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Synthesis, biological evaluation and molecular modeling of novel selective COX-2 inhibitors: sulfide, sulfoxide, and sulfone derivatives of 1,5-diarylpyrrol-3-substituted scaffold 1.1 Articolo in rivista 2019 Reale, A.; Brogi, S.; Chelini, A.; Paolino, M.; Di Capua, A.; Giuliani, G.; Cappelli, A.; Giorgi, G.; Chemi, G.; Grillo, A.; Valoti, M.; Sautebin, L.; Rossi, A.; Pace, S.; La Motta, C.; Di Cesare Mannelli, L.; Lucarini, E.; Ghelardini, C.; Anzini, M.
Gliotoxin from Aspergillus fumigatus Abrogates Leukotriene B4 Formation through Inhibition of Leukotriene A4 Hydrolase 1.1 Articolo in rivista 2019 König, Stefanie; Pace, Simona; Pein, Helmut; Heinekamp, Thorsten; Kramer, Jan; Romp, Erik; Straßburger, Maria; Troisi, Fabiana; Proschak, Anna; Dworschak, Jan; Scherlach, Kirstin; Rossi, Antonietta; Sautebin, Lidia; Haeggström, Jesper Z; Hertweck, Christian; Brakhage, Axel A; Gerstmeier, Jana; Proschak, Ewgenij; Werz, Oliver
Endogenous metabolites of vitamin E limit inflammation by targeting 5-lipoxygenase 1.1 Articolo in rivista 2018 Pein, Helmut; Ville, Alexia; Pace, Simona; Temml, Veronika; Garscha, Ulrike; Raasch, Martin; Alsabil, Khaled; Viault, Guillaume; Dinh, Chau-Phi; Guilet, David; Troisi, Fabiana; Neukirch, Konstantin; König, Stefanie; Bilancia, Rosella; Waltenberger, Birgit; Stuppner, Hermann; Wallert, Maria; Lorkowski, Stefan; Weinigel, Christina; Rummler, Silke; Birringer, Marc; Roviezzo, Fiorentina; Sautebin, Lidia; Helesbeux, Jean-Jacques; Séraphin, Denis; Mosig, Alexander S.; Schuster, Daniela; Rossi, Antonietta; Richomme, Pascal; Werz, Oliver; Koeberle, Andreas
Sex differences in prostaglandin biosynthesis in neutrophils during acute inflammation 1.1 Articolo in rivista 2017 Pace, Simona; Rossi, Antonietta; Krauth, Verena; Dehm, Friederike; Troisi, Fabiana; Bilancia, Rossella; Weinigel, Christina; Rummler, Silke; Werz, Oliver; Sautebin, Lidia
Pharmacological profile and efficiency in vivo of diflapolin, the first dual inhibitor of 5-lipoxygenase-activating protein and soluble epoxide hydrolase 1.1 Articolo in rivista 2017 Garscha, Ulrike; Romp, Erik; Pace, Simona; Rossi, Antonietta; Temml, Veronika; Schuster, Daniela; Kã¶nig, Stefanie; Gerstmeier, Jana; Liening, Stefanie; Werner, Markus; Atze, Heiner; Wittmann, Sandra; Weinigel, Christina; Rummler, Silke; Scriba, Gerhard K.; Sautebin, Lidia; Werz, Oliver
Sex-biased eicosanoid biology: impact for sex differences in inflammation and consequences for pharmacotherapy 1.1 Articolo in rivista 2017 Pace, Simona; Sautebin, Lidia; Werz, Oliver
Evaluation of Dual 5-Lipoxygenase/Microsomal Prostaglandin E2 Synthase-1 Inhibitory Effect of Natural and Synthetic Acronychia-Type Isoprenylated Acetophenones 1.1 Articolo in rivista 2017 Svouraki, Alexandra; Garscha, Ulrike; Kouloura, Eirini; Pace, Simona; Pergola, Carlo; Krauth, Verena; Rossi, Antonietta; Sautebin, Lidia; Halabalaki, Maria; Werz, Oliver; Gaboriaud Kolar, Nicolas; Skaltsounis, Alexios Leandros
Androgen-mediated sex bias impairs efficiency of leukotriene biosynthesis inhibitors in males 1.1 Articolo in rivista 2017 Pace, Simona; Pergola, Carlo; Dehm, Friederike; Rossi, Antonietta; Gerstmeier, Jana; Troisi, Fabiana; Pein, Helmut; Schaible, Anja M.; Weinigel, Christina; Rummler, Silke; Northoff, Hinnak; Laufer, Stefan; Maier, Thorsten J.; Rådmark, Olof; Samuelsson, Bengt; Koeberle, Andreas; Sautebin, Lidia; Werz, Oliver
Vitamin A regulates Akt signaling through the phospholipid fatty acid composition 1.1 Articolo in rivista 2017 Pein, Helmut; Koeberle, Solveigh C.; Voelkel, Maria; Schneider, Freya; Rossi, Antonietta; Thürmer, Maria; Loeser, Konstantin; Sautebin, Lidia; Morrison, Helen; Werz, Oliver; Koeberle, Andreas
Capitolo 42 del Trattato di Farmacologia. Farmaci per la terapia della gotta 2.1 Contributo in volume (Capitolo o Saggio) 2016 Sautebin, Lidia; Rossi, Antonietta
BRP-187: A potent inhibitor of leukotriene biosynthesis that acts through impeding the dynamic 5-lipoxygenase/5-lipoxygenase-activating protein (FLAP) complex assembly 1.1 Articolo in rivista 2016 Garscha, Ulrike; Voelker, Susanna; Pace, Simona; Gerstmeier, Jana; Emini, Besa; Liening, Stefanie; Rossi, Antonietta; Weinigel, Christina; Rummler, Silke; Schubert, Ulrich S; Scriba, Gerhard K. E; Çelikoğlu, Erşan; Çalışkan, Burcu; Banoglu, Erden; Sautebin, Lidia; Werz, Oliver
Synthesis and biological evaluation of fluorinated 1,5-diarylpyrrole-3-alkoxyethyl ether derivatives as selective COX-2 inhibitors endowed with anti-inflammatory activity 1.1 Articolo in rivista 2016 Di Capua, Angela; Sticozzi, Claudia; Brogi, Simone; Brindisi, Margherita; Cappelli, Andrea; Sautebin, Lidia; Rossi, Antonietta; Pace, Simona; Ghelardini, Carla; Di Cesare Mannelli, Lorenzo; Valacchi, Giuseppe; Giorgi, Gianluca; Giordani, Antonio; Poce, Giovanna; Biava, Mariangela; Anzini, Maurizio
Use of Mometasone furoate in prolonged treatment of experimental spinal cord injury in mice: A comparative study of three different glucocorticoids 1.1 Articolo in rivista 2015 Galuppo, Maria; Rossi, Antonietta; Giacoppo, Sabrina; Pace, Simona; Bramanti, Placido; Sautebin, Lidia; Mazzon, Emanuela
SAR Studies on Curcumin's Pro-inflammatory Targets: Discovery of Prenylated Pyrazolocurcuminoids as Potent and Selective Novel Inhibitors of 5-Lipoxygenase. 1.1 Articolo in rivista 2014 Koeberle, A; Muñoz, E; Appendino, Gb; Minassi, A; Pace, Simona; Rossi, Antonietta; Weinigel, C; Barz, D; Sautebin, Lidia; Caprioglio, D; Collado, Ja; Werz, O.
The novel benzimidazole derivative BRP-7 inhibits leukotriene biosynthesis in vitro and in vivo by targeting 5-lipoxygenase-activating protein (FLAP). 1.1 Articolo in rivista 2014 Pergola, C; Gerstmeier, J; Mönch, B; Çalışkan, B; Luderer, S; Weinigel, C; Barz, D; Maczewsky, J; Pace, Simona; Rossi, Antonietta; Sautebin, Lidia; Banoglu, E; Werz, O.
Enhancing the pharmacodynamic profile of a class of selective COX-2 inhibiting nitric oxide donors. 1.1 Articolo in rivista 2014 Biava, M; Battilocchio, C; Poce, G; Alfonso, S; Consalvi, S; Di Capua, A; Calderone, V; Martelli, A; Testai, L; Sautebin, Lidia; Rossi, Antonietta; Ghelardini, C; Di Cesare Mannelli, L; Giordani, A; Persiani, S; Colovic, M; Dovizio, M; Patrignani, P; Anzini, M.
In vivo sex differences in leukotriene biosynthesis in zymosan-induced peritonitis. 1.1 Articolo in rivista 2014 Rossi, Antonietta; Pergola, C; Pace, Simona; Rådmark, O; Werz, O; Sautebin, Lidia
BRP-7, a novel benzimidazole-based chemotype targeting 5-lipoxygenase-activating protein, inhibits leukotriene biosynthesis in experimental models of acute inflammation in vivo. 4.2 Abstract in Atti di convegno 2013 Rossi, Antonietta; Maczewsky, J.; Pace, Simona; Pergola, C; Çalışkan, B; Banoglu, E; Werz, O; Sautebin, Lidia
“Il nuovo sistema di Cosmetovigilanza secondo il Regolamento 1223/2009: le iniziative del Ministero della Salute” 8.02 Comunicazioni a Convegni o Seminari 2013 Sautebin, Lidia
In vivo differences in leukotriene biosynthesis in zymosan-induced peritonitis: role of resident peritoneal macrophages. 4.2 Abstract in Atti di convegno 2013 Rossi, Antonietta; Pace, Simona; Pergola, C; Maczewsky, J; Rǻdmark, O; Samuelsson, B; Werz, O; Sautebin, Lidia
Mostrati risultati da 1 a 20 di 183
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