SANTAGADA, VINCENZO
SANTAGADA, VINCENZO
DIPARTIMENTO DI FARMACIA
A convenient synthesis by microwave heating and pharmacological evaluation of novel benzoyltriazole and saccharine derivatives as 5-HT1A receptor ligands.
2002 Caliendo, Giuseppe; Fiorino, Ferdinando; Perissutti, Elisa; Severino, Beatrice; Daniela, Scolaro; Stefania, Gessi; Elena, Cattabriga; Pier Andrea, Borea; Santagada, Vincenzo
Enhanced activity of a hydrogen sulphide-releasing derivative of mesalamine (ATB-429) in a mouse model of colitis
2007 Fiorucci, S; Orlandi, S; Mencarelli, A; Caliendo, Giuseppe; Santagada, Vincenzo; Distrutti, E; Santucci, L; Cirino, Giuseppe; Wallace, J. L.
Synthesis and biological activity of tripeptide FR113680 analogues containing unconventional amino acids.
1995 Caliendo, Giuseppe; Calignano, Antonio; Grieco, Paolo; Mancuso, F; Perissutti, Elisa; Santini, A; Santagada, Vincenzo
Synthesis by microwave irradiation and binding properties of novel 5-HT1A receptor ligands.
2001 Caliendo, Giuseppe; Fiorino, Ferdinando; Perissutti, Elisa; Severino, Beatrice; Gessi, S; Cattabriga, E; Borea, P. A.; Santagada, Vincenzo
Foye's Principi di Chimica Farmaceutica
2014 R., Amoroso; D., Barlocco; Caliendo, Giuseppe; Ritieni, Alberto; Novellino, Ettore; Santagada, Vincenzo; P., Diana; R., Di Santo; B., Gatto; S., Grasso; S., Moro; Mn, Romanelli; S., Guglielmo; V., De Filippis; D., Dalzoppo
Synthesis and in Vitro Activities of Highly Potent Selective Tripeptide Antagonists of the Neurokinin NK-1 Receptor.
1995 Caliendo, Giuseppe; Calignano, Antonio; Greco, Giovanni; Grieco, Paolo; Mancuso, F.; Perissutti, Elisa; Santagada, Vincenzo; Novellino, Ettore
Molecular Structure and Conformation of the (Z) and (E) Geometric Isomers of 2-(2-Phenylbenzylidene)-3-quinuclidinone.
1995 Santini, Antonello; Benedetti, Ettore; Pedone, Carlo; Giordano, M.; Caliendo, Giuseppe; Santagada, Vincenzo; Grieco, Paolo; Greco, Giovanni
Opioid pseudopeptides containing heteroaromatic or heteroaliphatic nuclei
2000 Balboni, G.; Salvadori, S.; Guerrini, R.; Bianchi, C.; Santagada, V.; Caliendo, Giuseppe; Bryant, S. D.; Lazarus, L. H.
Synthesis and Biological Activity of Benzotriazole Derivatives Structurally Related to Trazodone.
1995 Caliendo, Giuseppe; DI CARLO, Raffaele; Greco, Giovanni; Meli, Rosaria; Novellino, Ettore; Perissutti, Elisa; Santagada, Vincenzo
Synthesis, Local Anesthetic Activity and QSAR Studies for a Set of N-[2-(alkylamino)-ethyl]benzotriazol-X-yl Acetamides.
1995 Caliendo, Giuseppe; DI CARLO, Raffaele; Greco, Giovanni; Meli, Rosaria; Novellino, Ettore; Perissutti, Elisa; Santagada, Vincenzo
Synthesis and Antiinflammatory-Analgesic Profile of 1-Methyl-2-(4-X-benzoyl)imidazole-5-carboxylic Acids.
1995 Caliendo, Giuseppe; Cirino, Giuseppe; Greco, Giovanni; Novellino, Ettore; Perissutti, Elisa; Pinto, A.; Santagada, Vincenzo; Silipo, Carlo; Sorrentino, Ludovico
Synthesis and muscarinic receptor binding profiles of antagonist benzotriazole derivatives
1993 Cappello, B.; Greco, Giovanni; Novellino, Ettore; Perissutti, Elisa; Santagada, Vincenzo; Silipo, C.; Vittoria, A.; Di Carlo, R.; Meli, Rosaria; Muccioli, G.
Structure-Affinity Relationship Studies on Benzotriazole Derivatives Binding to 5-HT Receptor Subtypes.
1996 Caliendo, Giuseppe; Greco, Giovanni; Grieco, Paolo; Novellino, Ettore; Perissutti, Elisa; Santagada, Vincenzo; Barbarulo, D.; Esposito, E.; De Blasi, A.
Anti-inflammatory peptides: an update and future perspectives
2002 Santagada, Vincenzo; Ialenti, A.; Metafora, S.; Caliendo, G.; Maffia, P.; Morelli, F.; DE ROSA, R.; DE MARIA, S.; Carten, AND M.
Conformational analysis of three NK1 tripeptide antagonists: A proton nuclear magnetic resonance study
1997 Caliendo, Giuseppe; Grieco, Paolo; Perissutti, Elisa; Santagada, Vincenzo; Saviano, G.; Tancredi, T.; Temussi, P. A.
Bromazepam determination in human plasma by high-performance liquid chromatography coupled to tandem mass spectrometry: a highly sensitive and specific tool for bioequivalence studies
2004 T. L., Laurito; G. D., Mendes; Santagada, Vincenzo; Caliendo, Giuseppe; M. E. A., DE MORAES; G., DE NUCCI
Synthesis and Binding Affinities for 5-HT1A, 5-HT2A and 5-HT2C receptors of a series of 1- and 2-(4-arylpiperazinylalkyl)-4-(benzoyl)-1,2,3-triazole derivatives.
1999 Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; Santagada, Vincenzo; Albrizio, Stefania; Spadola, L.; Bruni, G.; Romeo, M. R.
Protease-activated receptor-2 activation improves efficiency of experimental ischemic preconditioning
2002 C., Napoli; F., DE NIGRIS; C., Cicala; Wallace, J. L.; M. R., Bucci; Bonaduce, Domenico; G., Caliendo; M., Condorelli; Santagada, Vincenzo; Cirino, Giuseppe
Comparative bioavailability of two losartan formulations in healthy human volunteers after a single dose administration.
2006 Oliveira, Ch; MEDEIROS SILVA, R; Santagada, Vincenzo; Caliendo, Giuseppe; Perissutti, Elisa; PRADO GALOPPO, M; MARCONDES REZENDE, V; BARRIENTOS ASTIGARRAGA, Re; Duarte, Mendes; DE NUCCI, G.
Synthesis of benzamide derivatives and their evaluation as antiprion agents
2012 Fiorino, Ferdinando; M., Eiden; A., Giese; Severino, Beatrice; A., Esposito; M. H., Groschup; Perissutti, Elisa; Magli, Elisa; Incisivo, GIUSEPPINA MARIA; Ciano, Antonio; Frecentese, Francesco; H. A., Kretzschmar; J., Wagner; Santagada, Vincenzo; Caliendo, Giuseppe
| Titolo | Tipologia | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|---|
| A convenient synthesis by microwave heating and pharmacological evaluation of novel benzoyltriazole and saccharine derivatives as 5-HT1A receptor ligands. | 1.1 Articolo in rivista | 2002 | Caliendo, Giuseppe; Fiorino, Ferdinando; Perissutti, Elisa; Severino, Beatrice; Daniela, Scolaro; Stefania, Gessi; Elena, Cattabriga; Pier Andrea, Borea; Santagada, Vincenzo | |
| Enhanced activity of a hydrogen sulphide-releasing derivative of mesalamine (ATB-429) in a mouse model of colitis | 1.1 Articolo in rivista | 2007 | Fiorucci, S; Orlandi, S; Mencarelli, A; Caliendo, Giuseppe; Santagada, Vincenzo; Distrutti, E; Santucci, L; Cirino, Giuseppe; Wallace, J. L. | |
| Synthesis and biological activity of tripeptide FR113680 analogues containing unconventional amino acids. | 1.1 Articolo in rivista | 1995 | Caliendo, Giuseppe; Calignano, Antonio; Grieco, Paolo; Mancuso, F; Perissutti, Elisa; Santini, A; Santagada, Vincenzo | |
| Synthesis by microwave irradiation and binding properties of novel 5-HT1A receptor ligands. | 1.1 Articolo in rivista | 2001 | Caliendo, Giuseppe; Fiorino, Ferdinando; Perissutti, Elisa; Severino, Beatrice; Gessi, S; Cattabriga, E; Borea, P. A.; Santagada, Vincenzo | |
| Foye's Principi di Chimica Farmaceutica | 3.8 Traduzione di libro | 2014 | R., Amoroso; D., Barlocco; Caliendo, Giuseppe; Ritieni, Alberto; Novellino, Ettore; Santagada, Vincenzo; P., Diana; R., Di Santo; B., Gatto; S., Grasso; S., Moro; Mn, Romanelli; S., Guglielmo; V., De Filippis; D., Dalzoppo | |
| Synthesis and in Vitro Activities of Highly Potent Selective Tripeptide Antagonists of the Neurokinin NK-1 Receptor. | 1.1 Articolo in rivista | 1995 | Caliendo, Giuseppe; Calignano, Antonio; Greco, Giovanni; Grieco, Paolo; Mancuso, F.; Perissutti, Elisa; Santagada, Vincenzo; Novellino, Ettore | |
| Molecular Structure and Conformation of the (Z) and (E) Geometric Isomers of 2-(2-Phenylbenzylidene)-3-quinuclidinone. | 1.1 Articolo in rivista | 1995 | Santini, Antonello; Benedetti, Ettore; Pedone, Carlo; Giordano, M.; Caliendo, Giuseppe; Santagada, Vincenzo; Grieco, Paolo; Greco, Giovanni | |
| Opioid pseudopeptides containing heteroaromatic or heteroaliphatic nuclei | 1.1 Articolo in rivista | 2000 | Balboni, G.; Salvadori, S.; Guerrini, R.; Bianchi, C.; Santagada, V.; Caliendo, Giuseppe; Bryant, S. D.; Lazarus, L. H. | |
| Synthesis and Biological Activity of Benzotriazole Derivatives Structurally Related to Trazodone. | 1.1 Articolo in rivista | 1995 | Caliendo, Giuseppe; DI CARLO, Raffaele; Greco, Giovanni; Meli, Rosaria; Novellino, Ettore; Perissutti, Elisa; Santagada, Vincenzo | |
| Synthesis, Local Anesthetic Activity and QSAR Studies for a Set of N-[2-(alkylamino)-ethyl]benzotriazol-X-yl Acetamides. | 1.1 Articolo in rivista | 1995 | Caliendo, Giuseppe; DI CARLO, Raffaele; Greco, Giovanni; Meli, Rosaria; Novellino, Ettore; Perissutti, Elisa; Santagada, Vincenzo | |
| Synthesis and Antiinflammatory-Analgesic Profile of 1-Methyl-2-(4-X-benzoyl)imidazole-5-carboxylic Acids. | 1.1 Articolo in rivista | 1995 | Caliendo, Giuseppe; Cirino, Giuseppe; Greco, Giovanni; Novellino, Ettore; Perissutti, Elisa; Pinto, A.; Santagada, Vincenzo; Silipo, Carlo; Sorrentino, Ludovico | |
| Synthesis and muscarinic receptor binding profiles of antagonist benzotriazole derivatives | 1.1 Articolo in rivista | 1993 | Cappello, B.; Greco, Giovanni; Novellino, Ettore; Perissutti, Elisa; Santagada, Vincenzo; Silipo, C.; Vittoria, A.; Di Carlo, R.; Meli, Rosaria; Muccioli, G. | |
| Structure-Affinity Relationship Studies on Benzotriazole Derivatives Binding to 5-HT Receptor Subtypes. | 1.1 Articolo in rivista | 1996 | Caliendo, Giuseppe; Greco, Giovanni; Grieco, Paolo; Novellino, Ettore; Perissutti, Elisa; Santagada, Vincenzo; Barbarulo, D.; Esposito, E.; De Blasi, A. | |
| Anti-inflammatory peptides: an update and future perspectives | 2.1 Contributo in volume (Capitolo o Saggio) | 2002 | Santagada, Vincenzo; Ialenti, A.; Metafora, S.; Caliendo, G.; Maffia, P.; Morelli, F.; DE ROSA, R.; DE MARIA, S.; Carten, AND M. | |
| Conformational analysis of three NK1 tripeptide antagonists: A proton nuclear magnetic resonance study | 1.1 Articolo in rivista | 1997 | Caliendo, Giuseppe; Grieco, Paolo; Perissutti, Elisa; Santagada, Vincenzo; Saviano, G.; Tancredi, T.; Temussi, P. A. | |
| Bromazepam determination in human plasma by high-performance liquid chromatography coupled to tandem mass spectrometry: a highly sensitive and specific tool for bioequivalence studies | 1.1 Articolo in rivista | 2004 | T. L., Laurito; G. D., Mendes; Santagada, Vincenzo; Caliendo, Giuseppe; M. E. A., DE MORAES; G., DE NUCCI | |
| Synthesis and Binding Affinities for 5-HT1A, 5-HT2A and 5-HT2C receptors of a series of 1- and 2-(4-arylpiperazinylalkyl)-4-(benzoyl)-1,2,3-triazole derivatives. | 1.1 Articolo in rivista | 1999 | Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; Santagada, Vincenzo; Albrizio, Stefania; Spadola, L.; Bruni, G.; Romeo, M. R. | |
| Protease-activated receptor-2 activation improves efficiency of experimental ischemic preconditioning | 1.1 Articolo in rivista | 2002 | C., Napoli; F., DE NIGRIS; C., Cicala; Wallace, J. L.; M. R., Bucci; Bonaduce, Domenico; G., Caliendo; M., Condorelli; Santagada, Vincenzo; Cirino, Giuseppe | |
| Comparative bioavailability of two losartan formulations in healthy human volunteers after a single dose administration. | 1.1 Articolo in rivista | 2006 | Oliveira, Ch; MEDEIROS SILVA, R; Santagada, Vincenzo; Caliendo, Giuseppe; Perissutti, Elisa; PRADO GALOPPO, M; MARCONDES REZENDE, V; BARRIENTOS ASTIGARRAGA, Re; Duarte, Mendes; DE NUCCI, G. | |
| Synthesis of benzamide derivatives and their evaluation as antiprion agents | 1.1 Articolo in rivista | 2012 | Fiorino, Ferdinando; M., Eiden; A., Giese; Severino, Beatrice; A., Esposito; M. H., Groschup; Perissutti, Elisa; Magli, Elisa; Incisivo, GIUSEPPINA MARIA; Ciano, Antonio; Frecentese, Francesco; H. A., Kretzschmar; J., Wagner; Santagada, Vincenzo; Caliendo, Giuseppe |