bazzani, C; Grieco, Paolo; P, Novellino; E, Tomasi; A, Bertolini; A, Guarini
Inflamed phenotype of the mesenteric microcirculation of melanocortin type 3 receptor null mice after ischaemia-reperfusion 1.1 Articolo in rivista 2008 G., Leoni; H. B., Patel; Sampaio, A. L. F.; Gavins, F. N. E.; Grieco, Paolo; S. J., Getting; M., Perretti
Efficient Synthesis in Solid-Phase of Freidinger-like lactams by Microwave irradiation 4.1 Articoli in Atti di convegno 2005 T., Lama; P., Campiglia; L., Auriemma; GOMEZ MONTERREY, ISABEL MARIA; Carotenuto, Alfonso; Novellino, Ettore; Grieco, Paolo
The use of microwave irradiation in peptide chemistry 1.1 Articolo in rivista 2004 Grieco, Paolo