COSIMELLI, BARBARA
COSIMELLI, BARBARA
DIPARTIMENTO DI FARMACIA
Determination of the absolute configuration of the enantiomers of an oxadiazol-3-one calcium channel blocker, resolved by chiral HPLC, via concerted use of three chiroptical spectroscopies
2012 Giovanni Battista, Barrano; Salvatore, Caccamese; Cosimelli, Barbara; Frank J., Devlin; Elda, Severi; Domenico, Spinelli
Osteoblast differentiation and survival: A role for A2B adenosine receptor allosteric modulators
2014 Maria Letizia, Trincavelli; Simona, Daniele; Chiara, Giacomelli; Sabrina, Taliani; Federico Da, Settimo; Cosimelli, Barbara; Greco, Giovanni; Novellino, Ettore; Claudia, Martini
Preliminary Finding on a New Calcium Channel Entry Blocker Chemotype: 5,6-Diamino-4-hydroxy-2-mercaptopyrimidine Derivatives
2011 Cosimelli, Barbara; Elda, Severi; Novellino, Ettore; Anna, Cavaccini; Cataldi, Mauro; Roberta, Budriesi; Matteo, Micucci; Alberto, Chiarini; Pierfranco, Ioan
Zinc phthalocyanines and corresponding conjugates, their preparation and use in photodynamic therapy and as diagnostic agents.
1999 Roncucci, G; Dei, D; DE FILIPPIS, M. P.; Fantetti, L; Masini, I; Cosimelli, Barbara; Jori, G.
From the central benzodiazepine receptor to the adenosine receptors exploiting the 3-diketoindole moiety
2011 Cosimelli, Barbara
Synthesis and biological evaluation on human glioblastoma cells of novel pyrazolo[3,4-d]pyrimidine adenosine A(3) receptor antagonists
2010 Mugnaini, L.; La Motta, C.; Taliani, S; Simorini, F.; Salerno, S.; Marini, A. M.; Da Settimo, F.; Cosimelli, Barbara; Greco, Giovanni; Novellino, Ettore; Daniele, S.; Trincavelli, M. L.; Martini, C.
Chemistry of Substituted Pyrazolo[1,5-a]pyrimidines. Part 3. A Structural Correc¬tion of Pyrazolo[1,5-a][1,3]diazepine Derivative on the Basis of 13C NMR Spectroscopy.
1993 Chimichi, S; Cosimelli, Barbara; Bruni, F; Costanzo, A.
Inhibition of MDR1 activity in vitro by a novel class of diltiazem analogues: towards new candidates
2009 Viale, M.; Cordazzo, C.; Cosimelli, Barbara; de Totero, D.; Castagnola, P.; Aiello, C.; Cianfriglia, M.; Severi, E.; Petrillo, G.; Spinelli, D.
Chemistry of substituted pyrazolo[1,5-a]pyrimidines. Part 5. 7-Oxo-6-[pyrazol-3’(5’)-yl]-4,7-dihydropyrazolo[1,5-a]pyrimidines from 6-ethoxycarbonyl-7-(2-dimethylaminovinyl)-pyrazolo[1,5-a]pyrimidines: elucidation of the reaction mechanism through NMR spectroscopy and X-Ray diffraction analysis.
1996 Chimichi, S; Bruni, F; Cosimelli, Barbara; Selleri, S; Valle, G.
Substituent effect on the redox potential of some substituted (aryl)(2-nitrobenzo[b]thiophen-3-yl)amines.
2001 Cosimelli, Barbara; Spinelli, D; Costanzo, F; Tonelli, D; Lamartina, L; Sarva', M. C.; Seeber, R.
Modulation of A2B adenosine receptor by 1-Benzyl-3-ketoindole derivatives
2013 S., Taliani; M. L., Trincavelli; Cosimelli, Barbara; Laneri, Sonia; E., Severi; E., Barresi; I., Pugliesi; S., Daniele; C., Giacomelli; Greco, Giovanni; Novellino, Ettore; C., Martini; F., Da Settimo
3-Aryl-[1,2,4]triazino[4,3-a]benzimidazol-4(10H)-one: a novel template for the design of highly selective A2B adenosine receptor antagonists
2012 Taliani, S.; Pugliesi, I.; Barresi, E.; Salerno, S.; Simorini, F.; La Motta, C.; Marini, A. M.; Da Settimo, F.; Cosconati, S.; Marinelli, Luciana; Cosimelli, Barbara; Greco, Giovanni; Novellino, Ettore; Daniele, S.; Trincavelli, M. L.; Martini, C.
Regioselective Synthesis of 4-Acetyl- and 5-Acetyl-3-methylisoxazole: their Conversion into Silyl- and Methyl Enol Ethers.
1992 Chimichi, S; Cosimelli, Barbara
Ring-ring Interconversions. Part 3. On the effect of the substituents on the thiazole moiety in the ring-opening/ring-closing reactions of nitrosoimidazo[2,1-b][1,3]thiazoles with hydrochloric acid.
2000 Billi, R; Cosimelli, Barbara; Leoni, A; Spinelli, D.
Derivatives of 4-Amino-6-hydroxy-2-mercaptopyrimidine as Novel, Potent, and Selective A3 Adenosine Receptor Antagonists
2008 Cosimelli, Barbara; Greco, Giovanni; Ehlardo, M.; Novellino, Ettore; Da Settimo, F.; Taliani, S.; La Motta, C.; Bellandi, M.; Tuccinardi, T.; Martinelli, A.; Ciampi, O.; Trincavelli, M. L.; Martini, C.
L-Type calcium channel blockers: from diltiazem to 1,2,4-oxadiazol-5-ones via thiazinooxadiazol-3-one derivatives
2009 Budriesi, R.; Cosimelli, Barbara; Ioan, P.; Ugenti, P.; Carosati, E.; Frosini, M.; Fusi, F.; Spisani, R.; Saponara, S.; Corda, G.; Cruciani, G.; Novellino, Ettore; Spinelli, D.; Chiarini, A.
A New Synthetic Route to 2,2’:5’,2”-Terthiophene-5-derivatives to Conjugate with Proteins and Monoclonal Antibodies.
1996 Cosimelli, Barbara; Neri, D; Roncucci, G.
Ring opening of 2-substituted 4-nitrothiophenes with pyrrolidine. Access to new functionalized nitro-unsaturated building blocks.
2001 Dell'Erba, C; Gabellini, A; Novi, M; Petrillo, G; Tavani, C; Cosimelli, Barbara; Spinelli, D.
Synthesis and antimycotic activity of new unsymmetrical substituted zinc phthalocyanines.
2003 Cosimelli, Barbara; Roncucci, G; Dei, D; Fantetti, L; Ferroni, F; Ricci, M; Spinelli, D.
New Fluorescent 2-Phenylindolglyoxylamide Derivatives as Probes Targeting the Peripheral-Type Benzodiazepine Receptor: Design, Synthesis and Biological Evaluation.
2007 Taliani, S.; Simorini, F.; Sergianni, V.; LA MOTTA, C.; DA SETTIMO, F.; Cosimelli, Barbara; ABIGNENTE DI FRASSELLO, Enrico; Greco, Giovanni; Novellino, Ettore; Rossi, L.; Gremigni, V.; Spinetti, F.; Chelli, B.; Martini, C.
| Titolo | Tipologia | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|---|
| Determination of the absolute configuration of the enantiomers of an oxadiazol-3-one calcium channel blocker, resolved by chiral HPLC, via concerted use of three chiroptical spectroscopies | 8.02 Comunicazioni a Convegni o Seminari | 2012 | Giovanni Battista, Barrano; Salvatore, Caccamese; Cosimelli, Barbara; Frank J., Devlin; Elda, Severi; Domenico, Spinelli | |
| Osteoblast differentiation and survival: A role for A2B adenosine receptor allosteric modulators | 1.1 Articolo in rivista | 2014 | Maria Letizia, Trincavelli; Simona, Daniele; Chiara, Giacomelli; Sabrina, Taliani; Federico Da, Settimo; Cosimelli, Barbara; Greco, Giovanni; Novellino, Ettore; Claudia, Martini | |
| Preliminary Finding on a New Calcium Channel Entry Blocker Chemotype: 5,6-Diamino-4-hydroxy-2-mercaptopyrimidine Derivatives | 1.1 Articolo in rivista | 2011 | Cosimelli, Barbara; Elda, Severi; Novellino, Ettore; Anna, Cavaccini; Cataldi, Mauro; Roberta, Budriesi; Matteo, Micucci; Alberto, Chiarini; Pierfranco, Ioan | |
| Zinc phthalocyanines and corresponding conjugates, their preparation and use in photodynamic therapy and as diagnostic agents. | 6.1 Brevetto | 1999 | Roncucci, G; Dei, D; DE FILIPPIS, M. P.; Fantetti, L; Masini, I; Cosimelli, Barbara; Jori, G. | |
| From the central benzodiazepine receptor to the adenosine receptors exploiting the 3-diketoindole moiety | 8.02 Comunicazioni a Convegni o Seminari | 2011 | Cosimelli, Barbara | |
| Synthesis and biological evaluation on human glioblastoma cells of novel pyrazolo[3,4-d]pyrimidine adenosine A(3) receptor antagonists | 4.3 Poster | 2010 | Mugnaini, L.; La Motta, C.; Taliani, S; Simorini, F.; Salerno, S.; Marini, A. M.; Da Settimo, F.; Cosimelli, Barbara; Greco, Giovanni; Novellino, Ettore; Daniele, S.; Trincavelli, M. L.; Martini, C. | |
| Chemistry of Substituted Pyrazolo[1,5-a]pyrimidines. Part 3. A Structural Correc¬tion of Pyrazolo[1,5-a][1,3]diazepine Derivative on the Basis of 13C NMR Spectroscopy. | 1.1 Articolo in rivista | 1993 | Chimichi, S; Cosimelli, Barbara; Bruni, F; Costanzo, A. | |
| Inhibition of MDR1 activity in vitro by a novel class of diltiazem analogues: towards new candidates | 1.1 Articolo in rivista | 2009 | Viale, M.; Cordazzo, C.; Cosimelli, Barbara; de Totero, D.; Castagnola, P.; Aiello, C.; Cianfriglia, M.; Severi, E.; Petrillo, G.; Spinelli, D. | |
| Chemistry of substituted pyrazolo[1,5-a]pyrimidines. Part 5. 7-Oxo-6-[pyrazol-3’(5’)-yl]-4,7-dihydropyrazolo[1,5-a]pyrimidines from 6-ethoxycarbonyl-7-(2-dimethylaminovinyl)-pyrazolo[1,5-a]pyrimidines: elucidation of the reaction mechanism through NMR spectroscopy and X-Ray diffraction analysis. | 1.1 Articolo in rivista | 1996 | Chimichi, S; Bruni, F; Cosimelli, Barbara; Selleri, S; Valle, G. | |
| Substituent effect on the redox potential of some substituted (aryl)(2-nitrobenzo[b]thiophen-3-yl)amines. | 1.1 Articolo in rivista | 2001 | Cosimelli, Barbara; Spinelli, D; Costanzo, F; Tonelli, D; Lamartina, L; Sarva', M. C.; Seeber, R. | |
| Modulation of A2B adenosine receptor by 1-Benzyl-3-ketoindole derivatives | 1.1 Articolo in rivista | 2013 | S., Taliani; M. L., Trincavelli; Cosimelli, Barbara; Laneri, Sonia; E., Severi; E., Barresi; I., Pugliesi; S., Daniele; C., Giacomelli; Greco, Giovanni; Novellino, Ettore; C., Martini; F., Da Settimo | |
| 3-Aryl-[1,2,4]triazino[4,3-a]benzimidazol-4(10H)-one: a novel template for the design of highly selective A2B adenosine receptor antagonists | 4.3 Poster | 2012 | Taliani, S.; Pugliesi, I.; Barresi, E.; Salerno, S.; Simorini, F.; La Motta, C.; Marini, A. M.; Da Settimo, F.; Cosconati, S.; Marinelli, Luciana; Cosimelli, Barbara; Greco, Giovanni; Novellino, Ettore; Daniele, S.; Trincavelli, M. L.; Martini, C. | |
| Regioselective Synthesis of 4-Acetyl- and 5-Acetyl-3-methylisoxazole: their Conversion into Silyl- and Methyl Enol Ethers. | 1.1 Articolo in rivista | 1992 | Chimichi, S; Cosimelli, Barbara | |
| Ring-ring Interconversions. Part 3. On the effect of the substituents on the thiazole moiety in the ring-opening/ring-closing reactions of nitrosoimidazo[2,1-b][1,3]thiazoles with hydrochloric acid. | 1.1 Articolo in rivista | 2000 | Billi, R; Cosimelli, Barbara; Leoni, A; Spinelli, D. | |
| Derivatives of 4-Amino-6-hydroxy-2-mercaptopyrimidine as Novel, Potent, and Selective A3 Adenosine Receptor Antagonists | 1.1 Articolo in rivista | 2008 | Cosimelli, Barbara; Greco, Giovanni; Ehlardo, M.; Novellino, Ettore; Da Settimo, F.; Taliani, S.; La Motta, C.; Bellandi, M.; Tuccinardi, T.; Martinelli, A.; Ciampi, O.; Trincavelli, M. L.; Martini, C. | |
| L-Type calcium channel blockers: from diltiazem to 1,2,4-oxadiazol-5-ones via thiazinooxadiazol-3-one derivatives | 1.1 Articolo in rivista | 2009 | Budriesi, R.; Cosimelli, Barbara; Ioan, P.; Ugenti, P.; Carosati, E.; Frosini, M.; Fusi, F.; Spisani, R.; Saponara, S.; Corda, G.; Cruciani, G.; Novellino, Ettore; Spinelli, D.; Chiarini, A. | |
| A New Synthetic Route to 2,2’:5’,2”-Terthiophene-5-derivatives to Conjugate with Proteins and Monoclonal Antibodies. | 1.1 Articolo in rivista | 1996 | Cosimelli, Barbara; Neri, D; Roncucci, G. | |
| Ring opening of 2-substituted 4-nitrothiophenes with pyrrolidine. Access to new functionalized nitro-unsaturated building blocks. | 1.1 Articolo in rivista | 2001 | Dell'Erba, C; Gabellini, A; Novi, M; Petrillo, G; Tavani, C; Cosimelli, Barbara; Spinelli, D. | |
| Synthesis and antimycotic activity of new unsymmetrical substituted zinc phthalocyanines. | 1.1 Articolo in rivista | 2003 | Cosimelli, Barbara; Roncucci, G; Dei, D; Fantetti, L; Ferroni, F; Ricci, M; Spinelli, D. | |
| New Fluorescent 2-Phenylindolglyoxylamide Derivatives as Probes Targeting the Peripheral-Type Benzodiazepine Receptor: Design, Synthesis and Biological Evaluation. | 1.1 Articolo in rivista | 2007 | Taliani, S.; Simorini, F.; Sergianni, V.; LA MOTTA, C.; DA SETTIMO, F.; Cosimelli, Barbara; ABIGNENTE DI FRASSELLO, Enrico; Greco, Giovanni; Novellino, Ettore; Rossi, L.; Gremigni, V.; Spinetti, F.; Chelli, B.; Martini, C. |