CALIENDO, GIUSEPPE
CALIENDO, GIUSEPPE
DIPARTIMENTO DI FARMACIA
pH-dependence of hydrophobic parameters in sets of ionizable drugs
1985 LA ROTONDA, MARIA IMMACOLATA; G., Amato; Barbato, Francesco; Caliendo, Giuseppe; C., Silipo; A., Vittoria
Relationships between log D and Rm values in a set of beta adrenoceptor bloking agents
1991 Barbato, Francesco; Caliendo, Giuseppe; Cappello, Brunella; LA ROTONDA, MARIA IMMACOLATA
Substrate specificity of recombinant dengue 2 virus NS2B-NS3protease: Influence of natural and unnatural basic amino acidson hydrolysis of synthetic fluorescent substrates
2007 I. E., Gouvea; M. A., Izidoro; W. A. S., Judice; M. H. S., Cezari; Caliendo, Giuseppe; Santagada, Vincenzo; C. N. D., dos Santos; M. H., Queiroz; M. A., Juliano; P. R., Young; D. P., Fairlie; L., Juliano
The application of microwave irradiation as new convenient synthetic procedure in drug discovery
2002 Santagada, Vincenzo; Perissutti, Elisa; Caliendo, Giuseppe
A convenient strategy of dimerization by microwave heating and using 2,5-diketopiperazine as scaffold.
2003 Santagada, Vincenzo; Fiorino, Ferdinando; Perissutti, Elisa; Severino, Beatrice; Terracciano, Sara; Cirino, Giuseppe; Caliendo, Giuseppe
Markedly Reduced Toxicity of a Hydrogen Sulfide-Releasing Derivative of Naproxen (ATB-346)
2010 Wallace, J. L.; Caliendo, Giuseppe; Santagada, Vincenzo; Cirino, Giuseppe
Enhanced activity of a hydrogen sulphide-releasing derivative of mesalamine (ATB-429) in a mouse model of colitis
2007 Fiorucci, S; Orlandi, S; Mencarelli, A; Caliendo, Giuseppe; Santagada, Vincenzo; Distrutti, E; Santucci, L; Cirino, Giuseppe; Wallace, J. L.
Design of inhibitors for human tissue kallikrein using non-natural aromatic and basic amino acids.
2002 Daniel C., Pimenta; Robson L., Melo; Caliendo, Giuseppe; Santagada, Vincenzo; Fiorino, Ferdinando; Severino, Beatrice; Gilberto De, Nucci; Luiz, Juliano; Maria, A. J. u. l. i. a. n. o.
Synthesis and structure-activity of antisense peptides corresponding to the region for CaM-binding domain of the inducible nitric oxide synthase
2000 Sautebin, L.; Rombol, L.; DI ROSA, M.; Caliendo, Giuseppe; Perissutti, Elisa; Grieco, G.; Severino, Beatrice; Santagada, Vincenzo
Synthesis and trazodone-like pharmacological profile of 1- and 2-[3-[4(X)-1-piperazinyl]-propyl]-benzotriazoles
1993 Caliendo, Giuseppe; Di Carlo, R.; Meli, Rosaria; Perissutti, Elisa; Santagada, Vincenzo; Silipo, C.; Vittoria, A.
Pharmacological dissection of vascular effects caused by activation of protease-activated receptor 1 and 2 in anesthetized rats
2001 Cicala, Carla; S., Morello; Santagada, Vincenzo; Caliendo, Giuseppe; L., Sorrentino; Cirino, Giuseppe
The nitric oxide related therapeutic phenomenon: a challenging task.
2002 Cirino, Giuseppe; Santagada, Vincenzo; Caliendo, Giuseppe
13C-NMR and 1H-NMR chemical shifts in a correlation analysis of benzotriazole derivatives active as plant growth regulators
1988 Sparatore, F.; Caliendo, Giuseppe; La Rotonda, M. I.; Novellino, Ettore; Silipo, C.; Vittoria, A.
73) Protease-activated receptor-2 activation improves efficiency of experimental ischemic preconditioning and reduces cardiac inflammation.
2002 C., Napoli; F., DE NIGRIS; C., Cicala; Wallace, J. L.; M. R., Bucci; Bonaduce, Domenico; Caliendo, Giuseppe; M., Condorelli; V., Santagada; Cirino, Giuseppe
Synthesis and hydrolysis by cathepsin B of fluorogenic substrates with the general structure benzoyl-X-ARG-MCA containing non-natural basic amino acids at position X
2001 Melo, R. L.; BARBOSA POZZO, R. C.; Alves, L. C. E.; Perissutti, E; Caliendo, G; Santagada, V; Juliano, L; Juliano, M. A.
Synthesis of new 1,2,3-benzotriazin-4-one-arylpiperazine derivatives as 5-HT1A serotonin receptor ligands.
2000 Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; Santagada, Vincenzo; Severino, Beatrice; Bruni, G; Romeo, M. R.
Synthesis and in vitro activities of NK-1 antagonists derived from L-Triptophan.
1997 Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; Santagada, Vincenzo; Calignano, Antonio; Mancuso, F.; Albrizio, Stefania
Synthesis and vasorelaxant activity of new 1,4-benzoxazine derivatives potassium channel openers.
2002 Caliendo, Giuseppe; Perissutti, Elisa; Santagada, Vincenzo; Fiorino, Ferdinando; Severino, Beatrice; D'EMMANUELE DI VILLA BIANCA, Roberta; Laura, Lippolis; Aldo, Pinto; Sorrentino, Raffaella
Minimal structural requirements for agonist activity of PAR-2 activating peptides.
2002 Santagada, Vincenzo; Caliendo, Giuseppe; Severino, Beatrice; Perissutti, Elisa; Fiorino, Ferdinando; Cicala, Carla; De Filippis, V; Cirino, Giuseppe
Synthesis of substituted benzamides as anti-inflammatory agents that inhibit preferentially cyclooxygenase 1 but do not cause gastric damage.
2001 Caliendo, Giuseppe; Santagada, Vincenzo; Perissutti, Elisa; Severino, Beatrice; Fiorino, Ferdinando; Warner, T. D.; Wallace, J. L.; Ifa, D. R.; Antunes, E; Cirino, Giuseppe; de Nucci, G.
Titolo | Tipologia | Data di pubblicazione | Autore(i) | File |
---|---|---|---|---|
pH-dependence of hydrophobic parameters in sets of ionizable drugs | 4.1 Articoli in Atti di convegno | 1985 | LA ROTONDA, MARIA IMMACOLATA; G., Amato; Barbato, Francesco; Caliendo, Giuseppe; C., Silipo; A., Vittoria | |
Relationships between log D and Rm values in a set of beta adrenoceptor bloking agents | 4.1 Articoli in Atti di convegno | 1991 | Barbato, Francesco; Caliendo, Giuseppe; Cappello, Brunella; LA ROTONDA, MARIA IMMACOLATA | |
Substrate specificity of recombinant dengue 2 virus NS2B-NS3protease: Influence of natural and unnatural basic amino acidson hydrolysis of synthetic fluorescent substrates | 1.1 Articolo in rivista | 2007 | I. E., Gouvea; M. A., Izidoro; W. A. S., Judice; M. H. S., Cezari; Caliendo, Giuseppe; Santagada, Vincenzo; C. N. D., dos Santos; M. H., Queiroz; M. A., Juliano; P. R., Young; D. P., Fairlie; L., Juliano | |
The application of microwave irradiation as new convenient synthetic procedure in drug discovery | 1.1 Articolo in rivista | 2002 | Santagada, Vincenzo; Perissutti, Elisa; Caliendo, Giuseppe | |
A convenient strategy of dimerization by microwave heating and using 2,5-diketopiperazine as scaffold. | 1.1 Articolo in rivista | 2003 | Santagada, Vincenzo; Fiorino, Ferdinando; Perissutti, Elisa; Severino, Beatrice; Terracciano, Sara; Cirino, Giuseppe; Caliendo, Giuseppe | |
Markedly Reduced Toxicity of a Hydrogen Sulfide-Releasing Derivative of Naproxen (ATB-346) | 1.1 Articolo in rivista | 2010 | Wallace, J. L.; Caliendo, Giuseppe; Santagada, Vincenzo; Cirino, Giuseppe | |
Enhanced activity of a hydrogen sulphide-releasing derivative of mesalamine (ATB-429) in a mouse model of colitis | 1.1 Articolo in rivista | 2007 | Fiorucci, S; Orlandi, S; Mencarelli, A; Caliendo, Giuseppe; Santagada, Vincenzo; Distrutti, E; Santucci, L; Cirino, Giuseppe; Wallace, J. L. | |
Design of inhibitors for human tissue kallikrein using non-natural aromatic and basic amino acids. | 1.1 Articolo in rivista | 2002 | Daniel C., Pimenta; Robson L., Melo; Caliendo, Giuseppe; Santagada, Vincenzo; Fiorino, Ferdinando; Severino, Beatrice; Gilberto De, Nucci; Luiz, Juliano; Maria, A. J. u. l. i. a. n. o. | |
Synthesis and structure-activity of antisense peptides corresponding to the region for CaM-binding domain of the inducible nitric oxide synthase | 1.1 Articolo in rivista | 2000 | Sautebin, L.; Rombol, L.; DI ROSA, M.; Caliendo, Giuseppe; Perissutti, Elisa; Grieco, G.; Severino, Beatrice; Santagada, Vincenzo | |
Synthesis and trazodone-like pharmacological profile of 1- and 2-[3-[4(X)-1-piperazinyl]-propyl]-benzotriazoles | 1.1 Articolo in rivista | 1993 | Caliendo, Giuseppe; Di Carlo, R.; Meli, Rosaria; Perissutti, Elisa; Santagada, Vincenzo; Silipo, C.; Vittoria, A. | |
Pharmacological dissection of vascular effects caused by activation of protease-activated receptor 1 and 2 in anesthetized rats | 1.1 Articolo in rivista | 2001 | Cicala, Carla; S., Morello; Santagada, Vincenzo; Caliendo, Giuseppe; L., Sorrentino; Cirino, Giuseppe | |
The nitric oxide related therapeutic phenomenon: a challenging task. | 1.1 Articolo in rivista | 2002 | Cirino, Giuseppe; Santagada, Vincenzo; Caliendo, Giuseppe | |
13C-NMR and 1H-NMR chemical shifts in a correlation analysis of benzotriazole derivatives active as plant growth regulators | 1.1 Articolo in rivista | 1988 | Sparatore, F.; Caliendo, Giuseppe; La Rotonda, M. I.; Novellino, Ettore; Silipo, C.; Vittoria, A. | |
73) Protease-activated receptor-2 activation improves efficiency of experimental ischemic preconditioning and reduces cardiac inflammation. | 1.1 Articolo in rivista | 2002 | C., Napoli; F., DE NIGRIS; C., Cicala; Wallace, J. L.; M. R., Bucci; Bonaduce, Domenico; Caliendo, Giuseppe; M., Condorelli; V., Santagada; Cirino, Giuseppe | |
Synthesis and hydrolysis by cathepsin B of fluorogenic substrates with the general structure benzoyl-X-ARG-MCA containing non-natural basic amino acids at position X | 1.1 Articolo in rivista | 2001 | Melo, R. L.; BARBOSA POZZO, R. C.; Alves, L. C. E.; Perissutti, E; Caliendo, G; Santagada, V; Juliano, L; Juliano, M. A. | |
Synthesis of new 1,2,3-benzotriazin-4-one-arylpiperazine derivatives as 5-HT1A serotonin receptor ligands. | 1.1 Articolo in rivista | 2000 | Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; Santagada, Vincenzo; Severino, Beatrice; Bruni, G; Romeo, M. R. | |
Synthesis and in vitro activities of NK-1 antagonists derived from L-Triptophan. | 1.1 Articolo in rivista | 1997 | Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; Santagada, Vincenzo; Calignano, Antonio; Mancuso, F.; Albrizio, Stefania | |
Synthesis and vasorelaxant activity of new 1,4-benzoxazine derivatives potassium channel openers. | 1.1 Articolo in rivista | 2002 | Caliendo, Giuseppe; Perissutti, Elisa; Santagada, Vincenzo; Fiorino, Ferdinando; Severino, Beatrice; D'EMMANUELE DI VILLA BIANCA, Roberta; Laura, Lippolis; Aldo, Pinto; Sorrentino, Raffaella | |
Minimal structural requirements for agonist activity of PAR-2 activating peptides. | 1.1 Articolo in rivista | 2002 | Santagada, Vincenzo; Caliendo, Giuseppe; Severino, Beatrice; Perissutti, Elisa; Fiorino, Ferdinando; Cicala, Carla; De Filippis, V; Cirino, Giuseppe | |
Synthesis of substituted benzamides as anti-inflammatory agents that inhibit preferentially cyclooxygenase 1 but do not cause gastric damage. | 1.1 Articolo in rivista | 2001 | Caliendo, Giuseppe; Santagada, Vincenzo; Perissutti, Elisa; Severino, Beatrice; Fiorino, Ferdinando; Warner, T. D.; Wallace, J. L.; Ifa, D. R.; Antunes, E; Cirino, Giuseppe; de Nucci, G. |