Sfoglia per Autore
Functional Selectivity Revealed by N-Methylation Scanning of Human Urotensin II and Related Peptides
2019 Merlino, Francesco; Billard, Etienne; Yousif, Ali Munaim; Di Maro, Salvatore; Brancaccio, Diego; Abate, Luigi; Carotenuto, Alfonso; Bellavita, Rosa; d'Emmanuele di Villa Bianca, Roberta; Santicioli, Paolo; Marinelli, Luciana; Novellino, Ettore; Hébert, Terence; Lubell, William D; Chatenet, David; Grieco, Paolo
Urotensin-II-Targeted Liposomes as a New Drug Delivery System towards Prostate and Colon Cancer Cells
2019 Zappavigna, S.; Abate, M.; Cossu, A. M.; Lusa, S.; Campani, V.; Scotti, L.; Luce, A.; Yousif, A. M.; Merlino, F.; Grieco, P.; De Rosa, G.; Caraglia, M.
Boosting Fmoc Solid-Phase Peptide Synthesis by Ultrasonication
2019 Merlino, F.; Tomassi, S.; Yousif, A. M.; Messere, A.; Marinelli, L.; Grieco, P.; Novellino, E.; Cosconati, S.; Di Maro, S.
Urokinase receptor derived peptides as potent inhibitors of the formyl peptide receptor type 1-triggered cell migration
2018 Yousif, Ali Munaim; Ingangi, Vincenzo; Merlino, Francesco; Brancaccio, Diego; Minopoli, Michele; Bellavita, Rosa; Novellino, Ettore; Carriero, Maria Vincenza; Carotenuto, Alfonso; Grieco, Paolo
Development of Macrocyclic Peptidomimetics Containing Constrained α,α-Dialkylated Amino Acids with Potent and Selective Activity at Human Melanocortin Receptors
2018 Merlino, Francesco; Zhou, Yang; Cai, Minying; Carotenuto, Alfonso; Yousif, Ali M; Brancaccio, Diego; Di Maro, Salvatore; Zappavigna, Silvia; Limatola, Antonio; Novellino, Ettore; Grieco, Paolo; Hruby, Victor J
Glycine-replaced derivatives of [Pro3,DLeu9]TL, a temporin L analogue: Evaluation of antimicrobial, cytotoxic and hemolytic activities
2017 Merlino, Francesco; Carotenuto, Alfonso; Casciaro, Bruno; Martora, Francesca; Loffredo, Maria Rosa; Di Grazia, Antonio; Yousif, Ali M.; Brancaccio, Diego; Palomba, Luciana; Novellino, Ettore; Galdiero, Massimiliano; Iovene, Maria Rosaria; Mangoni, Maria L.; Grieco, Paolo
Structure-Activity Study of the Peptides P5U and Urantide by the Development of Analogues Containing Uncoded Amino Acids at Position9
2016 Merlino, Francesco; Brancaccio, Diego; Yousif, ALI MUNAIM; Piras, Linda; Campiglia, Pietro; GOMEZ MONTERREY, ISABEL MARIA; Santicioli, Paolo; Meini, Stefania; Maggi, Carlo A.; Novellino, Ettore; Carotenuto, Alfonso; Grieco, Paolo
Treatment with a Urokinase Receptor-derived Cyclized Peptide Improves Experimental Colitis by Preventing Monocyte Recruitment and Macrophage Polarization
2016 Genua, Marco; Ingangi, Vincenzo; Fonteyne, Philippe; Piontini, Andrea; Yousif, ALI MUNAIM; Merlino, Francesco; Grieco, Paolo; Malesci, Alberto; Carriero, Maria V; Danese, Silvio
The urokinase receptor-derived cyclic peptide [SRSRY] suppresses neovascularization and intravasation of osteosarcoma and chondrosarcoma cells
2016 Ingangi, Vincenzo; Bifulco, Katia; Yousif, ALI MUNAIM; Ragone, Concetta; Motti, MARIA LETIZIA; Rea, Domenica; Minopoli, Michele; Botti, Giovanni; Scognamiglio, Giuseppe; Fazioli, Flavio; Gallo, Michele; De Chiara, Annarosaria; Arra, Claudio; Grieco, Paolo; Carriero, Maria Vincenza
Urotensin II(4-11) Azasulfuryl Peptides: Synthesis and Biological Activity
2016 Merlino, Francesco; Yousif, ALI MUNAIM; Billard, Étienne; Dufour Gallant, Julien; Turcotte, Stéphane; Grieco, Paolo; Chatenet, David; Lubell, William D.
Screening Platform toward New Anti-HIV Aptamers Set on Molecular Docking and Fluorescence Quenching Techniques
2016 Oliviero, G; Stornaiuolo, M; D'Atri, V; Nici, F; Yousif, Am; D'Errico, S; Piccialli, G; Mayol, L; Novellino, E; Marinelli, L; Grieco, P; Carotenuto, A; Noppen, S; Liekens, S; Balzarini, J; Borbone, N
Screening Platform toward New Anti-HIV Aptamers Set on Molecular Docking and Fluorescence Quenching Techniques
2016 Oliviero, Giorgia; Stornaiuolo, Mariano; D'Atri, Valentina; Nici, Fabrizia; Yousif, ALI MUNAIM; D'Errico, Stefano; Piccialli, Gennaro; Mayol, Luciano; Novellino, Ettore; Marinelli, Luciana; Grieco, Paolo; Carotenuto, Alfonso; Noppen, Sam; Liekens, Sandra; Balzarini, Jan; Borbone, Nicola
Cyclization of the urokinase receptor-derived Ser-Arg-Ser-Arg-Tyr peptide generates a potent inhibitor of trans-endothelial migration of monocytes
2015 Yousif, ALI MUNAIM; Minopoli, Michele; Bifulco, Katia; Ingangi, Vincenzo; Di Carluccio, Gioconda; Merlino, Francesco; Motti, MARIA LETIZIA; Grieco, Paolo; Carriero, Maria Vincenza
An investigation into the origin of the biased agonism associated with the urotensin II receptor activation
2015 Brancaccio, Diego; Merlino, Francesco; Limatola, Antonio; Yousif, ALI MUNAIM; GOMEZ MONTERREY, ISABEL MARIA; Campiglia, Pietro; Novellino, Ettore; Grieco, Paolo; Carotenuto, Alfonso
Discovery of Novel Potent and Selective Agonists at the Melanocortin-3 Receptor
2015 Carotenuto, Alfonso; Merlino, Francesco; Cai, Minying; Brancaccio, Diego; Yousif, ALI MUNAIM; Novellino, Ettore; Hruby, Victor J.; Grieco, Paolo
Urotensin II receptor determines prognosis of bladder cancer regulating cell motility/invasion
2014 Renato, Franco; Silvia, Zappavigna; Vincenzo, Gigantino; Amalia, Luce; Monica, Cantile; Margherita, Cerrone; Gaetano, Facchini; Sisto, Perdonà; Sandro, Pignata; Giuseppe Di, Lorenzo; Sergio, Chieffi; Giovanni, Vitale; Marco De, Sio; Alessandro, Sgambato; Gerardo, Botti; Yousif, ALI MUNAIM; Novellino, Ettore; Grieco, Paolo; Michele, Caraglia
Lead Optimization of P5U and Urantide: Discovery of Novel Potent Ligands at the Urotensin-II Receptor
2014 Carotenuto, Alfonso; Auriemma, Luigia; Merlino, Francesco; Yousif, ALI MUNAIM; Marasco, Daniela; Limatola, Antonio; Pietro, Campiglia; GOMEZ MONTERREY, ISABEL MARIA; Paolo, Santicioli; Stefania, Meini; Carlo A., Maggi; Novellino, Ettore; Grieco, Paolo
Urotensin-II Ligands: An Overview from Peptide to Nonpeptide Structures
2013 Merlino, Francesco; DI MARO, Salvatore; Yousif, ALI MUNAIM; Michele, Caraglia; Grieco, Paolo
Design, synthesis, and conformational analysis of Melanotropin analogues of MTII and SHU9119.
2013 Grieco, Paolo; Yousif, ALI MUNAIM; Carotenuto, Alfonso; Limatola, Antonio; Brancaccio, Diego; Novellino, Ettore; V. J., Hruby
Discovery of New Potent Ligands at Human Urotensin-II Receptor
2013 Yousif, ALI MUNAIM; Merlino, Francesco; Carotenuto, Alfonso; Limatola, Antonio; Paolo, Santicioli; Campiglia, Pietro; Meini, Stefania; Maggi Carlo, A.; Novellino, Ettore; Grieco, Paolo
Titolo | Tipologia | Data di pubblicazione | Autore(i) | File |
---|---|---|---|---|
Functional Selectivity Revealed by N-Methylation Scanning of Human Urotensin II and Related Peptides | 1.1 Articolo in rivista | 2019 | Merlino, Francesco; Billard, Etienne; Yousif, Ali Munaim; Di Maro, Salvatore; Brancaccio, Diego; Abate, Luigi; Carotenuto, Alfonso; Bellavita, Rosa; d'Emmanuele di Villa Bianca, Roberta; Santicioli, Paolo; Marinelli, Luciana; Novellino, Ettore; Hébert, Terence; Lubell, William D; Chatenet, David; Grieco, Paolo | |
Urotensin-II-Targeted Liposomes as a New Drug Delivery System towards Prostate and Colon Cancer Cells | 1.1 Articolo in rivista | 2019 | Zappavigna, S.; Abate, M.; Cossu, A. M.; Lusa, S.; Campani, V.; Scotti, L.; Luce, A.; Yousif, A. M.; Merlino, F.; Grieco, P.; De Rosa, G.; Caraglia, M. | |
Boosting Fmoc Solid-Phase Peptide Synthesis by Ultrasonication | 1.1 Articolo in rivista | 2019 | Merlino, F.; Tomassi, S.; Yousif, A. M.; Messere, A.; Marinelli, L.; Grieco, P.; Novellino, E.; Cosconati, S.; Di Maro, S. | |
Urokinase receptor derived peptides as potent inhibitors of the formyl peptide receptor type 1-triggered cell migration | 1.1 Articolo in rivista | 2018 | Yousif, Ali Munaim; Ingangi, Vincenzo; Merlino, Francesco; Brancaccio, Diego; Minopoli, Michele; Bellavita, Rosa; Novellino, Ettore; Carriero, Maria Vincenza; Carotenuto, Alfonso; Grieco, Paolo | |
Development of Macrocyclic Peptidomimetics Containing Constrained α,α-Dialkylated Amino Acids with Potent and Selective Activity at Human Melanocortin Receptors | 1.1 Articolo in rivista | 2018 | Merlino, Francesco; Zhou, Yang; Cai, Minying; Carotenuto, Alfonso; Yousif, Ali M; Brancaccio, Diego; Di Maro, Salvatore; Zappavigna, Silvia; Limatola, Antonio; Novellino, Ettore; Grieco, Paolo; Hruby, Victor J | |
Glycine-replaced derivatives of [Pro3,DLeu9]TL, a temporin L analogue: Evaluation of antimicrobial, cytotoxic and hemolytic activities | 1.1 Articolo in rivista | 2017 | Merlino, Francesco; Carotenuto, Alfonso; Casciaro, Bruno; Martora, Francesca; Loffredo, Maria Rosa; Di Grazia, Antonio; Yousif, Ali M.; Brancaccio, Diego; Palomba, Luciana; Novellino, Ettore; Galdiero, Massimiliano; Iovene, Maria Rosaria; Mangoni, Maria L.; Grieco, Paolo | |
Structure-Activity Study of the Peptides P5U and Urantide by the Development of Analogues Containing Uncoded Amino Acids at Position9 | 1.1 Articolo in rivista | 2016 | Merlino, Francesco; Brancaccio, Diego; Yousif, ALI MUNAIM; Piras, Linda; Campiglia, Pietro; GOMEZ MONTERREY, ISABEL MARIA; Santicioli, Paolo; Meini, Stefania; Maggi, Carlo A.; Novellino, Ettore; Carotenuto, Alfonso; Grieco, Paolo | |
Treatment with a Urokinase Receptor-derived Cyclized Peptide Improves Experimental Colitis by Preventing Monocyte Recruitment and Macrophage Polarization | 1.1 Articolo in rivista | 2016 | Genua, Marco; Ingangi, Vincenzo; Fonteyne, Philippe; Piontini, Andrea; Yousif, ALI MUNAIM; Merlino, Francesco; Grieco, Paolo; Malesci, Alberto; Carriero, Maria V; Danese, Silvio | |
The urokinase receptor-derived cyclic peptide [SRSRY] suppresses neovascularization and intravasation of osteosarcoma and chondrosarcoma cells | 1.1 Articolo in rivista | 2016 | Ingangi, Vincenzo; Bifulco, Katia; Yousif, ALI MUNAIM; Ragone, Concetta; Motti, MARIA LETIZIA; Rea, Domenica; Minopoli, Michele; Botti, Giovanni; Scognamiglio, Giuseppe; Fazioli, Flavio; Gallo, Michele; De Chiara, Annarosaria; Arra, Claudio; Grieco, Paolo; Carriero, Maria Vincenza | |
Urotensin II(4-11) Azasulfuryl Peptides: Synthesis and Biological Activity | 1.1 Articolo in rivista | 2016 | Merlino, Francesco; Yousif, ALI MUNAIM; Billard, Étienne; Dufour Gallant, Julien; Turcotte, Stéphane; Grieco, Paolo; Chatenet, David; Lubell, William D. | |
Screening Platform toward New Anti-HIV Aptamers Set on Molecular Docking and Fluorescence Quenching Techniques | 1.1 Articolo in rivista | 2016 | Oliviero, G; Stornaiuolo, M; D'Atri, V; Nici, F; Yousif, Am; D'Errico, S; Piccialli, G; Mayol, L; Novellino, E; Marinelli, L; Grieco, P; Carotenuto, A; Noppen, S; Liekens, S; Balzarini, J; Borbone, N | |
Screening Platform toward New Anti-HIV Aptamers Set on Molecular Docking and Fluorescence Quenching Techniques | 1.1 Articolo in rivista | 2016 | Oliviero, Giorgia; Stornaiuolo, Mariano; D'Atri, Valentina; Nici, Fabrizia; Yousif, ALI MUNAIM; D'Errico, Stefano; Piccialli, Gennaro; Mayol, Luciano; Novellino, Ettore; Marinelli, Luciana; Grieco, Paolo; Carotenuto, Alfonso; Noppen, Sam; Liekens, Sandra; Balzarini, Jan; Borbone, Nicola | |
Cyclization of the urokinase receptor-derived Ser-Arg-Ser-Arg-Tyr peptide generates a potent inhibitor of trans-endothelial migration of monocytes | 1.1 Articolo in rivista | 2015 | Yousif, ALI MUNAIM; Minopoli, Michele; Bifulco, Katia; Ingangi, Vincenzo; Di Carluccio, Gioconda; Merlino, Francesco; Motti, MARIA LETIZIA; Grieco, Paolo; Carriero, Maria Vincenza | |
An investigation into the origin of the biased agonism associated with the urotensin II receptor activation | 1.1 Articolo in rivista | 2015 | Brancaccio, Diego; Merlino, Francesco; Limatola, Antonio; Yousif, ALI MUNAIM; GOMEZ MONTERREY, ISABEL MARIA; Campiglia, Pietro; Novellino, Ettore; Grieco, Paolo; Carotenuto, Alfonso | |
Discovery of Novel Potent and Selective Agonists at the Melanocortin-3 Receptor | 1.1 Articolo in rivista | 2015 | Carotenuto, Alfonso; Merlino, Francesco; Cai, Minying; Brancaccio, Diego; Yousif, ALI MUNAIM; Novellino, Ettore; Hruby, Victor J.; Grieco, Paolo | |
Urotensin II receptor determines prognosis of bladder cancer regulating cell motility/invasion | 1.1 Articolo in rivista | 2014 | Renato, Franco; Silvia, Zappavigna; Vincenzo, Gigantino; Amalia, Luce; Monica, Cantile; Margherita, Cerrone; Gaetano, Facchini; Sisto, Perdonà; Sandro, Pignata; Giuseppe Di, Lorenzo; Sergio, Chieffi; Giovanni, Vitale; Marco De, Sio; Alessandro, Sgambato; Gerardo, Botti; Yousif, ALI MUNAIM; Novellino, Ettore; Grieco, Paolo; Michele, Caraglia | |
Lead Optimization of P5U and Urantide: Discovery of Novel Potent Ligands at the Urotensin-II Receptor | 1.1 Articolo in rivista | 2014 | Carotenuto, Alfonso; Auriemma, Luigia; Merlino, Francesco; Yousif, ALI MUNAIM; Marasco, Daniela; Limatola, Antonio; Pietro, Campiglia; GOMEZ MONTERREY, ISABEL MARIA; Paolo, Santicioli; Stefania, Meini; Carlo A., Maggi; Novellino, Ettore; Grieco, Paolo | |
Urotensin-II Ligands: An Overview from Peptide to Nonpeptide Structures | 1.1 Articolo in rivista | 2013 | Merlino, Francesco; DI MARO, Salvatore; Yousif, ALI MUNAIM; Michele, Caraglia; Grieco, Paolo | |
Design, synthesis, and conformational analysis of Melanotropin analogues of MTII and SHU9119. | 4.1 Articoli in Atti di convegno | 2013 | Grieco, Paolo; Yousif, ALI MUNAIM; Carotenuto, Alfonso; Limatola, Antonio; Brancaccio, Diego; Novellino, Ettore; V. J., Hruby | |
Discovery of New Potent Ligands at Human Urotensin-II Receptor | 1.5 Abstract in rivista | 2013 | Yousif, ALI MUNAIM; Merlino, Francesco; Carotenuto, Alfonso; Limatola, Antonio; Paolo, Santicioli; Campiglia, Pietro; Meini, Stefania; Maggi Carlo, A.; Novellino, Ettore; Grieco, Paolo |
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