COSIMELLI, BARBARA
COSIMELLI, BARBARA
DIPARTIMENTO DI FARMACIA
Chemistry of Substituted Pyrazolo[1,5-a]pyrimidines. Part 4. A Structural Correction of a Series of Pyrazolo[5',1':2,3]pyrimido[5,4-d][1,3]diazepines on the Basis of NMR Spectroscopy and X-Ray Diffraction Analysis.
1994 Chimichi, S; Cosimelli, Barbara; Bruni, F; Selleri, S; Costanzo, A; Guerrini, G; Valle, G.
Determination of the absolute configuration of the enantiomers of an oxadiazol-3-one calcium channel blocker, resolved by chiral HPLC, via concerted use of three chiroptical spectroscopies
2012 Giovanni Battista, Barrano; Salvatore, Caccamese; Cosimelli, Barbara; Frank J., Devlin; Elda, Severi; Domenico, Spinelli
3-Aryl-[1,2,4]triazino[4,3-a]benzimidazol-4(10H)-one: a novel template for the design of highly selective A2B adenosine receptor antagonists
2012 Taliani, S.; Pugliesi, I.; Barresi, E.; Simorini, F.; Salerno, S.; La Motta, C.; Marini, A. M.; Cosimelli, Barbara; Cosconati, S.; DI MARO, Salvatore; Marinelli, Luciana; Daniele, S.; Trincavelli, M. L.; Greco, Giovanni; Novellino, Ettore; Martini, C.; Da Settimo, F.
Synthesis, Citotoxicity and Apoptosis Induction in Human Tumor Cells by Geiparvarin Analogues
2004 Viola, G; Vedaldi, D; Dall'Acqua, F; Basso, G; Disaro', S; Spinelli, M; Cosimelli, Barbara; Boccalini, M; Chimichi, S.
Derivatives of benzimidazol-2-ylquinoline and benzimidazol-2-ylisoquinoline as selective A1 adenosine receptor antagonists with stimulant activity on human colon motility
2011 Cosimelli, Barbara; S., Taliani; Greco, Giovanni; Novellino, Ettore; A., Sala; E., Severi; F., Da Settimo; C., La Motta; I., Pugliesi; L., Antonioli; M., Fornai; R., Colucci; C., Blandizzi; S., Daniele; M. L., Trincavelli; C., Martini
Chemistry of Substituted Pyrazolo[1,5-a]pyrimidines. Part 3. A Structural Correc¬tion of Pyrazolo[1,5-a][1,3]diazepine Derivative on the Basis of 13C NMR Spectroscopy.
1993 Chimichi, S; Cosimelli, Barbara; Bruni, F; Costanzo, A.
Ring-ring Interconversions. Part 3. On the effect of the substituents on the thiazole moiety in the ring-opening/ring-closing reactions of nitrosoimidazo[2,1-b][1,3]thiazoles with hydrochloric acid.
2000 Billi, R; Cosimelli, Barbara; Leoni, A; Spinelli, D.
New results on the reactivity of 5,6-diamino-4-hydroxy-2-mercaptopyrimidine
2004 Cosimelli, Barbara; Iadanza, M; Spisani, R; Novellino, Ettore
From the central benzodiazepine receptor to the adenosine receptors exploiting the 3-diketoindole moiety
2011 Cosimelli, Barbara
Zinc phthalocyanines and corresponding conjugates, their preparation and use in photodynamic therapy and as diagnostic agents.
1999 Roncucci, G; Dei, D; DE FILIPPIS, M. P.; Fantetti, L; Masini, I; Cosimelli, Barbara; Jori, G.
2-Phenyl[1,2,3]triazolo[1,2-a][1,2,4]benzotriazin-1-one derivatives as a new class of adenosine receptor antagonists
2005 Primofiore, G.; Da Settimo, F.; Taliani, S.; Sergianni, V.; Simorini, F.; La Motta, C.; Marini, A. M.; Tuscano, D.; Martini, C.; Greco, Giovanni; Cosimelli, Barbara; Novellino, Ettore
Pyrazolo[1,5-a]pyrido[3,4-e]pyrimidine: A New Heterocyclic Ring System.
1990 Bruni, F; Chimichi, S; Cosimelli, Barbara; Costanzo, A; Guerrini, G; Selleri, S.
Inhibition of MDR1 activity in vitro by a novel class of diltiazem analogues: towards new candidates
2009 Viale, M.; Cordazzo, C.; Cosimelli, Barbara; de Totero, D.; Castagnola, P.; Aiello, C.; Cianfriglia, M.; Severi, E.; Petrillo, G.; Spinelli, D.
First example of Diels-Alder reaction of 4-(1-ethenylsubstituted)-3-methylisoxazoles with acetylenedicarboxylate
2008 Chimichi, S.; Cosimelli, Barbara; Boccalini, M.; Matteucci A., Messaoudi A.
Discovery of novel and cardioselective diltiazem-like calcium channel blockers via virtual screening.
2008 Carosati, E.; Budriesi, R.; Ioan, P.; Ugenti, P.; Frosini, M.; Fusi, F.; Corda, G.; Cosimelli, Barbara; Spinelli, D.; Chiarini, A.; Cruciani, G.
A New Entry to Pyrazolo[1,5-a]pyrido[3,4-e]pyrimidine Derivatives.
1990 Bruni, F; Chimichi, S; Cosimelli, Barbara; Costanzo, A; Guerrini, G; Selleri, S.
Tertiary amides with a five-membered heteroaromatic ring as new probes for the translocator protein
2011 Cosimelli, Barbara; F., Simorini; S., Taliani; C., La Motta; F., Da Settimo; E., Severi; Greco, Giovanni; Novellino, Ettore; B., Costa; E., Da Pozzo; S., Bendinelli; C., Martini
L-Type calcium channel blockers: from diltiazem to 1,2,4-oxadiazol-5-ones via thiazinooxadiazol-3-one derivatives
2009 Budriesi, R.; Cosimelli, Barbara; Ioan, P.; Ugenti, P.; Carosati, E.; Frosini, M.; Fusi, F.; Spisani, R.; Saponara, S.; Corda, G.; Cruciani, G.; Novellino, Ettore; Spinelli, D.; Chiarini, A.
Allosteric Modulators of Human A2B Adenosine Receptor
2014 Maria Letizia, Trincavelli; Chiara, Giacomelli; Simona, Daniele; Sabrina, Taliania; Cosimelli, Barbara; Laneri, Sonia; Elda, Severi; Elisabetta, Barresi; Isabella, Pugliesi; Greco, Giovanni; Novellino, Ettore; Federico Da, Settimo; Claudia, Martini
From the Pharmacophore to the Homology Model of the Benzodiazepine Receptor: The Indolyglyoxylamides Affair.
2012 Cosimelli, Barbara; Cosconati, S.; Marinelli, Luciana; Novellino, Ettore; Greco, Giovanni
| Titolo | Tipologia | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|---|
| Chemistry of Substituted Pyrazolo[1,5-a]pyrimidines. Part 4. A Structural Correction of a Series of Pyrazolo[5',1':2,3]pyrimido[5,4-d][1,3]diazepines on the Basis of NMR Spectroscopy and X-Ray Diffraction Analysis. | 1.1 Articolo in rivista | 1994 | Chimichi, S; Cosimelli, Barbara; Bruni, F; Selleri, S; Costanzo, A; Guerrini, G; Valle, G. | |
| Determination of the absolute configuration of the enantiomers of an oxadiazol-3-one calcium channel blocker, resolved by chiral HPLC, via concerted use of three chiroptical spectroscopies | 8.02 Comunicazioni a Convegni o Seminari | 2012 | Giovanni Battista, Barrano; Salvatore, Caccamese; Cosimelli, Barbara; Frank J., Devlin; Elda, Severi; Domenico, Spinelli | |
| 3-Aryl-[1,2,4]triazino[4,3-a]benzimidazol-4(10H)-one: a novel template for the design of highly selective A2B adenosine receptor antagonists | 1.1 Articolo in rivista | 2012 | Taliani, S.; Pugliesi, I.; Barresi, E.; Simorini, F.; Salerno, S.; La Motta, C.; Marini, A. M.; Cosimelli, Barbara; Cosconati, S.; DI MARO, Salvatore; Marinelli, Luciana; Daniele, S.; Trincavelli, M. L.; Greco, Giovanni; Novellino, Ettore; Martini, C.; Da Settimo, F. | |
| Synthesis, Citotoxicity and Apoptosis Induction in Human Tumor Cells by Geiparvarin Analogues | 1.1 Articolo in rivista | 2004 | Viola, G; Vedaldi, D; Dall'Acqua, F; Basso, G; Disaro', S; Spinelli, M; Cosimelli, Barbara; Boccalini, M; Chimichi, S. | |
| Derivatives of benzimidazol-2-ylquinoline and benzimidazol-2-ylisoquinoline as selective A1 adenosine receptor antagonists with stimulant activity on human colon motility | 1.1 Articolo in rivista | 2011 | Cosimelli, Barbara; S., Taliani; Greco, Giovanni; Novellino, Ettore; A., Sala; E., Severi; F., Da Settimo; C., La Motta; I., Pugliesi; L., Antonioli; M., Fornai; R., Colucci; C., Blandizzi; S., Daniele; M. L., Trincavelli; C., Martini | |
| Chemistry of Substituted Pyrazolo[1,5-a]pyrimidines. Part 3. A Structural Correc¬tion of Pyrazolo[1,5-a][1,3]diazepine Derivative on the Basis of 13C NMR Spectroscopy. | 1.1 Articolo in rivista | 1993 | Chimichi, S; Cosimelli, Barbara; Bruni, F; Costanzo, A. | |
| Ring-ring Interconversions. Part 3. On the effect of the substituents on the thiazole moiety in the ring-opening/ring-closing reactions of nitrosoimidazo[2,1-b][1,3]thiazoles with hydrochloric acid. | 1.1 Articolo in rivista | 2000 | Billi, R; Cosimelli, Barbara; Leoni, A; Spinelli, D. | |
| New results on the reactivity of 5,6-diamino-4-hydroxy-2-mercaptopyrimidine | 1.1 Articolo in rivista | 2004 | Cosimelli, Barbara; Iadanza, M; Spisani, R; Novellino, Ettore | |
| From the central benzodiazepine receptor to the adenosine receptors exploiting the 3-diketoindole moiety | 8.02 Comunicazioni a Convegni o Seminari | 2011 | Cosimelli, Barbara | |
| Zinc phthalocyanines and corresponding conjugates, their preparation and use in photodynamic therapy and as diagnostic agents. | 6.1 Brevetto | 1999 | Roncucci, G; Dei, D; DE FILIPPIS, M. P.; Fantetti, L; Masini, I; Cosimelli, Barbara; Jori, G. | |
| 2-Phenyl[1,2,3]triazolo[1,2-a][1,2,4]benzotriazin-1-one derivatives as a new class of adenosine receptor antagonists | 4.1 Articoli in Atti di convegno | 2005 | Primofiore, G.; Da Settimo, F.; Taliani, S.; Sergianni, V.; Simorini, F.; La Motta, C.; Marini, A. M.; Tuscano, D.; Martini, C.; Greco, Giovanni; Cosimelli, Barbara; Novellino, Ettore | |
| Pyrazolo[1,5-a]pyrido[3,4-e]pyrimidine: A New Heterocyclic Ring System. | 1.1 Articolo in rivista | 1990 | Bruni, F; Chimichi, S; Cosimelli, Barbara; Costanzo, A; Guerrini, G; Selleri, S. | |
| Inhibition of MDR1 activity in vitro by a novel class of diltiazem analogues: towards new candidates | 1.1 Articolo in rivista | 2009 | Viale, M.; Cordazzo, C.; Cosimelli, Barbara; de Totero, D.; Castagnola, P.; Aiello, C.; Cianfriglia, M.; Severi, E.; Petrillo, G.; Spinelli, D. | |
| First example of Diels-Alder reaction of 4-(1-ethenylsubstituted)-3-methylisoxazoles with acetylenedicarboxylate | 1.1 Articolo in rivista | 2008 | Chimichi, S.; Cosimelli, Barbara; Boccalini, M.; Matteucci A., Messaoudi A. | |
| Discovery of novel and cardioselective diltiazem-like calcium channel blockers via virtual screening. | 1.1 Articolo in rivista | 2008 | Carosati, E.; Budriesi, R.; Ioan, P.; Ugenti, P.; Frosini, M.; Fusi, F.; Corda, G.; Cosimelli, Barbara; Spinelli, D.; Chiarini, A.; Cruciani, G. | |
| A New Entry to Pyrazolo[1,5-a]pyrido[3,4-e]pyrimidine Derivatives. | 1.1 Articolo in rivista | 1990 | Bruni, F; Chimichi, S; Cosimelli, Barbara; Costanzo, A; Guerrini, G; Selleri, S. | |
| Tertiary amides with a five-membered heteroaromatic ring as new probes for the translocator protein | 1.1 Articolo in rivista | 2011 | Cosimelli, Barbara; F., Simorini; S., Taliani; C., La Motta; F., Da Settimo; E., Severi; Greco, Giovanni; Novellino, Ettore; B., Costa; E., Da Pozzo; S., Bendinelli; C., Martini | |
| L-Type calcium channel blockers: from diltiazem to 1,2,4-oxadiazol-5-ones via thiazinooxadiazol-3-one derivatives | 1.1 Articolo in rivista | 2009 | Budriesi, R.; Cosimelli, Barbara; Ioan, P.; Ugenti, P.; Carosati, E.; Frosini, M.; Fusi, F.; Spisani, R.; Saponara, S.; Corda, G.; Cruciani, G.; Novellino, Ettore; Spinelli, D.; Chiarini, A. | |
| Allosteric Modulators of Human A2B Adenosine Receptor | 1.1 Articolo in rivista | 2014 | Maria Letizia, Trincavelli; Chiara, Giacomelli; Simona, Daniele; Sabrina, Taliania; Cosimelli, Barbara; Laneri, Sonia; Elda, Severi; Elisabetta, Barresi; Isabella, Pugliesi; Greco, Giovanni; Novellino, Ettore; Federico Da, Settimo; Claudia, Martini | |
| From the Pharmacophore to the Homology Model of the Benzodiazepine Receptor: The Indolyglyoxylamides Affair. | 1.1 Articolo in rivista | 2012 | Cosimelli, Barbara; Cosconati, S.; Marinelli, Luciana; Novellino, Ettore; Greco, Giovanni |