COSIMELLI, BARBARA
COSIMELLI, BARBARA
DIPARTIMENTO DI FARMACIA
Chemistry of Substituted Pyrazolo[1,5-a]pyrimidines. Part 4. A Structural Correction of a Series of Pyrazolo[5',1':2,3]pyrimido[5,4-d][1,3]diazepines on the Basis of NMR Spectroscopy and X-Ray Diffraction Analysis.
1994 Chimichi, S; Cosimelli, Barbara; Bruni, F; Selleri, S; Costanzo, A; Guerrini, G; Valle, G.
Determination of the absolute configuration of the enantiomers of an oxadiazol-3-one calcium channel blocker, resolved by chiral HPLC, via concerted use of three chiroptical spectroscopies
2012 Giovanni Battista, Barrano; Salvatore, Caccamese; Cosimelli, Barbara; Frank J., Devlin; Elda, Severi; Domenico, Spinelli
Synthesis, Citotoxicity and Apoptosis Induction in Human Tumor Cells by Geiparvarin Analogues
2004 Viola, G; Vedaldi, D; Dall'Acqua, F; Basso, G; Disaro', S; Spinelli, M; Cosimelli, Barbara; Boccalini, M; Chimichi, S.
Chemistry of Substituted Pyrazolo[1,5-a]pyrimidines. Part 3. A Structural Correc¬tion of Pyrazolo[1,5-a][1,3]diazepine Derivative on the Basis of 13C NMR Spectroscopy.
1993 Chimichi, S; Cosimelli, Barbara; Bruni, F; Costanzo, A.
Ring-ring Interconversions. Part 3. On the effect of the substituents on the thiazole moiety in the ring-opening/ring-closing reactions of nitrosoimidazo[2,1-b][1,3]thiazoles with hydrochloric acid.
2000 Billi, R; Cosimelli, Barbara; Leoni, A; Spinelli, D.
Zinc phthalocyanines and corresponding conjugates, their preparation and use in photodynamic therapy and as diagnostic agents.
1999 Roncucci, G; Dei, D; DE FILIPPIS, M. P.; Fantetti, L; Masini, I; Cosimelli, Barbara; Jori, G.
Inhibition of MDR1 activity in vitro by a novel class of diltiazem analogues: towards new candidates
2009 Viale, M.; Cordazzo, C.; Cosimelli, Barbara; de Totero, D.; Castagnola, P.; Aiello, C.; Cianfriglia, M.; Severi, E.; Petrillo, G.; Spinelli, D.
First example of Diels-Alder reaction of 4-(1-ethenylsubstituted)-3-methylisoxazoles with acetylenedicarboxylate
2008 Chimichi, S.; Cosimelli, Barbara; Boccalini, M.; Matteucci A., Messaoudi A.
Discovery of novel and cardioselective diltiazem-like calcium channel blockers via virtual screening.
2008 Carosati, E.; Budriesi, R.; Ioan, P.; Ugenti, P.; Frosini, M.; Fusi, F.; Corda, G.; Cosimelli, Barbara; Spinelli, D.; Chiarini, A.; Cruciani, G.
A New Entry to Pyrazolo[1,5-a]pyrido[3,4-e]pyrimidine Derivatives.
1990 Bruni, F; Chimichi, S; Cosimelli, Barbara; Costanzo, A; Guerrini, G; Selleri, S.
Tertiary amides with a five-membered heteroaromatic ring as new probes for the translocator protein
2011 Cosimelli, Barbara; F., Simorini; S., Taliani; C., La Motta; F., Da Settimo; E., Severi; Greco, Giovanni; Novellino, Ettore; B., Costa; E., Da Pozzo; S., Bendinelli; C., Martini
L-Type calcium channel blockers: from diltiazem to 1,2,4-oxadiazol-5-ones via thiazinooxadiazol-3-one derivatives
2009 Budriesi, R.; Cosimelli, Barbara; Ioan, P.; Ugenti, P.; Carosati, E.; Frosini, M.; Fusi, F.; Spisani, R.; Saponara, S.; Corda, G.; Cruciani, G.; Novellino, Ettore; Spinelli, D.; Chiarini, A.
Allosteric Modulators of Human A2B Adenosine Receptor
2014 Maria Letizia, Trincavelli; Chiara, Giacomelli; Simona, Daniele; Sabrina, Taliania; Cosimelli, Barbara; Laneri, Sonia; Elda, Severi; Elisabetta, Barresi; Isabella, Pugliesi; Greco, Giovanni; Novellino, Ettore; Federico Da, Settimo; Claudia, Martini
From the Pharmacophore to the Homology Model of the Benzodiazepine Receptor: The Indolyglyoxylamides Affair.
2012 Cosimelli, Barbara; Cosconati, S.; Marinelli, Luciana; Novellino, Ettore; Greco, Giovanni
Modulation of A2B adenosine receptor by 1-Benzyl-3-ketoindole derivatives
2013 S., Taliani; M. L., Trincavelli; Cosimelli, Barbara; Laneri, Sonia; E., Severi; E., Barresi; I., Pugliesi; S., Daniele; C., Giacomelli; Greco, Giovanni; Novellino, Ettore; C., Martini; F., Da Settimo
Absolute configuration and biological profile of two thiazinooxadiazol-3-ones with L-type calcium channel activity: a study of the structural effects
2012 Ioan, P.; Ciogli, A.; Sirci, F.; Budriesi, R.; Cosimelli, Barbara; Pierini, M.; Severi, E.; Chiarini, A.; Cruciani, G.; Gasparrini, F.; Spinelli, D.; Carosati, E.
Ring-ring Interconversions of Nitrosoimidazoles. The Effect of Some Condensed Six-membered Rings on the Reactivity.
2000 Billi, R; Cosimelli, Barbara; Spinelli, D; Andreani, A; Leoni, A.
On the Nitration of 5-Phenyl- and 3-Methyl-5-phenylisoxazole.
1989 Chimichi, S; Cosimelli, Barbara
Alkali-metal Complexes with Neutral Molecular Receptors containing Nitrogen Donor Atoms: a Crystallographic and Multinuclear Magnetic Resonance Study.
1991 DI VAIRA, M; Cosimelli, Barbara; Mani, F; Stoppioni, P.
Regioselective Synthesis of 4-Acetyl- and 5-Acetyl-3-methylisoxazole: their Conversion into Silyl- and Methyl Enol Ethers.
1992 Chimichi, S; Cosimelli, Barbara
| Titolo | Tipologia | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|---|
| Chemistry of Substituted Pyrazolo[1,5-a]pyrimidines. Part 4. A Structural Correction of a Series of Pyrazolo[5',1':2,3]pyrimido[5,4-d][1,3]diazepines on the Basis of NMR Spectroscopy and X-Ray Diffraction Analysis. | 1.1 Articolo in rivista | 1994 | Chimichi, S; Cosimelli, Barbara; Bruni, F; Selleri, S; Costanzo, A; Guerrini, G; Valle, G. | |
| Determination of the absolute configuration of the enantiomers of an oxadiazol-3-one calcium channel blocker, resolved by chiral HPLC, via concerted use of three chiroptical spectroscopies | 8.02 Comunicazioni a Convegni o Seminari | 2012 | Giovanni Battista, Barrano; Salvatore, Caccamese; Cosimelli, Barbara; Frank J., Devlin; Elda, Severi; Domenico, Spinelli | |
| Synthesis, Citotoxicity and Apoptosis Induction in Human Tumor Cells by Geiparvarin Analogues | 1.1 Articolo in rivista | 2004 | Viola, G; Vedaldi, D; Dall'Acqua, F; Basso, G; Disaro', S; Spinelli, M; Cosimelli, Barbara; Boccalini, M; Chimichi, S. | |
| Chemistry of Substituted Pyrazolo[1,5-a]pyrimidines. Part 3. A Structural Correc¬tion of Pyrazolo[1,5-a][1,3]diazepine Derivative on the Basis of 13C NMR Spectroscopy. | 1.1 Articolo in rivista | 1993 | Chimichi, S; Cosimelli, Barbara; Bruni, F; Costanzo, A. | |
| Ring-ring Interconversions. Part 3. On the effect of the substituents on the thiazole moiety in the ring-opening/ring-closing reactions of nitrosoimidazo[2,1-b][1,3]thiazoles with hydrochloric acid. | 1.1 Articolo in rivista | 2000 | Billi, R; Cosimelli, Barbara; Leoni, A; Spinelli, D. | |
| Zinc phthalocyanines and corresponding conjugates, their preparation and use in photodynamic therapy and as diagnostic agents. | 6.1 Brevetto | 1999 | Roncucci, G; Dei, D; DE FILIPPIS, M. P.; Fantetti, L; Masini, I; Cosimelli, Barbara; Jori, G. | |
| Inhibition of MDR1 activity in vitro by a novel class of diltiazem analogues: towards new candidates | 1.1 Articolo in rivista | 2009 | Viale, M.; Cordazzo, C.; Cosimelli, Barbara; de Totero, D.; Castagnola, P.; Aiello, C.; Cianfriglia, M.; Severi, E.; Petrillo, G.; Spinelli, D. | |
| First example of Diels-Alder reaction of 4-(1-ethenylsubstituted)-3-methylisoxazoles with acetylenedicarboxylate | 1.1 Articolo in rivista | 2008 | Chimichi, S.; Cosimelli, Barbara; Boccalini, M.; Matteucci A., Messaoudi A. | |
| Discovery of novel and cardioselective diltiazem-like calcium channel blockers via virtual screening. | 1.1 Articolo in rivista | 2008 | Carosati, E.; Budriesi, R.; Ioan, P.; Ugenti, P.; Frosini, M.; Fusi, F.; Corda, G.; Cosimelli, Barbara; Spinelli, D.; Chiarini, A.; Cruciani, G. | |
| A New Entry to Pyrazolo[1,5-a]pyrido[3,4-e]pyrimidine Derivatives. | 1.1 Articolo in rivista | 1990 | Bruni, F; Chimichi, S; Cosimelli, Barbara; Costanzo, A; Guerrini, G; Selleri, S. | |
| Tertiary amides with a five-membered heteroaromatic ring as new probes for the translocator protein | 1.1 Articolo in rivista | 2011 | Cosimelli, Barbara; F., Simorini; S., Taliani; C., La Motta; F., Da Settimo; E., Severi; Greco, Giovanni; Novellino, Ettore; B., Costa; E., Da Pozzo; S., Bendinelli; C., Martini | |
| L-Type calcium channel blockers: from diltiazem to 1,2,4-oxadiazol-5-ones via thiazinooxadiazol-3-one derivatives | 1.1 Articolo in rivista | 2009 | Budriesi, R.; Cosimelli, Barbara; Ioan, P.; Ugenti, P.; Carosati, E.; Frosini, M.; Fusi, F.; Spisani, R.; Saponara, S.; Corda, G.; Cruciani, G.; Novellino, Ettore; Spinelli, D.; Chiarini, A. | |
| Allosteric Modulators of Human A2B Adenosine Receptor | 1.1 Articolo in rivista | 2014 | Maria Letizia, Trincavelli; Chiara, Giacomelli; Simona, Daniele; Sabrina, Taliania; Cosimelli, Barbara; Laneri, Sonia; Elda, Severi; Elisabetta, Barresi; Isabella, Pugliesi; Greco, Giovanni; Novellino, Ettore; Federico Da, Settimo; Claudia, Martini | |
| From the Pharmacophore to the Homology Model of the Benzodiazepine Receptor: The Indolyglyoxylamides Affair. | 1.1 Articolo in rivista | 2012 | Cosimelli, Barbara; Cosconati, S.; Marinelli, Luciana; Novellino, Ettore; Greco, Giovanni | |
| Modulation of A2B adenosine receptor by 1-Benzyl-3-ketoindole derivatives | 1.1 Articolo in rivista | 2013 | S., Taliani; M. L., Trincavelli; Cosimelli, Barbara; Laneri, Sonia; E., Severi; E., Barresi; I., Pugliesi; S., Daniele; C., Giacomelli; Greco, Giovanni; Novellino, Ettore; C., Martini; F., Da Settimo | |
| Absolute configuration and biological profile of two thiazinooxadiazol-3-ones with L-type calcium channel activity: a study of the structural effects | 1.1 Articolo in rivista | 2012 | Ioan, P.; Ciogli, A.; Sirci, F.; Budriesi, R.; Cosimelli, Barbara; Pierini, M.; Severi, E.; Chiarini, A.; Cruciani, G.; Gasparrini, F.; Spinelli, D.; Carosati, E. | |
| Ring-ring Interconversions of Nitrosoimidazoles. The Effect of Some Condensed Six-membered Rings on the Reactivity. | 1.1 Articolo in rivista | 2000 | Billi, R; Cosimelli, Barbara; Spinelli, D; Andreani, A; Leoni, A. | |
| On the Nitration of 5-Phenyl- and 3-Methyl-5-phenylisoxazole. | 1.1 Articolo in rivista | 1989 | Chimichi, S; Cosimelli, Barbara | |
| Alkali-metal Complexes with Neutral Molecular Receptors containing Nitrogen Donor Atoms: a Crystallographic and Multinuclear Magnetic Resonance Study. | 1.1 Articolo in rivista | 1991 | DI VAIRA, M; Cosimelli, Barbara; Mani, F; Stoppioni, P. | |
| Regioselective Synthesis of 4-Acetyl- and 5-Acetyl-3-methylisoxazole: their Conversion into Silyl- and Methyl Enol Ethers. | 1.1 Articolo in rivista | 1992 | Chimichi, S; Cosimelli, Barbara |