CALIENDO, GIUSEPPE
CALIENDO, GIUSEPPE
DIPARTIMENTO DI FARMACIA
Relationships between log D and Rm values in a set of beta adrenoceptor bloking agents
1991 Barbato, Francesco; Caliendo, Giuseppe; Cappello, Brunella; LA ROTONDA, MARIA IMMACOLATA
le microonde nella sintesi organica. fondamenti e applicazioni in chimica farmaceutica
2008 Santagada, Vincenzo; Caliendo, Giuseppe; Perissutti, Elisa
Foye's Principi di Chimica Farmaceutica
2014 R., Amoroso; D., Barlocco; Caliendo, Giuseppe; Ritieni, Alberto; Novellino, Ettore; Santagada, Vincenzo; P., Diana; R., Di Santo; B., Gatto; S., Grasso; S., Moro; Mn, Romanelli; S., Guglielmo; V., De Filippis; D., Dalzoppo
73) Protease-activated receptor-2 activation improves efficiency of experimental ischemic preconditioning and reduces cardiac inflammation.
2002 C., Napoli; F., DE NIGRIS; C., Cicala; Wallace, J. L.; M. R., Bucci; Bonaduce, Domenico; Caliendo, Giuseppe; M., Condorelli; V., Santagada; Cirino, Giuseppe
In vitro mutagenicity of anti-inflammatory parsalmide analogues PA7, PA10, and PA31 triggered by biotransformation into hydroxy derivatives
2006 Cardoso, Hs; Bicalho, B; Genari, P; Santagada, Vincenzo; Caliendo, Giuseppe; Perissutti, Elisa; Donato, Jl; DE NUCCI, G.
Synthesis and antimicrobial activities of 5-amidobenzotriazole derivatives
1990 Caliendo, Giuseppe; Novellino, Ettore; Saliocco, G.; Santagada, Vincenzo; Silipo, V.; Vittoria, A.
A convenient synthesis by microwave heating and pharmacological evaluation of novel benzoyltriazole and saccharine derivatives as 5-HT1A receptor ligands.
2002 Caliendo, Giuseppe; Fiorino, Ferdinando; Perissutti, Elisa; Severino, Beatrice; Daniela, Scolaro; Stefania, Gessi; Elena, Cattabriga; Pier Andrea, Borea; Santagada, Vincenzo
Structure-Affinity Relationship Studies on Benzotriazole Derivatives Binding to 5-HT Receptor Subtypes.
1996 Caliendo, Giuseppe; Greco, Giovanni; Grieco, Paolo; Novellino, Ettore; Perissutti, Elisa; Santagada, Vincenzo; Barbarulo, D.; Esposito, E.; De Blasi, A.
Design of inhibitors for human tissue kallikrein using non-natural aromatic and basic amino acids.
2002 Daniel C., Pimenta; Robson L., Melo; Caliendo, Giuseppe; Santagada, Vincenzo; Fiorino, Ferdinando; Severino, Beatrice; Gilberto De, Nucci; Luiz, Juliano; Maria, A. J. u. l. i. a. n. o.
Markedly Reduced Toxicity of a Hydrogen Sulfide-Releasing Derivative of Naproxen (ATB-346)
2010 Wallace, J. L.; Caliendo, Giuseppe; Santagada, Vincenzo; Cirino, Giuseppe
Solid-State Structure and Conformation of (Z)-2-(Phenylbenzylidene)-3-quinuclidinone, an Intermediate in the Synthesis of Quinuclidine Derivatives
1994 Santini, Antonello; Pedone, Carlo; Benedetti, Ettore; Silipo, Carlo; Vittoria, Antonio; Caliendo, Giuseppe; Greco, Giovanni
PAR1 Antagonism Protects Against Experimental Liver Fibrosis. Role of Proteinase Receptors in Stellate Cell Activation
2004 Fiorucci, S.; Antonelli, E.; Distrutti, E.; Severino, Beatrice; Fiorentina, R.; Baldoni, M.; Caliendo, Giuseppe; Santagada, Vincenzo; Morelli, A.; Cirino, Giuseppe
Synthesis of new 1,2,3-benzotriazin-4-one-arylpiperazine derivatives as 5-HT1A serotonin receptor ligands.
2000 Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; Santagada, Vincenzo; Severino, Beatrice; Bruni, G; Romeo, M. R.
Pharmacokinetics of Dihydroergocristine and its major metabolite 8'-Hydroxy-Dihydroergocristine in Human plasma
2005 B., Bicalho; G. C., Guzzo; S., Lilla; H. O., DOS SANTOS; G. D., Mendes; Caliendo, Giuseppe; Perissutti, Elisa; Aiello, Anna; Luciano, Paolo; Santagada, Vincenzo; A. S., Pereira; G., DE NUCCIA
Na+/Ca2+ exchanger in Na+ efflux-Ca2+ influx mode of operation exerts a neuroprotective role in cellular models of in vitro anoxia and in vivo cerebral ischemia.
2002 Tortiglione, A.; Pignataro, Giuseppe; Minale, M.; Secondo, Agnese; Scorziello, Antonella; DI RENZO, GIANFRANCO MARIA LUIGI; Amoroso, S.; Caliendo, Giuseppe; Santagada, Vincenzo; Annunziato, Lucio
A convenient strategy of dimerization by microwave heating and using 2,5-diketopiperazine as scaffold.
2003 Santagada, Vincenzo; Fiorino, Ferdinando; Perissutti, Elisa; Severino, Beatrice; Terracciano, Sara; Cirino, Giuseppe; Caliendo, Giuseppe
Synthesis and antinociceptive Activity of Peptides Related to Interleukin-1b193-195 Lys-Pro-Thr.
1996 Caliendo, Giuseppe; Greco, Giovanni; Grieco, Paolo; Perissutti, Elisa; Santagada, Vincenzo; Ialenti, Armando; Maffia, Pasquale; Albrizio, Stefania; Santini, Antonello
Pyrrolobenzoxazepinone (PBO) Derivatives as Non-Nucleoside HIV-1 Reverse Transcriptase (RT) Inhibitors. Further Structure-Activity Relationship Studies and Identification of More Potent Broad Spectrum HIV-1 RT Inhibitors with Antiviral Activity.
1999 Campiani, G.; Morelli, Elena; Fabbrini, M.; Nacci, V.; Greco, Giovanni; Novellino, Ettore; Ramunno, A.; Maga, G.; Spadari, S.; Caliendo, Giuseppe; Bergamini, A.; Faggioli, E.; Uccella, I.; Bolacchi, F.; Marini, S.; Coletta, M.; Nacca, A.; Caccia, S.
Bromazepam determination in human plasma by high-performance liquid chromatography coupled to tandem mass spectrometry: a highly sensitive and specific tool for bioequivalence studies
2004 T. L., Laurito; G. D., Mendes; Santagada, Vincenzo; Caliendo, Giuseppe; M. E. A., DE MORAES; G., DE NUCCI
S1 subsite specificity of a recombinant cysteine proteinase, CPB, of Leishmania mexicana compared with cruzain, human cathepsin L and papain using substrates containing non-natural basic amino acids.
2001 Alves, L. C.; Melo, R. L.; Sanderson, S. J.; Mottram, J. C.; Coombs, G. H.; Caliendo, Giuseppe; Santagada, V.; Juliano, L.; Juliano, M. A.
| Titolo | Tipologia | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|---|
| Relationships between log D and Rm values in a set of beta adrenoceptor bloking agents | 4.1 Articoli in Atti di convegno | 1991 | Barbato, Francesco; Caliendo, Giuseppe; Cappello, Brunella; LA ROTONDA, MARIA IMMACOLATA | |
| le microonde nella sintesi organica. fondamenti e applicazioni in chimica farmaceutica | 3.1 Monografia o trattato scientifico | 2008 | Santagada, Vincenzo; Caliendo, Giuseppe; Perissutti, Elisa | |
| Foye's Principi di Chimica Farmaceutica | 3.8 Traduzione di libro | 2014 | R., Amoroso; D., Barlocco; Caliendo, Giuseppe; Ritieni, Alberto; Novellino, Ettore; Santagada, Vincenzo; P., Diana; R., Di Santo; B., Gatto; S., Grasso; S., Moro; Mn, Romanelli; S., Guglielmo; V., De Filippis; D., Dalzoppo | |
| 73) Protease-activated receptor-2 activation improves efficiency of experimental ischemic preconditioning and reduces cardiac inflammation. | 1.1 Articolo in rivista | 2002 | C., Napoli; F., DE NIGRIS; C., Cicala; Wallace, J. L.; M. R., Bucci; Bonaduce, Domenico; Caliendo, Giuseppe; M., Condorelli; V., Santagada; Cirino, Giuseppe | |
| In vitro mutagenicity of anti-inflammatory parsalmide analogues PA7, PA10, and PA31 triggered by biotransformation into hydroxy derivatives | 1.1 Articolo in rivista | 2006 | Cardoso, Hs; Bicalho, B; Genari, P; Santagada, Vincenzo; Caliendo, Giuseppe; Perissutti, Elisa; Donato, Jl; DE NUCCI, G. | |
| Synthesis and antimicrobial activities of 5-amidobenzotriazole derivatives | 1.1 Articolo in rivista | 1990 | Caliendo, Giuseppe; Novellino, Ettore; Saliocco, G.; Santagada, Vincenzo; Silipo, V.; Vittoria, A. | |
| A convenient synthesis by microwave heating and pharmacological evaluation of novel benzoyltriazole and saccharine derivatives as 5-HT1A receptor ligands. | 1.1 Articolo in rivista | 2002 | Caliendo, Giuseppe; Fiorino, Ferdinando; Perissutti, Elisa; Severino, Beatrice; Daniela, Scolaro; Stefania, Gessi; Elena, Cattabriga; Pier Andrea, Borea; Santagada, Vincenzo | |
| Structure-Affinity Relationship Studies on Benzotriazole Derivatives Binding to 5-HT Receptor Subtypes. | 1.1 Articolo in rivista | 1996 | Caliendo, Giuseppe; Greco, Giovanni; Grieco, Paolo; Novellino, Ettore; Perissutti, Elisa; Santagada, Vincenzo; Barbarulo, D.; Esposito, E.; De Blasi, A. | |
| Design of inhibitors for human tissue kallikrein using non-natural aromatic and basic amino acids. | 1.1 Articolo in rivista | 2002 | Daniel C., Pimenta; Robson L., Melo; Caliendo, Giuseppe; Santagada, Vincenzo; Fiorino, Ferdinando; Severino, Beatrice; Gilberto De, Nucci; Luiz, Juliano; Maria, A. J. u. l. i. a. n. o. | |
| Markedly Reduced Toxicity of a Hydrogen Sulfide-Releasing Derivative of Naproxen (ATB-346) | 1.1 Articolo in rivista | 2010 | Wallace, J. L.; Caliendo, Giuseppe; Santagada, Vincenzo; Cirino, Giuseppe | |
| Solid-State Structure and Conformation of (Z)-2-(Phenylbenzylidene)-3-quinuclidinone, an Intermediate in the Synthesis of Quinuclidine Derivatives | 1.1 Articolo in rivista | 1994 | Santini, Antonello; Pedone, Carlo; Benedetti, Ettore; Silipo, Carlo; Vittoria, Antonio; Caliendo, Giuseppe; Greco, Giovanni | |
| PAR1 Antagonism Protects Against Experimental Liver Fibrosis. Role of Proteinase Receptors in Stellate Cell Activation | 1.1 Articolo in rivista | 2004 | Fiorucci, S.; Antonelli, E.; Distrutti, E.; Severino, Beatrice; Fiorentina, R.; Baldoni, M.; Caliendo, Giuseppe; Santagada, Vincenzo; Morelli, A.; Cirino, Giuseppe | |
| Synthesis of new 1,2,3-benzotriazin-4-one-arylpiperazine derivatives as 5-HT1A serotonin receptor ligands. | 1.1 Articolo in rivista | 2000 | Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; Santagada, Vincenzo; Severino, Beatrice; Bruni, G; Romeo, M. R. | |
| Pharmacokinetics of Dihydroergocristine and its major metabolite 8'-Hydroxy-Dihydroergocristine in Human plasma | 1.1 Articolo in rivista | 2005 | B., Bicalho; G. C., Guzzo; S., Lilla; H. O., DOS SANTOS; G. D., Mendes; Caliendo, Giuseppe; Perissutti, Elisa; Aiello, Anna; Luciano, Paolo; Santagada, Vincenzo; A. S., Pereira; G., DE NUCCIA | |
| Na+/Ca2+ exchanger in Na+ efflux-Ca2+ influx mode of operation exerts a neuroprotective role in cellular models of in vitro anoxia and in vivo cerebral ischemia. | 1.1 Articolo in rivista | 2002 | Tortiglione, A.; Pignataro, Giuseppe; Minale, M.; Secondo, Agnese; Scorziello, Antonella; DI RENZO, GIANFRANCO MARIA LUIGI; Amoroso, S.; Caliendo, Giuseppe; Santagada, Vincenzo; Annunziato, Lucio | |
| A convenient strategy of dimerization by microwave heating and using 2,5-diketopiperazine as scaffold. | 1.1 Articolo in rivista | 2003 | Santagada, Vincenzo; Fiorino, Ferdinando; Perissutti, Elisa; Severino, Beatrice; Terracciano, Sara; Cirino, Giuseppe; Caliendo, Giuseppe | |
| Synthesis and antinociceptive Activity of Peptides Related to Interleukin-1b193-195 Lys-Pro-Thr. | 1.1 Articolo in rivista | 1996 | Caliendo, Giuseppe; Greco, Giovanni; Grieco, Paolo; Perissutti, Elisa; Santagada, Vincenzo; Ialenti, Armando; Maffia, Pasquale; Albrizio, Stefania; Santini, Antonello | |
| Pyrrolobenzoxazepinone (PBO) Derivatives as Non-Nucleoside HIV-1 Reverse Transcriptase (RT) Inhibitors. Further Structure-Activity Relationship Studies and Identification of More Potent Broad Spectrum HIV-1 RT Inhibitors with Antiviral Activity. | 1.1 Articolo in rivista | 1999 | Campiani, G.; Morelli, Elena; Fabbrini, M.; Nacci, V.; Greco, Giovanni; Novellino, Ettore; Ramunno, A.; Maga, G.; Spadari, S.; Caliendo, Giuseppe; Bergamini, A.; Faggioli, E.; Uccella, I.; Bolacchi, F.; Marini, S.; Coletta, M.; Nacca, A.; Caccia, S. | |
| Bromazepam determination in human plasma by high-performance liquid chromatography coupled to tandem mass spectrometry: a highly sensitive and specific tool for bioequivalence studies | 1.1 Articolo in rivista | 2004 | T. L., Laurito; G. D., Mendes; Santagada, Vincenzo; Caliendo, Giuseppe; M. E. A., DE MORAES; G., DE NUCCI | |
| S1 subsite specificity of a recombinant cysteine proteinase, CPB, of Leishmania mexicana compared with cruzain, human cathepsin L and papain using substrates containing non-natural basic amino acids. | 1.1 Articolo in rivista | 2001 | Alves, L. C.; Melo, R. L.; Sanderson, S. J.; Mottram, J. C.; Coombs, G. H.; Caliendo, Giuseppe; Santagada, V.; Juliano, L.; Juliano, M. A. |