CALIENDO, GIUSEPPE
CALIENDO, GIUSEPPE
DIPARTIMENTO DI FARMACIA
Synthesis and trazodone-like pharmacological profile of 1- and 2-[3-[4(X)-1-piperazinyl]-propyl]-benzotriazoles
1993 Caliendo, Giuseppe; Di Carlo, R.; Meli, Rosaria; Perissutti, Elisa; Santagada, Vincenzo; Silipo, C.; Vittoria, A.
Pharmacological evaluation of benzotriazole derivatives structurally related to trazodone
1992 Perissutti, Elisa; Meli, Rosaria; Maggetti, S.; Caliendo, Giuseppe; Cappello, B.; Silipo, C.; Vittoria, A.; Di Carlo, R.
Assessment of substitution in the second pharmacophore of Dmt-Tic analogues
2000 Santagada, V.; Balboni, G.; Caliendo, Giuseppe; Guerrini, R.; Salvadori, S.; Bianchi, C.; Bryant, S. D.; Lazarus, L. H.
Probing the shape of a hydrophobic pocket in the active site of delta-opioid antagonists
2001 Santagada, V; Caliendo, G; Severino, B; Perissutti, Elisa; E, Ceccarelli; F, Giusti; L, Mazzoni; Mr, Salvadori; S, Temussi; Pa,
Combined Use of Factorial Design and Comparative Molecular Field Analysis (CoMFA): a Case Study.
1994 Caliendo, Giuseppe; Greco, Giovanni; Novellino, Ettore; Perissutti, Elisa; Santagada, Vincenzo; Silipo, Carlo
Anti-inflammatory peptides: an update and future perspectives
2002 Santagada, Vincenzo; Ialenti, A.; Metafora, S.; Caliendo, G.; Maffia, P.; Morelli, F.; DE ROSA, R.; DE MARIA, S.; Carten, AND M.
The application of microwave irradiation as new convenient synthetic procedure in drug discovery
2002 Santagada, Vincenzo; Perissutti, Elisa; Caliendo, Giuseppe
Synthesis of substituted benzamides as anti-inflammatory agents that inhibit preferentially cyclooxygenase 1 but do not cause gastric damage.
2001 Caliendo, Giuseppe; Santagada, Vincenzo; Perissutti, Elisa; Severino, Beatrice; Fiorino, Ferdinando; Warner, T. D.; Wallace, J. L.; Ifa, D. R.; Antunes, E; Cirino, Giuseppe; de Nucci, G.
Preparation and local anesthetic activity of benzotriazinone and benzoyltriazole derivatives.
1999 Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; Santagada, Vincenzo; Meli, Rosaria; MATTACE RASO, Giuseppina; Zanesco, A; De Nucci, G.
A convenient synthesis by microwave irradiation of an active metabolite (EXP-3174) of losartan.
2003 Santagada, Vincenzo; Fiorino, Ferdinando; Perissutti, Elisa; Severino, Beatrice; Terracciano, Sara; Cleber Evandro, Teixeira; Caliendo, Giuseppe
A nitro-arginine derivative of trimebutine (NO2-Arg-Trim) attenuates pain induced by colorectal distension in conscious rats.
2009 Distrutti, E.; Mencarelli, A.; Renga, B.; Caliendo, Giuseppe; Santagada, Vincenzo; Severino, Beatrice; Fiorucci, S.
Relationships between log D and Rm values in a set of beta adrenoceptor bloking agents
1991 Barbato, Francesco; Caliendo, Giuseppe; Cappello, Brunella; LA ROTONDA, MARIA IMMACOLATA
73) Protease-activated receptor-2 activation improves efficiency of experimental ischemic preconditioning and reduces cardiac inflammation.
2002 C., Napoli; F., DE NIGRIS; C., Cicala; Wallace, J. L.; M. R., Bucci; Bonaduce, Domenico; Caliendo, Giuseppe; M., Condorelli; V., Santagada; Cirino, Giuseppe
le microonde nella sintesi organica. fondamenti e applicazioni in chimica farmaceutica
2008 Santagada, Vincenzo; Caliendo, Giuseppe; Perissutti, Elisa
PAR1 Antagonism Protects Against Experimental Liver Fibrosis. Role of Proteinase Receptors in Stellate Cell Activation
2004 Fiorucci, S.; Antonelli, E.; Distrutti, E.; Severino, Beatrice; Fiorentina, R.; Baldoni, M.; Caliendo, Giuseppe; Santagada, Vincenzo; Morelli, A.; Cirino, Giuseppe
Sequence and structure-activity relationship of a scorpion venom toxin with nitrergic activity in rabbit corpus cavernosum
2003 Teixeira, C. E.; Ifa, D. R.; Corso, G.; Santagada, V.; Caliendo, Giuseppe; Antunes, E.; DE NUCCI, G.
Structure-Affinity Relationship Studies on Benzotriazole Derivatives Binding to 5-HT Receptor Subtypes.
1996 Caliendo, Giuseppe; Greco, Giovanni; Grieco, Paolo; Novellino, Ettore; Perissutti, Elisa; Santagada, Vincenzo; Barbarulo, D.; Esposito, E.; De Blasi, A.
Comparative bioavailability of two losartan formulations in healthy human volunteers after a single dose administration.
2006 Oliveira, Ch; MEDEIROS SILVA, R; Santagada, Vincenzo; Caliendo, Giuseppe; Perissutti, Elisa; PRADO GALOPPO, M; MARCONDES REZENDE, V; BARRIENTOS ASTIGARRAGA, Re; Duarte, Mendes; DE NUCCI, G.
Synthesis and biological activity of pseudopeptides inhibitors of Ras farnesyl transferase containing unconventional amino acids.
1999 Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; De Luca, S; Giuliano, A; Santelli, G; Califano, D; Severino, Beatrice; Santagada, Vincenzo
Synthesis and Structure-Activity Relationships of Antiinflammatory 1-Methyl-2-(4-X-benzoyl)imidazole-5-acetic Acids.
1994 Caliendo, Giuseppe; Cirino, Giuseppe; Greco, Giovanni; Novellino, Ettore; Perissutti, Elisa; Pinto, A.; Santagada, Vincenzo; Silipo, Carlo; Sorrentino, Ludovico
| Titolo | Tipologia | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|---|
| Synthesis and trazodone-like pharmacological profile of 1- and 2-[3-[4(X)-1-piperazinyl]-propyl]-benzotriazoles | 1.1 Articolo in rivista | 1993 | Caliendo, Giuseppe; Di Carlo, R.; Meli, Rosaria; Perissutti, Elisa; Santagada, Vincenzo; Silipo, C.; Vittoria, A. | |
| Pharmacological evaluation of benzotriazole derivatives structurally related to trazodone | 1.1 Articolo in rivista | 1992 | Perissutti, Elisa; Meli, Rosaria; Maggetti, S.; Caliendo, Giuseppe; Cappello, B.; Silipo, C.; Vittoria, A.; Di Carlo, R. | |
| Assessment of substitution in the second pharmacophore of Dmt-Tic analogues | 1.1 Articolo in rivista | 2000 | Santagada, V.; Balboni, G.; Caliendo, Giuseppe; Guerrini, R.; Salvadori, S.; Bianchi, C.; Bryant, S. D.; Lazarus, L. H. | |
| Probing the shape of a hydrophobic pocket in the active site of delta-opioid antagonists | 1.1 Articolo in rivista | 2001 | Santagada, V; Caliendo, G; Severino, B; Perissutti, Elisa; E, Ceccarelli; F, Giusti; L, Mazzoni; Mr, Salvadori; S, Temussi; Pa, | |
| Combined Use of Factorial Design and Comparative Molecular Field Analysis (CoMFA): a Case Study. | 1.1 Articolo in rivista | 1994 | Caliendo, Giuseppe; Greco, Giovanni; Novellino, Ettore; Perissutti, Elisa; Santagada, Vincenzo; Silipo, Carlo | |
| Anti-inflammatory peptides: an update and future perspectives | 2.1 Contributo in volume (Capitolo o Saggio) | 2002 | Santagada, Vincenzo; Ialenti, A.; Metafora, S.; Caliendo, G.; Maffia, P.; Morelli, F.; DE ROSA, R.; DE MARIA, S.; Carten, AND M. | |
| The application of microwave irradiation as new convenient synthetic procedure in drug discovery | 1.1 Articolo in rivista | 2002 | Santagada, Vincenzo; Perissutti, Elisa; Caliendo, Giuseppe | |
| Synthesis of substituted benzamides as anti-inflammatory agents that inhibit preferentially cyclooxygenase 1 but do not cause gastric damage. | 1.1 Articolo in rivista | 2001 | Caliendo, Giuseppe; Santagada, Vincenzo; Perissutti, Elisa; Severino, Beatrice; Fiorino, Ferdinando; Warner, T. D.; Wallace, J. L.; Ifa, D. R.; Antunes, E; Cirino, Giuseppe; de Nucci, G. | |
| Preparation and local anesthetic activity of benzotriazinone and benzoyltriazole derivatives. | 1.1 Articolo in rivista | 1999 | Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; Santagada, Vincenzo; Meli, Rosaria; MATTACE RASO, Giuseppina; Zanesco, A; De Nucci, G. | |
| A convenient synthesis by microwave irradiation of an active metabolite (EXP-3174) of losartan. | 1.1 Articolo in rivista | 2003 | Santagada, Vincenzo; Fiorino, Ferdinando; Perissutti, Elisa; Severino, Beatrice; Terracciano, Sara; Cleber Evandro, Teixeira; Caliendo, Giuseppe | |
| A nitro-arginine derivative of trimebutine (NO2-Arg-Trim) attenuates pain induced by colorectal distension in conscious rats. | 1.1 Articolo in rivista | 2009 | Distrutti, E.; Mencarelli, A.; Renga, B.; Caliendo, Giuseppe; Santagada, Vincenzo; Severino, Beatrice; Fiorucci, S. | |
| Relationships between log D and Rm values in a set of beta adrenoceptor bloking agents | 4.1 Articoli in Atti di convegno | 1991 | Barbato, Francesco; Caliendo, Giuseppe; Cappello, Brunella; LA ROTONDA, MARIA IMMACOLATA | |
| 73) Protease-activated receptor-2 activation improves efficiency of experimental ischemic preconditioning and reduces cardiac inflammation. | 1.1 Articolo in rivista | 2002 | C., Napoli; F., DE NIGRIS; C., Cicala; Wallace, J. L.; M. R., Bucci; Bonaduce, Domenico; Caliendo, Giuseppe; M., Condorelli; V., Santagada; Cirino, Giuseppe | |
| le microonde nella sintesi organica. fondamenti e applicazioni in chimica farmaceutica | 3.1 Monografia o trattato scientifico | 2008 | Santagada, Vincenzo; Caliendo, Giuseppe; Perissutti, Elisa | |
| PAR1 Antagonism Protects Against Experimental Liver Fibrosis. Role of Proteinase Receptors in Stellate Cell Activation | 1.1 Articolo in rivista | 2004 | Fiorucci, S.; Antonelli, E.; Distrutti, E.; Severino, Beatrice; Fiorentina, R.; Baldoni, M.; Caliendo, Giuseppe; Santagada, Vincenzo; Morelli, A.; Cirino, Giuseppe | |
| Sequence and structure-activity relationship of a scorpion venom toxin with nitrergic activity in rabbit corpus cavernosum | 1.1 Articolo in rivista | 2003 | Teixeira, C. E.; Ifa, D. R.; Corso, G.; Santagada, V.; Caliendo, Giuseppe; Antunes, E.; DE NUCCI, G. | |
| Structure-Affinity Relationship Studies on Benzotriazole Derivatives Binding to 5-HT Receptor Subtypes. | 1.1 Articolo in rivista | 1996 | Caliendo, Giuseppe; Greco, Giovanni; Grieco, Paolo; Novellino, Ettore; Perissutti, Elisa; Santagada, Vincenzo; Barbarulo, D.; Esposito, E.; De Blasi, A. | |
| Comparative bioavailability of two losartan formulations in healthy human volunteers after a single dose administration. | 1.1 Articolo in rivista | 2006 | Oliveira, Ch; MEDEIROS SILVA, R; Santagada, Vincenzo; Caliendo, Giuseppe; Perissutti, Elisa; PRADO GALOPPO, M; MARCONDES REZENDE, V; BARRIENTOS ASTIGARRAGA, Re; Duarte, Mendes; DE NUCCI, G. | |
| Synthesis and biological activity of pseudopeptides inhibitors of Ras farnesyl transferase containing unconventional amino acids. | 1.1 Articolo in rivista | 1999 | Caliendo, Giuseppe; Fiorino, Ferdinando; Grieco, Paolo; Perissutti, Elisa; De Luca, S; Giuliano, A; Santelli, G; Califano, D; Severino, Beatrice; Santagada, Vincenzo | |
| Synthesis and Structure-Activity Relationships of Antiinflammatory 1-Methyl-2-(4-X-benzoyl)imidazole-5-acetic Acids. | 1.1 Articolo in rivista | 1994 | Caliendo, Giuseppe; Cirino, Giuseppe; Greco, Giovanni; Novellino, Ettore; Perissutti, Elisa; Pinto, A.; Santagada, Vincenzo; Silipo, Carlo; Sorrentino, Ludovico |