MERLINO, FRANCESCO
MERLINO, FRANCESCO
DIPARTIMENTO DI FARMACIA
Discovery of New Potent Ligands at Human Urotensin-II Receptor
2013 Yousif, ALI MUNAIM; Merlino, Francesco; Carotenuto, Alfonso; Limatola, Antonio; Paolo, Santicioli; Campiglia, Pietro; Meini, Stefania; Maggi Carlo, A.; Novellino, Ettore; Grieco, Paolo
Cyclization of the urokinase receptor-derived Ser-Arg-Ser-Arg-Tyr peptide generates a potent inhibitor of trans-endothelial migration of monocytes
2015 Yousif, ALI MUNAIM; Minopoli, Michele; Bifulco, Katia; Ingangi, Vincenzo; Di Carluccio, Gioconda; Merlino, Francesco; Motti, MARIA LETIZIA; Grieco, Paolo; Carriero, Maria Vincenza
Activation of Melanocortin Receptors MC1 and MC5 Attenuates Retinal Damage in Experimental Diabetic Retinopathy
2016 Rossi, S; Maisto, R; Gesualdo, C; Trotta, Mc; Ferraraccio, F; Kaneva, Mk; Getting, Sj; Surace, Enrico Maria; Testa, F; Simonelli, F; Grieco, Paolo; Merlino, Francesco; Perretti, M; D'Amico, M; Di Filippo, C. 2.
Urokinase receptor derived peptides as potent inhibitors of the formyl peptide receptor type 1-triggered cell migration
2018 Yousif, Ali Munaim; Ingangi, Vincenzo; Merlino, Francesco; Brancaccio, Diego; Minopoli, Michele; Bellavita, Rosa; Novellino, Ettore; Carriero, Maria Vincenza; Carotenuto, Alfonso; Grieco, Paolo
Treatment with a Urokinase Receptor-derived Cyclized Peptide Improves Experimental Colitis by Preventing Monocyte Recruitment and Macrophage Polarization
2016 Genua, Marco; Ingangi, Vincenzo; Fonteyne, Philippe; Piontini, Andrea; Yousif, ALI MUNAIM; Merlino, Francesco; Grieco, Paolo; Malesci, Alberto; Carriero, Maria V; Danese, Silvio
Synthesis and Pharmacological Evaluation of a Novel Peptide Based on Anemonia sulcata BDS-I Toxin as a New KV3.4 Inhibitor Exerting a Neuroprotective Effect Against Amyloid-β Peptide
2019 Ciccone, Roselia; Piccialli, Ilaria; Grieco, Paolo; Merlino, Francesco; Annunziato, Lucio; Pannaccione, Anna
HOST DEFENSE TEMPORIN 1 PEPTIDES AND THEIR POTENTIAL AS ANTIVIRAL AGENTS
2017 Palomba, Luciana; Merlino, Francesco; Zannella, Carla; Franci, Gianluigi; Galdiero, Stefania; Grieco, Paolo; Galdiero, Massimiliano
Urotensin II receptor expression in patients with ulcerative colitis: a pilot study
2020 Gravina, Antonietta G; Dallio, Marcello; Tuccillo, Concetta; Martorano, Marco; Abenavoli, Ludovico; Luzza, Francesco; Stiuso, Paola; Lama, Stefania; Grieco, Paolo; Merlino, Francesco; Caraglia, Michele; Loguercio, Carmelina; Federico, Alessandro
Breast tumor cell invasion and pro-invasive activity of cancer-associated fibroblasts co-targeted by novel urokinase-derived decapeptides
2020 Belli, S.; Franco, P.; Iommelli, F.; De Vincenzo, A.; Brancaccio, D.; Telesca, M.; Merlino, F.; Novellino, E.; Ranson, M.; Vecchio, S. D.; Grieco, P.; Carotenuto, A.; Stoppelli, M. P.
Novel anti-inflammatory and chondroprotective effects of the human melanocortin MC1 receptor agonist BMS-470539 dihydrochloride and human melanocortin MC3 receptor agonist PG-990 on lipopolysaccharide activated chondrocytes
2020 Can, V. C.; Locke, I. C.; Kaneva, M. K.; Kerrigan, M. J. P.; Merlino, F.; De Pascale, C.; Grieco, P.; Getting, S. J.
Urotensin-II-Targeted Liposomes as a New Drug Delivery System towards Prostate and Colon Cancer Cells
2019 Zappavigna, S.; Abate, M.; Cossu, A. M.; Lusa, S.; Campani, V.; Scotti, L.; Luce, A.; Yousif, A. M.; Merlino, F.; Grieco, P.; De Rosa, G.; Caraglia, M.
Novel α-MSH peptide analogues with broad spectrum antimicrobial activity.
2013 Grieco, Paolo; Carotenuto, Alfonso; L., Auriemma; Limatola, Antonio; DI MARO, Salvatore; Merlino, Francesco; M. L., Mangoni; V., Luca; A., Di Grazia; S., Gatti; P., Campiglia; GOMEZ MONTERREY, ISABEL MARIA; Novellino, Ettore; A., Catania
Novel temporin L antimicrobial peptides: promoting self-assembling by lipidic tags to tackle superbugs
2020 Bellavita, R.; Falanga, A.; Buommino, E.; Merlino, F.; Casciaro, B.; Cappiello, F.; Mangoni, M. L.; Novellino, E.; Catania, M. R.; Paolillo, R.; Grieco, P.; Galdiero, S.
The Outcomes of Decorated Prolines in the Discovery of Antimicrobial Peptides from Temporin-L
2019 Buommino, E.; Carotenuto, A.; Antignano, Mariarosaria; Bellavita, R.; Casciaro, Raffaella; Loffredo, MARIA ROSARIA; Merlino, F.; Novellino, E.; Mangoni, M. L.; Nocera, F. P.; Brancaccio, D.; Punzi, P.; Roversi, D.; Ingenito, R.; Bianchi, E.; Grieco, P.
An investigation into the origin of the biased agonism associated with the urotensin II receptor activation
2015 Brancaccio, Diego; Merlino, Francesco; Limatola, Antonio; Yousif, ALI MUNAIM; GOMEZ MONTERREY, ISABEL MARIA; Campiglia, Pietro; Novellino, Ettore; Grieco, Paolo; Carotenuto, Alfonso
Structure-Activity Study of the Peptides P5U and Urantide by the Development of Analogues Containing Uncoded Amino Acids at Position9
2016 Merlino, Francesco; Brancaccio, Diego; Yousif, ALI MUNAIM; Piras, Linda; Campiglia, Pietro; GOMEZ MONTERREY, ISABEL MARIA; Santicioli, Paolo; Meini, Stefania; Maggi, Carlo A.; Novellino, Ettore; Carotenuto, Alfonso; Grieco, Paolo
Lead Optimization of P5U and Urantide: Discovery of Novel Potent Ligands at the Urotensin-II Receptor
2014 Carotenuto, Alfonso; Auriemma, Luigia; Merlino, Francesco; Yousif, ALI MUNAIM; Marasco, Daniela; Limatola, Antonio; Pietro, Campiglia; GOMEZ MONTERREY, ISABEL MARIA; Paolo, Santicioli; Stefania, Meini; Carlo A., Maggi; Novellino, Ettore; Grieco, Paolo
New insight into the binding mode of peptides at urotensin-II receptor by Trp-constrained analogues of P5U and urantide.
2013 Carotenuto, Alfonso; L., Auriemma; Merlino, Francesco; Limatola, Antonio; P., Campiglia; GOMEZ MONTERREY, ISABEL MARIA; D'EMMANUELE DI VILLA BIANCA, Roberta; Brancaccio, Diego; P., Santicioli; S., Meini; Maggi, C. A.; Novellino, Ettore; Grieco, Paolo
Simultaneous Targeting of RGD-Integrins and Dual Murine Double Minute Proteins in Glioblastoma Multiforme
2018 Merlino, Francesco; Daniele, Simona; La Pietra, Valeria; Di Maro, Salvatore; Di Leva, Francesco Saverio; Brancaccio, Diego; Tomassi, Stefano; Giuntini, Stefano; Cerofolini, Linda; Fragai, Marco; Luchinat, Claudio; Reichart, Florian; Cavallini, Chiara; Costa, Barbara; Piccarducci, Rebecca; Taliani, Sabrina; Da Settimo, Federico; Martini, Claudia; Kessler, Horst; Novellino, Ettore; Marinelli, Luciana
Development of Macrocyclic Peptidomimetics Containing Constrained α,α-Dialkylated Amino Acids with Potent and Selective Activity at Human Melanocortin Receptors
2018 Merlino, Francesco; Zhou, Yang; Cai, Minying; Carotenuto, Alfonso; Yousif, Ali M; Brancaccio, Diego; Di Maro, Salvatore; Zappavigna, Silvia; Limatola, Antonio; Novellino, Ettore; Grieco, Paolo; Hruby, Victor J
| Titolo | Tipologia | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|---|
| Discovery of New Potent Ligands at Human Urotensin-II Receptor | 1.5 Abstract in rivista | 2013 | Yousif, ALI MUNAIM; Merlino, Francesco; Carotenuto, Alfonso; Limatola, Antonio; Paolo, Santicioli; Campiglia, Pietro; Meini, Stefania; Maggi Carlo, A.; Novellino, Ettore; Grieco, Paolo | |
| Cyclization of the urokinase receptor-derived Ser-Arg-Ser-Arg-Tyr peptide generates a potent inhibitor of trans-endothelial migration of monocytes | 1.1 Articolo in rivista | 2015 | Yousif, ALI MUNAIM; Minopoli, Michele; Bifulco, Katia; Ingangi, Vincenzo; Di Carluccio, Gioconda; Merlino, Francesco; Motti, MARIA LETIZIA; Grieco, Paolo; Carriero, Maria Vincenza | |
| Activation of Melanocortin Receptors MC1 and MC5 Attenuates Retinal Damage in Experimental Diabetic Retinopathy | 1.1 Articolo in rivista | 2016 | Rossi, S; Maisto, R; Gesualdo, C; Trotta, Mc; Ferraraccio, F; Kaneva, Mk; Getting, Sj; Surace, Enrico Maria; Testa, F; Simonelli, F; Grieco, Paolo; Merlino, Francesco; Perretti, M; D'Amico, M; Di Filippo, C. 2. | |
| Urokinase receptor derived peptides as potent inhibitors of the formyl peptide receptor type 1-triggered cell migration | 1.1 Articolo in rivista | 2018 | Yousif, Ali Munaim; Ingangi, Vincenzo; Merlino, Francesco; Brancaccio, Diego; Minopoli, Michele; Bellavita, Rosa; Novellino, Ettore; Carriero, Maria Vincenza; Carotenuto, Alfonso; Grieco, Paolo | |
| Treatment with a Urokinase Receptor-derived Cyclized Peptide Improves Experimental Colitis by Preventing Monocyte Recruitment and Macrophage Polarization | 1.1 Articolo in rivista | 2016 | Genua, Marco; Ingangi, Vincenzo; Fonteyne, Philippe; Piontini, Andrea; Yousif, ALI MUNAIM; Merlino, Francesco; Grieco, Paolo; Malesci, Alberto; Carriero, Maria V; Danese, Silvio | |
| Synthesis and Pharmacological Evaluation of a Novel Peptide Based on Anemonia sulcata BDS-I Toxin as a New KV3.4 Inhibitor Exerting a Neuroprotective Effect Against Amyloid-β Peptide | 1.1 Articolo in rivista | 2019 | Ciccone, Roselia; Piccialli, Ilaria; Grieco, Paolo; Merlino, Francesco; Annunziato, Lucio; Pannaccione, Anna | |
| HOST DEFENSE TEMPORIN 1 PEPTIDES AND THEIR POTENTIAL AS ANTIVIRAL AGENTS | 4.2 Abstract in Atti di convegno | 2017 | Palomba, Luciana; Merlino, Francesco; Zannella, Carla; Franci, Gianluigi; Galdiero, Stefania; Grieco, Paolo; Galdiero, Massimiliano | |
| Urotensin II receptor expression in patients with ulcerative colitis: a pilot study | 1.1 Articolo in rivista | 2020 | Gravina, Antonietta G; Dallio, Marcello; Tuccillo, Concetta; Martorano, Marco; Abenavoli, Ludovico; Luzza, Francesco; Stiuso, Paola; Lama, Stefania; Grieco, Paolo; Merlino, Francesco; Caraglia, Michele; Loguercio, Carmelina; Federico, Alessandro | |
| Breast tumor cell invasion and pro-invasive activity of cancer-associated fibroblasts co-targeted by novel urokinase-derived decapeptides | 1.1 Articolo in rivista | 2020 | Belli, S.; Franco, P.; Iommelli, F.; De Vincenzo, A.; Brancaccio, D.; Telesca, M.; Merlino, F.; Novellino, E.; Ranson, M.; Vecchio, S. D.; Grieco, P.; Carotenuto, A.; Stoppelli, M. P. | |
| Novel anti-inflammatory and chondroprotective effects of the human melanocortin MC1 receptor agonist BMS-470539 dihydrochloride and human melanocortin MC3 receptor agonist PG-990 on lipopolysaccharide activated chondrocytes | 1.1 Articolo in rivista | 2020 | Can, V. C.; Locke, I. C.; Kaneva, M. K.; Kerrigan, M. J. P.; Merlino, F.; De Pascale, C.; Grieco, P.; Getting, S. J. | |
| Urotensin-II-Targeted Liposomes as a New Drug Delivery System towards Prostate and Colon Cancer Cells | 1.1 Articolo in rivista | 2019 | Zappavigna, S.; Abate, M.; Cossu, A. M.; Lusa, S.; Campani, V.; Scotti, L.; Luce, A.; Yousif, A. M.; Merlino, F.; Grieco, P.; De Rosa, G.; Caraglia, M. | |
| Novel α-MSH peptide analogues with broad spectrum antimicrobial activity. | 1.1 Articolo in rivista | 2013 | Grieco, Paolo; Carotenuto, Alfonso; L., Auriemma; Limatola, Antonio; DI MARO, Salvatore; Merlino, Francesco; M. L., Mangoni; V., Luca; A., Di Grazia; S., Gatti; P., Campiglia; GOMEZ MONTERREY, ISABEL MARIA; Novellino, Ettore; A., Catania | |
| Novel temporin L antimicrobial peptides: promoting self-assembling by lipidic tags to tackle superbugs | 1.1 Articolo in rivista | 2020 | Bellavita, R.; Falanga, A.; Buommino, E.; Merlino, F.; Casciaro, B.; Cappiello, F.; Mangoni, M. L.; Novellino, E.; Catania, M. R.; Paolillo, R.; Grieco, P.; Galdiero, S. | |
| The Outcomes of Decorated Prolines in the Discovery of Antimicrobial Peptides from Temporin-L | 1.1 Articolo in rivista | 2019 | Buommino, E.; Carotenuto, A.; Antignano, Mariarosaria; Bellavita, R.; Casciaro, Raffaella; Loffredo, MARIA ROSARIA; Merlino, F.; Novellino, E.; Mangoni, M. L.; Nocera, F. P.; Brancaccio, D.; Punzi, P.; Roversi, D.; Ingenito, R.; Bianchi, E.; Grieco, P. | |
| An investigation into the origin of the biased agonism associated with the urotensin II receptor activation | 1.1 Articolo in rivista | 2015 | Brancaccio, Diego; Merlino, Francesco; Limatola, Antonio; Yousif, ALI MUNAIM; GOMEZ MONTERREY, ISABEL MARIA; Campiglia, Pietro; Novellino, Ettore; Grieco, Paolo; Carotenuto, Alfonso | |
| Structure-Activity Study of the Peptides P5U and Urantide by the Development of Analogues Containing Uncoded Amino Acids at Position9 | 1.1 Articolo in rivista | 2016 | Merlino, Francesco; Brancaccio, Diego; Yousif, ALI MUNAIM; Piras, Linda; Campiglia, Pietro; GOMEZ MONTERREY, ISABEL MARIA; Santicioli, Paolo; Meini, Stefania; Maggi, Carlo A.; Novellino, Ettore; Carotenuto, Alfonso; Grieco, Paolo | |
| Lead Optimization of P5U and Urantide: Discovery of Novel Potent Ligands at the Urotensin-II Receptor | 1.1 Articolo in rivista | 2014 | Carotenuto, Alfonso; Auriemma, Luigia; Merlino, Francesco; Yousif, ALI MUNAIM; Marasco, Daniela; Limatola, Antonio; Pietro, Campiglia; GOMEZ MONTERREY, ISABEL MARIA; Paolo, Santicioli; Stefania, Meini; Carlo A., Maggi; Novellino, Ettore; Grieco, Paolo | |
| New insight into the binding mode of peptides at urotensin-II receptor by Trp-constrained analogues of P5U and urantide. | 1.1 Articolo in rivista | 2013 | Carotenuto, Alfonso; L., Auriemma; Merlino, Francesco; Limatola, Antonio; P., Campiglia; GOMEZ MONTERREY, ISABEL MARIA; D'EMMANUELE DI VILLA BIANCA, Roberta; Brancaccio, Diego; P., Santicioli; S., Meini; Maggi, C. A.; Novellino, Ettore; Grieco, Paolo | |
| Simultaneous Targeting of RGD-Integrins and Dual Murine Double Minute Proteins in Glioblastoma Multiforme | 1.1 Articolo in rivista | 2018 | Merlino, Francesco; Daniele, Simona; La Pietra, Valeria; Di Maro, Salvatore; Di Leva, Francesco Saverio; Brancaccio, Diego; Tomassi, Stefano; Giuntini, Stefano; Cerofolini, Linda; Fragai, Marco; Luchinat, Claudio; Reichart, Florian; Cavallini, Chiara; Costa, Barbara; Piccarducci, Rebecca; Taliani, Sabrina; Da Settimo, Federico; Martini, Claudia; Kessler, Horst; Novellino, Ettore; Marinelli, Luciana | |
| Development of Macrocyclic Peptidomimetics Containing Constrained α,α-Dialkylated Amino Acids with Potent and Selective Activity at Human Melanocortin Receptors | 1.1 Articolo in rivista | 2018 | Merlino, Francesco; Zhou, Yang; Cai, Minying; Carotenuto, Alfonso; Yousif, Ali M; Brancaccio, Diego; Di Maro, Salvatore; Zappavigna, Silvia; Limatola, Antonio; Novellino, Ettore; Grieco, Paolo; Hruby, Victor J |