CANNALIRE, ROLANDO
CANNALIRE, ROLANDO
DIPARTIMENTO DI FARMACIA
New Pyrazolobenzothiazine Derivatives As Hepatitis C Virus NS5B Polymerase Palm Site I Inhibitors
2014 Manfroni, Giuseppe; Manvar, Dinesh; Barreca Maria, Letizia; Kaushik-Basu, Neerja; Leyssen, Pieter; Paeshuyse, Jan; Cannalire, Rolando; Iraci, Nunzio; Basu, Amartya; Chudaev, Maxim; Zamperini, Claudio; Dreassi, Elena; Sabatini, Stefano; Tabarrini, Oriana; Neyts, Johan; Cecchetti, Violetta
Tumour cell population growth inhibition and cell death induction of functionalized 6-aminoquinolone derivatives
2015 Franci, G; Manfroni, Giuseppe; Cannalire, Rolando; Felicetti, Tommaso; Tabarrini, Oriana; Salvato, A; Barreca, MARIA LETIZIA; Altucci, L; Cecchetti, Violetta
Structure-based insights into p38α MAPK: from crystal structures analysis to hit optimization
2015 Astolfi, Andrea; Barreca Maria, Letizia; Iraci, Nunzio; Cannalire, Rolando; Sabatini, Stefano; Manfroni, Giuseppe; Cecchetti, Violetta
Modifications on C6 and C7 Positions of 3-Phenylquinolone Efflux Pump Inhibitors Led to Potent and Safe Antimycobacterial Treatment Adjuvants
2019 Felicetti, T.; Machado, D.; Cannalire, R.; Astolfi, A.; Massari, S.; Tabarrini, O.; Manfroni, G.; Barreca, M. L.; Cecchetti, V.; Viveiros, M.; Sabatini, S.
Boosting Effect of 2-Phenylquinoline Efflux Inhibitors in Combination with Macrolides against Mycobacterium smegmatis and Mycobacterium avium
2015 Machado, Diana; Cannalire, Rolando; Santos Costa, Sofia; Manfroni, Giuseppe; Tabarrini, Oriana; Cecchetti, Violetta; Couto, Isabel; Viveiros, Miguel; Sabatini, Stefano
The Pyrazolobenzothiazine Core as a New Chemotype of p38 Alpha Mitogen-Activated Protein Kinase Inhibitors
2015 Sabatini, Stefano; Manfroni, Giuseppe; Barreca Maria, Letizia; Bauer Silke, M; Gargaro, Marco; Cannalire, Rolando; Astolfi, Andrea; Brea, Jose; Vacca, Carmine; Pirro, Matteo; Massari, Serena; Tabarrini, Oriana; Loza Maria, Isabel; Fallarino, Francesca; Laufer Stefan, A; Cecchetti, Violetta
The versatile nature of the 6-aminoquinolone scaffold: identification of submicromolar hepatitis C virus NS5B inhibitors
2014 Manfroni, Giuseppe; Cannalire, Rolando; Barreca Maria, Letizia; Kaushik-Basu, Neerja; Leyssen, Pieter; Winquist, Johan; Iraci, Nunzio; Manvar, Dinesh; Paeshuyse, Jan; Guhamazumder, Rupa; Basu, Amartya; Sabatini, Stefano; Tabarrini, Oriana; Danielson U., Helena; Neyts, Johan; Cecchetti, Violetta
Searching for Novel Inhibitors of the S. aureus NorA Efflux Pump: Synthesis and Biological Evaluation of the 3-Phenyl-1,4-benzothiazine Analogues
2017 Felicetti, Tommaso; Cannalire, Rolando; Burali, MARIA SOLE; Massari, Serena; Manfroni, Giuseppe; Barreca, MARIA LETIZIA; Tabarrini, Oriana; Schindler, Bryan D; Sabatini, Stefano; Kaatz, Glenn W; Cecchetti, Violetta
Natural isoflavone biochanin A as a template for the design of new and potent 3-phenylquinolone efflux inhibitors against Mycobacterium avium
2017 Cannalire, Rolando; Machado, Diana; Felicetti, Tommaso; Santos Costa, Sofia; Massari, Serena; Manfroni, Giuseppe; Barreca, Maria Letizia; Tabarrini, Oriana; Couto, Isabel; Viveiros, Miguel; Sabatini, Stefano; Cecchetti, Violetta
Advantageous Use of Ionic Liquids for the Synthesis of Pharmaceutically Relevant Quinolones
2018 Cannalire, Rolando; Tiecco, Matteo; Cecchetti, Violetta; Germani, Raimondo; Manfroni, Giuseppe
Studies on 2-phenylquinoline Staphylococcus aureus NorA efflux pump inhibitors: New insights on the C-6 position
2018 Felicetti, T.; Cannalire, R.; Nizi, M. G.; Tabarrini, O.; Massari, S.; Barreca, M. L.; Manfroni, G.; Schindler, B. D.; Cecchetti, V.; Kaatz, G. W.; Sabatini, S.
Broad spectrum anti-flavivirus pyridobenzothiazolones leading to less infective virions
2019 Cannalire, Rolando; Tarantino, D.; Piorkowski, G.; Carletti, T.; Massari, S.; Felicetti, T.; Barreca, M. L.; Sabatini, S.; Tabarrini, O.; Marcello, A.; Milani, M.; Cecchetti, V.; Mastrangelo, E.; Manfroni, G.; Querat, G.
Mode of action of the 2-phenylquinoline efflux inhibitor PQQ4R against Escherichia coli
2017 Machado, Diana; Fernandes, Laura; Costa, Sofia S.; Cannalire, Rolando; Manfroni, Giuseppe; Tabarrini, Oriana; Couto, Isabel; Sabatini, Stefano; Viveiros, Miguel
Visible-light photocatalytic functionalization of isocyanides for the synthesis of secondary amides and ketene aminals
2020 Cannalire, R.; Amato, J.; Summa, V.; Novellino, E.; Tron, G. C.; Giustiniano, M.
Structural Modifications of the Quinolin-4-yloxy Core to Obtain New Staphylococcus aureus NorA Inhibitors
2020 Cannalire, Rolando; Mangiaterra, Gianmarco; Felicetti, Tommaso; Astolfi, Andrea; Cedraro, Nicholas; Massari, Serena; Manfroni, Giuseppe; Tabarrini, Oriana; Vaiasicca, Salvatore; Letizia Barreca, Maria; Cecchetti, Violetta; Biavasco, Francesca; Sabatini, Stefano
SARS-CoV-2 Entry Inhibitors: Small Molecules and Peptides Targeting Virus or Host Cells
2020 Cannalire, Rolando; Stefanelli, Irina; Cerchia, Carmen; R Beccari, Andrea; Pelliccia, Sveva; Summa, Vincenzo
C-2 phenyl replacements to obtain potent quinoline-based Staphylococcus aureus NorA inhibitors
2020 Felicetti, Tommaso; Mangiaterra, Gianmarco; Cannalire, Rolando; Cedraro, Nicholas; Pietrella, Donatella; Astolfi, Andrea; Massari, Serena; Tabarrini, Oriana; Manfroni, Giuseppe; Letizia Barreca, Maria; Cecchetti, Violetta; Biavasco, Francesca; Sabatini, Stefano
Evolution of HCV NS4B Inhibitors
2019 Manfroni, Giuseppe; Cannalire, Rolando
Pyridobenzothiazolones Exert Potent Anti-Dengue Activity by Hampering Multiple Functions of NS5 Polymerase
2020 Cannalire, Rolando; Wing Ki Chan, Kitti; Sole Burali, Maria; Piaw Gwee, Chin; Wang, Sai; Astolfi, Andrea; Massari, Serena; Sabatini, Stefano; Tabarrini, Oriana; Mastrangelo, Eloise; Letizia Barreca, Maria; Cecchetti, Violetta; G Vasudevan, Subhash; Manfroni, Giuseppe
Broad-Spectrum Flavivirus Inhibitors: a Medicinal Chemistry Point of View
2020 Felicetti, Tommaso; Manfroni, Giuseppe; Cecchetti, Violetta; Cannalire, Rolando
| Titolo | Tipologia | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|---|
| New Pyrazolobenzothiazine Derivatives As Hepatitis C Virus NS5B Polymerase Palm Site I Inhibitors | 1.1 Articolo in rivista | 2014 | Manfroni, Giuseppe; Manvar, Dinesh; Barreca Maria, Letizia; Kaushik-Basu, Neerja; Leyssen, Pieter; Paeshuyse, Jan; Cannalire, Rolando; Iraci, Nunzio; Basu, Amartya; Chudaev, Maxim; Zamperini, Claudio; Dreassi, Elena; Sabatini, Stefano; Tabarrini, Oriana; Neyts, Johan; Cecchetti, Violetta | |
| Tumour cell population growth inhibition and cell death induction of functionalized 6-aminoquinolone derivatives | 1.1 Articolo in rivista | 2015 | Franci, G; Manfroni, Giuseppe; Cannalire, Rolando; Felicetti, Tommaso; Tabarrini, Oriana; Salvato, A; Barreca, MARIA LETIZIA; Altucci, L; Cecchetti, Violetta | |
| Structure-based insights into p38α MAPK: from crystal structures analysis to hit optimization | 4.3 Poster | 2015 | Astolfi, Andrea; Barreca Maria, Letizia; Iraci, Nunzio; Cannalire, Rolando; Sabatini, Stefano; Manfroni, Giuseppe; Cecchetti, Violetta | |
| Modifications on C6 and C7 Positions of 3-Phenylquinolone Efflux Pump Inhibitors Led to Potent and Safe Antimycobacterial Treatment Adjuvants | 1.1 Articolo in rivista | 2019 | Felicetti, T.; Machado, D.; Cannalire, R.; Astolfi, A.; Massari, S.; Tabarrini, O.; Manfroni, G.; Barreca, M. L.; Cecchetti, V.; Viveiros, M.; Sabatini, S. | |
| Boosting Effect of 2-Phenylquinoline Efflux Inhibitors in Combination with Macrolides against Mycobacterium smegmatis and Mycobacterium avium | 1.1 Articolo in rivista | 2015 | Machado, Diana; Cannalire, Rolando; Santos Costa, Sofia; Manfroni, Giuseppe; Tabarrini, Oriana; Cecchetti, Violetta; Couto, Isabel; Viveiros, Miguel; Sabatini, Stefano | |
| The Pyrazolobenzothiazine Core as a New Chemotype of p38 Alpha Mitogen-Activated Protein Kinase Inhibitors | 1.1 Articolo in rivista | 2015 | Sabatini, Stefano; Manfroni, Giuseppe; Barreca Maria, Letizia; Bauer Silke, M; Gargaro, Marco; Cannalire, Rolando; Astolfi, Andrea; Brea, Jose; Vacca, Carmine; Pirro, Matteo; Massari, Serena; Tabarrini, Oriana; Loza Maria, Isabel; Fallarino, Francesca; Laufer Stefan, A; Cecchetti, Violetta | |
| The versatile nature of the 6-aminoquinolone scaffold: identification of submicromolar hepatitis C virus NS5B inhibitors | 1.1 Articolo in rivista | 2014 | Manfroni, Giuseppe; Cannalire, Rolando; Barreca Maria, Letizia; Kaushik-Basu, Neerja; Leyssen, Pieter; Winquist, Johan; Iraci, Nunzio; Manvar, Dinesh; Paeshuyse, Jan; Guhamazumder, Rupa; Basu, Amartya; Sabatini, Stefano; Tabarrini, Oriana; Danielson U., Helena; Neyts, Johan; Cecchetti, Violetta | |
| Searching for Novel Inhibitors of the S. aureus NorA Efflux Pump: Synthesis and Biological Evaluation of the 3-Phenyl-1,4-benzothiazine Analogues | 1.1 Articolo in rivista | 2017 | Felicetti, Tommaso; Cannalire, Rolando; Burali, MARIA SOLE; Massari, Serena; Manfroni, Giuseppe; Barreca, MARIA LETIZIA; Tabarrini, Oriana; Schindler, Bryan D; Sabatini, Stefano; Kaatz, Glenn W; Cecchetti, Violetta | |
| Natural isoflavone biochanin A as a template for the design of new and potent 3-phenylquinolone efflux inhibitors against Mycobacterium avium | 1.1 Articolo in rivista | 2017 | Cannalire, Rolando; Machado, Diana; Felicetti, Tommaso; Santos Costa, Sofia; Massari, Serena; Manfroni, Giuseppe; Barreca, Maria Letizia; Tabarrini, Oriana; Couto, Isabel; Viveiros, Miguel; Sabatini, Stefano; Cecchetti, Violetta | |
| Advantageous Use of Ionic Liquids for the Synthesis of Pharmaceutically Relevant Quinolones | 1.1 Articolo in rivista | 2018 | Cannalire, Rolando; Tiecco, Matteo; Cecchetti, Violetta; Germani, Raimondo; Manfroni, Giuseppe | |
| Studies on 2-phenylquinoline Staphylococcus aureus NorA efflux pump inhibitors: New insights on the C-6 position | 1.1 Articolo in rivista | 2018 | Felicetti, T.; Cannalire, R.; Nizi, M. G.; Tabarrini, O.; Massari, S.; Barreca, M. L.; Manfroni, G.; Schindler, B. D.; Cecchetti, V.; Kaatz, G. W.; Sabatini, S. | |
| Broad spectrum anti-flavivirus pyridobenzothiazolones leading to less infective virions | 1.1 Articolo in rivista | 2019 | Cannalire, Rolando; Tarantino, D.; Piorkowski, G.; Carletti, T.; Massari, S.; Felicetti, T.; Barreca, M. L.; Sabatini, S.; Tabarrini, O.; Marcello, A.; Milani, M.; Cecchetti, V.; Mastrangelo, E.; Manfroni, G.; Querat, G. | |
| Mode of action of the 2-phenylquinoline efflux inhibitor PQQ4R against Escherichia coli | 1.1 Articolo in rivista | 2017 | Machado, Diana; Fernandes, Laura; Costa, Sofia S.; Cannalire, Rolando; Manfroni, Giuseppe; Tabarrini, Oriana; Couto, Isabel; Sabatini, Stefano; Viveiros, Miguel | |
| Visible-light photocatalytic functionalization of isocyanides for the synthesis of secondary amides and ketene aminals | 1.1 Articolo in rivista | 2020 | Cannalire, R.; Amato, J.; Summa, V.; Novellino, E.; Tron, G. C.; Giustiniano, M. | |
| Structural Modifications of the Quinolin-4-yloxy Core to Obtain New Staphylococcus aureus NorA Inhibitors | 1.1 Articolo in rivista | 2020 | Cannalire, Rolando; Mangiaterra, Gianmarco; Felicetti, Tommaso; Astolfi, Andrea; Cedraro, Nicholas; Massari, Serena; Manfroni, Giuseppe; Tabarrini, Oriana; Vaiasicca, Salvatore; Letizia Barreca, Maria; Cecchetti, Violetta; Biavasco, Francesca; Sabatini, Stefano | |
| SARS-CoV-2 Entry Inhibitors: Small Molecules and Peptides Targeting Virus or Host Cells | 1.1 Articolo in rivista | 2020 | Cannalire, Rolando; Stefanelli, Irina; Cerchia, Carmen; R Beccari, Andrea; Pelliccia, Sveva; Summa, Vincenzo | |
| C-2 phenyl replacements to obtain potent quinoline-based Staphylococcus aureus NorA inhibitors | 1.1 Articolo in rivista | 2020 | Felicetti, Tommaso; Mangiaterra, Gianmarco; Cannalire, Rolando; Cedraro, Nicholas; Pietrella, Donatella; Astolfi, Andrea; Massari, Serena; Tabarrini, Oriana; Manfroni, Giuseppe; Letizia Barreca, Maria; Cecchetti, Violetta; Biavasco, Francesca; Sabatini, Stefano | |
| Evolution of HCV NS4B Inhibitors | 2.1 Contributo in volume (Capitolo o Saggio) | 2019 | Manfroni, Giuseppe; Cannalire, Rolando | |
| Pyridobenzothiazolones Exert Potent Anti-Dengue Activity by Hampering Multiple Functions of NS5 Polymerase | 1.1 Articolo in rivista | 2020 | Cannalire, Rolando; Wing Ki Chan, Kitti; Sole Burali, Maria; Piaw Gwee, Chin; Wang, Sai; Astolfi, Andrea; Massari, Serena; Sabatini, Stefano; Tabarrini, Oriana; Mastrangelo, Eloise; Letizia Barreca, Maria; Cecchetti, Violetta; G Vasudevan, Subhash; Manfroni, Giuseppe | |
| Broad-Spectrum Flavivirus Inhibitors: a Medicinal Chemistry Point of View | 1.1 Articolo in rivista | 2020 | Felicetti, Tommaso; Manfroni, Giuseppe; Cecchetti, Violetta; Cannalire, Rolando |