Sfoglia per Autore
Theonella: A Treasure Trove of Structurally Unique and Biologically Active Sterols
2023 Festa, Carmen; DE MARINO, Simona; Zampella, Angela; Fiorucci, Stefano
Expanding the Library of 1,2,4-Oxadiazole Derivatives: Discovery of New Farnesoid X Receptor (FXR) Antagonists/Pregnane X Receptor (PXR) Agonists
2023 Finamore, Claudia; Festa, Carmen; Fiorillo, Bianca; Di Leva, Francesco Saverio; Roselli, Rosalinda; Marchianò, Silvia; Biagioli, Michele; Spinelli, Lucio; Fiorucci, Stefano; Limongelli, Vittorio; Zampella, Angela; DE MARINO, Simona
Guest Editor
2022 DE MARINO, Simona
Phytochemical Analysis of the Methanolic Extract and Essential Oil from Leaves of Industrial Hemp Futura 75 Cultivar: Isolation of a New Cannabinoid Derivative and Biological Profile Using Computational Approaches
2022 De Vita, Simona; Finamore, Claudia; Chini, Maria Giovanna; Saviano, Gabriella; De Felice, Vincenzo; De Marino, Simona; Lauro, Gianluigi; Casapullo, Agostino; Fantasma, Francesca; Trombetta, Federico; Bifulco, Giuseppe; Iorizzi, Maria
Discovering New G-Quadruplex DNA Catalysts in Enantioselective Sulfoxidation Reaction
2022 Festa, Carmen; Esposito, Veronica; Benigno, Daniela; DE MARINO, Simona; Zampella, Angela; Virgilio, Antonella; Galeone, Aldo
“Discovery of promising 1,2,4-oxadiazoles hits for the development of new anti-inflammatory agents interfering with eicosanoid biosynthesis pathways”
2021 Sciarretta, M; Potenza, M; Festa, C; Maione, F; Saviano, A; Chini, Mg; De Marino, S; D’Auria, Mv; Werz, O; Bifulco, G
Synergistic activity of a synthetic 1,2,4-oxadiazole-containing derivative and oxacillin against methicillin-resistant Staphylococcus aureus
2021 Buommino, Elisabetta; Sciarretta, Martina; Festa, Carmen; DE ROSA, Adriana; Piccolo, Marialuisa; DE MARINO, Simona; Maria, ; D’Auria., V.
Structure-based screening for the discovery of 1,2,4-oxadiazoles as promising hits for the development of new anti-inflammatory agents interfering with eicosanoid biosyn-thesis pathways
2021 Sciarretta, Martina; Saviano, Anella; Maione, Francesco; D'Auria, MARIA VALERIA; DE MARINO, Simona; Giordano, Assunta; Festa, Carmen
Biological Profile of Two Gentiana lutea L. Metabolites Using Computational Approaches and In Vitro Tests
2021 Finamore, Claudia; Festa, Carmen; DE MARINO, Simona; Russo, Roberto; Avagliano, Carmen; Calignano, Antonio
Synergism of a novel 1,2,4-oxadiazole-containing derivative with oxacillin against methicillin-resistant Staphylococcus aureus
2021 Buommino, Elisabetta; DE MARINO, Simona; Sciarretta, Martina; Piccolo, Marialuisa; Festa, Carmen; D'Auria, MARIA VALERIA
Design and synthesis of new potential inhibitors of proteins relevant to cancer insurgence.
2020 Sciarretta, M.; Potenza, M.; Festa, C.; Chini, M. G.; De Marino, S.; D’Auria, M. V.; Werz, O.; Bifulco, G.
Design and synthesis of hyodeoxycholic acid derivatives as GPBAR1 receptor modulators useful in the treatment of colon inflammation
2020 Finamore, C.; De Marino, S.; Cassiano, C.; Di Leva, F. S.; Limongelli, V.; Zampella, A.; Fiorucci, S.; Festa, C.
GPBAR1 activation by C6-substituted hyodeoxycholane analogues protect against colitis
2020 De Marino, S.; Finamore, C.; Biagioli, M.; Carino, A.; Marchiano, S.; Roselli, R.; Di Giorgio, C.; Bordoni, M.; Di Leva, F. S.; Novellino, E.; Cassiano, C.; Limongelli, V.; Zampella, A.; Festa, C.; Fiorucci, S.
Synthesis of new oxadiazole derivatives as potent and selective FXR antagonists
2019 Festa, Carmen; Finamore, Claudia; Di Leva, Francesco Saverio; Limongelli, Vittorio; Zampella, Angela; DE MARINO, Simona
Synthesis of new isoxazole derivatives as fxr agonists with improved pharmacokinetic properties
2019 Finamore, C.; Sepe, V.; Baronissi, G.; Cassiano, C.; Monti, M. C.; De Marino, S.; Novellino, E.; Limongelli, V.; Fiorucci, S.; Zampella, A.
Discovery of ((1,2,4-oxadiazol-5-yl)pyrrolidin-3-yl)ureidyl derivatives as selective non-steroidal agonists of the G-protein coupled bile acid receptor-1
2019 Di Leva, Francesco Saverio; Festa, Carmen; Carino, Adriana; De Marino, Simona; Marchianò, Silvia; Di Marino, Daniele; Finamore, Claudia; Monti, Maria Chiara; Zampella, Angela; Fiorucci, Stefano; Limongelli, Vittorio
Wound healing activity and phytochemical screening of purified fractions of Sempervivum tectorum L. leaves on HCT 116
2019 Cattaneo, Fabio; DE MARINO, Simona; Parisi, Melania; Festa, Carmen; Castaldo, Martina; Finamore, Claudia; Duraturo, Francesca; Zollo, Cristiana; Ammendola, Rosario; Zollo, Franco; Iorizzi, Maria
Phytochemical and biological studies of Nepeta asterotricha Rech. f. (Lamiaceae): Isolation of Nepetamoside
2019 Mostafa Goldansaz, Seyed; Festa, Carmen; Pagano, Ester; DE MARINO, Simona; Finamore, Claudia; Parisi, OLGA ALESSANDRA; Borrelli, Francesca; Sonboli, Ali; D'Auria, MARIA VALERIA
Chemistry and Pharmacology of GPBAR1 and FXR Selective Agonists, Dual Agonists, and Antagonists
2019 DE MARINO, Simona; Festa, Carmen; Sepe, Valentina; Zampella, Angela
Investigation around the Oxadiazole Core in the Discovery of a New Chemotype of Potent and Selective FXR Antagonists
2019 Festa, Carmen; Finamore, Claudia; Silvia Marchiano, †; Di Leva, Francesco Saverio; Carino, Adriana; Chiara Monti, Maria; del Gaudio, Federica; Ceccacci, Sara; Limongelli, Vittorio; Zampella, Angela; Fiorucci, Stefano; DE MARINO, Simona
Titolo | Tipologia | Data di pubblicazione | Autore(i) | File |
---|---|---|---|---|
Theonella: A Treasure Trove of Structurally Unique and Biologically Active Sterols | 1.1 Articolo in rivista | 2023 | Festa, Carmen; DE MARINO, Simona; Zampella, Angela; Fiorucci, Stefano | |
Expanding the Library of 1,2,4-Oxadiazole Derivatives: Discovery of New Farnesoid X Receptor (FXR) Antagonists/Pregnane X Receptor (PXR) Agonists | 1.1 Articolo in rivista | 2023 | Finamore, Claudia; Festa, Carmen; Fiorillo, Bianca; Di Leva, Francesco Saverio; Roselli, Rosalinda; Marchianò, Silvia; Biagioli, Michele; Spinelli, Lucio; Fiorucci, Stefano; Limongelli, Vittorio; Zampella, Angela; DE MARINO, Simona | |
Guest Editor | 8.06 Partecip. Editorial Board di riviste scientifiche | 2022 | DE MARINO, Simona | |
Phytochemical Analysis of the Methanolic Extract and Essential Oil from Leaves of Industrial Hemp Futura 75 Cultivar: Isolation of a New Cannabinoid Derivative and Biological Profile Using Computational Approaches | 1.1 Articolo in rivista | 2022 | De Vita, Simona; Finamore, Claudia; Chini, Maria Giovanna; Saviano, Gabriella; De Felice, Vincenzo; De Marino, Simona; Lauro, Gianluigi; Casapullo, Agostino; Fantasma, Francesca; Trombetta, Federico; Bifulco, Giuseppe; Iorizzi, Maria | |
Discovering New G-Quadruplex DNA Catalysts in Enantioselective Sulfoxidation Reaction | 1.1 Articolo in rivista | 2022 | Festa, Carmen; Esposito, Veronica; Benigno, Daniela; DE MARINO, Simona; Zampella, Angela; Virgilio, Antonella; Galeone, Aldo | |
“Discovery of promising 1,2,4-oxadiazoles hits for the development of new anti-inflammatory agents interfering with eicosanoid biosynthesis pathways” | 4.2 Abstract in Atti di convegno | 2021 | Sciarretta, M; Potenza, M; Festa, C; Maione, F; Saviano, A; Chini, Mg; De Marino, S; D’Auria, Mv; Werz, O; Bifulco, G | |
Synergistic activity of a synthetic 1,2,4-oxadiazole-containing derivative and oxacillin against methicillin-resistant Staphylococcus aureus | 4.2 Abstract in Atti di convegno | 2021 | Buommino, Elisabetta; Sciarretta, Martina; Festa, Carmen; DE ROSA, Adriana; Piccolo, Marialuisa; DE MARINO, Simona; Maria, ; D’Auria., V. | |
Structure-based screening for the discovery of 1,2,4-oxadiazoles as promising hits for the development of new anti-inflammatory agents interfering with eicosanoid biosyn-thesis pathways | 1.1 Articolo in rivista | 2021 | Sciarretta, Martina; Saviano, Anella; Maione, Francesco; D'Auria, MARIA VALERIA; DE MARINO, Simona; Giordano, Assunta; Festa, Carmen | |
Biological Profile of Two Gentiana lutea L. Metabolites Using Computational Approaches and In Vitro Tests | 1.1 Articolo in rivista | 2021 | Finamore, Claudia; Festa, Carmen; DE MARINO, Simona; Russo, Roberto; Avagliano, Carmen; Calignano, Antonio | |
Synergism of a novel 1,2,4-oxadiazole-containing derivative with oxacillin against methicillin-resistant Staphylococcus aureus | 1.1 Articolo in rivista | 2021 | Buommino, Elisabetta; DE MARINO, Simona; Sciarretta, Martina; Piccolo, Marialuisa; Festa, Carmen; D'Auria, MARIA VALERIA | |
Design and synthesis of new potential inhibitors of proteins relevant to cancer insurgence. | 4.2 Abstract in Atti di convegno | 2020 | Sciarretta, M.; Potenza, M.; Festa, C.; Chini, M. G.; De Marino, S.; D’Auria, M. V.; Werz, O.; Bifulco, G. | |
Design and synthesis of hyodeoxycholic acid derivatives as GPBAR1 receptor modulators useful in the treatment of colon inflammation | 4.2 Abstract in Atti di convegno | 2020 | Finamore, C.; De Marino, S.; Cassiano, C.; Di Leva, F. S.; Limongelli, V.; Zampella, A.; Fiorucci, S.; Festa, C. | |
GPBAR1 activation by C6-substituted hyodeoxycholane analogues protect against colitis | 1.1 Articolo in rivista | 2020 | De Marino, S.; Finamore, C.; Biagioli, M.; Carino, A.; Marchiano, S.; Roselli, R.; Di Giorgio, C.; Bordoni, M.; Di Leva, F. S.; Novellino, E.; Cassiano, C.; Limongelli, V.; Zampella, A.; Festa, C.; Fiorucci, S. | |
Synthesis of new oxadiazole derivatives as potent and selective FXR antagonists | 8.02 Comunicazioni a Convegni o Seminari | 2019 | Festa, Carmen; Finamore, Claudia; Di Leva, Francesco Saverio; Limongelli, Vittorio; Zampella, Angela; DE MARINO, Simona | |
Synthesis of new isoxazole derivatives as fxr agonists with improved pharmacokinetic properties | 4.2 Abstract in Atti di convegno | 2019 | Finamore, C.; Sepe, V.; Baronissi, G.; Cassiano, C.; Monti, M. C.; De Marino, S.; Novellino, E.; Limongelli, V.; Fiorucci, S.; Zampella, A. | |
Discovery of ((1,2,4-oxadiazol-5-yl)pyrrolidin-3-yl)ureidyl derivatives as selective non-steroidal agonists of the G-protein coupled bile acid receptor-1 | 1.1 Articolo in rivista | 2019 | Di Leva, Francesco Saverio; Festa, Carmen; Carino, Adriana; De Marino, Simona; Marchianò, Silvia; Di Marino, Daniele; Finamore, Claudia; Monti, Maria Chiara; Zampella, Angela; Fiorucci, Stefano; Limongelli, Vittorio | |
Wound healing activity and phytochemical screening of purified fractions of Sempervivum tectorum L. leaves on HCT 116 | 1.1 Articolo in rivista | 2019 | Cattaneo, Fabio; DE MARINO, Simona; Parisi, Melania; Festa, Carmen; Castaldo, Martina; Finamore, Claudia; Duraturo, Francesca; Zollo, Cristiana; Ammendola, Rosario; Zollo, Franco; Iorizzi, Maria | |
Phytochemical and biological studies of Nepeta asterotricha Rech. f. (Lamiaceae): Isolation of Nepetamoside | 1.1 Articolo in rivista | 2019 | Mostafa Goldansaz, Seyed; Festa, Carmen; Pagano, Ester; DE MARINO, Simona; Finamore, Claudia; Parisi, OLGA ALESSANDRA; Borrelli, Francesca; Sonboli, Ali; D'Auria, MARIA VALERIA | |
Chemistry and Pharmacology of GPBAR1 and FXR Selective Agonists, Dual Agonists, and Antagonists | 2.1 Contributo in volume (Capitolo o Saggio) | 2019 | DE MARINO, Simona; Festa, Carmen; Sepe, Valentina; Zampella, Angela | |
Investigation around the Oxadiazole Core in the Discovery of a New Chemotype of Potent and Selective FXR Antagonists | 1.1 Articolo in rivista | 2019 | Festa, Carmen; Finamore, Claudia; Silvia Marchiano, †; Di Leva, Francesco Saverio; Carino, Adriana; Chiara Monti, Maria; del Gaudio, Federica; Ceccacci, Sara; Limongelli, Vittorio; Zampella, Angela; Fiorucci, Stefano; DE MARINO, Simona |
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