SANTORO, MASSIMO

SANTORO, MASSIMO  

Dipartimento di Medicina molecolare e Biotecnologie mediche  

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NCOA4 links iron bioavailability to DNA metabolism 1.1 Articolo in rivista 2022 Federico, Giorgia; Carrillo, Federica; Dapporto, Francesca; Chiariello, Mario; Santoro, Massimo; Bellelli, Roberto; Carlomagno, Francesca
Discovery of pyrazolo-thieno[3,2-d]pyrimidinylamino-phenyl acetamides as type-II pan-tropomyosin receptor kinase (TRK) inhibitors: Design, synthesis, and biological evaluation 1.1 Articolo in rivista 2021 Yan, W.; Zhang, L.; Lv, F.; Moccia, M.; Carlomagno, F.; Landry, C.; Santoro, M.; Gosselet, F.; Frett, B.; Li, H. -Y.
Targeted activity of the small molecule kinase inhibitor Pz-1 towards RET and TRK kinases 1.1 Articolo in rivista 2021 Moccia, M.; Yang, D.; Lakkaniga, N. R.; Frett, B.; Mcconnell, N.; Zhang, L.; Brescia, A.; Federico, G.; Zhang, L.; Salerno, P.; Santoro, M.; Li, H. -Y.; Carlomagno, F.
Discovery of N-Trisubstituted Pyrimidine Derivatives as Type I RET and RET Gatekeeper Mutant Inhibitors with a Novel Kinase Binding Pose 1.1 Articolo in rivista 2022 Zhang, Lingtian; Moccia, Marialuisa; Briggs, David C; Bharate, Jaideep B; Lakkaniga, Naga Rajiv; Knowles, Phillip; Yan, Wei; Tran, Phuc; Kharbanda, Anupreet; Wang, Xiuqi; Leung, Yuet-Kin; Frett, Brendan; Santoro, Massimo; Mcdonald, Neil Q; Carlomagno, Francesca; Li, Hong-Yu
Chromatin and DNA methylation dynamics during retinoic acid-induced RET gene transcriptional activation in neuroblastoma cells. 1.1 Articolo in rivista 2011 Angrisano, Tiziana; Sacchetti, Silvana; Natale, Francesco; Cerrato, A.; Pero, Raffaela; Keller, Simona; Peluso, S.; Perillo, B.; Avvedimento, VITTORIO ENRICO; Fusco, Alfredo; Bruni, C.; Lembo, Francesca; Santoro, Massimo; Chiariotti, Lorenzo
The importance of the RET gene in thyroid cancer and therapeutic implications 1.1 Articolo in rivista 2021 Salvatore, D.; Santoro, M.; Schlumberger, M.
Signal Transducer and Activator of Transcription 1 Plays a Pivotal Role in RET/PTC3 Oncogene-induced Expression of Indoleamine 2,3-Dioxygenase 1 1.1 Articolo in rivista 2017 Moretti, Sonia; Menicali, Elisa; Nucci, Nicole; Voce, Pasquale; Colella, Renato; Melillo, ROSA MARINA; Liotti, Federica; Morelli, Silvia; Fallarino, Francesca; Macchiarulo, Antonio; Santoro, Massimo; Avenia, Nicola; Puxeddu, Efisio
A dual mechanism of activation of the sonic hedgehog pathway in anaplastic thyroid cancer: Crosstalk with RAS-BRAF-MEK pathway and ligand secretion by tumor stroma 1.1 Articolo in rivista 2018 Parascandolo, Alessia; Laukkanen, Mikko O.; de Rosa, Nancy; Ugolini, Clara; Cantisani, MARIA CARMELA; Cirafici, Anna Maria; Basolo, Fulvio; Santoro, Massimo; Castellone, Maria Domenica
Revised American Thyroid Association guidelines for the management of medullary thyroid carcinoma 1.1 Articolo in rivista 2015 Wells, Samuel A; Asa, Sylvia L; Dralle, Henning; Elisei, Rossella; Evans, Douglas B; Gagel, Robert F; Lee, Nancy; Machens, Andreas; Moley, Jeffrey F; Pacini, Furio; Raue, Friedhelm; Frank Raue, Karin; Robinson, Bruce; Rosenthal, M. Sara; Santoro, Massimo; Schlumberger, Martin; Shah, Manisha; Waguespack, Steven G.
Association between DNA methylation profile and malignancy in follicular-patterned thyroid neoplasms 1.1 Articolo in rivista 2019 Affinito, Ornella; Salerno, Paolo; D'Alessio, Alfonso Manuel; Cuomo, Mariella; Florio, Ermanno; Carlomagno, Francesca; Proietti, Agnese; Giannini, Riccardo; Basolo, Fulvio; Chiariotti, Lorenzo; Cocozza, Sergio; Santoro, Massimo
Protein kinase Calpha activation by RET: evidence for a negative feedback mechanism controlling RET tyrosine kinase 1.1 Articolo in rivista 2003 Andreozzi, F; Melillo, ROSA MARINA; Carlomagno, F; Oriente, Francesco; Miele, C; Fiory, Francesca; Santopietro, S; Castellone, Md; Beguinot, Francesco; Santoro, Massimo; Formisano, Pietro
NCOA4 Links Iron Bioavailability to DNA Metabolism 1.1 Articolo in rivista 2017 Federico, G; Bellelli, R; Nai, A; Silvestri, L; Camaschella, C; Iolascon, A; Santoro, M; Carlomagno, F
Cross talk between the bombesin neuropeptide receptor and Sonic hedgehog pathways in small cell lung carcinoma 1.1 Articolo in rivista 2015 Castellone, M. D; Laukkanen, M. O; Teramoto, H; Bellelli, Roberto; Alì, G; Fontanini, G; Santoro, Massimo; Gutkind, J. S.
Insights into Current Tropomyosin Receptor Kinase (TRK) Inhibitors: Development and Clinical Application 1.1 Articolo in rivista 2019 Yan, Wei; Lakkaniga, Naga Rajiv; Carlomagno, Francesca; Santoro, Massimo; Mcdonald, Neil Q.; Lv, Fengping; Gunaganti, Naresh; Frett, Brendan; Li, Hong-Yu
Bioisosteric discovery of npa101.3, a second-generation ret/vegfr2 inhibitor optimized for single-agent polypharmacology 1.1 Articolo in rivista 2020 Moccia, M.; Frett, B.; Zhang, L.; Lakkaniga, N. R.; Briggs, D. C.; Chauhan, R.; Brescia, A.; Federico, G.; Yan, W.; Santoro, M.; Mcdonald, N. Q.; Li, H. -Y.; Carlomagno, F.
Ret gene fusions in malignancies of the thyroid and other tissues 1.1 Articolo in rivista 2020 Santoro, M.; Moccia, M.; Federico, G.; Carlomagno, F.
Fragment-Based Discovery of a Dual pan-RET/VEGFR2 Kinase Inhibitor Optimized for Single-Agent Polypharmacology 1.1 Articolo in rivista 2015 Frett, Brendan; Carlomagno, Francesca; Moccia, Marialuisa; Brescia, Annalisa; Federico, Giorgia; De Falco, Valentina; Admire, Brittany; Chen, Zhongzhu; Qi, Wenqing; Santoro, Massimo; Li, Hong yu
The molecular basis for RET tyrosine-kinase inhibitors in thyroid cancer 1.1 Articolo in rivista 2017 De Falco, Valentina; Carlomagno, Francesca; Li, Hong-yu; Santoro, Massimo
Mast cells induce epithelial-to-mesenchymal transition and stem cell features in human thyroid cancer cells through an IL-8-Akt-Slug pathway. 1.1 Articolo in rivista 2015 Visciano, Carla; Liotti, Federica; Prevete, Nella; Cali', G; Franco, R; Collina, F; DE PAULIS, Amato; Marone, Gianni; Santoro, Massimo; Melillo, ROSA MARINA
Thyroid cell transformation inhibits the expression of a novel rat protein tyrosine phosphatase. 1.1 Articolo in rivista 1997 Zhang, L; Martelli, Ml; Battaglia, C; Trapasso, Serena; Tramontano, Donatella; Viglietto, G; Porcellini, Antonio; Santoro, Massimo; Fusco, Alfredo