DE MARINO, SIMONA
DE MARINO, SIMONA
Dipartimento di Farmacia
Phytochemical Analysis of the Methanolic Extract and Essential Oil from Leaves of Industrial Hemp Futura 75 Cultivar: Isolation of a New Cannabinoid Derivative and Biological Profile Using Computational Approaches
2022 De Vita, Simona; Finamore, Claudia; Chini, Maria Giovanna; Saviano, Gabriella; De Felice, Vincenzo; De Marino, Simona; Lauro, Gianluigi; Casapullo, Agostino; Fantasma, Francesca; Trombetta, Federico; Bifulco, Giuseppe; Iorizzi, Maria
Structure-based screening for the discovery of 1,2,4-oxadiazoles as promising hits for the development of new anti-inflammatory agents interfering with eicosanoid biosyn-thesis pathways
2021 Sciarretta, Martina; Saviano, Anella; Maione, Francesco; D'Auria, MARIA VALERIA; DE MARINO, Simona; Giordano, Assunta; Festa, Carmen
Synergism of a novel 1,2,4-oxadiazole-containing derivative with oxacillin against methicillin-resistant Staphylococcus aureus
2021 Buommino, Elisabetta; DE MARINO, Simona; Sciarretta, Martina; Piccolo, Marialuisa; Festa, Carmen; D'Auria, MARIA VALERIA
Synthesis of new isoxazole derivatives as fxr agonists with improved pharmacokinetic properties
2019 Finamore, C.; Sepe, V.; Baronissi, G.; Cassiano, C.; Monti, M. C.; De Marino, S.; Novellino, E.; Limongelli, V.; Fiorucci, S.; Zampella, A.
Design and synthesis of hyodeoxycholic acid derivatives as GPBAR1 receptor modulators useful in the treatment of colon inflammation
2020 Finamore, C.; De Marino, S.; Cassiano, C.; Di Leva, F. S.; Limongelli, V.; Zampella, A.; Fiorucci, S.; Festa, C.
Discovering New G-Quadruplex DNA Catalysts in Enantioselective Sulfoxidation Reaction
2022 Festa, Carmen; Esposito, Veronica; Benigno, Daniela; DE MARINO, Simona; Zampella, Angela; Virgilio, Antonella; Galeone, Aldo
“Discovery of promising 1,2,4-oxadiazoles hits for the development of new anti-inflammatory agents interfering with eicosanoid biosynthesis pathways”
2021 Sciarretta, M; Potenza, M; Festa, C; Maione, F; Saviano, A; Chini, Mg; De Marino, S; D’Auria, Mv; Werz, O; Bifulco, G
Design and synthesis of new potential inhibitors of proteins relevant to cancer insurgence.
2020 Sciarretta, M.; Potenza, M.; Festa, C.; Chini, M. G.; De Marino, S.; D’Auria, M. V.; Werz, O.; Bifulco, G.
Synergistic activity of a synthetic 1,2,4-oxadiazole-containing derivative and oxacillin against methicillin-resistant Staphylococcus aureus
2021 Buommino, Elisabetta; Sciarretta, Martina; Festa, Carmen; DE ROSA, Adriana; Piccolo, Marialuisa; DE MARINO, Simona; Maria, ; D’Auria., V.
Biological Profile of Two Gentiana lutea L. Metabolites Using Computational Approaches and In Vitro Tests
2021 Finamore, Claudia; Festa, Carmen; DE MARINO, Simona; Russo, Roberto; Avagliano, Carmen; Calignano, Antonio
Marine natural products as modulators of nuclear receptors
2012 D'Auria, MARIA VALERIA; DE MARINO, Simona; Sepe, Valentina; Zampella, Angela; Bifulco, G.; Renga, B.; D'Amore, C.; Fiorucci, S.; Debitus, C. .
Wound healing activity and phytochemical screening of purified fractions of Sempervivum tectorum L. leaves on HCT 116
2019 Cattaneo, Fabio; DE MARINO, Simona; Parisi, Melania; Festa, Carmen; Castaldo, Martina; Finamore, Claudia; Duraturo, Francesca; Zollo, Cristiana; Ammendola, Rosario; Zollo, Franco; Iorizzi, Maria
Isolation of Plakinamine I: a new steroidal alkaloid from the marine sponge Corticium sp. and synthesis of an analogue model compound
2005 Zampella, Angela; R., D'Orsi; Sepe, Valentina; DE MARINO, Simona; Borbone, Nicola; A., Valentin; C., Debitus; Zollo, Franco; D'Auria, MARIA VALERIA
Targeting bile acid receptors: discovery of a potent and selective Farnesoid X receptor agonist as a new lead in the pharmacological approach to liver diseases
2017 Festa, Carmen; DE MARINO, Simona; Carino, A.; Sepe, Valentina; Marchianò, S.; Cipriani, S.; Di Leva, Francesco Saverio; Limongelli, Vittorio; Monti, M. C.; Capolupo, A.; Distrutti, E.; Fiorucci, S.; Zampella, Angela
Investigation around the Oxadiazole Core in the Discovery of a New Chemotype of Potent and Selective FXR Antagonists
2019 Festa, Carmen; Finamore, Claudia; Silvia Marchiano, †; Di Leva, Francesco Saverio; Carino, Adriana; Chiara Monti, Maria; del Gaudio, Federica; Ceccacci, Sara; Limongelli, Vittorio; Zampella, Angela; Fiorucci, Stefano; DE MARINO, Simona
Exploitation of Cholane Scaffold for the Discovery of Potent and Selective Farnesoid X Receptor (FXR) and G-Protein Coupled Bile Acid Receptor 1 (GP-BAR1) Ligands
2014 Festa, Carmen; B., Renga; C., D’Amore; Sepe, Valentina; Finamore, Claudia; DE MARINO, Simona; A., Carino; M. C., Monti; Zampella, Angela; S., Fiorucci
Binding mechanism of the farnesoid X receptor marine antagonist suvanine reveals a strategy to forestall drug modulation on nuclear receptors. Design, synthesis, and biological evaluation of novel ligands
2013 Di Leva, Francesco Saverio; Festa, Carmen; C., D'Amore; DE MARINO, Simona; B., Renga; D'Auria, MARIA VALERIA; Novellino, Ettore; Limongelli, Vittorio; Zampella, Angela; S., Fiorucci
Discovery of ((1,2,4-oxadiazol-5-yl)pyrrolidin-3-yl)ureidyl derivatives as selective non-steroidal agonists of the G-protein coupled bile acid receptor-1
2019 Di Leva, Francesco Saverio; Festa, Carmen; Carino, Adriana; De Marino, Simona; Marchianò, Silvia; Di Marino, Daniele; Finamore, Claudia; Monti, Maria Chiara; Zampella, Angela; Fiorucci, Stefano; Limongelli, Vittorio
Marine and semi-synthetic hydroxysteroids as new scaffolds for pregnane x receptor modulation.
2014 Sepe, Valentina; Di Leva, Francesco Saverio; C., D’Amore; Festa, Carmen; DE MARINO, Simona; B., Renga; D'Auria, MARIA VALERIA; Novellino, Ettore; Limongelli, Vittorio; L., D’Souza; Zampella, Angela; S., Fiorucci
Antioxidant activity and chemical components as potential anticancer agents in the Olive leaf (Olea europaea L. cv. Leccino) decoction
2014 DE MARINO, Simona; Festa, Carmen; Zollo, Franco; A., Nini; L., Antenucci; G., Raimo; M., Iorizzi
Titolo | Tipologia | Data di pubblicazione | Autore(i) | File |
---|---|---|---|---|
Phytochemical Analysis of the Methanolic Extract and Essential Oil from Leaves of Industrial Hemp Futura 75 Cultivar: Isolation of a New Cannabinoid Derivative and Biological Profile Using Computational Approaches | 1.1 Articolo in rivista | 2022 | De Vita, Simona; Finamore, Claudia; Chini, Maria Giovanna; Saviano, Gabriella; De Felice, Vincenzo; De Marino, Simona; Lauro, Gianluigi; Casapullo, Agostino; Fantasma, Francesca; Trombetta, Federico; Bifulco, Giuseppe; Iorizzi, Maria | |
Structure-based screening for the discovery of 1,2,4-oxadiazoles as promising hits for the development of new anti-inflammatory agents interfering with eicosanoid biosyn-thesis pathways | 1.1 Articolo in rivista | 2021 | Sciarretta, Martina; Saviano, Anella; Maione, Francesco; D'Auria, MARIA VALERIA; DE MARINO, Simona; Giordano, Assunta; Festa, Carmen | |
Synergism of a novel 1,2,4-oxadiazole-containing derivative with oxacillin against methicillin-resistant Staphylococcus aureus | 1.1 Articolo in rivista | 2021 | Buommino, Elisabetta; DE MARINO, Simona; Sciarretta, Martina; Piccolo, Marialuisa; Festa, Carmen; D'Auria, MARIA VALERIA | |
Synthesis of new isoxazole derivatives as fxr agonists with improved pharmacokinetic properties | 4.2 Abstract in Atti di convegno | 2019 | Finamore, C.; Sepe, V.; Baronissi, G.; Cassiano, C.; Monti, M. C.; De Marino, S.; Novellino, E.; Limongelli, V.; Fiorucci, S.; Zampella, A. | |
Design and synthesis of hyodeoxycholic acid derivatives as GPBAR1 receptor modulators useful in the treatment of colon inflammation | 4.2 Abstract in Atti di convegno | 2020 | Finamore, C.; De Marino, S.; Cassiano, C.; Di Leva, F. S.; Limongelli, V.; Zampella, A.; Fiorucci, S.; Festa, C. | |
Discovering New G-Quadruplex DNA Catalysts in Enantioselective Sulfoxidation Reaction | 1.1 Articolo in rivista | 2022 | Festa, Carmen; Esposito, Veronica; Benigno, Daniela; DE MARINO, Simona; Zampella, Angela; Virgilio, Antonella; Galeone, Aldo | |
“Discovery of promising 1,2,4-oxadiazoles hits for the development of new anti-inflammatory agents interfering with eicosanoid biosynthesis pathways” | 4.2 Abstract in Atti di convegno | 2021 | Sciarretta, M; Potenza, M; Festa, C; Maione, F; Saviano, A; Chini, Mg; De Marino, S; D’Auria, Mv; Werz, O; Bifulco, G | |
Design and synthesis of new potential inhibitors of proteins relevant to cancer insurgence. | 4.2 Abstract in Atti di convegno | 2020 | Sciarretta, M.; Potenza, M.; Festa, C.; Chini, M. G.; De Marino, S.; D’Auria, M. V.; Werz, O.; Bifulco, G. | |
Synergistic activity of a synthetic 1,2,4-oxadiazole-containing derivative and oxacillin against methicillin-resistant Staphylococcus aureus | 4.2 Abstract in Atti di convegno | 2021 | Buommino, Elisabetta; Sciarretta, Martina; Festa, Carmen; DE ROSA, Adriana; Piccolo, Marialuisa; DE MARINO, Simona; Maria, ; D’Auria., V. | |
Biological Profile of Two Gentiana lutea L. Metabolites Using Computational Approaches and In Vitro Tests | 1.1 Articolo in rivista | 2021 | Finamore, Claudia; Festa, Carmen; DE MARINO, Simona; Russo, Roberto; Avagliano, Carmen; Calignano, Antonio | |
Marine natural products as modulators of nuclear receptors | 1.5 Abstract in rivista | 2012 | D'Auria, MARIA VALERIA; DE MARINO, Simona; Sepe, Valentina; Zampella, Angela; Bifulco, G.; Renga, B.; D'Amore, C.; Fiorucci, S.; Debitus, C. . | |
Wound healing activity and phytochemical screening of purified fractions of Sempervivum tectorum L. leaves on HCT 116 | 1.1 Articolo in rivista | 2019 | Cattaneo, Fabio; DE MARINO, Simona; Parisi, Melania; Festa, Carmen; Castaldo, Martina; Finamore, Claudia; Duraturo, Francesca; Zollo, Cristiana; Ammendola, Rosario; Zollo, Franco; Iorizzi, Maria | |
Isolation of Plakinamine I: a new steroidal alkaloid from the marine sponge Corticium sp. and synthesis of an analogue model compound | 1.1 Articolo in rivista | 2005 | Zampella, Angela; R., D'Orsi; Sepe, Valentina; DE MARINO, Simona; Borbone, Nicola; A., Valentin; C., Debitus; Zollo, Franco; D'Auria, MARIA VALERIA | |
Targeting bile acid receptors: discovery of a potent and selective Farnesoid X receptor agonist as a new lead in the pharmacological approach to liver diseases | 1.1 Articolo in rivista | 2017 | Festa, Carmen; DE MARINO, Simona; Carino, A.; Sepe, Valentina; Marchianò, S.; Cipriani, S.; Di Leva, Francesco Saverio; Limongelli, Vittorio; Monti, M. C.; Capolupo, A.; Distrutti, E.; Fiorucci, S.; Zampella, Angela | |
Investigation around the Oxadiazole Core in the Discovery of a New Chemotype of Potent and Selective FXR Antagonists | 1.1 Articolo in rivista | 2019 | Festa, Carmen; Finamore, Claudia; Silvia Marchiano, †; Di Leva, Francesco Saverio; Carino, Adriana; Chiara Monti, Maria; del Gaudio, Federica; Ceccacci, Sara; Limongelli, Vittorio; Zampella, Angela; Fiorucci, Stefano; DE MARINO, Simona | |
Exploitation of Cholane Scaffold for the Discovery of Potent and Selective Farnesoid X Receptor (FXR) and G-Protein Coupled Bile Acid Receptor 1 (GP-BAR1) Ligands | 1.1 Articolo in rivista | 2014 | Festa, Carmen; B., Renga; C., D’Amore; Sepe, Valentina; Finamore, Claudia; DE MARINO, Simona; A., Carino; M. C., Monti; Zampella, Angela; S., Fiorucci | |
Binding mechanism of the farnesoid X receptor marine antagonist suvanine reveals a strategy to forestall drug modulation on nuclear receptors. Design, synthesis, and biological evaluation of novel ligands | 1.1 Articolo in rivista | 2013 | Di Leva, Francesco Saverio; Festa, Carmen; C., D'Amore; DE MARINO, Simona; B., Renga; D'Auria, MARIA VALERIA; Novellino, Ettore; Limongelli, Vittorio; Zampella, Angela; S., Fiorucci | |
Discovery of ((1,2,4-oxadiazol-5-yl)pyrrolidin-3-yl)ureidyl derivatives as selective non-steroidal agonists of the G-protein coupled bile acid receptor-1 | 1.1 Articolo in rivista | 2019 | Di Leva, Francesco Saverio; Festa, Carmen; Carino, Adriana; De Marino, Simona; Marchianò, Silvia; Di Marino, Daniele; Finamore, Claudia; Monti, Maria Chiara; Zampella, Angela; Fiorucci, Stefano; Limongelli, Vittorio | |
Marine and semi-synthetic hydroxysteroids as new scaffolds for pregnane x receptor modulation. | 1.1 Articolo in rivista | 2014 | Sepe, Valentina; Di Leva, Francesco Saverio; C., D’Amore; Festa, Carmen; DE MARINO, Simona; B., Renga; D'Auria, MARIA VALERIA; Novellino, Ettore; Limongelli, Vittorio; L., D’Souza; Zampella, Angela; S., Fiorucci | |
Antioxidant activity and chemical components as potential anticancer agents in the Olive leaf (Olea europaea L. cv. Leccino) decoction | 1.1 Articolo in rivista | 2014 | DE MARINO, Simona; Festa, Carmen; Zollo, Franco; A., Nini; L., Antenucci; G., Raimo; M., Iorizzi |