Sfoglia per Autore
Chemistry and Pharmacology of GPBAR1 and FXR Selective Agonists, Dual Agonists, and Antagonists
2019 DE MARINO, Simona; Festa, Carmen; Sepe, Valentina; Zampella, Angela
Novel Isoxazole Derivatives with Potent FXR Agonistic Activity Prevent Acetaminophen-Induced Liver Injury
2019 Sepe, Valentina; Marchianò, Silvia; Finamore, Claudia; Baronissi, Giuliana; Di Leva, Francesco Saverio; Carino, Adriana; Biagioli, Michele; Fiorucci, Chiara; Cassiano, Chiara; Chiara Monti, Maria; del Gaudio, Federica; Novellino, Ettore; Limongelli, Vittorio; Fiorucci, Stefano; Zampella, Angela
Introduction of Nonacidic Side Chains on 6-Ethylcholane Scaffolds in the Identification of Potent Bile Acid Receptor Agonists with Improved Pharmacokinetic Properties
2019 Finamore, Claudia; Baronissi, Giuliana; Marchianò, Silvia; Di Leva, Francesco Saverio; Carino, Adriana; Chiara Monti, Maria; Limongelli, Vittorio; Zampella, Angela; Fiorucci, Stefano; Sepe, Valentina
Modification of semisynthetic bile acid derivatives as human receptor modulators
2018 Finamore, C.; Festa, C.; De Marino, S.; Fiorucci, S.; Zampella, A.; Sepe, V.
Synthesis of a new class of isoxazole derivatives with a dual FXR agonistic and COX-2 inhibitory activity
2018 Finamore, C.; Sepe, V.; Masullo, D.; Fiorucci, S.; Zampella, A.
Synthesis of a new class of isoxazole derivatives with a dual FXR agonistic and COX-2 inhibitory activity.
2018 Finamore, C.; Sepe, V.; Masullo, D.; Fiorucci, S.; Zampella, Angela
Farnesoid X receptor modulators 2014-present: a patent review
2018 Sepe, Valentina; Distrutti, Eleonora; Fiorucci, Stefano; Zampella, Angela
Identification of new GPBAR1 selective agonists containing an epoxide group on cholane side chains
2018 Sepe, Valentina; DE MARINO, Simona; Festa, Carmen; Finamore, Claudia; D'Auria, MARIA VALERIA; Fiorucci, Stefano; Zampella, Angela
Modification of semisynthetic bile acid derivatives as human receptor modulators
2018 Sepe, Valentina
Speculation on 6-ethylcholane scaffold in the discovery of novel FXR and GPBAR1 ligands.
2017 Finamore, C.; Festa C., C.; Sepe, V.; Carino, A.; Masullo, D.; Marchianò, S.; Monti, M. C.; Fiorucci, S.; Zampella, A.
2° International Summer School on Natural Products
2017 Costantino, Valeria; Oliviero, Giorgia; Tartaglione, Luciana; DE MARINO, Simona; Sepe, Valentina; Imperatore, Concetta
Epoxide functionalization on cholane side chains in the identification of G-protein coupled bile acid receptor (GPBAR1) selective agonists
2017 DE MARINO, Simona; Carino, Adriana; Masullo, Dario; Finamore, Claudia; Sepe, Valentina; Marchianò, Silvia; Di Leva, Francesco Saverio; Limongelli, Vittorio; Fiorucci, Stefano; Zampella, Angela
Targeting bile acid receptors: discovery of a potent and selective Farnesoid X receptor agonist as a new lead in the pharmacological approach to liver diseases
2017 Festa, Carmen; DE MARINO, Simona; Carino, A.; Sepe, Valentina; Marchianò, S.; Cipriani, S.; Di Leva, Francesco Saverio; Limongelli, Vittorio; Monti, M. C.; Capolupo, A.; Distrutti, E.; Fiorucci, S.; Zampella, Angela
Navigation in bile acid chemical space: discovery of novel FXR and GPBAR1 modulators
2016 Finamore, Claudia; Festa, Carmen; Sepe, Valentina; Carino, Adriana; Masullo, Dario; Marchianò, Silvia; Fiorucci, Stefano; Zampella, Angela
Rational Drug Design of New Selective Modulators of GPBAR1
2016 Zampella, Angela; Fiorucci, Stefano; Limongelli, Vittorio; D'Auria, MARIA VALERIA; DE MARINO, Simona; Sepe, Valentina; Festa, Carmen
Towards FXR selectivity: manipulation of 6-ethylcholane scaffold
2016 Sepe, Valentina; Festa, Carmen; Masullo, Dario; Renga, B.; Fiorucci, S.; Zampella, Angela; Finamore, Claudia
Investigation on bile acid receptor regulators. Discovery of cholanoic acid derivatives with dual G-protein coupled bile acid receptor 1 (GPBAR1) antagonistic and farnesoid X receptor (FXR) modulatory activity
2016 Sepe, Valentina; Renga, Barbara; Festa, Carmen; Finamore, Claudia; Masullo, Dario; Carino, Adriana; Cipriani, Sabrina; Distrutti, Eleonora; Fiorucci, Stefano; Zampella, Angela
Navigation in bile acid chemical space: discovery of novel FXR and GPBAR1 ligands
2016 Finamore, Claudia; Festa, Carmen; Renga, B; Sepe, Valentina; Carino, A; Masullo, Dario; Biagioli, M; Marchianò, S; Capolupo, A; Monti, Mc; Fiorucci, S; Zampella, Angela
Insights on FXR selective modulation. Speculation on bile acid chemical space in the discovery of potent and selective agonists
2016 Sepe, Valentina; Festa, Carmen; Renga, Barbara; Carino, Adriana; Cipriani, Sabrina; Finamore, Claudia; Masullo, Dario; Del Gaudio, Federica; Monti, Maria Chiara; Fiorucci, Stefano; Zampella, Angela
Bile acids derivatives in the selective modulation of FXR and GP-BAR1
2015 Finamore, Claudia; Sepe, Valentina; D’Amore, C.; Festa, Carmen; Renga, B.; DE MARINO, Simona; Zampella, Angela; Fiorucci, S.; Masullo, Dario
Titolo | Tipologia | Data di pubblicazione | Autore(i) | File |
---|---|---|---|---|
Chemistry and Pharmacology of GPBAR1 and FXR Selective Agonists, Dual Agonists, and Antagonists | 2.1 Contributo in volume (Capitolo o Saggio) | 2019 | DE MARINO, Simona; Festa, Carmen; Sepe, Valentina; Zampella, Angela | |
Novel Isoxazole Derivatives with Potent FXR Agonistic Activity Prevent Acetaminophen-Induced Liver Injury | 1.1 Articolo in rivista | 2019 | Sepe, Valentina; Marchianò, Silvia; Finamore, Claudia; Baronissi, Giuliana; Di Leva, Francesco Saverio; Carino, Adriana; Biagioli, Michele; Fiorucci, Chiara; Cassiano, Chiara; Chiara Monti, Maria; del Gaudio, Federica; Novellino, Ettore; Limongelli, Vittorio; Fiorucci, Stefano; Zampella, Angela | |
Introduction of Nonacidic Side Chains on 6-Ethylcholane Scaffolds in the Identification of Potent Bile Acid Receptor Agonists with Improved Pharmacokinetic Properties | 1.1 Articolo in rivista | 2019 | Finamore, Claudia; Baronissi, Giuliana; Marchianò, Silvia; Di Leva, Francesco Saverio; Carino, Adriana; Chiara Monti, Maria; Limongelli, Vittorio; Zampella, Angela; Fiorucci, Stefano; Sepe, Valentina | |
Modification of semisynthetic bile acid derivatives as human receptor modulators | 4.2 Abstract in Atti di convegno | 2018 | Finamore, C.; Festa, C.; De Marino, S.; Fiorucci, S.; Zampella, A.; Sepe, V. | |
Synthesis of a new class of isoxazole derivatives with a dual FXR agonistic and COX-2 inhibitory activity | 4.2 Abstract in Atti di convegno | 2018 | Finamore, C.; Sepe, V.; Masullo, D.; Fiorucci, S.; Zampella, A. | |
Synthesis of a new class of isoxazole derivatives with a dual FXR agonistic and COX-2 inhibitory activity. | 4.2 Abstract in Atti di convegno | 2018 | Finamore, C.; Sepe, V.; Masullo, D.; Fiorucci, S.; Zampella, Angela | |
Farnesoid X receptor modulators 2014-present: a patent review | 1.1 Articolo in rivista | 2018 | Sepe, Valentina; Distrutti, Eleonora; Fiorucci, Stefano; Zampella, Angela | |
Identification of new GPBAR1 selective agonists containing an epoxide group on cholane side chains | 4.2 Abstract in Atti di convegno | 2018 | Sepe, Valentina; DE MARINO, Simona; Festa, Carmen; Finamore, Claudia; D'Auria, MARIA VALERIA; Fiorucci, Stefano; Zampella, Angela | |
Modification of semisynthetic bile acid derivatives as human receptor modulators | 8.02 Comunicazioni a Convegni o Seminari | 2018 | Sepe, Valentina | |
Speculation on 6-ethylcholane scaffold in the discovery of novel FXR and GPBAR1 ligands. | 4.2 Abstract in Atti di convegno | 2017 | Finamore, C.; Festa C., C.; Sepe, V.; Carino, A.; Masullo, D.; Marchianò, S.; Monti, M. C.; Fiorucci, S.; Zampella, A. | |
2° International Summer School on Natural Products | 8.04 Convegni organizzati dalla struttura | 2017 | Costantino, Valeria; Oliviero, Giorgia; Tartaglione, Luciana; DE MARINO, Simona; Sepe, Valentina; Imperatore, Concetta | |
Epoxide functionalization on cholane side chains in the identification of G-protein coupled bile acid receptor (GPBAR1) selective agonists | 1.1 Articolo in rivista | 2017 | DE MARINO, Simona; Carino, Adriana; Masullo, Dario; Finamore, Claudia; Sepe, Valentina; Marchianò, Silvia; Di Leva, Francesco Saverio; Limongelli, Vittorio; Fiorucci, Stefano; Zampella, Angela | |
Targeting bile acid receptors: discovery of a potent and selective Farnesoid X receptor agonist as a new lead in the pharmacological approach to liver diseases | 1.1 Articolo in rivista | 2017 | Festa, Carmen; DE MARINO, Simona; Carino, A.; Sepe, Valentina; Marchianò, S.; Cipriani, S.; Di Leva, Francesco Saverio; Limongelli, Vittorio; Monti, M. C.; Capolupo, A.; Distrutti, E.; Fiorucci, S.; Zampella, Angela | |
Navigation in bile acid chemical space: discovery of novel FXR and GPBAR1 modulators | 4.2 Abstract in Atti di convegno | 2016 | Finamore, Claudia; Festa, Carmen; Sepe, Valentina; Carino, Adriana; Masullo, Dario; Marchianò, Silvia; Fiorucci, Stefano; Zampella, Angela | |
Rational Drug Design of New Selective Modulators of GPBAR1 | 4.2 Abstract in Atti di convegno | 2016 | Zampella, Angela; Fiorucci, Stefano; Limongelli, Vittorio; D'Auria, MARIA VALERIA; DE MARINO, Simona; Sepe, Valentina; Festa, Carmen | |
Towards FXR selectivity: manipulation of 6-ethylcholane scaffold | 4.2 Abstract in Atti di convegno | 2016 | Sepe, Valentina; Festa, Carmen; Masullo, Dario; Renga, B.; Fiorucci, S.; Zampella, Angela; Finamore, Claudia | |
Investigation on bile acid receptor regulators. Discovery of cholanoic acid derivatives with dual G-protein coupled bile acid receptor 1 (GPBAR1) antagonistic and farnesoid X receptor (FXR) modulatory activity | 1.1 Articolo in rivista | 2016 | Sepe, Valentina; Renga, Barbara; Festa, Carmen; Finamore, Claudia; Masullo, Dario; Carino, Adriana; Cipriani, Sabrina; Distrutti, Eleonora; Fiorucci, Stefano; Zampella, Angela | |
Navigation in bile acid chemical space: discovery of novel FXR and GPBAR1 ligands | 1.1 Articolo in rivista | 2016 | Finamore, Claudia; Festa, Carmen; Renga, B; Sepe, Valentina; Carino, A; Masullo, Dario; Biagioli, M; Marchianò, S; Capolupo, A; Monti, Mc; Fiorucci, S; Zampella, Angela | |
Insights on FXR selective modulation. Speculation on bile acid chemical space in the discovery of potent and selective agonists | 1.1 Articolo in rivista | 2016 | Sepe, Valentina; Festa, Carmen; Renga, Barbara; Carino, Adriana; Cipriani, Sabrina; Finamore, Claudia; Masullo, Dario; Del Gaudio, Federica; Monti, Maria Chiara; Fiorucci, Stefano; Zampella, Angela | |
Bile acids derivatives in the selective modulation of FXR and GP-BAR1 | 4.2 Abstract in Atti di convegno | 2015 | Finamore, Claudia; Sepe, Valentina; D’Amore, C.; Festa, Carmen; Renga, B.; DE MARINO, Simona; Zampella, Angela; Fiorucci, S.; Masullo, Dario |
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