COSIMELLI, BARBARA

COSIMELLI, BARBARA  

DIPARTIMENTO DI FARMACIA  

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Risultati 1 - 20 di 94 (tempo di esecuzione: 0.045 secondi).
Titolo Tipologia Data di pubblicazione Autore(i) File
Determination of the absolute configuration of the enantiomers of an oxadiazol-3-one calcium channel blocker, resolved by chiral HPLC, via concerted use of three chiroptical spectroscopies 8.02 Comunicazioni a Convegni o Seminari 2012 Giovanni Battista, Barrano; Salvatore, Caccamese; Cosimelli, Barbara; Frank J., Devlin; Elda, Severi; Domenico, Spinelli
Derivatives of benzimidazol-2-ylquinoline and benzimidazol-2-ylisoquinoline as selective A1 adenosine receptor antagonists with stimulant activity on human colon motility 1.1 Articolo in rivista 2011 Cosimelli, Barbara; S., Taliani; Greco, Giovanni; Novellino, Ettore; A., Sala; E., Severi; F., Da Settimo; C., La Motta; I., Pugliesi; L., Antonioli; M., Fornai; R., Colucci; C., Blandizzi; S., Daniele; M. L., Trincavelli; C., Martini
Natural and Synthetic Geiparvarins Are Strong and Selective MAO-B Inhibitors. Synthesis and SAR Studies. 1.1 Articolo in rivista 2002 Carotti, A; Carrieri, A; Chimichi, S; Boccalini, M; Cosimelli, Barbara; Gnerre, C; Carotti, A; Carrupt, P. A.; Testa, B.
A novel approach to the evaluation of the importance of steric and electronic effects in SNAr reactions: a computational, thermodynamic, 1H and 13C NMR study of “Meisenheimer-type” adducts in the benzo[b]thiophene series 1.1 Articolo in rivista 2010 Consiglio, G.; Cosimelli, Barbara; Guernelli, S.; Lanza, C. Z.; Sancassan, F.; Spinelli, D.; Stenta, M.
A New Convenient Route to 2-Oxoethoxycoumarins: Key Intermediates in the Synthesis of Natural Products. 1.1 Articolo in rivista 2002 Chimichi, S; Boccalini, M; Cosimelli, Barbara
Unambiguous Structure Determination of Some Pyrazolo[1,5-a]pyrimidine Derivatives by Multinuclear NMR Spectroscopy. 1.1 Articolo in rivista 1992 Chimichi, S; Cosimelli, Barbara; Bruni, F; Selleri, S.
On the reaction of 3-bromo-2-nitrobenzo[b]thiophene with some ortho-substituted anilines: an analysis of the products of reaction and of their NMR and MS properties 1.1 Articolo in rivista 2003 Cosimelli, Barbara; Lamartina, L; Lanza, C. Z.; Spinelli, D; Spisani, R; Vegna, F.
Synthesis and biological evaluation on human glioblastoma cells of novel pyrazolo[3,4-d]pyrimidine adenosine A(3) receptor antagonists 4.3 Poster 2010 Mugnaini, L.; La Motta, C.; Taliani, S; Simorini, F.; Salerno, S.; Marini, A. M.; Da Settimo, F.; Cosimelli, Barbara; Greco, Giovanni; Novellino, Ettore; Daniele, S.; Trincavelli, M. L.; Martini, C.
3-Aryl-[1,2,4]triazino[4,3-a]benzimidazol-4(10H)-one: a novel template for the design of highly selective A2B adenosine receptor antagonists 4.3 Poster 2012 Taliani, S.; Pugliesi, I.; Barresi, E.; Salerno, S.; Simorini, F.; La Motta, C.; Marini, A. M.; Da Settimo, F.; Cosconati, S.; Marinelli, Luciana; Cosimelli, Barbara; Greco, Giovanni; Novellino, Ettore; Daniele, S.; Trincavelli, M. L.; Martini, C.
Substituent effect on the electrochemical behaviour of some ortho-substituted (aryl)(2-nitrobenzo[b]thiophen-3-yl)amines. A combined experimental and computational study. 1.1 Articolo in rivista 2006 Bottoni, A; Cosimelli, Barbara; Scavetta, E; Spinelli, D; Spisani, R; Stenta, M; Tonelli, D.
Chemistry of Substituted Pyrazolo[1,5-a]pyrimidines. Part 3. A Structural Correc¬tion of Pyrazolo[1,5-a][1,3]diazepine Derivative on the Basis of 13C NMR Spectroscopy. 1.1 Articolo in rivista 1993 Chimichi, S; Cosimelli, Barbara; Bruni, F; Costanzo, A.
Calcium Channel Antagonists Discovered by a Multidisciplinary Approach. 1.1 Articolo in rivista 2006 Carosati, E; Cruciani, G; Chiarini, A; Budriesi, R; Ioan, P; Spisani, R; Spinelli, D; Cosimelli, Barbara; Fusi, F; Frosini, M; Matucci, R; Gasparrini, F; Ciogli, A; Stephens, P. J.; Devlin, F. J.
A New Class of Selective Myocardial Calcium Channel Modulators. 2. The Role of the Acetal Chain in Oxadiazol-3-one Derivatives 1.1 Articolo in rivista 2005 Budriesi, R; Carosati, E; Chiarini, A; Cosimelli, Barbara; Cruciani, G; Ioan, P; Spinelli, D; Spisani, R.
New 5-(2-ethenylsubstituted)-3(2H)-furanones with in vitro antiproliferative activity 1.1 Articolo in rivista 2003 Chimichi, S; Boccalini, M; Cosimelli, Barbara; Viola, G; Dallacqua, F.
Regioselective Synthesis of 4-Acetyl- and 5-Acetyl-3-methylisoxazole: their Conversion into Silyl- and Methyl Enol Ethers. 1.1 Articolo in rivista 1992 Chimichi, S; Cosimelli, Barbara
Ring-ring interconversion: the rearrangement of 6-(4-chlorophenyl)-3-methyl-5-nitrosoimidazo[2,1-b][1,3]thiazole into 8-(4-chlorophenyl)-8-hydroxy-5-methyl-8H-[1,4]thiazino[3,4-c][1,2,4]oxadiazol-3-one. Elucidation of the reaction product through spectroscopic and X-ray crystal structure analysis. 1.1 Articolo in rivista 1997 Andreani, A; Billi, R; Cosimelli, Barbara; Mugnoli, A; Rambaldi, M; Spinelli, D.
Ring opening of 2-substituted 4-nitrothiophenes with pyrrolidine. Access to new functionalized nitro-unsaturated building blocks. 1.1 Articolo in rivista 2001 Dell'Erba, C; Gabellini, A; Novi, M; Petrillo, G; Tavani, C; Cosimelli, Barbara; Spinelli, D.
Determination of the Absolute Configuration of a Chiral Oxadiazol-3-one Calcium Channel Blocker, Resolved by Using Chiral Chromatography, via Concerted Density Functional Theory Calculations of Its Vibrational Circular Dichroism, Electronic Circular Dichroism, and Optical Rotation. 1.1 Articolo in rivista 2007 Stephens, P. J.; Devlin, F. J.; Gasparrini, F; Ciogli, A; Spinelli, D; Cosimelli, Barbara
Diltiazem Analogues: The Last Ten Years on Structure Activity Relationships. 1.1 Articolo in rivista 2007 Budriesi, R; Cosimelli, Barbara; Ioan, P; Carosati, E; Ugenti, M. P.; Spisani, R.
New Fluorescent 2-Phenylindolglyoxylamide Derivatives as Probes Targeting the Peripheral-Type Benzodiazepine Receptor: Design, Synthesis and Biological Evaluation. 1.1 Articolo in rivista 2007 Taliani, S.; Simorini, F.; Sergianni, V.; LA MOTTA, C.; DA SETTIMO, F.; Cosimelli, Barbara; ABIGNENTE DI FRASSELLO, Enrico; Greco, Giovanni; Novellino, Ettore; Rossi, L.; Gremigni, V.; Spinetti, F.; Chelli, B.; Martini, C.