CALIENDO, GIUSEPPE

CALIENDO, GIUSEPPE  

DIPARTIMENTO DI FARMACIA  

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Synthesis and structure-activity of antisense peptides corresponding to the region for CaM-binding domain of the inducible nitric oxide synthase 1.1 Articolo in rivista 2000 Sautebin, L.; Rombol, L.; DI ROSA, M.; Caliendo, Giuseppe; Perissutti, Elisa; Grieco, G.; Severino, Beatrice; Santagada, Vincenzo
Human Tissue Kallikrein S1 Subsite Recognition of Non-Natural Basic Amino Acids 1.1 Articolo in rivista 2001 MELO ROBSON, L; POZZO ROSELI C., Barbosa; PIMENTA DANIEL, C; Perissutti, Elisa; Caliendo, Giuseppe; Santagada, Vincenzo; Juliano, Luiz; JULIANO MARIA, A.
Synthesis and Binding Affinities for 5-HT1A, 5-HT2A and 5-HT2C receptors of a series of 1- and 2-(4-arylpiperazinylalkyl)-4-(benzoyl)-1,2,3-triazole derivatives. 1.1 Articolo in rivista 1999 Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; Santagada, Vincenzo; Albrizio, Stefania; Spadola, L.; Bruni, G.; Romeo, M. R.
Phenol derived CVFM analogs inhibitors of ras farnesyl transferase possessing cellular in vitro activity. 1.1 Articolo in rivista 1998 Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; Ramunno, Anna; Santagada, Vincenzo; Albrizio, Stefania; Califano, D.; Giuliano, A.; Santelli, G.
Synthesis and in vitro activities of NK-1 antagonists derived from L-Triptophan. 1.1 Articolo in rivista 1997 Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; Santagada, Vincenzo; Calignano, Antonio; Mancuso, F.; Albrizio, Stefania
Synthesis of novel anti-inflammatory peptides derived from the amino-acid sequence of the bioactive protein SV-IV 1.1 Articolo in rivista 2001 Ialenti, Armando; Santagada, Vincenzo; Caliendo, Giuseppe; Severino, Beatrice; Fiorino, Ferdinando; Maffia, Pasquale; Ianaro, Angela; Morelli, F; DI MICCO, B; Carteni', M; Stiuso, P; Metafora, V; Metafora, S.
Probing the shape of a hydrophobic pocket in the active site of delta-opioid antagonists 1.1 Articolo in rivista 2001 Santagada, V; Caliendo, G; Severino, B; Perissutti, Elisa; E, Ceccarelli; F, Giusti; L, Mazzoni; Mr, Salvadori; S, Temussi; Pa,
Comparative bioavailability of two losartan formulations in healthy human volunteers after a single dose administration. 1.1 Articolo in rivista 2006 Oliveira, Ch; MEDEIROS SILVA, R; Santagada, Vincenzo; Caliendo, Giuseppe; Perissutti, Elisa; PRADO GALOPPO, M; MARCONDES REZENDE, V; BARRIENTOS ASTIGARRAGA, Re; Duarte, Mendes; DE NUCCI, G.
Synthesis, Pharmacological Evaluation, and Molecular Modeling Studies of Novel Peptidic CAAX Analogues as Farnesyl-Protein-Transferase Inhibitors 1.1 Articolo in rivista 2006 Santagada, Vincenzo; Caliendo, Giuseppe; Severino, Beatrice; Lavecchia, Antonio; Perissutti, Elisa; Fiorino, Ferdinando; Zampella, Angela; Sepe, Valentina; Califano, D.; Santelli, G.; Novellino, Ettore
Protease activated receptor-2 modulates myocardial ischemia reperfusion injury in the rat heart. 1.1 Articolo in rivista 2000 Napoli, C; Cicala, Carla; Wallace, J; DE NIGRIS, F; Santagada, V; Caliendo, G; Franconi, F; Ignarro, L; Cirino, Giuseppe
Synthesis and antinociceptive Activity of Peptides Related to Interleukin-1b193-195 Lys-Pro-Thr. 1.1 Articolo in rivista 1996 Caliendo, Giuseppe; Greco, Giovanni; Grieco, Paolo; Perissutti, Elisa; Santagada, Vincenzo; Ialenti, Armando; Maffia, Pasquale; Albrizio, Stefania; Santini, Antonello
Conformation-activity relationship of peptide T and new pseudocyclic hexapeptide analogs. 1.1 Articolo in rivista 2007 D'Ursi, A; Caliendo, Giuseppe; Perissutti, Elisa; Santagada, Vincenzo; Severino, Beatrice; Albrizio, Stefania; Bifulco, G; Spisani, S; Temussi, PIERO ANDREA
Combined Use of Factorial Design and Comparative Molecular Field Analysis (CoMFA): a Case Study. 1.1 Articolo in rivista 1994 Caliendo, Giuseppe; Greco, Giovanni; Novellino, Ettore; Perissutti, Elisa; Santagada, Vincenzo; Silipo, Carlo
Anti-inflammatory peptides: an update and future perspectives 2.1 Contributo in volume (Capitolo o Saggio) 2002 Santagada, Vincenzo; Ialenti, A.; Metafora, S.; Caliendo, G.; Maffia, P.; Morelli, F.; DE ROSA, R.; DE MARIA, S.; Carten, AND M.
Enhanced activity of a hydrogen sulphide-releasing derivative of mesalamine (ATB-429) in a mouse model of colitis 1.1 Articolo in rivista 2007 Fiorucci, S; Orlandi, S; Mencarelli, A; Caliendo, Giuseppe; Santagada, Vincenzo; Distrutti, E; Santucci, L; Cirino, Giuseppe; Wallace, J. L.
PAR1 Antagonism Protects Against Experimental Liver Fibrosis. Role of Proteinase Receptors in Stellate Cell Activation 1.1 Articolo in rivista 2004 Fiorucci, S.; Antonelli, E.; Distrutti, E.; Severino, Beatrice; Fiorentina, R.; Baldoni, M.; Caliendo, Giuseppe; Santagada, Vincenzo; Morelli, A.; Cirino, Giuseppe
A convenient strategy of dimerization by microwave heating and using 2,5-diketopiperazine as scaffold. 1.1 Articolo in rivista 2003 Santagada, Vincenzo; Fiorino, Ferdinando; Perissutti, Elisa; Severino, Beatrice; Terracciano, Sara; Cirino, Giuseppe; Caliendo, Giuseppe
A convenient synthesis by microwave irradiation of an active metabolite (EXP-3174) of losartan. 1.1 Articolo in rivista 2003 Santagada, Vincenzo; Fiorino, Ferdinando; Perissutti, Elisa; Severino, Beatrice; Terracciano, Sara; Cleber Evandro, Teixeira; Caliendo, Giuseppe
Microwave-enhanced solution coupling of the a,a-dialkyl amino acid, Aib 1.1 Articolo in rivista 2001 Santagada, Vincenzo; Fiorino, Ferdinando; Perissutti, Elisa; Severino, Beatrice; De Filippis, V; Vivenzio, B; Caliendo, Giuseppe
Gastrointestinal safety and anti-inflammatory effects of a hydrogen sulfide-releasing diclofenac derivative in the rat 1.1 Articolo in rivista 2007 Wallace, Jl; Caliendo, Giuseppe; Santagada, Vincenzo; Cirino, Giuseppe; Fiorucci, S.