CANNALIRE, ROLANDO
CANNALIRE, ROLANDO
Dipartimento di Farmacia
Isocyanide chemistry enabled by continuous flow technology
2022 Cerra, B.; Blondeau, C.; Cannalire, R.; Giustiniano, M.; Tali Shandiz, S.; Gioiello, A.
Photomicellar Catalyzed Synthesis of Amides from Isocyanides: Optimization, Scope, and NMR Studies of Photocatalyst/Surfactant Interactions
2021 Cannalire, Rolando; Santoro, Federica; Russo, Camilla; Graziani, Giulia; Cesare Tron, Gian; Carotenuto, Alfonso; Brancaccio, Diego; Giustiniano, Mariateresa
Easy access to α-ketoamides as SARS-CoV-2 and MERS Mpro inhibitors via the PADAM oxidation route
2022 Pelliccia, Sveva; Cerchia, Carmen; Esposito, Francesca; Cannalire, Rolando; Corona, Angela; Costanzi, Elisa; Kuzikov, Maria; Gribbon, Philip; Zaliani, Andrea; Brindisi, Margherita; Storici, Paola; Tramontano, Enzo; Summa, Vincenzo
Discovery of potent p38α MAPK inhibitors through a funnel like workflow combining in silico screening and in vitro validation
2019 Astolfi, Andrea; Kudolo, Mark; Brea, Jose; Manni, Giorgia; Manfroni, Giuseppe; Palazzotti, Deborah; Sabatini, Stefano; Cecchetti, Federica; Felicetti, Tommaso; Cannalire, Rolando; Massari, Serena; Tabarrini, Oriana; Loza, Maria Isabel; Fallarino, Francesca; Cecchetti, Violetta; Laufer, Stefan A; Barreca, Maria Letizia
Ethidium bromide exposure unmasks an antibiotic efflux system in Rhodococcus equi
2021 Rampacci, Elisa; Marenzoni, Maria Luisa; Cannalire, Rolando; Pietrella, Donatella; Sabatini, Stefano; Giovagnoli, Stefano; Felicetti, Tommaso; Pepe, Marco; Passamonti, Fabrizio
From Quinoline to Quinazoline-Based S. aureus NorA Efflux Pump Inhibitors by Coupling a Focused Scaffold Hopping Approach and a Pharmacophore Search
2021 Cedraro, Nicholas; Cannalire, Rolando; Astolfi, Andrea; Mangiaterra, Gianmarco; Felicetti, Tommaso; Vaiasicca, Salvatore; Cernicchi, Giada; Massari, Serena; Manfroni, Giuseppe; Tabarrini, Oriana; Cecchetti, Violetta; Barreca, Maria Letizia; Biavasco, Francesca; Sabatini, Stefano
Visible-Light Photocatalytic Ugi/Aza-Wittig Cascade towards 2-Aminomethyl-1,3,4-oxadiazole Derivatives
2021 Russo, C.; Cannalire, R.; Luciano, P.; Brunelli, F.; Tron, G. C.; Giustiniano, M.
Domino synthesis of 5-aminoimidazoles from Strecker multicomponent adducts via ytterbium-promoted isocyanide insertion/5-exo-dig cyclization
2022 Cannalire, Rolando; Russo, Camilla; Luciano, Paolo; Cerra, Bruno; Gioiello, Antimo; Brunelli, Francesca; Tron, Gian Cesare; Giustiniano, Mariateresa
An overview on small molecules acting as broad-spectrum agents for yellow fever infection
2022 Desantis, Jenny; Felicetti, Tommaso; Cannalire, Rolando
Visible-light photocatalytic metal-free multicomponent Ugi-like chemistry
2022 Russo, Camilla; Graziani, Giulia; Cannalire, Rolando; Cesare Tron, Gian; Giustiniano, Mariateresa
Natural Compounds Inhibit SARS-CoV-2 nsp13 Unwinding and ATPase Enzyme Activities
2022 Corona, Angela; Wycisk, Krzysztof; Talarico, Carmine; Manelfi, Candida; Milia, Jessica; Cannalire, Rolando; Esposito, Francesca; Gribbon, Philip; Zaliani, Andrea; Iaconis, Daniela; Beccari, Andrea R.; Summa, Vincenzo; Nowotny, Marcin; Tramontano, Enzo
A Focus on Severe Acute Respiratory Syndrome ( SARS ) Coronavirus ( SARS‐CoVs ) 1 and 2
2022 Cannalire, Rolando; Tramontano, Enzo; Summa, Vincenzo
Identification of Inhibitors of SARS-CoV-2 3CL-Pro Enzymatic Activity Using a Small Molecule in Vitro Repurposing Screen
2021 Kuzikov, M.; Costanzi, E.; Reinshagen, J.; Esposito, F.; Vangeel, L.; Wolf, M.; Ellinger, B.; Claussen, C.; Geisslinger, G.; Corona, A.; Iaconis, D.; Talarico, C.; Manelfi, C.; Cannalire, R.; Rossetti, G.; Gossen, J.; Albani, S.; Musiani, F.; Herzog, K.; Ye, Y.; Giabbai, B.; Demitri, N.; Jochmans, D.; Jonghe, S. D.; Rymenants, J.; Summa, V.; Tramontano, E.; Beccari, A. R.; Leyssen, P.; Storici, P.; Neyts, J.; Gribbon, P.; Zaliani, A.
Visible light photocatalysis in the late-stage functionalization of pharmaceutically relevant compounds
2021 Cannalire, R.; Pelliccia, S.; Sancineto, L.; Novellino, E.; Tron, G. C.; Giustiniano, M.
Functionalized 2,1-benzothiazine 2,2-dioxides as new inhibitors of Dengue NS5 RNA-dependent RNA polymerase
2018 Cannalire, Rolando; Delia, Tarantino; Andrea, Astolfi; Maria Letizia Barreca, ; Stefano, Sabatini; Serena, Massari; Oriana, Tabarrini; Mario, Milani; Gilles, Querat; Eloise, Mastrangelo; Giuseppe, Manfroni; Cecchetti, Violetta
A Journey around the Medicinal Chemistry of Hepatitis C Virus Inhibitors Targeting NS4B: From Target to Preclinical Drug Candidates
2016 Cannalire, Rolando; Barreca Maria, Letizia; Manfroni, Giuseppe; Cecchetti, Violetta
2-Phenylquinoline S. aureus NorA Efflux Pump Inhibitors: Evaluation of the Importance of Methoxy Group Introduction
2018 Felicetti, Tommaso; Cannalire, Rolando; Pietrella, Donatella; Latacz, Gniewomir; Lubelska, Annamaria; Manfroni, Giuseppe; Letizia Barreca, Maria; Massari, Serena; Tabarrini, Oriana; Kieć-Kononowicz, Katarzyna; Schindler, Bryan D.; Kaatz, Glenn W.; Cecchetti, Violetta; Sabatini, Stefano
Targeting flavivirus RNA dependent RNA polymerase through a pyridobenzothiazole inhibitor
2016 Tarantino, Delia; Cannalire, Rolando; Mastrangelo, Eloise; Croci, Romina; Querat, Gilles; Barreca Maria, Letizia; Bolognesi, Martino; Manfroni, Giuseppe; Cecchetti, Violetta; Milani, Mario
Targeting SARS-CoV-2 Proteases and Polymerase for COVID-19 Treatment: State of the Art and Future Opportunities
2020 Cannalire, Rolando; Cerchia, Carmen; Beccari, Andrea R; Di Leva, Francesco Saverio; Summa, Vincenzo
Broad-Spectrum Flavivirus Inhibitors: a Medicinal Chemistry Point of View
2020 Felicetti, Tommaso; Manfroni, Giuseppe; Cecchetti, Violetta; Cannalire, Rolando
| Titolo | Tipologia | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|---|
| Isocyanide chemistry enabled by continuous flow technology | 1.1 Articolo in rivista | 2022 | Cerra, B.; Blondeau, C.; Cannalire, R.; Giustiniano, M.; Tali Shandiz, S.; Gioiello, A. | |
| Photomicellar Catalyzed Synthesis of Amides from Isocyanides: Optimization, Scope, and NMR Studies of Photocatalyst/Surfactant Interactions | 1.1 Articolo in rivista | 2021 | Cannalire, Rolando; Santoro, Federica; Russo, Camilla; Graziani, Giulia; Cesare Tron, Gian; Carotenuto, Alfonso; Brancaccio, Diego; Giustiniano, Mariateresa | |
| Easy access to α-ketoamides as SARS-CoV-2 and MERS Mpro inhibitors via the PADAM oxidation route | 1.1 Articolo in rivista | 2022 | Pelliccia, Sveva; Cerchia, Carmen; Esposito, Francesca; Cannalire, Rolando; Corona, Angela; Costanzi, Elisa; Kuzikov, Maria; Gribbon, Philip; Zaliani, Andrea; Brindisi, Margherita; Storici, Paola; Tramontano, Enzo; Summa, Vincenzo | |
| Discovery of potent p38α MAPK inhibitors through a funnel like workflow combining in silico screening and in vitro validation | 1.1 Articolo in rivista | 2019 | Astolfi, Andrea; Kudolo, Mark; Brea, Jose; Manni, Giorgia; Manfroni, Giuseppe; Palazzotti, Deborah; Sabatini, Stefano; Cecchetti, Federica; Felicetti, Tommaso; Cannalire, Rolando; Massari, Serena; Tabarrini, Oriana; Loza, Maria Isabel; Fallarino, Francesca; Cecchetti, Violetta; Laufer, Stefan A; Barreca, Maria Letizia | |
| Ethidium bromide exposure unmasks an antibiotic efflux system in Rhodococcus equi | 1.1 Articolo in rivista | 2021 | Rampacci, Elisa; Marenzoni, Maria Luisa; Cannalire, Rolando; Pietrella, Donatella; Sabatini, Stefano; Giovagnoli, Stefano; Felicetti, Tommaso; Pepe, Marco; Passamonti, Fabrizio | |
| From Quinoline to Quinazoline-Based S. aureus NorA Efflux Pump Inhibitors by Coupling a Focused Scaffold Hopping Approach and a Pharmacophore Search | 1.1 Articolo in rivista | 2021 | Cedraro, Nicholas; Cannalire, Rolando; Astolfi, Andrea; Mangiaterra, Gianmarco; Felicetti, Tommaso; Vaiasicca, Salvatore; Cernicchi, Giada; Massari, Serena; Manfroni, Giuseppe; Tabarrini, Oriana; Cecchetti, Violetta; Barreca, Maria Letizia; Biavasco, Francesca; Sabatini, Stefano | |
| Visible-Light Photocatalytic Ugi/Aza-Wittig Cascade towards 2-Aminomethyl-1,3,4-oxadiazole Derivatives | 1.1 Articolo in rivista | 2021 | Russo, C.; Cannalire, R.; Luciano, P.; Brunelli, F.; Tron, G. C.; Giustiniano, M. | |
| Domino synthesis of 5-aminoimidazoles from Strecker multicomponent adducts via ytterbium-promoted isocyanide insertion/5-exo-dig cyclization | 1.1 Articolo in rivista | 2022 | Cannalire, Rolando; Russo, Camilla; Luciano, Paolo; Cerra, Bruno; Gioiello, Antimo; Brunelli, Francesca; Tron, Gian Cesare; Giustiniano, Mariateresa | |
| An overview on small molecules acting as broad-spectrum agents for yellow fever infection | 1.1 Articolo in rivista | 2022 | Desantis, Jenny; Felicetti, Tommaso; Cannalire, Rolando | |
| Visible-light photocatalytic metal-free multicomponent Ugi-like chemistry | 1.1 Articolo in rivista | 2022 | Russo, Camilla; Graziani, Giulia; Cannalire, Rolando; Cesare Tron, Gian; Giustiniano, Mariateresa | |
| Natural Compounds Inhibit SARS-CoV-2 nsp13 Unwinding and ATPase Enzyme Activities | 1.1 Articolo in rivista | 2022 | Corona, Angela; Wycisk, Krzysztof; Talarico, Carmine; Manelfi, Candida; Milia, Jessica; Cannalire, Rolando; Esposito, Francesca; Gribbon, Philip; Zaliani, Andrea; Iaconis, Daniela; Beccari, Andrea R.; Summa, Vincenzo; Nowotny, Marcin; Tramontano, Enzo | |
| A Focus on Severe Acute Respiratory Syndrome ( SARS ) Coronavirus ( SARS‐CoVs ) 1 and 2 | 3.1 Monografia o trattato scientifico | 2022 | Cannalire, Rolando; Tramontano, Enzo; Summa, Vincenzo | |
| Identification of Inhibitors of SARS-CoV-2 3CL-Pro Enzymatic Activity Using a Small Molecule in Vitro Repurposing Screen | 1.1 Articolo in rivista | 2021 | Kuzikov, M.; Costanzi, E.; Reinshagen, J.; Esposito, F.; Vangeel, L.; Wolf, M.; Ellinger, B.; Claussen, C.; Geisslinger, G.; Corona, A.; Iaconis, D.; Talarico, C.; Manelfi, C.; Cannalire, R.; Rossetti, G.; Gossen, J.; Albani, S.; Musiani, F.; Herzog, K.; Ye, Y.; Giabbai, B.; Demitri, N.; Jochmans, D.; Jonghe, S. D.; Rymenants, J.; Summa, V.; Tramontano, E.; Beccari, A. R.; Leyssen, P.; Storici, P.; Neyts, J.; Gribbon, P.; Zaliani, A. | |
| Visible light photocatalysis in the late-stage functionalization of pharmaceutically relevant compounds | 1.1 Articolo in rivista | 2021 | Cannalire, R.; Pelliccia, S.; Sancineto, L.; Novellino, E.; Tron, G. C.; Giustiniano, M. | |
| Functionalized 2,1-benzothiazine 2,2-dioxides as new inhibitors of Dengue NS5 RNA-dependent RNA polymerase | 1.1 Articolo in rivista | 2018 | Cannalire, Rolando; Delia, Tarantino; Andrea, Astolfi; Maria Letizia Barreca, ; Stefano, Sabatini; Serena, Massari; Oriana, Tabarrini; Mario, Milani; Gilles, Querat; Eloise, Mastrangelo; Giuseppe, Manfroni; Cecchetti, Violetta | |
| A Journey around the Medicinal Chemistry of Hepatitis C Virus Inhibitors Targeting NS4B: From Target to Preclinical Drug Candidates | 1.1 Articolo in rivista | 2016 | Cannalire, Rolando; Barreca Maria, Letizia; Manfroni, Giuseppe; Cecchetti, Violetta | |
| 2-Phenylquinoline S. aureus NorA Efflux Pump Inhibitors: Evaluation of the Importance of Methoxy Group Introduction | 1.1 Articolo in rivista | 2018 | Felicetti, Tommaso; Cannalire, Rolando; Pietrella, Donatella; Latacz, Gniewomir; Lubelska, Annamaria; Manfroni, Giuseppe; Letizia Barreca, Maria; Massari, Serena; Tabarrini, Oriana; Kieć-Kononowicz, Katarzyna; Schindler, Bryan D.; Kaatz, Glenn W.; Cecchetti, Violetta; Sabatini, Stefano | |
| Targeting flavivirus RNA dependent RNA polymerase through a pyridobenzothiazole inhibitor | 1.1 Articolo in rivista | 2016 | Tarantino, Delia; Cannalire, Rolando; Mastrangelo, Eloise; Croci, Romina; Querat, Gilles; Barreca Maria, Letizia; Bolognesi, Martino; Manfroni, Giuseppe; Cecchetti, Violetta; Milani, Mario | |
| Targeting SARS-CoV-2 Proteases and Polymerase for COVID-19 Treatment: State of the Art and Future Opportunities | 1.1 Articolo in rivista | 2020 | Cannalire, Rolando; Cerchia, Carmen; Beccari, Andrea R; Di Leva, Francesco Saverio; Summa, Vincenzo | |
| Broad-Spectrum Flavivirus Inhibitors: a Medicinal Chemistry Point of View | 1.1 Articolo in rivista | 2020 | Felicetti, Tommaso; Manfroni, Giuseppe; Cecchetti, Violetta; Cannalire, Rolando |