COSIMELLI, BARBARA
COSIMELLI, BARBARA
DIPARTIMENTO DI FARMACIA
Determination of the absolute configuration of the enantiomers of an oxadiazol-3-one calcium channel blocker, resolved by chiral HPLC, via concerted use of three chiroptical spectroscopies
2012 Giovanni Battista, Barrano; Salvatore, Caccamese; Cosimelli, Barbara; Frank J., Devlin; Elda, Severi; Domenico, Spinelli
Chemistry of Substituted Pyrazolo[1,5-a]pyrimidines. Part 4. A Structural Correction of a Series of Pyrazolo[5',1':2,3]pyrimido[5,4-d][1,3]diazepines on the Basis of NMR Spectroscopy and X-Ray Diffraction Analysis.
1994 Chimichi, S; Cosimelli, Barbara; Bruni, F; Selleri, S; Costanzo, A; Guerrini, G; Valle, G.
Playing with Opening and Closing of Heterocycles: Using the Cusmano-Ruccia Reaction to Develop a Novel Class of Oxadiazolothiazinones, Active as Calcium Channel Modulators and P-Glycoprotein Inhibitors
2014 Domenico, Spinelli; Roberta, Budriesi; Cosimelli, Barbara; Elda, Severi; Matteo, Micucci; Massimo, Baroni; Fabio, Fusi; Pierfranco, Ioan; Simon, Cross; Maria, Frosini; Simona, Saponara; Rosanna, Matucci; Camillo, Rosano; Maurizio, Viale; Alberto, Chiarini; Emanuele, Carosati
Preliminary Finding on a New Calcium Channel Entry Blocker Chemotype: 5,6-Diamino-4-hydroxy-2-mercaptopyrimidine Derivatives
2011 Cosimelli, Barbara; Elda, Severi; Novellino, Ettore; Anna, Cavaccini; Cataldi, Mauro; Roberta, Budriesi; Matteo, Micucci; Alberto, Chiarini; Pierfranco, Ioan
A New Convenient Route to 2-Oxoethoxycoumarins: Key Intermediates in the Synthesis of Natural Products.
2002 Chimichi, S; Boccalini, M; Cosimelli, Barbara
Refinement of the Benzodiazepine Receptor Site Topology by Structure-Activity Relationships of New N-(Heteroarylmethyl)indol-3-ylglyoxylamides.
2006 Primofiore, G; Da, Settimo; F, Marini; A. M, Taliani; S, ; La, Motta; C, Simorini; Novellino, Ettore; E, ; Greco, Giovanni; Cosimelli, Barbara; Ehlardo, Marina; Sala, Annalisa; A, Besnard; F, Montali; M, Martini
Ring-ring interconversions. Part 2. Effect of the Substituent on the Rearrangement of 6-Aryl-3-methyl-5-nitrosoimidazo[2,1-b][1,3]thiazoles into 8-Aryl-8-hydroxy-5-methyl-8H-[1,4]thiazino[3,4-c][1,2,4]oxadiazol-3-ones. A Novel Class of Potential Antitumor Agents.
1999 Billi, R; Cosimelli, Barbara; Spinelli, D; Rambaldi, M.
ABCB1 Structural Models, Molecular Docking, and Synthesis of New Oxadiazolothiazin-3-one Inhibitors
2013 C., Rosano; M., Viale; Cosimelli, Barbara; E., Severi; R., Gangemi; A., Ciogli; D., De Totero; D., Spinelli
Mononuclear Heterocyclic Rearrangements. Part 16. Kinetic Study of the Rearrangement of Some ortho-Substituted Z-Phenylhydrazones of 3-Benzoyl-5-phenyl-1,2,4-oxadiazole into 2-Aryl-4-benzoylamino-5-phenyl-1,2,3-triazoles in Dioxane-Water and in Benzene.
1999 Frenna, V; Macaluso, G; Consiglio, G; Cosimelli, Barbara; Spinelli, D.
First example of Diels-Alder reaction of 4-(1-ethenylsubstituted)-3-methylisoxazoles with acetylenedicarboxylate
2008 Chimichi, S.; Cosimelli, Barbara; Boccalini, M.; Matteucci A., Messaoudi A.
Derivatives of 4-Amino-6-hydroxy-2-mercaptopyrimidine as Novel, Potent, and Selective A3 Adenosine Receptor Antagonists
2008 Cosimelli, Barbara; Greco, Giovanni; Ehlardo, M.; Novellino, Ettore; Da Settimo, F.; Taliani, S.; La Motta, C.; Bellandi, M.; Tuccinardi, T.; Martinelli, A.; Ciampi, O.; Trincavelli, M. L.; Martini, C.
ortho-Substituted (aryl)(3-nitrobenzo[b]thiophen-2-yl)amines: study of the electrochemical behavior
2009 Cosimelli, Barbara; Lanza, C. Z.; Scavetta, E.; Severi, E.; Spinelli, D.; Stenta, M.; Tonelli, D.
High Affinity Central Benzodiazepine Receptor Ligands: Synthesis and Biological Evaluation of a Series of Phenyltriazolobenzotriazindione Derivatives (PTBTs)
2005 Primofiore, G; DA SETTIMO, F; Taliani, S; Salerno, S; Novellino, Ettore; Greco, Giovanni; Cosimelli, Barbara; Besnard, F; Costa, C; Montali, M; Martini, C.
Alkali-metal Complexes with Neutral Molecular Receptors containing Nitrogen Donor Atoms: a Crystallographic and Multinuclear Magnetic Resonance Study.
1991 DI VAIRA, M; Cosimelli, Barbara; Mani, F; Stoppioni, P.
Novel N-Substituted Indol-3-ylglyoxylamides Probing the LDi and L1/L2 Lipophilic Regions of the Benzodiazepine Receptor Site in Search for Subtype-Selective Ligands.
2007 Primofiore, G.; Taliani, S.; Da Settimo, F.; Marini, A. M.; La Motta, C.; Simorini, F.; Patrizi, M. P.; Sergianni, V.; Novellino, Ettore; Greco, Giovanni; Cosimelli, Barbara; Calderone, V.; Montali, M.; Besnard, F.; Martini, C.
Determination of the Absolute Configuration of a Chiral Oxadiazol-3-one Calcium Channel Blocker, Resolved by Using Chiral Chromatography, via Concerted Density Functional Theory Calculations of Its Vibrational Circular Dichroism, Electronic Circular Dichroism, and Optical Rotation.
2007 Stephens, P. J.; Devlin, F. J.; Gasparrini, F; Ciogli, A; Spinelli, D; Cosimelli, Barbara
The First Kinetic Evidence for Acid Catalysis in a Monocyclic Rearrangement of Heterocycles: Conversion of the Z-Phenylhydrazone of 5-Amino-3-benzoyl-1,2,4-oxadiazole into N,5-Diphenyl-2H-1,2,3-triazol-4-ylurea
2002 Cosimelli, Barbara; Frenna, V; Guernelli, S; Lanza, C. Z.; Macaluso, G; Petrillo, G; Spinelli, D.
8H-Pyrazolo[5',1':2,3]pyrimido[5,4-d][1,2]diazepine: A New Tricyclic System.
1993 Bruni, F; Cosimelli, Barbara; Costanzo, A; Guerrini, G; Selleri, S.
A convenient synthesis of psoralens.
2002 Chimichi, S; Boccalini, M; Cosimelli, Barbara; Viola, G; Vedaldi, D; Dall'Acqua, F.
Ring-ring Interconversions of Nitrosoimidazoles. The Effect of Some Condensed Six-membered Rings on the Reactivity.
2000 Billi, R; Cosimelli, Barbara; Spinelli, D; Andreani, A; Leoni, A.