Sfoglia per Autore
Preparation of arylaminocarbonyl pyrrolo-fused tricyclic sulfonamides as inhibitors of hepatitis B virus
2019 De Francesco, Raffaele; Donnici, Lorena; Guidotti, Luca; Iannacone, Matteo; Di Fabio, Romano; Summa, Vincenzo; Prandi, Adolfo; Randazzo, Pietro; Gornati, Davide; Grillo, Alessandro; Ferrante, Luca; Bencheva, Leda Ivanova; De Matteo, Marilenia; Ferrara, Marco
Synthesis and biological evaluation of RGD–cryptophycin conjugates for targeted drug delivery
2019 Borbely, A.; Figueras, E.; Martins, A.; Esposito, S.; Auciello, G.; Monteagudo, E.; Di Marco, A.; Summa, V.; Cordella, P.; Perego, R.; Kemker, I.; Frese, M.; Gallinari, P.; Steinkuhler, C.; Sewald, N.
6-Bromoindirubin-3′-oxime intercepts GSK3 signaling to promote and enhance skeletal muscle differentiation affecting miR-206 expression in mice
2019 Ragozzino, E.; Brancaccio, M.; Di Costanzo, A.; Scalabri, F.; Andolfi, G.; Wanderlingh, L. G.; Patriarca, E. J.; Minchiotti, G.; Altamura, S.; Varrone, F.; Summa, V.
Application of an in Vitro Blood-Brain Barrier Model in the Selection of Experimental Drug Candidates for the Treatment of Huntington's Disease
2019 Di Marco, A.; Gonzalez Paz, O.; Fini, I.; Vignone, D.; Cellucci, A.; Battista, M. R.; Auciello, G.; Orsatti, L.; Zini, M.; Monteagudo, E.; Khetarpal, V.; Rose, M.; Dominguez, C.; Herbst, T.; Toledo-Sherman, L.; Summa, V.; Munoz-Sanjuan, I.
Synthesis and Evaluation of Bifunctional Aminothiazoles as Antiretrovirals Targeting the HIV-1 Nucleocapsid Protein
2019 Mori, M.; Dasso Lang, M. C.; Saladini, F.; Palombi, N.; Kovalenko, L.; De Forni, D.; Poddesu, B.; Friggeri, L.; Giannini, A.; Malancona, S.; Summa, V.; Zazzi, M.; Mely, Y.; Botta, M.
Design, Synthesis, and Biological Evaluation of New 1-(Aryl-1 H-pyrrolyl)(phenyl)methyl-1 H-imidazole Derivatives as Antiprotozoal Agents
2019 Saccoliti, F.; Madia, V. N.; Tudino, V.; De Leo, A.; Pescatori, L.; Messore, A.; De Vita, D.; Scipione, L.; Brun, R.; Kaiser, M.; Maser, P.; Calvet, C. M.; Jennings, G. K.; Podust, L. M.; Pepe, G.; Cirilli, R.; Faggi, C.; Di Marco, A.; Battista, M. R.; Summa, V.; Costi, R.; Di Santo, R.
Improved Selective Class i HDAC and Novel Selective HDAC3 Inhibitors: Beyond Hydroxamic Acids and Benzamides
2019 Bresciani, A.; Ontoria, J. M.; Biancofiore, I.; Cellucci, A.; Ciammaichella, A.; Di Marco, A.; Ferrigno, F.; Francone, A.; Malancona, S.; Monteagudo, E.; Nizi, E.; Pace, P.; Ponzi, S.; Rossetti, I.; Veneziano, M.; Summa, V.; Harper, S.
Preparation of arylaminocarbonyl bicyclic sulfonamides as inhibitors of hepatitis B virus
2019 De Francesco, Raffaele; Prandi, Adolfo; Randazzo, Pietro; Donnici, Lorena; Guidotti, Luca; Iannacone, Matteo; Di Fabio, Romano; Summa, Vincenzo; Bencheva, Leda Ivanova; De Matteo, Marilenia; Ferrante, Luca
A novel method using nuclear magnetic resonance for plasma protein binding assessment in drug discovery programs
2019 Gallo, M.; Matteucci, S.; Alaimo, N.; Pitti, E.; Orsale, M. V.; Summa, V.; Cicero, D. O.; Monteagudo, E.
Preparation of arylaminocarbonyl bicyclic sulfonamides as inhibitors of hepatitis B virus
2019 De Francesco, Raffaele; Donnici, Lorena; Guidotti, Luca; Iannacone, Matteo; Di Fabio, Romano; Summa, Vincenzo; Bencheva, Leda Ivanova; De Matteo, Marilenia; Ferrante, Luca; Prandi, Adolfo; Randazzo, Pietro
Salivary metabolome and soccer match: Challenges for understanding exercise induced changes
2019 Pitti, E.; Petrella, G.; Di Marino, S.; Summa, V.; Perrone, M.; D'Ottavio, S.; Bernardini, A.; Cicero, D. O.
Structure-Based Identification of HIV-1 Nucleocapsid Protein Inhibitors Active against Wild-Type and Drug-Resistant HIV-1 Strains
2018 Mori, ; Kovalenko, ; Malancona, ; Saladini, ; De, Forni; Pires, ; Humbert, ; Real, ; Botzanowski, ; Cianferani, ; Giannini, ; Dasso, Lang; M., C.; Cugia, ; Poddesu, ; Lori, ; Zazzi, ; Harper, ; Steven, ; Summa, V; Mely, ; Y, ; Botta,
Early metabolic response to acute myocardial ischaemia in patients undergoing elective coronary angioplasty
2018 Di Marino, S; Viceconte, N; Lembo, A; Summa, V; Tanzilli, G; Raparelli, V; Truscelli, G; Mangieri, E; Gaudio, C; Cicero, D O
Discovery of 2-(1H-imidazo-2-yl)piperazines as a new class of potent and non-cytotoxic inhibitors of Trypanosoma brucei growth in vitro
2018 Ferrigno, F.; Biancofiore, I.; Malancona, S.; Ponzi, S.; Paonessa, G.; Graziani, R.; Bresciani, A.; Gennari, N.; Di Marco, A.; Kaiser, M.; Summa, V.; Harper, S.; Ontoria, J. M.
Largazole analogues as histone deacetylases inhibitors and anticancer agents: an overview on structure‐activity relationships
2017 G, Poli; R Di, Fabio; L, Ferrante; Summa, V; M, Botta
Heterocyclic compounds used in the treatment of kinetoplastid infection and their preparation
2017 Biancofiore, Ilaria; Ciammaichella, Alina; Ferrigno, Federica; Harper, Steven; Malancona, Savina; Ontoria Ontoria, Jesus Maria; Paonessa, Giacomo; Ponzi, Simona; Summa, Vincenzo
Preparation of dihydroxypyridinylpyrimidinecarboxamide derivatives for use as HIV-1 nucleocapsid inhibitors
2016 Botta, ; M, ; Mori, ; M, ; Saladini, ; F, ; Zazzi, ; M, ; Fezzardi, ; P, ; Harper, ; S, ; Malancona, ; S, ; Santoriello, ; M, ; Summa, V; De, Forni; D, ; Kovalenko, ; L, ; Mely, ; Y, ; Pires, ; M, ; Real, ; E, ; Lyonnais, ; S, ; Mirambeau, ; G,
A small sided game session affects salivary metabolite levels in young soccer players
2016 Cicero, ; D., O.; Di, Marino; Dinallo, ; Pieri, ; Summa, V; Desideri, ; Bernardini, ; Perondi, ; D'Ottavio,
Discovery of a selective series of inhibitors of Plasmodium falciparum HDACs
2016 Ontoriajm, ; G Paonessa, G; Ponzi, S; Ferrigno, F; Nizi, E; Biancofiore, I; Malancona, S; Graziani, R; Roberts, D; Willis, P; Bresciani, A; Nadia Gennari, N; Cecchetti, O; Monteagudo, E; Orsale, Mv; Veneziano, M; Di Marco, A; Cellucci, A; Laufer, R; Sergio Altamura, S; Summa, V; Harper, S
P2‐Quinazolinones and Bis‐Macrocycles as New Templates for Next‐Generation Hepatitis C Virus NS3/4a Protease Inhibitors: Discovery of MK‐2748 and MK‐6325
2015 Rudd, Mt; Butcher, Jw; Nguyen, Kt; Mcintyre, Cj; Romano, Jj; Gilbert, Kf; Bush, Kj; Liverton, Nj; Holloway, Mk; Harper, S; Ferrara, M; Difilippo, M; Summa, V; Swestock, J; Fritzen, J; Carroll, S; Burlein, C; Dimuzio, Jm; Gates, A; Graham, ; Qian Huang, Dj; Mcclain, S; Mchale, C; Stahlhut, Mw; Black, S; Chase, R; Soriano, A; Fandozzi, C; Taylor, A; Trainor, N; Olsen, Db; Coleman, Pj; Ludmerer, Sw; Mccauley, Ja
| Titolo | Tipologia | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|---|
| Preparation of arylaminocarbonyl pyrrolo-fused tricyclic sulfonamides as inhibitors of hepatitis B virus | 6.1 Brevetto | 2019 | De Francesco, Raffaele; Donnici, Lorena; Guidotti, Luca; Iannacone, Matteo; Di Fabio, Romano; Summa, Vincenzo; Prandi, Adolfo; Randazzo, Pietro; Gornati, Davide; Grillo, Alessandro; Ferrante, Luca; Bencheva, Leda Ivanova; De Matteo, Marilenia; Ferrara, Marco | |
| Synthesis and biological evaluation of RGD–cryptophycin conjugates for targeted drug delivery | 1.1 Articolo in rivista | 2019 | Borbely, A.; Figueras, E.; Martins, A.; Esposito, S.; Auciello, G.; Monteagudo, E.; Di Marco, A.; Summa, V.; Cordella, P.; Perego, R.; Kemker, I.; Frese, M.; Gallinari, P.; Steinkuhler, C.; Sewald, N. | |
| 6-Bromoindirubin-3′-oxime intercepts GSK3 signaling to promote and enhance skeletal muscle differentiation affecting miR-206 expression in mice | 1.1 Articolo in rivista | 2019 | Ragozzino, E.; Brancaccio, M.; Di Costanzo, A.; Scalabri, F.; Andolfi, G.; Wanderlingh, L. G.; Patriarca, E. J.; Minchiotti, G.; Altamura, S.; Varrone, F.; Summa, V. | |
| Application of an in Vitro Blood-Brain Barrier Model in the Selection of Experimental Drug Candidates for the Treatment of Huntington's Disease | 1.1 Articolo in rivista | 2019 | Di Marco, A.; Gonzalez Paz, O.; Fini, I.; Vignone, D.; Cellucci, A.; Battista, M. R.; Auciello, G.; Orsatti, L.; Zini, M.; Monteagudo, E.; Khetarpal, V.; Rose, M.; Dominguez, C.; Herbst, T.; Toledo-Sherman, L.; Summa, V.; Munoz-Sanjuan, I. | |
| Synthesis and Evaluation of Bifunctional Aminothiazoles as Antiretrovirals Targeting the HIV-1 Nucleocapsid Protein | 1.1 Articolo in rivista | 2019 | Mori, M.; Dasso Lang, M. C.; Saladini, F.; Palombi, N.; Kovalenko, L.; De Forni, D.; Poddesu, B.; Friggeri, L.; Giannini, A.; Malancona, S.; Summa, V.; Zazzi, M.; Mely, Y.; Botta, M. | |
| Design, Synthesis, and Biological Evaluation of New 1-(Aryl-1 H-pyrrolyl)(phenyl)methyl-1 H-imidazole Derivatives as Antiprotozoal Agents | 1.1 Articolo in rivista | 2019 | Saccoliti, F.; Madia, V. N.; Tudino, V.; De Leo, A.; Pescatori, L.; Messore, A.; De Vita, D.; Scipione, L.; Brun, R.; Kaiser, M.; Maser, P.; Calvet, C. M.; Jennings, G. K.; Podust, L. M.; Pepe, G.; Cirilli, R.; Faggi, C.; Di Marco, A.; Battista, M. R.; Summa, V.; Costi, R.; Di Santo, R. | |
| Improved Selective Class i HDAC and Novel Selective HDAC3 Inhibitors: Beyond Hydroxamic Acids and Benzamides | 1.1 Articolo in rivista | 2019 | Bresciani, A.; Ontoria, J. M.; Biancofiore, I.; Cellucci, A.; Ciammaichella, A.; Di Marco, A.; Ferrigno, F.; Francone, A.; Malancona, S.; Monteagudo, E.; Nizi, E.; Pace, P.; Ponzi, S.; Rossetti, I.; Veneziano, M.; Summa, V.; Harper, S. | |
| Preparation of arylaminocarbonyl bicyclic sulfonamides as inhibitors of hepatitis B virus | 6.1 Brevetto | 2019 | De Francesco, Raffaele; Prandi, Adolfo; Randazzo, Pietro; Donnici, Lorena; Guidotti, Luca; Iannacone, Matteo; Di Fabio, Romano; Summa, Vincenzo; Bencheva, Leda Ivanova; De Matteo, Marilenia; Ferrante, Luca | |
| A novel method using nuclear magnetic resonance for plasma protein binding assessment in drug discovery programs | 1.1 Articolo in rivista | 2019 | Gallo, M.; Matteucci, S.; Alaimo, N.; Pitti, E.; Orsale, M. V.; Summa, V.; Cicero, D. O.; Monteagudo, E. | |
| Preparation of arylaminocarbonyl bicyclic sulfonamides as inhibitors of hepatitis B virus | 6.1 Brevetto | 2019 | De Francesco, Raffaele; Donnici, Lorena; Guidotti, Luca; Iannacone, Matteo; Di Fabio, Romano; Summa, Vincenzo; Bencheva, Leda Ivanova; De Matteo, Marilenia; Ferrante, Luca; Prandi, Adolfo; Randazzo, Pietro | |
| Salivary metabolome and soccer match: Challenges for understanding exercise induced changes | 1.1 Articolo in rivista | 2019 | Pitti, E.; Petrella, G.; Di Marino, S.; Summa, V.; Perrone, M.; D'Ottavio, S.; Bernardini, A.; Cicero, D. O. | |
| Structure-Based Identification of HIV-1 Nucleocapsid Protein Inhibitors Active against Wild-Type and Drug-Resistant HIV-1 Strains | 1.1 Articolo in rivista | 2018 | Mori, ; Kovalenko, ; Malancona, ; Saladini, ; De, Forni; Pires, ; Humbert, ; Real, ; Botzanowski, ; Cianferani, ; Giannini, ; Dasso, Lang; M., C.; Cugia, ; Poddesu, ; Lori, ; Zazzi, ; Harper, ; Steven, ; Summa, V; Mely, ; Y, ; Botta, | |
| Early metabolic response to acute myocardial ischaemia in patients undergoing elective coronary angioplasty | 1.1 Articolo in rivista | 2018 | Di Marino, S; Viceconte, N; Lembo, A; Summa, V; Tanzilli, G; Raparelli, V; Truscelli, G; Mangieri, E; Gaudio, C; Cicero, D O | |
| Discovery of 2-(1H-imidazo-2-yl)piperazines as a new class of potent and non-cytotoxic inhibitors of Trypanosoma brucei growth in vitro | 1.1 Articolo in rivista | 2018 | Ferrigno, F.; Biancofiore, I.; Malancona, S.; Ponzi, S.; Paonessa, G.; Graziani, R.; Bresciani, A.; Gennari, N.; Di Marco, A.; Kaiser, M.; Summa, V.; Harper, S.; Ontoria, J. M. | |
| Largazole analogues as histone deacetylases inhibitors and anticancer agents: an overview on structure‐activity relationships | 1.1 Articolo in rivista | 2017 | G, Poli; R Di, Fabio; L, Ferrante; Summa, V; M, Botta | |
| Heterocyclic compounds used in the treatment of kinetoplastid infection and their preparation | 6.1 Brevetto | 2017 | Biancofiore, Ilaria; Ciammaichella, Alina; Ferrigno, Federica; Harper, Steven; Malancona, Savina; Ontoria Ontoria, Jesus Maria; Paonessa, Giacomo; Ponzi, Simona; Summa, Vincenzo | |
| Preparation of dihydroxypyridinylpyrimidinecarboxamide derivatives for use as HIV-1 nucleocapsid inhibitors | 6.1 Brevetto | 2016 | Botta, ; M, ; Mori, ; M, ; Saladini, ; F, ; Zazzi, ; M, ; Fezzardi, ; P, ; Harper, ; S, ; Malancona, ; S, ; Santoriello, ; M, ; Summa, V; De, Forni; D, ; Kovalenko, ; L, ; Mely, ; Y, ; Pires, ; M, ; Real, ; E, ; Lyonnais, ; S, ; Mirambeau, ; G, | |
| A small sided game session affects salivary metabolite levels in young soccer players | 1.1 Articolo in rivista | 2016 | Cicero, ; D., O.; Di, Marino; Dinallo, ; Pieri, ; Summa, V; Desideri, ; Bernardini, ; Perondi, ; D'Ottavio, | |
| Discovery of a selective series of inhibitors of Plasmodium falciparum HDACs | 1.1 Articolo in rivista | 2016 | Ontoriajm, ; G Paonessa, G; Ponzi, S; Ferrigno, F; Nizi, E; Biancofiore, I; Malancona, S; Graziani, R; Roberts, D; Willis, P; Bresciani, A; Nadia Gennari, N; Cecchetti, O; Monteagudo, E; Orsale, Mv; Veneziano, M; Di Marco, A; Cellucci, A; Laufer, R; Sergio Altamura, S; Summa, V; Harper, S | |
| P2‐Quinazolinones and Bis‐Macrocycles as New Templates for Next‐Generation Hepatitis C Virus NS3/4a Protease Inhibitors: Discovery of MK‐2748 and MK‐6325 | 1.1 Articolo in rivista | 2015 | Rudd, Mt; Butcher, Jw; Nguyen, Kt; Mcintyre, Cj; Romano, Jj; Gilbert, Kf; Bush, Kj; Liverton, Nj; Holloway, Mk; Harper, S; Ferrara, M; Difilippo, M; Summa, V; Swestock, J; Fritzen, J; Carroll, S; Burlein, C; Dimuzio, Jm; Gates, A; Graham, ; Qian Huang, Dj; Mcclain, S; Mchale, C; Stahlhut, Mw; Black, S; Chase, R; Soriano, A; Fandozzi, C; Taylor, A; Trainor, N; Olsen, Db; Coleman, Pj; Ludmerer, Sw; Mccauley, Ja |
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