COSIMELLI, BARBARA
COSIMELLI, BARBARA
DIPARTIMENTO DI FARMACIA
On the Nitration of 5-Phenyl- and 3-Methyl-5-phenylisoxazole.
1989 Chimichi, S; Cosimelli, Barbara
3-Aryl-[1,2,4]triazino[4,3-a]benzimidazol-4(10H)-one: a novel template for the design of highly selective A2B adenosine receptor antagonists
2012 Taliani, S.; Pugliesi, I.; Barresi, E.; Salerno, S.; Simorini, F.; La Motta, C.; Marini, A. M.; Da Settimo, F.; Cosconati, S.; Marinelli, Luciana; Cosimelli, Barbara; Greco, Giovanni; Novellino, Ettore; Daniele, S.; Trincavelli, M. L.; Martini, C.
Regioselective Synthesis of 4-Acetyl- and 5-Acetyl-3-methylisoxazole: their Conversion into Silyl- and Methyl Enol Ethers.
1992 Chimichi, S; Cosimelli, Barbara
A New Synthetic Route to 2,2’:5’,2”-Terthiophene-5-derivatives to Conjugate with Proteins and Monoclonal Antibodies.
1996 Cosimelli, Barbara; Neri, D; Roncucci, G.
Absolute configuration and biological profile of two thiazinooxadiazol-3-ones with L-type calcium channel activity: a study of the structural effects
2012 Ioan, P.; Ciogli, A.; Sirci, F.; Budriesi, R.; Cosimelli, Barbara; Pierini, M.; Severi, E.; Chiarini, A.; Cruciani, G.; Gasparrini, F.; Spinelli, D.; Carosati, E.
8H-Pyrazolo[5',1':2,3]pyrimido[5,4-d][1,2]diazepine: A New Tricyclic System.
1993 Bruni, F; Cosimelli, Barbara; Costanzo, A; Guerrini, G; Selleri, S.
Carbon-13 NMR Studies on Azolopyridines. 3-The Isothiazolopyridine Systems.
1994 Chimichi, S; Cosimelli, Barbara; Tedeschi, P; Ponticelli, F.
Playing with Opening and Closing of Heterocycles: Using the Cusmano-Ruccia Reaction to Develop a Novel Class of Oxadiazolothiazinones, Active as Calcium Channel Modulators and P-Glycoprotein Inhibitors
2014 Domenico, Spinelli; Roberta, Budriesi; Cosimelli, Barbara; Elda, Severi; Matteo, Micucci; Massimo, Baroni; Fabio, Fusi; Pierfranco, Ioan; Simon, Cross; Maria, Frosini; Simona, Saponara; Rosanna, Matucci; Camillo, Rosano; Maurizio, Viale; Alberto, Chiarini; Emanuele, Carosati
2-Phenyl[1,2,3]triazolo[1,2-a][1,2,4]benzotriazin-1-one derivatives as a new class of adenosine receptor antagonists
2005 Primofiore, G.; Da Settimo, F.; Taliani, S.; Sergianni, V.; Simorini, F.; La Motta, C.; Marini, A. M.; Tuscano, D.; Martini, C.; Greco, Giovanni; Cosimelli, Barbara; Novellino, Ettore
Complete 1H (600 MHz) and 13C NMR Spectral Assignment of 3,4-bis[(3,4-Dimethoxyphenyl)methyl]dihydro-(3R-trans)-2(3H)-furanone (Matairesinol Dimethyl Ether), a Naturally Occurring Dibenzylbutyrolactone Lignan.
1993 Chimichi, S; Cosimelli, Barbara; BAMBAGIOTTI ALBERTI, M; Coran, S. A.; Vincieri, F. F.
Osteoblast differentiation and survival: A role for A2B adenosine receptor allosteric modulators
2014 Maria Letizia, Trincavelli; Simona, Daniele; Chiara, Giacomelli; Sabrina, Taliani; Federico Da, Settimo; Cosimelli, Barbara; Greco, Giovanni; Novellino, Ettore; Claudia, Martini
L-Type calcium channel blockers: from diltiazem to 1,2,4-oxadiazol-5-ones via thiazinooxadiazol-3-one derivatives
2009 Budriesi, R.; Cosimelli, Barbara; Ioan, P.; Ugenti, P.; Carosati, E.; Frosini, M.; Fusi, F.; Spisani, R.; Saponara, S.; Corda, G.; Cruciani, G.; Novellino, Ettore; Spinelli, D.; Chiarini, A.
Studies in organic mass spectrometry. Part 24 Electron ionization mass spectra of some aryl(2-nitrobenzo[b]thiophen-3-yl)amines.
1999 Avellone, G; Ceraulo, L; Lamartina, L; Cosimelli, Barbara; Spinelli, D; Zuppiroli, L.
Tertiary amides with a five-membered heteroaromatic ring as new probes for the translocator protein
2011 Cosimelli, Barbara; F., Simorini; S., Taliani; C., La Motta; F., Da Settimo; E., Severi; Greco, Giovanni; Novellino, Ettore; B., Costa; E., Da Pozzo; S., Bendinelli; C., Martini
Natural and Synthetic Geiparvarins Are Strong and Selective MAO-B Inhibitors. Synthesis and SAR Studies.
2002 Carotti, A; Carrieri, A; Chimichi, S; Boccalini, M; Cosimelli, Barbara; Gnerre, C; Carotti, A; Carrupt, P. A.; Testa, B.
From the Pharmacophore to the Homology Model of the Benzodiazepine Receptor: The Indolyglyoxylamides Affair.
2012 Cosimelli, Barbara; Cosconati, S.; Marinelli, Luciana; Novellino, Ettore; Greco, Giovanni
Preliminary Finding on a New Calcium Channel Entry Blocker Chemotype: 5,6-Diamino-4-hydroxy-2-mercaptopyrimidine Derivatives
2011 Cosimelli, Barbara; Elda, Severi; Novellino, Ettore; Anna, Cavaccini; Cataldi, Mauro; Roberta, Budriesi; Matteo, Micucci; Alberto, Chiarini; Pierfranco, Ioan
Modulation of A2B adenosine receptor by 1-Benzyl-3-ketoindole derivatives
2013 S., Taliani; M. L., Trincavelli; Cosimelli, Barbara; Laneri, Sonia; E., Severi; E., Barresi; I., Pugliesi; S., Daniele; C., Giacomelli; Greco, Giovanni; Novellino, Ettore; C., Martini; F., Da Settimo
Design, synthesis and biological evaluation of novel N-alkyl- and N-acyl-(7-substituted-2-phenylimidazo[1,2-a][1,3,5]triazin-4-yl)amines (ITAs) as novel A1 adenosine receptor antagonists
2002 Novellino, E.; ABIGNENTE DI FRASSELLO, Enrico; Cosimelli, B.; Greco, Giovanni; Iadanza, M.; Laneri, S.; Lavecchia, A.; Rimoli, M. G.; DA SETTIMO, F.; Primofiore, G.; Tuscano, D.; Martini, C.
From the central benzodiazepine receptor to the adenosine receptors exploiting the 3-diketoindole moiety
2011 Cosimelli, Barbara
| Titolo | Tipologia | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|---|
| On the Nitration of 5-Phenyl- and 3-Methyl-5-phenylisoxazole. | 1.1 Articolo in rivista | 1989 | Chimichi, S; Cosimelli, Barbara | |
| 3-Aryl-[1,2,4]triazino[4,3-a]benzimidazol-4(10H)-one: a novel template for the design of highly selective A2B adenosine receptor antagonists | 4.3 Poster | 2012 | Taliani, S.; Pugliesi, I.; Barresi, E.; Salerno, S.; Simorini, F.; La Motta, C.; Marini, A. M.; Da Settimo, F.; Cosconati, S.; Marinelli, Luciana; Cosimelli, Barbara; Greco, Giovanni; Novellino, Ettore; Daniele, S.; Trincavelli, M. L.; Martini, C. | |
| Regioselective Synthesis of 4-Acetyl- and 5-Acetyl-3-methylisoxazole: their Conversion into Silyl- and Methyl Enol Ethers. | 1.1 Articolo in rivista | 1992 | Chimichi, S; Cosimelli, Barbara | |
| A New Synthetic Route to 2,2’:5’,2”-Terthiophene-5-derivatives to Conjugate with Proteins and Monoclonal Antibodies. | 1.1 Articolo in rivista | 1996 | Cosimelli, Barbara; Neri, D; Roncucci, G. | |
| Absolute configuration and biological profile of two thiazinooxadiazol-3-ones with L-type calcium channel activity: a study of the structural effects | 1.1 Articolo in rivista | 2012 | Ioan, P.; Ciogli, A.; Sirci, F.; Budriesi, R.; Cosimelli, Barbara; Pierini, M.; Severi, E.; Chiarini, A.; Cruciani, G.; Gasparrini, F.; Spinelli, D.; Carosati, E. | |
| 8H-Pyrazolo[5',1':2,3]pyrimido[5,4-d][1,2]diazepine: A New Tricyclic System. | 1.1 Articolo in rivista | 1993 | Bruni, F; Cosimelli, Barbara; Costanzo, A; Guerrini, G; Selleri, S. | |
| Carbon-13 NMR Studies on Azolopyridines. 3-The Isothiazolopyridine Systems. | 1.1 Articolo in rivista | 1994 | Chimichi, S; Cosimelli, Barbara; Tedeschi, P; Ponticelli, F. | |
| Playing with Opening and Closing of Heterocycles: Using the Cusmano-Ruccia Reaction to Develop a Novel Class of Oxadiazolothiazinones, Active as Calcium Channel Modulators and P-Glycoprotein Inhibitors | 1.1 Articolo in rivista | 2014 | Domenico, Spinelli; Roberta, Budriesi; Cosimelli, Barbara; Elda, Severi; Matteo, Micucci; Massimo, Baroni; Fabio, Fusi; Pierfranco, Ioan; Simon, Cross; Maria, Frosini; Simona, Saponara; Rosanna, Matucci; Camillo, Rosano; Maurizio, Viale; Alberto, Chiarini; Emanuele, Carosati | |
| 2-Phenyl[1,2,3]triazolo[1,2-a][1,2,4]benzotriazin-1-one derivatives as a new class of adenosine receptor antagonists | 4.1 Articoli in Atti di convegno | 2005 | Primofiore, G.; Da Settimo, F.; Taliani, S.; Sergianni, V.; Simorini, F.; La Motta, C.; Marini, A. M.; Tuscano, D.; Martini, C.; Greco, Giovanni; Cosimelli, Barbara; Novellino, Ettore | |
| Complete 1H (600 MHz) and 13C NMR Spectral Assignment of 3,4-bis[(3,4-Dimethoxyphenyl)methyl]dihydro-(3R-trans)-2(3H)-furanone (Matairesinol Dimethyl Ether), a Naturally Occurring Dibenzylbutyrolactone Lignan. | 1.1 Articolo in rivista | 1993 | Chimichi, S; Cosimelli, Barbara; BAMBAGIOTTI ALBERTI, M; Coran, S. A.; Vincieri, F. F. | |
| Osteoblast differentiation and survival: A role for A2B adenosine receptor allosteric modulators | 1.1 Articolo in rivista | 2014 | Maria Letizia, Trincavelli; Simona, Daniele; Chiara, Giacomelli; Sabrina, Taliani; Federico Da, Settimo; Cosimelli, Barbara; Greco, Giovanni; Novellino, Ettore; Claudia, Martini | |
| L-Type calcium channel blockers: from diltiazem to 1,2,4-oxadiazol-5-ones via thiazinooxadiazol-3-one derivatives | 1.1 Articolo in rivista | 2009 | Budriesi, R.; Cosimelli, Barbara; Ioan, P.; Ugenti, P.; Carosati, E.; Frosini, M.; Fusi, F.; Spisani, R.; Saponara, S.; Corda, G.; Cruciani, G.; Novellino, Ettore; Spinelli, D.; Chiarini, A. | |
| Studies in organic mass spectrometry. Part 24 Electron ionization mass spectra of some aryl(2-nitrobenzo[b]thiophen-3-yl)amines. | 1.1 Articolo in rivista | 1999 | Avellone, G; Ceraulo, L; Lamartina, L; Cosimelli, Barbara; Spinelli, D; Zuppiroli, L. | |
| Tertiary amides with a five-membered heteroaromatic ring as new probes for the translocator protein | 1.1 Articolo in rivista | 2011 | Cosimelli, Barbara; F., Simorini; S., Taliani; C., La Motta; F., Da Settimo; E., Severi; Greco, Giovanni; Novellino, Ettore; B., Costa; E., Da Pozzo; S., Bendinelli; C., Martini | |
| Natural and Synthetic Geiparvarins Are Strong and Selective MAO-B Inhibitors. Synthesis and SAR Studies. | 1.1 Articolo in rivista | 2002 | Carotti, A; Carrieri, A; Chimichi, S; Boccalini, M; Cosimelli, Barbara; Gnerre, C; Carotti, A; Carrupt, P. A.; Testa, B. | |
| From the Pharmacophore to the Homology Model of the Benzodiazepine Receptor: The Indolyglyoxylamides Affair. | 1.1 Articolo in rivista | 2012 | Cosimelli, Barbara; Cosconati, S.; Marinelli, Luciana; Novellino, Ettore; Greco, Giovanni | |
| Preliminary Finding on a New Calcium Channel Entry Blocker Chemotype: 5,6-Diamino-4-hydroxy-2-mercaptopyrimidine Derivatives | 1.1 Articolo in rivista | 2011 | Cosimelli, Barbara; Elda, Severi; Novellino, Ettore; Anna, Cavaccini; Cataldi, Mauro; Roberta, Budriesi; Matteo, Micucci; Alberto, Chiarini; Pierfranco, Ioan | |
| Modulation of A2B adenosine receptor by 1-Benzyl-3-ketoindole derivatives | 1.1 Articolo in rivista | 2013 | S., Taliani; M. L., Trincavelli; Cosimelli, Barbara; Laneri, Sonia; E., Severi; E., Barresi; I., Pugliesi; S., Daniele; C., Giacomelli; Greco, Giovanni; Novellino, Ettore; C., Martini; F., Da Settimo | |
| Design, synthesis and biological evaluation of novel N-alkyl- and N-acyl-(7-substituted-2-phenylimidazo[1,2-a][1,3,5]triazin-4-yl)amines (ITAs) as novel A1 adenosine receptor antagonists | 1.1 Articolo in rivista | 2002 | Novellino, E.; ABIGNENTE DI FRASSELLO, Enrico; Cosimelli, B.; Greco, Giovanni; Iadanza, M.; Laneri, S.; Lavecchia, A.; Rimoli, M. G.; DA SETTIMO, F.; Primofiore, G.; Tuscano, D.; Martini, C. | |
| From the central benzodiazepine receptor to the adenosine receptors exploiting the 3-diketoindole moiety | 8.02 Comunicazioni a Convegni o Seminari | 2011 | Cosimelli, Barbara |