Sfoglia per Autore
Photo-Flow Technology for Chemical Rearrangements: A Powerful Tool to Generate Pharmaceutically Relevant Compounds
2023 Alfano, A. I.; Pelliccia, S.; Rossino, G.; Chianese, O.; Summa, V.; Collina, S.; Brindisi, M.
Broad-spectrum coronavirus 3C-like protease peptidomimetic inhibitors effectively block SARS-CoV-2 replication in cells: Design, synthesis, biological evaluation, and X-ray structure determination
2023 Stefanelli, Irina; Corona, Angela; Cerchia, Carmen; Cassese, Emilia; Improta, Salvatore; Costanzi, Elisa; Pelliccia, Sveva; Morasso, Stefano; Esposito, Francesca; Paulis, Annalaura; Scognamiglio, Sante; Di Leva, Francesco Saverio; Storici, Paola; Brindisi, Margherita; Tramontano, Enzo; Cannalire, Rolando; Summa, Vincenzo
Continuous-Flow Technology for Chemical Rearrangements: A Powerful Tool to Generate Pharmaceutically Relevant Compounds
2023 Alfano, Antonella Ilenia; Pelliccia, Sveva; Rossino, Giacomo; Chianese, Orazio; Summa, Vincenzo; Collina, Simona; Brindisi, Margherita
Rejuvenating the [1, 2, 3]-triazolo [1,5-a]quinoxalin-4(5H)-one scaffold: Synthesis and derivatization in a sustainable guise and preliminary antimicrobial evaluation
2023 Pelliccia, Sveva; Alfano, Antonella Ilenia; Gomes Da Assunção, Beatriz Ramos; Turco, Luigia; Lembo, Francesca; Summa, Vincenzo; Buommino, Elisabetta; Brindisi, Margherita
Amide Bonds Meet Flow Chemistry: A Journey into Methodologies and Sustainable Evolution
2022 Alfano, A. L.; Lange, H.; Brindisi, M.
Chasing a Breath of Fresh Air in Cystic Fibrosis (CF): Therapeutic Potential of Selective HDAC6 Inhibitors to Tackle Multiple Pathways in CF Pathophysiology
2022 Barone, S.; Cassese, E.; Alfano, A. I.; Brindisi, M.; Summa, V.
Editorial: Multi-target directed ligands for the treatment of cancer
2022 Brindisi, Margherita; Kessler, Sonja M; Kumar, Vinod; Zwergel, Clemens
Efficacy of selective histone deacetylase 6 inhibition in mouse models of Pseudomonas aeruginosa infection: A new glimpse for reducing inflammation and infection in cystic fibrosis
2022 Brindisi, Margherita; Barone, Simona; Rossi, Alice; Cassese, Emilia; Del Gaudio, Nunzio; Feliz Morel, Álvaro Javier; Filocamo, Gessica; Alberico, Alessia; De Fino, Ida; Gugliandolo, Davide; Babaei, Mehrad; Bove, Guglielmo; Croce, Martina; Montesano, Camilla; Altucci, Lucia; Bragonzi, Alessandra; Summa, Vincenzo
Easy access to α-ketoamides as SARS-CoV-2 and MERS Mpro inhibitors via the PADAM oxidation route
2022 Pelliccia, Sveva; Cerchia, Carmen; Esposito, Francesca; Cannalire, Rolando; Corona, Angela; Costanzi, Elisa; Kuzikov, Maria; Gribbon, Philip; Zaliani, Andrea; Brindisi, Margherita; Storici, Paola; Tramontano, Enzo; Summa, Vincenzo
Mechanochemical Fischer indolisation: an eco-friendly design for a timeless reaction
2022 Porcheddu, A.; Mocci, R.; Brindisi, M.; Cuccu, F.; Fattuoni, C.; Delogu, F.; Colacino, E.; D'Auria, M. V.
Coupling Interrupted Fischer and Multicomponent Joullié-Ugi to Chase Chemical Diversity: from Batch to Sustainable Flow Synthesis of Peptidomimetics
2021 Alfano, A. I.; Buommino, E.; Ferraro, M. G.; Irace, C.; Zampella, A.; Lange, H.; Brindisi, M.
Novel quinolone-based potent and selective HDAC6 inhibitors: Synthesis, molecular modeling studies and biological investigation
2021 Relitti, N.; Saraswati, A. P.; Chemi, G.; Brindisi, M.; Brogi, S.; Herp, D.; Schmidtkunz, K.; Saccoccia, F.; Ruberti, G.; Ulivieri, C.; Vanni, F.; Sarno, F.; Altucci, L.; Lamponi, S.; Jung, M.; Gemma, S.; Butini, S.; Campiani, G.
Flow synthesis approaches to privileged scaffolds - recent routes reviewed for green and sustainable aspects
2021 Alfano, A. I.; Brindisi, M.; Lange, H.
Urea Derivatives in Modern Drug Discovery and Medicinal Chemistry
2020 Ghosh, A. K.; Brindisi, M.
Targeting Endocannabinoid Metabolism: an Arrow with Multiple Tips Against Multiple Sclerosis
2020 Maramai, S.; Brindisi, M.
Drug Development and Medicinal Chemistry Efforts toward SARS-Coronavirus and Covid-19 Therapeutics
2020 Ghosh, A. K.; Brindisi, M.; Shahabi, D.; Chapman, M. E.; Mesecar, A. D.
Autophagy modulators for the treatment of oral and esophageal squamous cell carcinomas
2020 Khan, T.; Relitti, N.; Brindisi, M.; Magnano, S.; Zisterer, D.; Gemma, S.; Butini, S.; Campiani, G.
Harnessing interrupted Fischer in continuous flow: sustainable synthesis of (spiro)indolenine and (spiro)indoline privileged scaffolds
2020 Alfano, Antonella Ilenia; Zampella, Angela; Novellino, Ettore; Brindisi, Margherita; Lange, Heiko
Spiroindoline-Capped Selective HDAC6 Inhibitors: Design, Synthesis, Structural Analysis, and Biological Evaluation
2020 Saraswati, A Prasanth; Relitti, Nicola; Brindisi, Margherita; Osko, Jeremy D; Chemi, Giulia; Federico, Stefano; Grillo, Alessandro; Brogi, Simone; Mccabe, Niamh H; Turkington, Richard C; Ibrahim, Ola; O'Sullivan, Jeffrey; Lamponi, Stefania; Ghanim, Magda; Kelly, Vincent P; Zisterer, Daniela; Amet, Rebecca; Hannon Barroeta, Patricia; Vanni, Francesca; Ulivieri, Cristina; Herp, Daniel; Sarno, Federica; Di Costanzo, Antonella; Saccoccia, Fulvio; Ruberti, Giovina; Jung, Manfred; Altucci, Lucia; Gemma, Sandra; Butini, Stefania; Christianson, David W; Campiani, Giuseppe
Old but Gold: Tracking the New Guise of Histone Deacetylase 6 (HDAC6) Enzyme as a Biomarker and Therapeutic Target in Rare Diseases
2020 Brindisi, Margherita; Saraswati, A Prasanth; Brogi, Simone; Gemma, Sandra; Butini, Stefania; Campiani, Giuseppe
| Titolo | Tipologia | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|---|
| Photo-Flow Technology for Chemical Rearrangements: A Powerful Tool to Generate Pharmaceutically Relevant Compounds | 1.1 Articolo in rivista | 2023 | Alfano, A. I.; Pelliccia, S.; Rossino, G.; Chianese, O.; Summa, V.; Collina, S.; Brindisi, M. | |
| Broad-spectrum coronavirus 3C-like protease peptidomimetic inhibitors effectively block SARS-CoV-2 replication in cells: Design, synthesis, biological evaluation, and X-ray structure determination | 1.1 Articolo in rivista | 2023 | Stefanelli, Irina; Corona, Angela; Cerchia, Carmen; Cassese, Emilia; Improta, Salvatore; Costanzi, Elisa; Pelliccia, Sveva; Morasso, Stefano; Esposito, Francesca; Paulis, Annalaura; Scognamiglio, Sante; Di Leva, Francesco Saverio; Storici, Paola; Brindisi, Margherita; Tramontano, Enzo; Cannalire, Rolando; Summa, Vincenzo | |
| Continuous-Flow Technology for Chemical Rearrangements: A Powerful Tool to Generate Pharmaceutically Relevant Compounds | 1.1 Articolo in rivista | 2023 | Alfano, Antonella Ilenia; Pelliccia, Sveva; Rossino, Giacomo; Chianese, Orazio; Summa, Vincenzo; Collina, Simona; Brindisi, Margherita | |
| Rejuvenating the [1, 2, 3]-triazolo [1,5-a]quinoxalin-4(5H)-one scaffold: Synthesis and derivatization in a sustainable guise and preliminary antimicrobial evaluation | 1.1 Articolo in rivista | 2023 | Pelliccia, Sveva; Alfano, Antonella Ilenia; Gomes Da Assunção, Beatriz Ramos; Turco, Luigia; Lembo, Francesca; Summa, Vincenzo; Buommino, Elisabetta; Brindisi, Margherita | |
| Amide Bonds Meet Flow Chemistry: A Journey into Methodologies and Sustainable Evolution | 1.1 Articolo in rivista | 2022 | Alfano, A. L.; Lange, H.; Brindisi, M. | |
| Chasing a Breath of Fresh Air in Cystic Fibrosis (CF): Therapeutic Potential of Selective HDAC6 Inhibitors to Tackle Multiple Pathways in CF Pathophysiology | 1.1 Articolo in rivista | 2022 | Barone, S.; Cassese, E.; Alfano, A. I.; Brindisi, M.; Summa, V. | |
| Editorial: Multi-target directed ligands for the treatment of cancer | 1.1 Articolo in rivista | 2022 | Brindisi, Margherita; Kessler, Sonja M; Kumar, Vinod; Zwergel, Clemens | |
| Efficacy of selective histone deacetylase 6 inhibition in mouse models of Pseudomonas aeruginosa infection: A new glimpse for reducing inflammation and infection in cystic fibrosis | 1.1 Articolo in rivista | 2022 | Brindisi, Margherita; Barone, Simona; Rossi, Alice; Cassese, Emilia; Del Gaudio, Nunzio; Feliz Morel, Álvaro Javier; Filocamo, Gessica; Alberico, Alessia; De Fino, Ida; Gugliandolo, Davide; Babaei, Mehrad; Bove, Guglielmo; Croce, Martina; Montesano, Camilla; Altucci, Lucia; Bragonzi, Alessandra; Summa, Vincenzo | |
| Easy access to α-ketoamides as SARS-CoV-2 and MERS Mpro inhibitors via the PADAM oxidation route | 1.1 Articolo in rivista | 2022 | Pelliccia, Sveva; Cerchia, Carmen; Esposito, Francesca; Cannalire, Rolando; Corona, Angela; Costanzi, Elisa; Kuzikov, Maria; Gribbon, Philip; Zaliani, Andrea; Brindisi, Margherita; Storici, Paola; Tramontano, Enzo; Summa, Vincenzo | |
| Mechanochemical Fischer indolisation: an eco-friendly design for a timeless reaction | 1.1 Articolo in rivista | 2022 | Porcheddu, A.; Mocci, R.; Brindisi, M.; Cuccu, F.; Fattuoni, C.; Delogu, F.; Colacino, E.; D'Auria, M. V. | |
| Coupling Interrupted Fischer and Multicomponent Joullié-Ugi to Chase Chemical Diversity: from Batch to Sustainable Flow Synthesis of Peptidomimetics | 1.1 Articolo in rivista | 2021 | Alfano, A. I.; Buommino, E.; Ferraro, M. G.; Irace, C.; Zampella, A.; Lange, H.; Brindisi, M. | |
| Novel quinolone-based potent and selective HDAC6 inhibitors: Synthesis, molecular modeling studies and biological investigation | 1.1 Articolo in rivista | 2021 | Relitti, N.; Saraswati, A. P.; Chemi, G.; Brindisi, M.; Brogi, S.; Herp, D.; Schmidtkunz, K.; Saccoccia, F.; Ruberti, G.; Ulivieri, C.; Vanni, F.; Sarno, F.; Altucci, L.; Lamponi, S.; Jung, M.; Gemma, S.; Butini, S.; Campiani, G. | |
| Flow synthesis approaches to privileged scaffolds - recent routes reviewed for green and sustainable aspects | 1.8 Articolo in rassegna (review) | 2021 | Alfano, A. I.; Brindisi, M.; Lange, H. | |
| Urea Derivatives in Modern Drug Discovery and Medicinal Chemistry | 1.1 Articolo in rivista | 2020 | Ghosh, A. K.; Brindisi, M. | |
| Targeting Endocannabinoid Metabolism: an Arrow with Multiple Tips Against Multiple Sclerosis | 1.1 Articolo in rivista | 2020 | Maramai, S.; Brindisi, M. | |
| Drug Development and Medicinal Chemistry Efforts toward SARS-Coronavirus and Covid-19 Therapeutics | 1.1 Articolo in rivista | 2020 | Ghosh, A. K.; Brindisi, M.; Shahabi, D.; Chapman, M. E.; Mesecar, A. D. | |
| Autophagy modulators for the treatment of oral and esophageal squamous cell carcinomas | 1.1 Articolo in rivista | 2020 | Khan, T.; Relitti, N.; Brindisi, M.; Magnano, S.; Zisterer, D.; Gemma, S.; Butini, S.; Campiani, G. | |
| Harnessing interrupted Fischer in continuous flow: sustainable synthesis of (spiro)indolenine and (spiro)indoline privileged scaffolds | 1.1 Articolo in rivista | 2020 | Alfano, Antonella Ilenia; Zampella, Angela; Novellino, Ettore; Brindisi, Margherita; Lange, Heiko | |
| Spiroindoline-Capped Selective HDAC6 Inhibitors: Design, Synthesis, Structural Analysis, and Biological Evaluation | 1.1 Articolo in rivista | 2020 | Saraswati, A Prasanth; Relitti, Nicola; Brindisi, Margherita; Osko, Jeremy D; Chemi, Giulia; Federico, Stefano; Grillo, Alessandro; Brogi, Simone; Mccabe, Niamh H; Turkington, Richard C; Ibrahim, Ola; O'Sullivan, Jeffrey; Lamponi, Stefania; Ghanim, Magda; Kelly, Vincent P; Zisterer, Daniela; Amet, Rebecca; Hannon Barroeta, Patricia; Vanni, Francesca; Ulivieri, Cristina; Herp, Daniel; Sarno, Federica; Di Costanzo, Antonella; Saccoccia, Fulvio; Ruberti, Giovina; Jung, Manfred; Altucci, Lucia; Gemma, Sandra; Butini, Stefania; Christianson, David W; Campiani, Giuseppe | |
| Old but Gold: Tracking the New Guise of Histone Deacetylase 6 (HDAC6) Enzyme as a Biomarker and Therapeutic Target in Rare Diseases | 1.1 Articolo in rivista | 2020 | Brindisi, Margherita; Saraswati, A Prasanth; Brogi, Simone; Gemma, Sandra; Butini, Stefania; Campiani, Giuseppe |
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